| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 6V6OC | P00533 | 701 | 1011 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 3.6437 | 14.2137 | BLBplus | -122.87, 171.43 | 70.23, 18.79 | -66.69, 140.71 | 67.25, 92.35 | 81.97, -11.3 | out-out | out | 14.2607 | Saltbr-out | 13.5365 | HRD-in | -75.21, -54.45 | 82.69, -13.83 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.7798 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 118.15 | APE8-dihe-in | -81.1, 67.37 | APE8-rot-na | 31.91 | APE67-dihe-in | -73.98, -4.02 | -53.95, -44.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.2764 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | C | 327.0 | 297.0 | 12 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 6v6o | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OD | P00533 | 701 | 1014 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 3.8632 | 14.1094 | BLBplus | -124.4, 171.55 | 69.25, 17.62 | -67.5, 139.98 | 64.11, 93.51 | 81.27, -10.57 | out-out | out | 14.2978 | Saltbr-out | 13.5608 | HRD-in | -74.72, -54.65 | 82.6, -12.74 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.694 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -74.63, -11.25 | APE9-dihe-in | -98.47, 121.43 | APE8-dihe-in | -79.76, 67.8 | APE8-rot-na | 32.25 | APE67-dihe-in | -74.09, -4.64 | -53.64, -43.16 | APE12-dist-na | 18.5142 | APE11-dist-na | 15.9087 | APE10-dist-na | 11.5368 | APE9-dist-in | 7.9994 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | D | 327.0 | 314.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6v6o | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OE | P00533 | 701 | 1014 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 3.7621 | 14.1256 | BLBplus | -123.9, 171.7 | 69.62, 18.55 | -66.64, 139.7 | 64.92, 95.49 | 81.38, -10.3 | out-out | out | 14.0102 | Saltbr-out | 14.5062 | HRD-in | -75.07, -55.34 | 81.99, -12.92 | out-out-none | SNCoon | out-none | ActLoopNT-out | 6.8972 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -28.58 | APE9-dihe-in | -100.13, 119.03 | APE8-dihe-in | -80.06, 70.49 | APE8-rot-na | 32.0 | APE67-dihe-in | -73.71, -4.57 | -52.25, -42.58 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.8528 | APE9-dist-in | 7.8342 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | E | 327.0 | 303.0 | 11 | 30 | 19 | 11 | [[712, 970]] | 1.0 | 6v6o | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OH | P00533 | 700 | 1014 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 3.651 | 13.9842 | BLBplus | -123.38, 171.8 | 70.53, 19.82 | -66.37, 140.7 | 65.92, 91.26 | 79.41, -10.87 | out-out | out | 13.6988 | Saltbr-out | 12.8647 | HRD-in | -75.67, -55.2 | 81.77, -12.73 | out-out-none | SNCoon | out-none | ActLoopNT-out | 6.8501 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -16.84 | APE9-dihe-in | -111.7, 114.25 | APE8-dihe-in | -84.18, 71.19 | APE8-rot-na | 31.92 | APE67-dihe-in | -73.23, -5.03 | -51.26, -41.97 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.2277 | APE9-dist-in | 7.798 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | H | 327.0 | 299.0 | 11 | 30 | 19 | 11 | [[712, 970]] | 1.0 | 6v6o | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OA | P00533 | 701 | 1007 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 5.2979 | 16.7269 | BLBtrans | -121.65, 172.71 | 69.64, 21.71 | -62.97, 137.24 | 151.72, 75.2 | 80.63, -10.98 | out-out | out | 14.3912 | Saltbr-out | 13.4198 | HRD-in | -75.85, -53.93 | 83.31, -13.79 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8089 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.46, -8.8 | APE9-dihe-in | -105.55, 118.94 | APE8-dihe-in | -80.71, 68.41 | APE8-rot-na | 31.83 | APE67-dihe-in | -75.0, -4.07 | -53.04, -43.94 | APE12-dist-na | 17.1716 | APE11-dist-na | 14.8931 | APE10-dist-na | 10.7033 | APE9-dist-in | 7.8108 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | A | 327.0 | 307.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6v6o | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OB | P00533 | 701 | 1014 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 5.7535 | 16.8597 | BLBtrans | -121.27, 172.7 | 70.02, 21.31 | -63.98, 138.97 | 154.89, 75.61 | 80.68, -11.77 | out-out | out | 14.1922 | Saltbr-out | 13.3835 | HRD-in | -75.47, -53.91 | 84.16, -12.57 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.4558 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -76.92, -9.63 | APE9-dihe-in | -88.61, 118.08 | APE8-dihe-in | -81.24, 68.33 | APE8-rot-na | 32.0 | APE67-dihe-in | -74.5, -4.48 | -53.39, -42.67 | APE12-dist-na | 18.8815 | APE11-dist-na | 15.8867 | APE10-dist-na | 11.3814 | APE9-dist-out | 8.3009 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | B | 327.0 | 314.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6v6o | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OF | P00533 | 701 | 1012 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 5.9053 | 17.2423 | BLBtrans | -120.46, 172.23 | 70.73, 22.19 | -64.5, 139.46 | 157.13, 75.08 | 81.89, -12.08 | out-out | out | 13.7421 | Saltbr-out | 12.6104 | HRD-in | -74.49, -52.75 | 85.72, -15.71 | out-out-none | SNCoon | out-none | ActLoopNT-out | 6.8108 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.82 | APE8-dihe-in | -82.55, 69.28 | APE8-rot-na | 31.97 | APE67-dihe-in | -74.52, -5.14 | -52.67, -43.32 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.827 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | F | 327.0 | 299.0 | 13 | 30 | 17 | 13 | [[712, 970]] | 1.0 | 6v6o | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OG | P00533 | 701 | 1009 | 1210.0 | QQM:1301 | Type1 | Inactive | DFGin | 5.5503 | 16.2142 | BLBtrans | -119.98, -175.83 | 64.58, 23.85 | -74.9, 132.09 | 162.27, 73.99 | 101.97, 164.72 | out-out | out | 13.3633 | Saltbr-out | 11.5722 | HRD-in | -77.28, -50.81 | 78.9, -9.78 | out-out-none | SNCoon | out-none | ActLoopNT-out | 9.86 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 124.89 | APE8-dihe-in | -78.97, 76.25 | APE8-rot-na | 32.23 | APE67-dihe-in | -70.7, -0.71 | -59.43, -44.63 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.9465 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | G | 327.0 | 294.0 | 15 | 30 | 15 | 15 | [[712, 970]] | 1.0 | 6v6o | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 6V6OC | P00533 | 701 | 1011 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 3.6437 | 14.2137 | BLBplus | -122.87, 171.43 | 70.23, 18.79 | -66.69, 140.71 | 67.25, 92.35 | 81.97, -11.3 | out-out | out | 14.2607 | Saltbr-out | 13.5365 | HRD-in | -75.21, -54.45 | 82.69, -13.83 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.7798 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 118.15 | APE8-dihe-in | -81.1, 67.37 | APE8-rot-na | 31.91 | APE67-dihe-in | -73.98, -4.02 | -53.95, -44.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.2764 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | C | 327.0 | 297.0 | 12 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 6v6o | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OD | P00533 | 701 | 1014 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 3.8632 | 14.1094 | BLBplus | -124.4, 171.55 | 69.25, 17.62 | -67.5, 139.98 | 64.11, 93.51 | 81.27, -10.57 | out-out | out | 14.2978 | Saltbr-out | 13.5608 | HRD-in | -74.72, -54.65 | 82.6, -12.74 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.694 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -74.63, -11.25 | APE9-dihe-in | -98.47, 121.43 | APE8-dihe-in | -79.76, 67.8 | APE8-rot-na | 32.25 | APE67-dihe-in | -74.09, -4.64 | -53.64, -43.16 | APE12-dist-na | 18.5142 | APE11-dist-na | 15.9087 | APE10-dist-na | 11.5368 | APE9-dist-in | 7.9994 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | D | 327.0 | 314.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6v6o | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OE | P00533 | 701 | 1014 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 3.7621 | 14.1256 | BLBplus | -123.9, 171.7 | 69.62, 18.55 | -66.64, 139.7 | 64.92, 95.49 | 81.38, -10.3 | out-out | out | 14.0102 | Saltbr-out | 14.5062 | HRD-in | -75.07, -55.34 | 81.99, -12.92 | out-out-none | SNCoon | out-none | ActLoopNT-out | 6.8972 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -28.58 | APE9-dihe-in | -100.13, 119.03 | APE8-dihe-in | -80.06, 70.49 | APE8-rot-na | 32.0 | APE67-dihe-in | -73.71, -4.57 | -52.25, -42.58 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.8528 | APE9-dist-in | 7.8342 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | E | 327.0 | 303.0 | 11 | 30 | 19 | 11 | [[712, 970]] | 1.0 | 6v6o | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OH | P00533 | 700 | 1014 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 3.651 | 13.9842 | BLBplus | -123.38, 171.8 | 70.53, 19.82 | -66.37, 140.7 | 65.92, 91.26 | 79.41, -10.87 | out-out | out | 13.6988 | Saltbr-out | 12.8647 | HRD-in | -75.67, -55.2 | 81.77, -12.73 | out-out-none | SNCoon | out-none | ActLoopNT-out | 6.8501 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -16.84 | APE9-dihe-in | -111.7, 114.25 | APE8-dihe-in | -84.18, 71.19 | APE8-rot-na | 31.92 | APE67-dihe-in | -73.23, -5.03 | -51.26, -41.97 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.2277 | APE9-dist-in | 7.798 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | H | 327.0 | 299.0 | 11 | 30 | 19 | 11 | [[712, 970]] | 1.0 | 6v6o | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OA | P00533 | 701 | 1007 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 5.2979 | 16.7269 | BLBtrans | -121.65, 172.71 | 69.64, 21.71 | -62.97, 137.24 | 151.72, 75.2 | 80.63, -10.98 | out-out | out | 14.3912 | Saltbr-out | 13.4198 | HRD-in | -75.85, -53.93 | 83.31, -13.79 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8089 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.46, -8.8 | APE9-dihe-in | -105.55, 118.94 | APE8-dihe-in | -80.71, 68.41 | APE8-rot-na | 31.83 | APE67-dihe-in | -75.0, -4.07 | -53.04, -43.94 | APE12-dist-na | 17.1716 | APE11-dist-na | 14.8931 | APE10-dist-na | 10.7033 | APE9-dist-in | 7.8108 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | A | 327.0 | 307.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6v6o | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OB | P00533 | 701 | 1014 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 5.7535 | 16.8597 | BLBtrans | -121.27, 172.7 | 70.02, 21.31 | -63.98, 138.97 | 154.89, 75.61 | 80.68, -11.77 | out-out | out | 14.1922 | Saltbr-out | 13.3835 | HRD-in | -75.47, -53.91 | 84.16, -12.57 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.4558 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -76.92, -9.63 | APE9-dihe-in | -88.61, 118.08 | APE8-dihe-in | -81.24, 68.33 | APE8-rot-na | 32.0 | APE67-dihe-in | -74.5, -4.48 | -53.39, -42.67 | APE12-dist-na | 18.8815 | APE11-dist-na | 15.8867 | APE10-dist-na | 11.3814 | APE9-dist-out | 8.3009 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | B | 327.0 | 314.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6v6o | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OF | P00533 | 701 | 1012 | 1210.0 | QQM:1202 | Type1 | Inactive | DFGin | 5.9053 | 17.2423 | BLBtrans | -120.46, 172.23 | 70.73, 22.19 | -64.5, 139.46 | 157.13, 75.08 | 81.89, -12.08 | out-out | out | 13.7421 | Saltbr-out | 12.6104 | HRD-in | -74.49, -52.75 | 85.72, -15.71 | out-out-none | SNCoon | out-none | ActLoopNT-out | 6.8108 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.82 | APE8-dihe-in | -82.55, 69.28 | APE8-rot-na | 31.97 | APE67-dihe-in | -74.52, -5.14 | -52.67, -43.32 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.827 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | F | 327.0 | 299.0 | 13 | 30 | 17 | 13 | [[712, 970]] | 1.0 | 6v6o | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6V6OG | P00533 | 701 | 1009 | 1210.0 | QQM:1301 | Type1 | Inactive | DFGin | 5.5503 | 16.2142 | BLBtrans | -119.98, -175.83 | 64.58, 23.85 | -74.9, 132.09 | 162.27, 73.99 | 101.97, 164.72 | out-out | out | 13.3633 | Saltbr-out | 11.5722 | HRD-in | -77.28, -50.81 | 78.9, -9.78 | out-out-none | SNCoon | out-none | ActLoopNT-out | 9.86 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 124.89 | APE8-dihe-in | -78.97, 76.25 | APE8-rot-na | 32.23 | APE67-dihe-in | -70.7, -0.71 | -59.43, -44.63 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.9465 | T790M,V948R | None | None | XRAY | 2.1 | 0.196 | 0.221 | G | 327.0 | 294.0 | 15 | 30 | 15 | 15 | [[712, 970]] | 1.0 | 6v6o | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6e-88 | 300.6 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|