| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| OTHER | GAK | GAK_HUMAN | 5Y7ZA | O14976 | 25 | 335 | 1311.0 | IRE:60401 | Type1 | Inactive | DFGin | 6.1831 | 14.3017 | ABAminus | -120.31, -65.73 | -84.03, 133.07 | -132.73, 38.63 | 297.55, 94.83 | -80.73, -23.71 | in-in | in | 9.3299 | Saltbr-in | 2.6528 | HRD-in | -76.12, -47.1 | 64.19, -3.41 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.6933 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -90.58, 12.1 | APE9-dihe-na | -127.21, 155.97 | APE8-dihe-in | -88.88, 126.92 | APE8-rot-in | 301.28 | APE67-dihe-in | -75.82, -11.44 | -39.58, -53.85 | APE12-dist-in | 11.6752 | APE11-dist-in | 8.7406 | APE10-dist-in | 4.1646 | APE9-dist-in | 4.1456 | None | None | None | XRAY | 2.804 | 0.235 | 0.288 | A | 313.0 | 311.0 | 0 | 40 | 40 | 0 | [[40, 313]] | 1.0 | 5y7z | OTHER_GAK_HUMAN | CAMK | 4e-44 | 157.2 | 3.0 | 252.0 | 250.0 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173.0 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| OTHER | GAK | GAK_HUMAN | 5Y7ZB | O14976 | 25 | 335 | 1311.0 | IRE:60401 | Type1 | Inactive | DFGin | 6.185 | 14.3005 | ABAminus | -126.63, -59.42 | -85.24, 119.57 | -121.34, 32.24 | 292.7, 91.36 | -76.51, -21.75 | in-in | in | 8.9976 | Saltbr-in | 3.3359 | HRD-in | -76.77, -44.95 | 63.95, -6.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7625 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.15, 9.34 | APE9-dihe-na | -125.96, 148.71 | APE8-dihe-in | -79.22, 127.62 | APE8-rot-in | 300.16 | APE67-dihe-in | -76.26, -13.67 | -39.68, -52.24 | APE12-dist-in | 11.7706 | APE11-dist-in | 8.7646 | APE10-dist-in | 4.2306 | APE9-dist-in | 4.0018 | None | None | None | XRAY | 2.804 | 0.235 | 0.288 | B | 313.0 | 311.0 | 0 | 40 | 40 | 0 | [[40, 313]] | 1.0 | 5y7z | OTHER_GAK_HUMAN | CAMK | 4e-44 | 157.2 | 3.0 | 252.0 | 250.0 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173.0 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| OTHER | GAK | GAK_HUMAN | 5Y7ZA | O14976 | 25 | 335 | 1311.0 | IRE:60401 | Type1 | Inactive | DFGin | 6.1831 | 14.3017 | ABAminus | -120.31, -65.73 | -84.03, 133.07 | -132.73, 38.63 | 297.55, 94.83 | -80.73, -23.71 | in-in | in | 9.3299 | Saltbr-in | 2.6528 | HRD-in | -76.12, -47.1 | 64.19, -3.41 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.6933 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -90.58, 12.1 | APE9-dihe-na | -127.21, 155.97 | APE8-dihe-in | -88.88, 126.92 | APE8-rot-in | 301.28 | APE67-dihe-in | -75.82, -11.44 | -39.58, -53.85 | APE12-dist-in | 11.6752 | APE11-dist-in | 8.7406 | APE10-dist-in | 4.1646 | APE9-dist-in | 4.1456 | None | None | None | XRAY | 2.804 | 0.235 | 0.288 | A | 313.0 | 311.0 | 0 | 40 | 40 | 0 | [[40, 313]] | 1.0 | 5y7z | Homo sapiens | OTHER_GAK_HUMAN | CAMK | 4e-44 | 157.2 | 3.0 | 252.0 | 250.0 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173.0 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| OTHER | GAK | GAK_HUMAN | 5Y7ZB | O14976 | 25 | 335 | 1311.0 | IRE:60401 | Type1 | Inactive | DFGin | 6.185 | 14.3005 | ABAminus | -126.63, -59.42 | -85.24, 119.57 | -121.34, 32.24 | 292.7, 91.36 | -76.51, -21.75 | in-in | in | 8.9976 | Saltbr-in | 3.3359 | HRD-in | -76.77, -44.95 | 63.95, -6.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7625 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -88.15, 9.34 | APE9-dihe-na | -125.96, 148.71 | APE8-dihe-in | -79.22, 127.62 | APE8-rot-in | 300.16 | APE67-dihe-in | -76.26, -13.67 | -39.68, -52.24 | APE12-dist-in | 11.7706 | APE11-dist-in | 8.7646 | APE10-dist-in | 4.2306 | APE9-dist-in | 4.0018 | None | None | None | XRAY | 2.804 | 0.235 | 0.288 | B | 313.0 | 311.0 | 0 | 40 | 40 | 0 | [[40, 313]] | 1.0 | 5y7z | Homo sapiens | OTHER_GAK_HUMAN | CAMK | 4e-44 | 157.2 | 3.0 | 252.0 | 250.0 | 190 | 191 | 192 | 194 | 196 | 69 | 85 | 89 | 170 | 172 | 171 | 173.0 | 245 | 230 | 225 | 224 | 223 | 222 | 221 | 220 | 219 | 124 | Cyclin-G-associated kinase |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|