| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | BMX | BMX_HUMAN | 3SXRA | P51813 | 411 | 671 | 675.0 | 1N1:60001 | Type1 | Inactive | DFGinter | 7.8824 | 8.1671 | BABtrans | -93.57, 121.18 | -103.19, -9.04 | -51.22, 114.45 | 184.77, 74.21 | 62.74, 18.94 | out-out | out | 10.805 | Saltbr-out | 7.5586 | HRD-out | -99.0, 124.02 | -80.22, -7.53 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8353 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -95.14, 119.04 | APE9-dihe-in | -94.0, 160.01 | APE8-dihe-in | -48.96, 127.48 | APE8-rot-na | 331.52 | APE67-dihe-in | -68.66, -11.59 | -65.07, -24.25 | APE12-dist-na | 10.0286 | APE11-dist-na | 7.5492 | APE10-dist-na | 12.0421 | APE9-dist-in | 5.1857 | Q432K,Q611M,D617T,Q620E | None | None | XRAY | 2.4 | 0.189 | 0.231 | A | 268.0 | 257.0 | 4 | 29 | 29 | 0 | [[417, 668]] | 1.0 | 3sxr | TYR_BMX_HUMAN | TYR | 3.1e-93 | 317.8 | 1.0 | 260.0 | 260.0 | 553 | 554 | 555 | 557 | 559 | 445 | 460 | 464 | 533 | 535 | 534 | 536.0 | 594 | 582 | 577 | 576 | 575 | 574 | 573 | 572 | 571 | 490 | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BMX | BMX_HUMAN | 3SXRB | P51813 | 411 | 671 | 675.0 | 1N1:60002 | Type1 | Inactive | DFGinter | 7.7085 | 8.2724 | BABtrans | -92.79, 121.27 | -96.68, -12.13 | -49.05, 115.54 | 186.98, 71.37 | 61.78, 19.24 | out-out | out | 10.8028 | Saltbr-out | 8.0973 | HRD-out | -100.92, 124.05 | -80.64, -7.7 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8449 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -93.81, 125.57 | APE9-dihe-in | -101.37, 158.16 | APE8-dihe-in | -49.48, 128.1 | APE8-rot-na | 332.21 | APE67-dihe-in | -66.79, -11.14 | -62.63, -27.73 | APE12-dist-na | 9.9457 | APE11-dist-na | 7.4465 | APE10-dist-na | 11.9437 | APE9-dist-in | 5.1904 | Q432K,Q611M,D617T,Q620E | None | None | XRAY | 2.4 | 0.189 | 0.231 | B | 268.0 | 255.0 | 6 | 29 | 29 | 0 | [[417, 668]] | 1.0 | 3sxr | TYR_BMX_HUMAN | TYR | 3.1e-93 | 317.8 | 1.0 | 260.0 | 260.0 | 553 | 554 | 555 | 557 | 559 | 445 | 460 | 464 | 533 | 535 | 534 | 536.0 | 594 | 582 | 577 | 576 | 575 | 574 | 573 | 572 | 571 | 490 | Cytoplasmic tyrosine-protein kinase BMX |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | BMX | BMX_HUMAN | 3SXRA | P51813 | 411 | 671 | 675.0 | 1N1:60001 | Type1 | Inactive | DFGinter | 7.8824 | 8.1671 | BABtrans | -93.57, 121.18 | -103.19, -9.04 | -51.22, 114.45 | 184.77, 74.21 | 62.74, 18.94 | out-out | out | 10.805 | Saltbr-out | 7.5586 | HRD-out | -99.0, 124.02 | -80.22, -7.53 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8353 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -95.14, 119.04 | APE9-dihe-in | -94.0, 160.01 | APE8-dihe-in | -48.96, 127.48 | APE8-rot-na | 331.52 | APE67-dihe-in | -68.66, -11.59 | -65.07, -24.25 | APE12-dist-na | 10.0286 | APE11-dist-na | 7.5492 | APE10-dist-na | 12.0421 | APE9-dist-in | 5.1857 | Q432K,Q611M,D617T,Q620E | None | None | XRAY | 2.4 | 0.189 | 0.231 | A | 268.0 | 257.0 | 4 | 29 | 29 | 0 | [[417, 668]] | 1.0 | 3sxr | Homo sapiens | TYR_BMX_HUMAN | TYR | 3.1e-93 | 317.8 | 1.0 | 260.0 | 260.0 | 553 | 554 | 555 | 557 | 559 | 445 | 460 | 464 | 533 | 535 | 534 | 536.0 | 594 | 582 | 577 | 576 | 575 | 574 | 573 | 572 | 571 | 490 | Cytoplasmic tyrosine-protein kinase BMX |
| TYR | BMX | BMX_HUMAN | 3SXRB | P51813 | 411 | 671 | 675.0 | 1N1:60002 | Type1 | Inactive | DFGinter | 7.7085 | 8.2724 | BABtrans | -92.79, 121.27 | -96.68, -12.13 | -49.05, 115.54 | 186.98, 71.37 | 61.78, 19.24 | out-out | out | 10.8028 | Saltbr-out | 8.0973 | HRD-out | -100.92, 124.05 | -80.64, -7.7 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8449 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -93.81, 125.57 | APE9-dihe-in | -101.37, 158.16 | APE8-dihe-in | -49.48, 128.1 | APE8-rot-na | 332.21 | APE67-dihe-in | -66.79, -11.14 | -62.63, -27.73 | APE12-dist-na | 9.9457 | APE11-dist-na | 7.4465 | APE10-dist-na | 11.9437 | APE9-dist-in | 5.1904 | Q432K,Q611M,D617T,Q620E | None | None | XRAY | 2.4 | 0.189 | 0.231 | B | 268.0 | 255.0 | 6 | 29 | 29 | 0 | [[417, 668]] | 1.0 | 3sxr | Homo sapiens | TYR_BMX_HUMAN | TYR | 3.1e-93 | 317.8 | 1.0 | 260.0 | 260.0 | 553 | 554 | 555 | 557 | 559 | 445 | 460 | 464 | 533 | 535 | 534 | 536.0 | 594 | 582 | 577 | 576 | 575 | 574 | 573 | 572 | 571 | 490 | Cytoplasmic tyrosine-protein kinase BMX |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|