| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK10 | MK10_HUMAN | 4H3BA | P53779 | 45 | 400 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 4.7159 | 14.0293 | BLBplus | -123.41, 176.65 | 67.2, 22.96 | -66.31, 128.63 | 45.16, 92.75 | 81.86, 0.06 | in-in | in | 9.2114 | Saltbr-in | 2.8204 | HRD-in | -72.51, -55.43 | 76.6, -32.39 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.9841 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -127.64, 145.01 | APE9-dihe-na | -67.81, 151.17 | APE8-dihe-out | -78.78, -22.86 | APE8-rot-in | 318.88 | APE67-dihe-in | -63.25, -19.39 | -46.58, -43.53 | APE12-dist-out | 19.3539 | APE11-dist-out | 15.0583 | APE10-dist-out | 16.389 | APE9-dist-out | 10.9806 | None | None | None | XRAY | 2.08 | 0.187 | 0.235 | A | 356.0 | 351.0 | 5 | 27 | 27 | 0 | [[64, 359]] | 1.0 | 4h3b | CMGC_MAPK10_HUMAN | CMGC | 1.3e-85 | 293.2 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 4H3BC | P53779 | 45 | 400 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 4.6314 | 13.9911 | BLBplus | -121.69, 179.82 | 65.29, 21.46 | -67.38, 128.27 | 47.58, 92.38 | 80.35, 1.93 | in-in | in | 9.2365 | Saltbr-in | 2.9366 | HRD-in | -73.51, -54.45 | 77.5, -31.66 | in-out-out | SNCioo | out-out | ActLoopNT-out | 11.1023 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -132.97, 144.71 | APE9-dihe-na | -66.82, 150.47 | APE8-dihe-out | -80.28, -21.43 | APE8-rot-in | 321.01 | APE67-dihe-in | -63.29, -18.12 | -48.05, -42.67 | APE12-dist-out | 19.4345 | APE11-dist-out | 15.119 | APE10-dist-out | 16.3515 | APE9-dist-out | 10.9652 | None | None | None | XRAY | 2.08 | 0.187 | 0.235 | C | 356.0 | 351.0 | 5 | 27 | 27 | 0 | [[64, 359]] | 1.0 | 4h3b | CMGC_MAPK10_HUMAN | CMGC | 1.3e-85 | 293.2 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK10 | MK10_HUMAN | 4H3BA | P53779 | 45 | 400 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 4.7159 | 14.0293 | BLBplus | -123.41, 176.65 | 67.2, 22.96 | -66.31, 128.63 | 45.16, 92.75 | 81.86, 0.06 | in-in | in | 9.2114 | Saltbr-in | 2.8204 | HRD-in | -72.51, -55.43 | 76.6, -32.39 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.9841 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -127.64, 145.01 | APE9-dihe-na | -67.81, 151.17 | APE8-dihe-out | -78.78, -22.86 | APE8-rot-in | 318.88 | APE67-dihe-in | -63.25, -19.39 | -46.58, -43.53 | APE12-dist-out | 19.3539 | APE11-dist-out | 15.0583 | APE10-dist-out | 16.389 | APE9-dist-out | 10.9806 | None | None | None | XRAY | 2.08 | 0.187 | 0.235 | A | 356.0 | 351.0 | 5 | 27 | 27 | 0 | [[64, 359]] | 1.0 | 4h3b | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.3e-85 | 293.2 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 4H3BC | P53779 | 45 | 400 | 464.0 | No_ligand | No_ligand | Inactive | DFGin | 4.6314 | 13.9911 | BLBplus | -121.69, 179.82 | 65.29, 21.46 | -67.38, 128.27 | 47.58, 92.38 | 80.35, 1.93 | in-in | in | 9.2365 | Saltbr-in | 2.9366 | HRD-in | -73.51, -54.45 | 77.5, -31.66 | in-out-out | SNCioo | out-out | ActLoopNT-out | 11.1023 | ActLoopCT-out | nonTYR | APEdihe_aaoii | APEdist_oooo | APE10-dihe-na | -132.97, 144.71 | APE9-dihe-na | -66.82, 150.47 | APE8-dihe-out | -80.28, -21.43 | APE8-rot-in | 321.01 | APE67-dihe-in | -63.29, -18.12 | -48.05, -42.67 | APE12-dist-out | 19.4345 | APE11-dist-out | 15.119 | APE10-dist-out | 16.3515 | APE9-dist-out | 10.9652 | None | None | None | XRAY | 2.08 | 0.187 | 0.235 | C | 356.0 | 351.0 | 5 | 27 | 27 | 0 | [[64, 359]] | 1.0 | 4h3b | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.3e-85 | 293.2 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|