| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR3 | FGFR3_HUMAN | 6PNXA | P22607 | 456 | 757 | 806.0 | ACP:801 | ATPlike | Inactive | DFGin | 5.1832 | 13.2568 | BLAplus | -117.43, 165.96 | 59.53, 36.21 | -90.35, -22.61 | 56.49, 88.29 | -100.71, 20.75 | in-out | in | 7.758 | Saltbr-out | 3.8922 | HRD-in | -72.74, -43.96 | 72.66, -12.59 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.6112 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 61.32, -168.18 | APE9-dihe-in | -95.45, 138.6 | APE8-dihe-in | -83.08, 62.92 | APE8-rot-na | 32.84 | APE67-dihe-in | -77.59, -4.01 | -63.19, -31.79 | APE12-dist-na | 17.76 | APE11-dist-na | 14.3869 | APE10-dist-na | 16.4747 | APE9-dist-in | 7.9796 | C482A,C582S,R669E | None | None | XRAY | 2.199 | 0.195 | 0.23 | A | 324.0 | 291.0 | 11 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6pnx | TYR_FGFR3_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | 6PNXB | P22607 | 455 | 756 | 806.0 | ACP:801 | ATPlike | Inactive | DFGin | 5.1024 | 12.8796 | BLAplus | -116.22, 163.18 | 57.59, 45.48 | -96.33, -11.84 | 56.51, 88.18 | -107.89, 22.55 | in-in | in | 7.3718 | Saltbr-in | 2.3809 | HRD-in | -94.02, -38.66 | 69.29, -17.12 | in-out-out | SNCioo | out-out | ActLoopNT-out | 4.1485 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 54.33, 74.29 | APE9-dihe-in | -157.39, 146.53 | APE8-dihe-in | -79.85, 92.16 | APE8-rot-na | 29.38 | APE67-dihe-in | -64.97, -14.94 | -62.55, -40.44 | APE12-dist-na | 17.5294 | APE11-dist-na | 16.9582 | APE10-dist-na | 14.6317 | APE9-dist-in | 7.491 | C482A,C582S,R669E | None | None | XRAY | 2.199 | 0.195 | 0.23 | B | 324.0 | 294.0 | 8 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6pnx | TYR_FGFR3_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR3 | FGFR3_HUMAN | 6PNXA | P22607 | 456 | 757 | 806.0 | ACP:801 | ATPlike | Inactive | DFGin | 5.1832 | 13.2568 | BLAplus | -117.43, 165.96 | 59.53, 36.21 | -90.35, -22.61 | 56.49, 88.29 | -100.71, 20.75 | in-out | in | 7.758 | Saltbr-out | 3.8922 | HRD-in | -72.74, -43.96 | 72.66, -12.59 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.6112 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 61.32, -168.18 | APE9-dihe-in | -95.45, 138.6 | APE8-dihe-in | -83.08, 62.92 | APE8-rot-na | 32.84 | APE67-dihe-in | -77.59, -4.01 | -63.19, -31.79 | APE12-dist-na | 17.76 | APE11-dist-na | 14.3869 | APE10-dist-na | 16.4747 | APE9-dist-in | 7.9796 | C482A,C582S,R669E | None | None | XRAY | 2.199 | 0.195 | 0.23 | A | 324.0 | 291.0 | 11 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6pnx | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | 6PNXB | P22607 | 455 | 756 | 806.0 | ACP:801 | ATPlike | Inactive | DFGin | 5.1024 | 12.8796 | BLAplus | -116.22, 163.18 | 57.59, 45.48 | -96.33, -11.84 | 56.51, 88.18 | -107.89, 22.55 | in-in | in | 7.3718 | Saltbr-in | 2.3809 | HRD-in | -94.02, -38.66 | 69.29, -17.12 | in-out-out | SNCioo | out-out | ActLoopNT-out | 4.1485 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 54.33, 74.29 | APE9-dihe-in | -157.39, 146.53 | APE8-dihe-in | -79.85, 92.16 | APE8-rot-na | 29.38 | APE67-dihe-in | -64.97, -14.94 | -62.55, -40.44 | APE12-dist-na | 17.5294 | APE11-dist-na | 16.9582 | APE10-dist-na | 14.6317 | APE9-dist-in | 7.491 | C482A,C582S,R669E | None | None | XRAY | 2.199 | 0.195 | 0.23 | B | 324.0 | 294.0 | 8 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6pnx | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|