| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| OTHER | AAK1 | AAK1_MOUSE | 7RJ6A | Q3UHJ0 | 26 | 330 | 959.0 | YFV:401 | Type1 | Active | DFGin | 6.5122 | 13.3768 | BLAminus | -125.62, 169.71 | 67.71, 96.16 | -104.68, 24.3 | 300.02, 93.63 | -68.93, -22.4 | in-in | in | 8.5967 | Saltbr-in | 2.7099 | HRD-in | -65.12, -47.31 | 74.51, -5.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8935 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -105.26, -12.99 | APE9-dihe-na | -116.7, 155.82 | APE8-dihe-in | -97.42, 121.54 | APE8-rot-in | 304.46 | APE67-dihe-in | -58.17, -28.42 | -45.34, -49.66 | APE12-dist-in | 12.1363 | APE11-dist-in | 8.6182 | APE10-dist-in | 4.2728 | APE9-dist-in | 3.6627 | None | None | None | XRAY | 2.132 | 0.202 | 0.215 | A | 318.0 | 305.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj6 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| OTHER | AAK1 | AAK1_MOUSE | 7RJ6B | Q3UHJ0 | 32 | 330 | 959.0 | 5OI:401 | Type1 | Active | DFGin | 6.386 | 13.2644 | BLAminus | -136.98, -179.6 | 61.47, 90.79 | -102.58, 19.8 | 300.28, 93.44 | -74.01, -20.13 | in-in | in | 8.7043 | Saltbr-in | 2.7308 | HRD-in | -65.76, -48.0 | 74.66, -11.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8975 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.51, -10.49 | APE9-dihe-na | -120.36, 163.0 | APE8-dihe-in | -104.78, 122.31 | APE8-rot-in | 303.78 | APE67-dihe-in | -58.21, -28.47 | -45.49, -49.71 | APE12-dist-in | 11.9714 | APE11-dist-in | 8.4144 | APE10-dist-in | 4.1372 | APE9-dist-in | 3.7792 | None | None | None | XRAY | 2.132 | 0.202 | 0.215 | B | 318.0 | 299.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj6 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| OTHER | AAK1 | AAK1_MOUSE | 7RJ6A | Q3UHJ0 | 26 | 330 | 959.0 | YFV:401 | Type1 | Active | DFGin | 6.5122 | 13.3768 | BLAminus | -125.62, 169.71 | 67.71, 96.16 | -104.68, 24.3 | 300.02, 93.63 | -68.93, -22.4 | in-in | in | 8.5967 | Saltbr-in | 2.7099 | HRD-in | -65.12, -47.31 | 74.51, -5.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8935 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -105.26, -12.99 | APE9-dihe-na | -116.7, 155.82 | APE8-dihe-in | -97.42, 121.54 | APE8-rot-in | 304.46 | APE67-dihe-in | -58.17, -28.42 | -45.34, -49.66 | APE12-dist-in | 12.1363 | APE11-dist-in | 8.6182 | APE10-dist-in | 4.2728 | APE9-dist-in | 3.6627 | None | None | None | XRAY | 2.132 | 0.202 | 0.215 | A | 318.0 | 305.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj6 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| OTHER | AAK1 | AAK1_MOUSE | 7RJ6B | Q3UHJ0 | 32 | 330 | 959.0 | 5OI:401 | Type1 | Active | DFGin | 6.386 | 13.2644 | BLAminus | -136.98, -179.6 | 61.47, 90.79 | -102.58, 19.8 | 300.28, 93.44 | -74.01, -20.13 | in-in | in | 8.7043 | Saltbr-in | 2.7308 | HRD-in | -65.76, -48.0 | 74.66, -11.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8975 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.51, -10.49 | APE9-dihe-na | -120.36, 163.0 | APE8-dihe-in | -104.78, 122.31 | APE8-rot-in | 303.78 | APE67-dihe-in | -58.21, -28.47 | -45.49, -49.71 | APE12-dist-in | 11.9714 | APE11-dist-in | 8.4144 | APE10-dist-in | 4.1372 | APE9-dist-in | 3.7792 | None | None | None | XRAY | 2.132 | 0.202 | 0.215 | B | 318.0 | 299.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj6 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |