| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 7OZFAAA | P11362 | 465 | 765 | 822.0 | 466:801 | Type1 | Inactive | DFGin | 5.2955 | 13.468 | BLAplus | -117.68, 161.62 | 66.46, 36.41 | -95.38, -7.29 | 57.95, 82.09 | -95.91, -11.26 | in-in | in | 7.8017 | Saltbr-in | 3.0344 | HRD-in | -74.16, -54.6 | 82.1, -14.72 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -100.26, 162.73 | APE9-dihe-in | -101.57, 112.99 | APE8-dihe-out | -53.92, -25.84 | APE8-rot-na | 335.55 | APE67-dihe-in | -73.42, -8.15 | -56.91, -22.71 | APE12-dist-na | 20.3344 | APE11-dist-na | 21.6782 | APE10-dist-na | 20.2 | APE9-dist-out | 11.7273 | None | None | None | XRAY | 1.82 | 0.206 | 0.242 | AAA | 309.0 | 288.0 | 13 | 30 | 25 | 5 | [[478, 756]] | 1.0 | 7ozf | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 7OZFBBB | P11362 | 460 | 763 | 822.0 | 466:801 | Type1 | Inactive | DFGin | 5.2534 | 13.0233 | BLAplus | -116.0, 158.26 | 69.37, 33.48 | -90.88, -17.29 | 57.42, 83.97 | -77.99, -12.47 | in-in | in | 7.6429 | Saltbr-in | 2.9656 | HRD-in | -73.91, -57.88 | 84.04, -15.02 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -115.71, 160.57 | APE9-dihe-in | -98.6, 110.79 | APE8-dihe-out | -55.8, -24.65 | APE8-rot-na | 332.84 | APE67-dihe-in | -74.09, -8.17 | -55.72, -20.54 | APE12-dist-na | 20.458 | APE11-dist-na | 21.8593 | APE10-dist-na | 20.1777 | APE9-dist-out | 11.6515 | None | None | None | XRAY | 1.82 | 0.206 | 0.242 | BBB | 309.0 | 282.0 | 22 | 30 | 25 | 5 | [[478, 756]] | 1.0 | 7ozf | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 7OZFAAA | P11362 | 465 | 765 | 822.0 | 466:801 | Type1 | Inactive | DFGin | 5.2955 | 13.468 | BLAplus | -117.68, 161.62 | 66.46, 36.41 | -95.38, -7.29 | 57.95, 82.09 | -95.91, -11.26 | in-in | in | 7.8017 | Saltbr-in | 3.0344 | HRD-in | -74.16, -54.6 | 82.1, -14.72 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -100.26, 162.73 | APE9-dihe-in | -101.57, 112.99 | APE8-dihe-out | -53.92, -25.84 | APE8-rot-na | 335.55 | APE67-dihe-in | -73.42, -8.15 | -56.91, -22.71 | APE12-dist-na | 20.3344 | APE11-dist-na | 21.6782 | APE10-dist-na | 20.2 | APE9-dist-out | 11.7273 | None | None | None | XRAY | 1.82 | 0.206 | 0.242 | AAA | 309.0 | 288.0 | 13 | 30 | 25 | 5 | [[478, 756]] | 1.0 | 7ozf | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 7OZFBBB | P11362 | 460 | 763 | 822.0 | 466:801 | Type1 | Inactive | DFGin | 5.2534 | 13.0233 | BLAplus | -116.0, 158.26 | 69.37, 33.48 | -90.88, -17.29 | 57.42, 83.97 | -77.99, -12.47 | in-in | in | 7.6429 | Saltbr-in | 2.9656 | HRD-in | -73.91, -57.88 | 84.04, -15.02 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -115.71, 160.57 | APE9-dihe-in | -98.6, 110.79 | APE8-dihe-out | -55.8, -24.65 | APE8-rot-na | 332.84 | APE67-dihe-in | -74.09, -8.17 | -55.72, -20.54 | APE12-dist-na | 20.458 | APE11-dist-na | 21.8593 | APE10-dist-na | 20.1777 | APE9-dist-out | 11.6515 | None | None | None | XRAY | 1.82 | 0.206 | 0.242 | BBB | 309.0 | 282.0 | 22 | 30 | 25 | 5 | [[478, 756]] | 1.0 | 7ozf | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|