| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWLA | P11362 | 465 | 765 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2596 | 13.1901 | BLAplus | -120.07, 160.93 | 64.42, 29.27 | -80.33, -20.1 | 51.65, 89.33 | -96.98, 0.13 | in-in | in | 7.7737 | Saltbr-in | 2.9039 | HRD-in | -75.31, -52.96 | 79.05, -10.93 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.242 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -109.23, 163.46 | APE9-dihe-in | -103.38, 113.99 | APE8-dihe-out | -51.08, -26.28 | APE8-rot-na | 327.94 | APE67-dihe-in | -75.8, -7.21 | -59.7, -19.52 | APE12-dist-na | 19.715 | APE11-dist-na | 21.1796 | APE10-dist-na | 19.602 | APE9-dist-out | 11.6028 | C488A,C584S | None | None | XRAY | 2.193 | 0.209 | 0.256 | A | 317.0 | 282.0 | 19 | 30 | 27 | 3 | [[478, 756]] | 1.0 | 4rwl | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWLB | P11362 | 458 | 764 | 822.0 | 3ZC:801 | Type1.5_Back | Inactive | DFGin | 5.5749 | 12.8603 | BLBplus | -118.6, 158.89 | 63.82, 31.02 | -77.01, 152.77 | 46.13, 88.04 | 75.46, -144.53 | in-in | in | 7.8641 | Saltbr-in | 2.7141 | HRD-in | -76.64, -55.25 | 80.83, -9.47 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -108.43, 164.04 | APE9-dihe-in | -102.17, 112.77 | APE8-dihe-out | -51.59, -26.38 | APE8-rot-na | 327.68 | APE67-dihe-in | -76.33, -6.25 | -60.23, -17.85 | APE12-dist-na | 20.4616 | APE11-dist-na | 21.2659 | APE10-dist-na | 19.7485 | APE9-dist-out | 11.5255 | C488A,C584S | None | None | XRAY | 2.193 | 0.209 | 0.256 | B | 317.0 | 285.0 | 22 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4rwl | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWLA | P11362 | 465 | 765 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2596 | 13.1901 | BLAplus | -120.07, 160.93 | 64.42, 29.27 | -80.33, -20.1 | 51.65, 89.33 | -96.98, 0.13 | in-in | in | 7.7737 | Saltbr-in | 2.9039 | HRD-in | -75.31, -52.96 | 79.05, -10.93 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.242 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -109.23, 163.46 | APE9-dihe-in | -103.38, 113.99 | APE8-dihe-out | -51.08, -26.28 | APE8-rot-na | 327.94 | APE67-dihe-in | -75.8, -7.21 | -59.7, -19.52 | APE12-dist-na | 19.715 | APE11-dist-na | 21.1796 | APE10-dist-na | 19.602 | APE9-dist-out | 11.6028 | C488A,C584S | None | None | XRAY | 2.193 | 0.209 | 0.256 | A | 317.0 | 282.0 | 19 | 30 | 27 | 3 | [[478, 756]] | 1.0 | 4rwl | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWLB | P11362 | 458 | 764 | 822.0 | 3ZC:801 | Type1.5_Back | Inactive | DFGin | 5.5749 | 12.8603 | BLBplus | -118.6, 158.89 | 63.82, 31.02 | -77.01, 152.77 | 46.13, 88.04 | 75.46, -144.53 | in-in | in | 7.8641 | Saltbr-in | 2.7141 | HRD-in | -76.64, -55.25 | 80.83, -9.47 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -108.43, 164.04 | APE9-dihe-in | -102.17, 112.77 | APE8-dihe-out | -51.59, -26.38 | APE8-rot-na | 327.68 | APE67-dihe-in | -76.33, -6.25 | -60.23, -17.85 | APE12-dist-na | 20.4616 | APE11-dist-na | 21.2659 | APE10-dist-na | 19.7485 | APE9-dist-out | 11.5255 | C488A,C584S | None | None | XRAY | 2.193 | 0.209 | 0.256 | B | 317.0 | 285.0 | 22 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4rwl | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|