| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | TEK | TIE2_HUMAN | 6MWEA | Q02763 | 816 | 1122 | 1124.0 | 919:1203 | Type2 | Inactive | DFGout | 13.3535 | 10.6059 | BBAminus | -139.56, 179.54 | -155.41, 121.99 | -100.36, 10.81 | 282.44, 103.03 | 91.89, 0.35 | in-in | in | 7.5591 | Saltbr-in | 2.4825 | HRD-in | -71.19, -54.67 | 81.44, -10.36 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.5425 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | -91.4, -5.72 | APE9-dihe-out | -57.22, -41.43 | APE8-dihe-out | -59.21, -21.01 | APE8-rot-na | 337.82 | APE67-dihe-in | -71.75, -11.24 | -48.45, -35.17 | APE12-dist-na | 11.3805 | APE11-dist-na | 8.608 | APE10-dist-na | 12.5606 | APE9-dist-out | 10.785 | None | None | None | XRAY | 2.05 | 0.149 | 0.166 | A | 317.0 | 292.0 | 15 | 27 | 25 | 2 | [[824, 1094]] | 1.0 | 6mwe | TYR_TEK_HUMAN | TYR | 7.5e-91 | 310.0 | 1.0 | 260.0 | 260.0 | 981 | 982 | 983 | 985 | 987 | 855 | 872 | 876 | 961 | 963 | 962 | 964.0 | 1020 | 1008 | 1003 | 1002 | 1001 | 1000 | 999 | 998 | 997 | 903 | Angiopoietin-1 receptor |
| TYR | TEK | TIE2_HUMAN | 6MWEB | Q02763 | 816 | 1122 | 1124.0 | 919:1203 | Type2 | Inactive | DFGout | 13.3959 | 10.5044 | BBAminus | -136.71, -178.85 | -151.95, 121.17 | -94.08, 7.28 | 284.75, 97.66 | 92.39, -1.76 | in-in | in | 7.559 | Saltbr-in | 2.5849 | HRD-in | -68.95, -51.62 | 79.52, -11.84 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.4156 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | -91.44, -0.78 | APE9-dihe-out | -58.14, -40.06 | APE8-dihe-out | -58.25, -21.33 | APE8-rot-na | 337.67 | APE67-dihe-in | -69.06, -11.94 | -47.55, -40.23 | APE12-dist-na | 10.9599 | APE11-dist-na | 7.9391 | APE10-dist-na | 11.8184 | APE9-dist-out | 10.9023 | None | None | None | XRAY | 2.05 | 0.149 | 0.166 | B | 317.0 | 290.0 | 17 | 27 | 24 | 3 | [[824, 1094]] | 1.0 | 6mwe | TYR_TEK_HUMAN | TYR | 7.5e-91 | 310.0 | 1.0 | 260.0 | 260.0 | 981 | 982 | 983 | 985 | 987 | 855 | 872 | 876 | 961 | 963 | 962 | 964.0 | 1020 | 1008 | 1003 | 1002 | 1001 | 1000 | 999 | 998 | 997 | 903 | Angiopoietin-1 receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | TEK | TIE2_HUMAN | 6MWEA | Q02763 | 816 | 1122 | 1124.0 | 919:1203 | Type2 | Inactive | DFGout | 13.3535 | 10.6059 | BBAminus | -139.56, 179.54 | -155.41, 121.99 | -100.36, 10.81 | 282.44, 103.03 | 91.89, 0.35 | in-in | in | 7.5591 | Saltbr-in | 2.4825 | HRD-in | -71.19, -54.67 | 81.44, -10.36 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.5425 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | -91.4, -5.72 | APE9-dihe-out | -57.22, -41.43 | APE8-dihe-out | -59.21, -21.01 | APE8-rot-na | 337.82 | APE67-dihe-in | -71.75, -11.24 | -48.45, -35.17 | APE12-dist-na | 11.3805 | APE11-dist-na | 8.608 | APE10-dist-na | 12.5606 | APE9-dist-out | 10.785 | None | None | None | XRAY | 2.05 | 0.149 | 0.166 | A | 317.0 | 292.0 | 15 | 27 | 25 | 2 | [[824, 1094]] | 1.0 | 6mwe | Homo sapiens | TYR_TEK_HUMAN | TYR | 7.5e-91 | 310.0 | 1.0 | 260.0 | 260.0 | 981 | 982 | 983 | 985 | 987 | 855 | 872 | 876 | 961 | 963 | 962 | 964.0 | 1020 | 1008 | 1003 | 1002 | 1001 | 1000 | 999 | 998 | 997 | 903 | Angiopoietin-1 receptor |
| TYR | TEK | TIE2_HUMAN | 6MWEB | Q02763 | 816 | 1122 | 1124.0 | 919:1203 | Type2 | Inactive | DFGout | 13.3959 | 10.5044 | BBAminus | -136.71, -178.85 | -151.95, 121.17 | -94.08, 7.28 | 284.75, 97.66 | 92.39, -1.76 | in-in | in | 7.559 | Saltbr-in | 2.5849 | HRD-in | -68.95, -51.62 | 79.52, -11.84 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.4156 | ActLoopCT-out | TYR | APEdihe_oooai | APEdist_aaao | APE10-dihe-out | -91.44, -0.78 | APE9-dihe-out | -58.14, -40.06 | APE8-dihe-out | -58.25, -21.33 | APE8-rot-na | 337.67 | APE67-dihe-in | -69.06, -11.94 | -47.55, -40.23 | APE12-dist-na | 10.9599 | APE11-dist-na | 7.9391 | APE10-dist-na | 11.8184 | APE9-dist-out | 10.9023 | None | None | None | XRAY | 2.05 | 0.149 | 0.166 | B | 317.0 | 290.0 | 17 | 27 | 24 | 3 | [[824, 1094]] | 1.0 | 6mwe | Homo sapiens | TYR_TEK_HUMAN | TYR | 7.5e-91 | 310.0 | 1.0 | 260.0 | 260.0 | 981 | 982 | 983 | 985 | 987 | 855 | 872 | 876 | 961 | 963 | 962 | 964.0 | 1020 | 1008 | 1003 | 1002 | 1001 | 1000 | 999 | 998 | 997 | 903 | Angiopoietin-1 receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|