| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 3KY2A | P11362 | 458 | 764 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1417 | 13.3026 | BLAplus | -122.69, 172.32 | 46.54, 42.6 | -95.25, -13.81 | 55.54, 83.43 | -110.08, 21.37 | in-in | in | 7.9833 | Saltbr-in | 2.7043 | HRD-in | -54.04, -52.31 | 78.54, -4.33 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9047 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.74, 144.51 | APE9-dihe-in | -109.2, 106.89 | APE8-dihe-out | -56.11, -24.62 | APE8-rot-na | 329.61 | APE67-dihe-in | -74.45, -13.88 | -60.05, -25.51 | APE12-dist-na | 17.0264 | APE11-dist-na | 19.6184 | APE10-dist-na | 16.6111 | APE9-dist-out | 11.1393 | C488A,C584S | None | None | XRAY | 2.7 | 0.206 | 0.252 | A | 317.0 | 305.0 | 2 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3ky2 | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3KY2B | P11362 | 460 | 763 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.3065 | 13.1313 | BLAplus | -120.14, 165.15 | 53.12, 37.21 | -90.32, -21.71 | 57.04, 89.19 | -96.69, 4.05 | in-in | in | 7.7505 | Saltbr-in | 2.873 | HRD-in | -63.32, -45.74 | 74.66, -3.4 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -103.35, 149.7 | APE9-dihe-in | -86.12, 120.09 | APE8-dihe-out | -58.71, -15.12 | APE8-rot-na | 326.3 | APE67-dihe-in | -64.29, -14.63 | -68.37, -29.74 | APE12-dist-na | 19.9297 | APE11-dist-na | 21.2795 | APE10-dist-na | 19.8376 | APE9-dist-out | 11.7932 | C488A,C584S | None | None | XRAY | 2.7 | 0.206 | 0.252 | B | 317.0 | 280.0 | 24 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 3ky2 | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 3KY2A | P11362 | 458 | 764 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1417 | 13.3026 | BLAplus | -122.69, 172.32 | 46.54, 42.6 | -95.25, -13.81 | 55.54, 83.43 | -110.08, 21.37 | in-in | in | 7.9833 | Saltbr-in | 2.7043 | HRD-in | -54.04, -52.31 | 78.54, -4.33 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9047 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.74, 144.51 | APE9-dihe-in | -109.2, 106.89 | APE8-dihe-out | -56.11, -24.62 | APE8-rot-na | 329.61 | APE67-dihe-in | -74.45, -13.88 | -60.05, -25.51 | APE12-dist-na | 17.0264 | APE11-dist-na | 19.6184 | APE10-dist-na | 16.6111 | APE9-dist-out | 11.1393 | C488A,C584S | None | None | XRAY | 2.7 | 0.206 | 0.252 | A | 317.0 | 305.0 | 2 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3ky2 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3KY2B | P11362 | 460 | 763 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.3065 | 13.1313 | BLAplus | -120.14, 165.15 | 53.12, 37.21 | -90.32, -21.71 | 57.04, 89.19 | -96.69, 4.05 | in-in | in | 7.7505 | Saltbr-in | 2.873 | HRD-in | -63.32, -45.74 | 74.66, -3.4 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -103.35, 149.7 | APE9-dihe-in | -86.12, 120.09 | APE8-dihe-out | -58.71, -15.12 | APE8-rot-na | 326.3 | APE67-dihe-in | -64.29, -14.63 | -68.37, -29.74 | APE12-dist-na | 19.9297 | APE11-dist-na | 21.2795 | APE10-dist-na | 19.8376 | APE9-dist-out | 11.7932 | C488A,C584S | None | None | XRAY | 2.7 | 0.206 | 0.252 | B | 317.0 | 280.0 | 24 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 3ky2 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|