| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 5O49A | P11362 | 464 | 764 | 822.0 | 9K5:801 | Type1 | Inactive | DFGin | 5.2397 | 13.6382 | BLAplus | -124.98, 161.58 | 68.85, 20.17 | -74.75, -11.05 | 61.69, 77.84 | -110.93, 4.69 | in-out | in | 8.1254 | Saltbr-out | 5.5459 | HRD-in | -64.73, -48.02 | 76.28, -6.18 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.7824 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.25, 168.76 | APE9-dihe-in | -119.19, 119.01 | APE8-dihe-out | -64.8, -20.97 | APE8-rot-na | 343.93 | APE67-dihe-in | -73.72, -10.74 | -55.47, -23.05 | APE12-dist-na | 19.5652 | APE11-dist-na | 21.14 | APE10-dist-na | 19.4995 | APE9-dist-out | 11.833 | C488A,C584S | None | None | XRAY | 1.91 | 0.2 | 0.22 | A | 309.0 | 289.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5o49 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5O49B | P11362 | 460 | 765 | 822.0 | 9K5:801 | Type1 | Inactive | DFGin | 5.6188 | 12.9288 | BLAplus | -126.58, 172.58 | 67.38, 24.13 | -84.06, -18.33 | 50.82, 87.05 | -104.51, 13.86 | in-out | in | 7.6377 | Saltbr-out | 4.5004 | HRD-in | -61.81, -47.66 | 75.62, -5.93 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -110.43, 163.49 | APE9-dihe-in | -105.31, 114.78 | APE8-dihe-out | -56.47, -25.97 | APE8-rot-na | 333.8 | APE67-dihe-in | -70.86, -8.05 | -56.14, -23.8 | APE12-dist-na | 19.0124 | APE11-dist-na | 20.4124 | APE10-dist-na | 18.7866 | APE9-dist-out | 11.7226 | C488A,C584S | None | None | XRAY | 1.91 | 0.2 | 0.22 | B | 309.0 | 286.0 | 20 | 30 | 25 | 5 | [[478, 756]] | 1.0 | 5o49 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 5O49A | P11362 | 464 | 764 | 822.0 | 9K5:801 | Type1 | Inactive | DFGin | 5.2397 | 13.6382 | BLAplus | -124.98, 161.58 | 68.85, 20.17 | -74.75, -11.05 | 61.69, 77.84 | -110.93, 4.69 | in-out | in | 8.1254 | Saltbr-out | 5.5459 | HRD-in | -64.73, -48.02 | 76.28, -6.18 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.7824 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.25, 168.76 | APE9-dihe-in | -119.19, 119.01 | APE8-dihe-out | -64.8, -20.97 | APE8-rot-na | 343.93 | APE67-dihe-in | -73.72, -10.74 | -55.47, -23.05 | APE12-dist-na | 19.5652 | APE11-dist-na | 21.14 | APE10-dist-na | 19.4995 | APE9-dist-out | 11.833 | C488A,C584S | None | None | XRAY | 1.91 | 0.2 | 0.22 | A | 309.0 | 289.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5o49 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5O49B | P11362 | 460 | 765 | 822.0 | 9K5:801 | Type1 | Inactive | DFGin | 5.6188 | 12.9288 | BLAplus | -126.58, 172.58 | 67.38, 24.13 | -84.06, -18.33 | 50.82, 87.05 | -104.51, 13.86 | in-out | in | 7.6377 | Saltbr-out | 4.5004 | HRD-in | -61.81, -47.66 | 75.62, -5.93 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -110.43, 163.49 | APE9-dihe-in | -105.31, 114.78 | APE8-dihe-out | -56.47, -25.97 | APE8-rot-na | 333.8 | APE67-dihe-in | -70.86, -8.05 | -56.14, -23.8 | APE12-dist-na | 19.0124 | APE11-dist-na | 20.4124 | APE10-dist-na | 18.7866 | APE9-dist-out | 11.7226 | C488A,C584S | None | None | XRAY | 1.91 | 0.2 | 0.22 | B | 309.0 | 286.0 | 20 | 30 | 25 | 5 | [[478, 756]] | 1.0 | 5o49 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|