| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PRKACA | KAPCA_MOUSE | 6MM6C | P05132 | 19 | 351 | 351.0 | ANP:60402 | ATPlike | Inactive | DFGin | 6.7799 | 16.0821 | ABAminus | -110.74, -8.1 | -141.78, 125.75 | -126.67, 17.79 | 291.81, 81.75 | -52.6, -43.19 | out-out | out | 10.4027 | Saltbr-out | 4.4909 | HRD-in | -64.73, -48.52 | 44.91, 28.18 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8769 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -155.16, 154.51 | APE9-dihe-na | 131.73, -155.42 | APE8-dihe-in | -119.09, 141.73 | APE8-rot-out | 198.33 | APE67-dihe-in | -57.79, -26.12 | -45.84, -50.95 | APE12-dist-in | 8.5303 | APE11-dist-in | 11.8147 | APE10-dist-in | 6.3058 | APE9-dist-in | 4.5025 | None | TPO198,SEP339 | TPO198,SEP339 | XRAY | 2.39 | 0.225 | 0.261 | C | 339.0 | 322.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6mm6 | Mus musculus | AGC_PRKACA_MOUSE | AGC | 1.3e-94 | 322.1 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_MOUSE | 6MM6E | P05132 | 19 | 351 | 351.0 | ANP:60401 | ATPlike | Inactive | DFGin | 6.7325 | 15.9653 | ABAminus | -112.26, -9.59 | -137.74, 126.1 | -127.73, 18.87 | 290.52, 82.39 | -53.04, -44.19 | out-out | out | 10.2709 | Saltbr-out | 5.278 | HRD-in | -66.74, -47.88 | 44.41, 27.02 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8731 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -157.27, 155.34 | APE9-dihe-na | 128.78, -154.8 | APE8-dihe-in | -120.26, 141.99 | APE8-rot-out | 197.33 | APE67-dihe-in | -57.79, -26.44 | -45.46, -51.33 | APE12-dist-in | 8.4779 | APE11-dist-in | 11.8514 | APE10-dist-in | 6.3306 | APE9-dist-in | 4.4228 | None | TPO198,SEP339 | TPO198,SEP339 | XRAY | 2.39 | 0.225 | 0.261 | E | 339.0 | 320.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6mm6 | Mus musculus | AGC_PRKACA_MOUSE | AGC | 1.3e-94 | 322.1 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PRKACA | KAPCA_MOUSE | 6MM6C | P05132 | 19 | 351 | 351.0 | ANP:60402 | ATPlike | Inactive | DFGin | 6.7799 | 16.0821 | ABAminus | -110.74, -8.1 | -141.78, 125.75 | -126.67, 17.79 | 291.81, 81.75 | -52.6, -43.19 | out-out | out | 10.4027 | Saltbr-out | 4.4909 | HRD-in | -64.73, -48.52 | 44.91, 28.18 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8769 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -155.16, 154.51 | APE9-dihe-na | 131.73, -155.42 | APE8-dihe-in | -119.09, 141.73 | APE8-rot-out | 198.33 | APE67-dihe-in | -57.79, -26.12 | -45.84, -50.95 | APE12-dist-in | 8.5303 | APE11-dist-in | 11.8147 | APE10-dist-in | 6.3058 | APE9-dist-in | 4.5025 | None | TPO198,SEP339 | TPO198,SEP339 | XRAY | 2.39 | 0.225 | 0.261 | C | 339.0 | 322.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6mm6 | Mus musculus | AGC_PRKACA_MOUSE | AGC | 1.3e-94 | 322.1 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_MOUSE | 6MM6E | P05132 | 19 | 351 | 351.0 | ANP:60401 | ATPlike | Inactive | DFGin | 6.7325 | 15.9653 | ABAminus | -112.26, -9.59 | -137.74, 126.1 | -127.73, 18.87 | 290.52, 82.39 | -53.04, -44.19 | out-out | out | 10.2709 | Saltbr-out | 5.278 | HRD-in | -66.74, -47.88 | 44.41, 27.02 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8731 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -157.27, 155.34 | APE9-dihe-na | 128.78, -154.8 | APE8-dihe-in | -120.26, 141.99 | APE8-rot-out | 197.33 | APE67-dihe-in | -57.79, -26.44 | -45.46, -51.33 | APE12-dist-in | 8.4779 | APE11-dist-in | 11.8514 | APE10-dist-in | 6.3306 | APE9-dist-in | 4.4228 | None | TPO198,SEP339 | TPO198,SEP339 | XRAY | 2.39 | 0.225 | 0.261 | E | 339.0 | 320.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6mm6 | Mus musculus | AGC_PRKACA_MOUSE | AGC | 1.3e-94 | 322.1 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |