| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFA | P36897 | 171 | 500 | 503.0 | JZO:1 | Type1.5_Back | Active | DFGin | 6.1932 | 12.9048 | BLAminus | -150.7, 165.18 | 67.92, 79.43 | -90.06, 14.08 | 309.25, 11.69 | -44.14, -39.87 | in-in | in | 8.1956 | Saltbr-in | 2.8368 | HRD-in | -56.75, -49.06 | 70.7, 0.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9397 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -96.99, 164.53 | APE9-dihe-na | 104.66, 167.11 | APE8-dihe-in | -69.97, 124.0 | APE8-rot-in | 297.54 | APE67-dihe-in | -37.23, -57.4 | -40.07, -69.34 | APE12-dist-in | 11.4628 | APE11-dist-in | 12.1707 | APE10-dist-in | 6.1624 | APE9-dist-in | 3.7623 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | A | 342.0 | 328.0 | 2 | 32 | 30 | 2 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFB | P36897 | 171 | 501 | 503.0 | JZO:2 | Type1.5_Back | Active | DFGin | 6.0248 | 12.6274 | BLAminus | -135.28, -176.57 | 58.41, 88.07 | -103.95, 28.48 | 315.03, 7.91 | -62.87, -35.81 | in-in | in | 8.1446 | Saltbr-in | 2.6009 | HRD-in | -81.18, -54.27 | 77.68, -8.36 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9703 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.7, -176.11 | APE9-dihe-na | 95.21, 172.61 | APE8-dihe-in | -76.23, 133.32 | APE8-rot-in | 308.48 | APE67-dihe-in | -45.62, -25.89 | -46.72, -68.47 | APE12-dist-in | 11.5191 | APE11-dist-in | 11.4129 | APE10-dist-in | 5.9541 | APE9-dist-in | 3.7322 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | B | 342.0 | 324.0 | 7 | 32 | 29 | 3 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFC | P36897 | 171 | 500 | 503.0 | JZO:3 | Type1.5_Back | Active | DFGin | 6.6922 | 12.959 | BLAminus | -135.28, 165.04 | 69.33, 88.35 | -106.61, 31.51 | 302.0, 1.76 | -58.82, -55.68 | in-in | in | 8.0361 | Saltbr-in | 2.3791 | HRD-in | -81.96, -30.19 | 61.27, -12.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8972 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -114.43, -160.74 | APE9-dihe-na | 83.32, -178.05 | APE8-dihe-in | -94.01, 131.52 | APE8-rot-in | 317.12 | APE67-dihe-in | -41.44, -18.99 | -53.51, -67.7 | APE12-dist-in | 10.7421 | APE11-dist-in | 11.8422 | APE10-dist-in | 6.2245 | APE9-dist-in | 3.8557 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | C | 342.0 | 330.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFD | P36897 | 171 | 500 | 503.0 | JZO:4 | Type1.5_Back | Active | DFGin | 6.8886 | 12.9989 | BLAminus | -135.85, -173.78 | 57.12, 75.33 | -93.52, 22.15 | 298.91, 178.96 | -63.23, -14.31 | in-in | in | 8.2643 | Saltbr-in | 2.8937 | HRD-in | -62.47, -52.01 | 74.47, -2.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.771 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.66, 172.34 | APE9-dihe-na | 99.39, 173.59 | APE8-dihe-in | -80.33, 105.05 | APE8-rot-in | 316.25 | APE67-dihe-in | -46.61, -41.72 | -34.28, -49.6 | APE12-dist-in | 12.0425 | APE11-dist-in | 12.0502 | APE10-dist-in | 6.3267 | APE9-dist-in | 4.0441 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | D | 342.0 | 330.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFE | P36897 | 171 | 500 | 503.0 | JZO:5 | Type1.5_Back | Active | DFGin | 6.468 | 12.9815 | BLAminus | -143.17, -179.95 | 57.87, 88.27 | -108.02, 21.93 | 307.67, 3.89 | -69.37, -7.25 | in-in | in | 8.0283 | Saltbr-in | 2.8557 | HRD-in | -68.17, -50.18 | 73.66, 3.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9023 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.74, 177.4 | APE9-dihe-na | 104.24, -175.74 | APE8-dihe-in | -89.11, 123.84 | APE8-rot-in | 292.33 | APE67-dihe-in | -50.81, -36.21 | -50.11, -48.46 | APE12-dist-in | 9.931 | APE11-dist-in | 12.0011 | APE10-dist-in | 6.2167 | APE9-dist-in | 3.7965 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | E | 342.0 | 330.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | 3kcf | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFA | P36897 | 171 | 500 | 503.0 | JZO:1 | Type1.5_Back | Active | DFGin | 6.1932 | 12.9048 | BLAminus | -150.7, 165.18 | 67.92, 79.43 | -90.06, 14.08 | 309.25, 11.69 | -44.14, -39.87 | in-in | in | 8.1956 | Saltbr-in | 2.8368 | HRD-in | -56.75, -49.06 | 70.7, 0.3 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9397 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -96.99, 164.53 | APE9-dihe-na | 104.66, 167.11 | APE8-dihe-in | -69.97, 124.0 | APE8-rot-in | 297.54 | APE67-dihe-in | -37.23, -57.4 | -40.07, -69.34 | APE12-dist-in | 11.4628 | APE11-dist-in | 12.1707 | APE10-dist-in | 6.1624 | APE9-dist-in | 3.7623 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | A | 342.0 | 328.0 | 2 | 32 | 30 | 2 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFB | P36897 | 171 | 501 | 503.0 | JZO:2 | Type1.5_Back | Active | DFGin | 6.0248 | 12.6274 | BLAminus | -135.28, -176.57 | 58.41, 88.07 | -103.95, 28.48 | 315.03, 7.91 | -62.87, -35.81 | in-in | in | 8.1446 | Saltbr-in | 2.6009 | HRD-in | -81.18, -54.27 | 77.68, -8.36 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9703 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.7, -176.11 | APE9-dihe-na | 95.21, 172.61 | APE8-dihe-in | -76.23, 133.32 | APE8-rot-in | 308.48 | APE67-dihe-in | -45.62, -25.89 | -46.72, -68.47 | APE12-dist-in | 11.5191 | APE11-dist-in | 11.4129 | APE10-dist-in | 5.9541 | APE9-dist-in | 3.7322 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | B | 342.0 | 324.0 | 7 | 32 | 29 | 3 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFC | P36897 | 171 | 500 | 503.0 | JZO:3 | Type1.5_Back | Active | DFGin | 6.6922 | 12.959 | BLAminus | -135.28, 165.04 | 69.33, 88.35 | -106.61, 31.51 | 302.0, 1.76 | -58.82, -55.68 | in-in | in | 8.0361 | Saltbr-in | 2.3791 | HRD-in | -81.96, -30.19 | 61.27, -12.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8972 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -114.43, -160.74 | APE9-dihe-na | 83.32, -178.05 | APE8-dihe-in | -94.01, 131.52 | APE8-rot-in | 317.12 | APE67-dihe-in | -41.44, -18.99 | -53.51, -67.7 | APE12-dist-in | 10.7421 | APE11-dist-in | 11.8422 | APE10-dist-in | 6.2245 | APE9-dist-in | 3.8557 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | C | 342.0 | 330.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFD | P36897 | 171 | 500 | 503.0 | JZO:4 | Type1.5_Back | Active | DFGin | 6.8886 | 12.9989 | BLAminus | -135.85, -173.78 | 57.12, 75.33 | -93.52, 22.15 | 298.91, 178.96 | -63.23, -14.31 | in-in | in | 8.2643 | Saltbr-in | 2.8937 | HRD-in | -62.47, -52.01 | 74.47, -2.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.771 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.66, 172.34 | APE9-dihe-na | 99.39, 173.59 | APE8-dihe-in | -80.33, 105.05 | APE8-rot-in | 316.25 | APE67-dihe-in | -46.61, -41.72 | -34.28, -49.6 | APE12-dist-in | 12.0425 | APE11-dist-in | 12.0502 | APE10-dist-in | 6.3267 | APE9-dist-in | 4.0441 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | D | 342.0 | 330.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | 3KCFE | P36897 | 171 | 500 | 503.0 | JZO:5 | Type1.5_Back | Active | DFGin | 6.468 | 12.9815 | BLAminus | -143.17, -179.95 | 57.87, 88.27 | -108.02, 21.93 | 307.67, 3.89 | -69.37, -7.25 | in-in | in | 8.0283 | Saltbr-in | 2.8557 | HRD-in | -68.17, -50.18 | 73.66, 3.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9023 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.74, 177.4 | APE9-dihe-na | 104.24, -175.74 | APE8-dihe-in | -89.11, 123.84 | APE8-rot-in | 292.33 | APE67-dihe-in | -50.81, -36.21 | -50.11, -48.46 | APE12-dist-in | 9.931 | APE11-dist-in | 12.0011 | APE10-dist-in | 6.2167 | APE9-dist-in | 3.7965 | None | None | None | XRAY | 2.8 | 0.237 | 0.278 | E | 342.0 | 330.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | 3kcf | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 4.9e-85 | 291.2 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|