| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 7OZBAAA | P11362 | 464 | 765 | 822.0 | 47I:801 | Type1 | Inactive | DFGin | 5.1652 | 13.2255 | BLAplus | -113.5, 164.02 | 64.24, 28.44 | -81.1, -17.3 | 55.31, 86.35 | -99.81, -4.02 | in-in | in | 7.6783 | Saltbr-in | 3.0354 | HRD-in | -68.22, -55.33 | 81.75, -15.47 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6293 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.53, 159.74 | APE9-dihe-in | -101.43, 112.26 | APE8-dihe-out | -54.35, -25.93 | APE8-rot-na | 332.55 | APE67-dihe-in | -70.65, -7.52 | -55.15, -25.11 | APE12-dist-na | 19.2916 | APE11-dist-na | 20.7453 | APE10-dist-na | 19.1948 | APE9-dist-out | 11.6637 | C488A,C584S | None | None | XRAY | 1.71 | 0.211 | 0.244 | AAA | 309.0 | 288.0 | 14 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 7ozb | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 7OZBBBB | P11362 | 460 | 764 | 822.0 | 47I:801 | Type1 | Inactive | DFGin | 5.2201 | 12.8529 | BLAplus | -116.55, 158.6 | 67.07, 25.64 | -79.35, -20.91 | 57.12, 84.44 | -89.98, -6.37 | in-in | in | 7.6315 | Saltbr-in | 2.9829 | HRD-in | -68.5, -59.33 | 86.86, -18.0 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.1932 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -112.69, 159.38 | APE9-dihe-in | -99.92, 110.92 | APE8-dihe-out | -56.91, -22.49 | APE8-rot-na | 333.27 | APE67-dihe-in | -69.35, -9.22 | -56.3, -24.07 | APE12-dist-na | 19.5566 | APE11-dist-na | 20.9014 | APE10-dist-na | 19.3195 | APE9-dist-out | 11.5573 | C488A,C584S | None | None | XRAY | 1.71 | 0.211 | 0.244 | BBB | 309.0 | 291.0 | 14 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 7ozb | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 7OZBAAA | P11362 | 464 | 765 | 822.0 | 47I:801 | Type1 | Inactive | DFGin | 5.1652 | 13.2255 | BLAplus | -113.5, 164.02 | 64.24, 28.44 | -81.1, -17.3 | 55.31, 86.35 | -99.81, -4.02 | in-in | in | 7.6783 | Saltbr-in | 3.0354 | HRD-in | -68.22, -55.33 | 81.75, -15.47 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6293 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.53, 159.74 | APE9-dihe-in | -101.43, 112.26 | APE8-dihe-out | -54.35, -25.93 | APE8-rot-na | 332.55 | APE67-dihe-in | -70.65, -7.52 | -55.15, -25.11 | APE12-dist-na | 19.2916 | APE11-dist-na | 20.7453 | APE10-dist-na | 19.1948 | APE9-dist-out | 11.6637 | C488A,C584S | None | None | XRAY | 1.71 | 0.211 | 0.244 | AAA | 309.0 | 288.0 | 14 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 7ozb | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 7OZBBBB | P11362 | 460 | 764 | 822.0 | 47I:801 | Type1 | Inactive | DFGin | 5.2201 | 12.8529 | BLAplus | -116.55, 158.6 | 67.07, 25.64 | -79.35, -20.91 | 57.12, 84.44 | -89.98, -6.37 | in-in | in | 7.6315 | Saltbr-in | 2.9829 | HRD-in | -68.5, -59.33 | 86.86, -18.0 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.1932 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -112.69, 159.38 | APE9-dihe-in | -99.92, 110.92 | APE8-dihe-out | -56.91, -22.49 | APE8-rot-na | 333.27 | APE67-dihe-in | -69.35, -9.22 | -56.3, -24.07 | APE12-dist-na | 19.5566 | APE11-dist-na | 20.9014 | APE10-dist-na | 19.3195 | APE9-dist-out | 11.5573 | C488A,C584S | None | None | XRAY | 1.71 | 0.211 | 0.244 | BBB | 309.0 | 291.0 | 14 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 7ozb | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|