| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 6XVAA | P10721 | 569 | 931 | 976.0 | O2K:61001 | Type2 | Inactive | DFGout | 15.5521 | 9.8729 | BBAminus | -130.9, -166.53 | -160.13, 95.6 | -61.57, -39.69 | 279.99, 84.81 | 51.06, -112.95 | in-in | in | 7.6706 | Saltbr-in | 2.8122 | HRD-in | -65.74, -44.71 | 75.29, -12.36 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4556 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -123.89, 95.77 | APE9-dihe-in | -112.54, 151.67 | APE8-dihe-in | -83.56, 70.47 | APE8-rot-na | 31.96 | APE67-dihe-in | -64.92, -13.68 | -47.25, -45.59 | APE12-dist-na | 16.2504 | APE11-dist-na | 13.1008 | APE10-dist-na | 11.1871 | APE9-dist-in | 7.9038 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.3 | 0.198 | 0.245 | A | 328.0 | 285.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 6xva | TYR_KIT_HUMAN | TYR | 2.4e-104 | 354.2 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 6XVAB | P10721 | 577 | 931 | 976.0 | O2K:61001 | Type2 | Inactive | DFGout | 15.832 | 9.9461 | BBAminus | -129.58, -168.14 | -159.52, 95.6 | -60.13, -40.05 | 280.9, 81.98 | 51.8, -114.7 | in-in | in | 7.838 | Saltbr-in | 2.8735 | HRD-in | -67.63, -49.04 | 76.72, -12.76 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.2998 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -120.1, 96.88 | APE9-dihe-in | -113.3, 152.94 | APE8-dihe-in | -84.37, 70.57 | APE8-rot-na | 30.8 | APE67-dihe-in | -65.41, -13.28 | -47.31, -45.65 | APE12-dist-na | 16.5272 | APE11-dist-na | 13.1483 | APE10-dist-na | 11.3543 | APE9-dist-in | 7.935 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.3 | 0.198 | 0.245 | B | 328.0 | 277.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 6xva | TYR_KIT_HUMAN | TYR | 2.4e-104 | 354.2 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 6XVAA | P10721 | 569 | 931 | 976.0 | O2K:61001 | Type2 | Inactive | DFGout | 15.5521 | 9.8729 | BBAminus | -130.9, -166.53 | -160.13, 95.6 | -61.57, -39.69 | 279.99, 84.81 | 51.06, -112.95 | in-in | in | 7.6706 | Saltbr-in | 2.8122 | HRD-in | -65.74, -44.71 | 75.29, -12.36 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.4556 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -123.89, 95.77 | APE9-dihe-in | -112.54, 151.67 | APE8-dihe-in | -83.56, 70.47 | APE8-rot-na | 31.96 | APE67-dihe-in | -64.92, -13.68 | -47.25, -45.59 | APE12-dist-na | 16.2504 | APE11-dist-na | 13.1008 | APE10-dist-na | 11.1871 | APE9-dist-in | 7.9038 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.3 | 0.198 | 0.245 | A | 328.0 | 285.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 6xva | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.4e-104 | 354.2 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 6XVAB | P10721 | 577 | 931 | 976.0 | O2K:61001 | Type2 | Inactive | DFGout | 15.832 | 9.9461 | BBAminus | -129.58, -168.14 | -159.52, 95.6 | -60.13, -40.05 | 280.9, 81.98 | 51.8, -114.7 | in-in | in | 7.838 | Saltbr-in | 2.8735 | HRD-in | -67.63, -49.04 | 76.72, -12.76 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.2998 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -120.1, 96.88 | APE9-dihe-in | -113.3, 152.94 | APE8-dihe-in | -84.37, 70.57 | APE8-rot-na | 30.8 | APE67-dihe-in | -65.41, -13.28 | -47.31, -45.65 | APE12-dist-na | 16.5272 | APE11-dist-na | 13.1483 | APE10-dist-na | 11.3543 | APE9-dist-in | 7.935 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.3 | 0.198 | 0.245 | B | 328.0 | 277.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 6xva | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.4e-104 | 354.2 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|