| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 6XV9A | P10721 | 566 | 931 | 976.0 | O35:61001 | Type2 | Inactive | DFGout | 15.5426 | 9.7475 | BBAminus | -131.58, -169.39 | -156.72, 93.49 | -62.05, -42.03 | 282.46, 88.43 | 48.41, -104.01 | in-in | in | 7.6893 | Saltbr-in | 2.8319 | HRD-in | -69.28, -49.38 | 72.93, -5.84 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.311 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.37, 97.09 | APE9-dihe-in | -112.0, 148.71 | APE8-dihe-in | -81.81, 67.27 | APE8-rot-na | 29.88 | APE67-dihe-in | -63.86, -9.66 | -46.65, -44.91 | APE12-dist-na | 16.5786 | APE11-dist-na | 13.1347 | APE10-dist-na | 10.916 | APE9-dist-in | 7.6291 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 3.38 | 0.197 | 0.247 | A | 328.0 | 288.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 6xv9 | TYR_KIT_HUMAN | TYR | 2.4e-104 | 354.2 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 6XV9B | P10721 | 572 | 931 | 976.0 | O35:61001 | Type2 | Inactive | DFGout | 15.678 | 9.7703 | BBAminus | -131.94, -171.98 | -157.03, 93.9 | -61.83, -41.64 | 282.16, 88.18 | 48.65, -104.6 | in-in | in | 7.7333 | Saltbr-in | 2.8538 | HRD-in | -68.86, -49.09 | 75.5, -9.43 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.206 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -118.51, 98.6 | APE9-dihe-in | -113.58, 149.31 | APE8-dihe-in | -82.14, 67.2 | APE8-rot-na | 30.55 | APE67-dihe-in | -64.65, -9.32 | -46.19, -45.23 | APE12-dist-na | 16.7634 | APE11-dist-na | 13.3341 | APE10-dist-na | 11.1489 | APE9-dist-in | 7.7545 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 3.38 | 0.197 | 0.247 | B | 328.0 | 282.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 6xv9 | TYR_KIT_HUMAN | TYR | 2.4e-104 | 354.2 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 6XV9A | P10721 | 566 | 931 | 976.0 | O35:61001 | Type2 | Inactive | DFGout | 15.5426 | 9.7475 | BBAminus | -131.58, -169.39 | -156.72, 93.49 | -62.05, -42.03 | 282.46, 88.43 | 48.41, -104.01 | in-in | in | 7.6893 | Saltbr-in | 2.8319 | HRD-in | -69.28, -49.38 | 72.93, -5.84 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.311 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.37, 97.09 | APE9-dihe-in | -112.0, 148.71 | APE8-dihe-in | -81.81, 67.27 | APE8-rot-na | 29.88 | APE67-dihe-in | -63.86, -9.66 | -46.65, -44.91 | APE12-dist-na | 16.5786 | APE11-dist-na | 13.1347 | APE10-dist-na | 10.916 | APE9-dist-in | 7.6291 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 3.38 | 0.197 | 0.247 | A | 328.0 | 288.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 6xv9 | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.4e-104 | 354.2 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 6XV9B | P10721 | 572 | 931 | 976.0 | O35:61001 | Type2 | Inactive | DFGout | 15.678 | 9.7703 | BBAminus | -131.94, -171.98 | -157.03, 93.9 | -61.83, -41.64 | 282.16, 88.18 | 48.65, -104.6 | in-in | in | 7.7333 | Saltbr-in | 2.8538 | HRD-in | -68.86, -49.09 | 75.5, -9.43 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.206 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -118.51, 98.6 | APE9-dihe-in | -113.58, 149.31 | APE8-dihe-in | -82.14, 67.2 | APE8-rot-na | 30.55 | APE67-dihe-in | -64.65, -9.32 | -46.19, -45.23 | APE12-dist-na | 16.7634 | APE11-dist-na | 13.3341 | APE10-dist-na | 11.1489 | APE9-dist-in | 7.7545 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 3.38 | 0.197 | 0.247 | B | 328.0 | 282.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 6xv9 | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.4e-104 | 354.2 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|