| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 3JS2A | P11362 | 464 | 765 | 822.0 | VM1:801 | Type1 | Inactive | DFGin | 5.153 | 13.3035 | BLAplus | -121.66, 167.26 | 60.21, 27.33 | -82.6, -17.8 | 54.2, 84.02 | -103.88, 10.59 | in-in | in | 7.7242 | Saltbr-in | 3.0512 | HRD-in | -72.72, -56.56 | 85.97, -17.24 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9689 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.37, 154.98 | APE9-dihe-in | -92.36, 117.27 | APE8-dihe-out | -54.75, -26.7 | APE8-rot-na | 329.63 | APE67-dihe-in | -71.32, -6.64 | -59.57, -19.47 | APE12-dist-na | 19.1598 | APE11-dist-na | 20.7834 | APE10-dist-na | 19.3186 | APE9-dist-out | 11.8143 | C488A,C584S | None | None | XRAY | 2.2 | 0.216 | 0.259 | A | 317.0 | 295.0 | 7 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3js2 | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3JS2B | P11362 | 459 | 762 | 822.0 | VM1:801 | Type1 | Inactive | DFGin | 5.166 | 12.9148 | BLAplus | -117.79, 168.89 | 57.38, 26.57 | -81.81, -21.58 | 58.31, 81.41 | -101.15, 4.46 | in-in | in | 7.4152 | Saltbr-in | 2.8977 | HRD-in | -70.61, -55.45 | 85.21, -19.22 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.3884 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -105.77, 164.88 | APE9-dihe-in | -101.88, 109.77 | APE8-dihe-out | -47.5, -33.8 | APE8-rot-na | 323.58 | APE67-dihe-in | -71.37, -10.85 | -58.97, -16.94 | APE12-dist-na | 19.4281 | APE11-dist-na | 20.9341 | APE10-dist-na | 19.561 | APE9-dist-out | 11.7757 | C488A,C584S | None | None | XRAY | 2.2 | 0.216 | 0.259 | B | 317.0 | 291.0 | 13 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3js2 | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 3JS2A | P11362 | 464 | 765 | 822.0 | VM1:801 | Type1 | Inactive | DFGin | 5.153 | 13.3035 | BLAplus | -121.66, 167.26 | 60.21, 27.33 | -82.6, -17.8 | 54.2, 84.02 | -103.88, 10.59 | in-in | in | 7.7242 | Saltbr-in | 3.0512 | HRD-in | -72.72, -56.56 | 85.97, -17.24 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9689 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.37, 154.98 | APE9-dihe-in | -92.36, 117.27 | APE8-dihe-out | -54.75, -26.7 | APE8-rot-na | 329.63 | APE67-dihe-in | -71.32, -6.64 | -59.57, -19.47 | APE12-dist-na | 19.1598 | APE11-dist-na | 20.7834 | APE10-dist-na | 19.3186 | APE9-dist-out | 11.8143 | C488A,C584S | None | None | XRAY | 2.2 | 0.216 | 0.259 | A | 317.0 | 295.0 | 7 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3js2 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3JS2B | P11362 | 459 | 762 | 822.0 | VM1:801 | Type1 | Inactive | DFGin | 5.166 | 12.9148 | BLAplus | -117.79, 168.89 | 57.38, 26.57 | -81.81, -21.58 | 58.31, 81.41 | -101.15, 4.46 | in-in | in | 7.4152 | Saltbr-in | 2.8977 | HRD-in | -70.61, -55.45 | 85.21, -19.22 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.3884 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -105.77, 164.88 | APE9-dihe-in | -101.88, 109.77 | APE8-dihe-out | -47.5, -33.8 | APE8-rot-na | 323.58 | APE67-dihe-in | -71.37, -10.85 | -58.97, -16.94 | APE12-dist-na | 19.4281 | APE11-dist-na | 20.9341 | APE10-dist-na | 19.561 | APE9-dist-out | 11.7757 | C488A,C584S | None | None | XRAY | 2.2 | 0.216 | 0.259 | B | 317.0 | 291.0 | 13 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3js2 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|