| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 3G0FA | P10721 | 566 | 930 | 976.0 | B49:9001 | Type1 | Inactive | DFGout | 15.9324 | 11.0239 | BBAminus | -133.24, 143.68 | -91.38, 106.1 | -85.13, 9.55 | 260.45, 86.5 | -43.92, 131.31 | in-in | in | 7.3079 | Saltbr-in | 2.8577 | HRD-out | -104.98, 124.53 | -81.9, 0.65 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.723 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -98.6, 122.46 | APE9-dihe-in | -125.81, 152.57 | APE8-dihe-in | -80.31, 82.53 | APE8-rot-na | 33.57 | APE67-dihe-in | -64.38, -18.09 | -77.28, -33.89 | APE12-dist-na | 17.5119 | APE11-dist-na | 13.7561 | APE10-dist-na | 12.6611 | APE9-dist-in | 7.4975 | D816H | None | None | XRAY | 2.6 | 0.212 | 0.255 | A | 336.0 | 291.0 | 16 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 3g0f | TYR_KIT_HUMAN | TYR | 9.5e-102 | 346.0 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 3G0FB | P10721 | 564 | 930 | 976.0 | B49:9001 | Type1 | Inactive | DFGout | 16.0247 | 10.6077 | BBAminus | -141.97, 146.96 | -100.97, 117.58 | -98.35, 1.5 | 249.66, 85.76 | -37.59, 131.92 | in-in | in | 7.3721 | Saltbr-in | 2.8397 | HRD-out | -103.28, 116.42 | -91.73, 18.13 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.63 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.56, 113.86 | APE9-dihe-in | -119.17, 158.81 | APE8-dihe-in | -86.16, 69.24 | APE8-rot-na | 31.3 | APE67-dihe-in | -71.68, -15.15 | -66.98, -25.93 | APE12-dist-na | 16.5739 | APE11-dist-na | 13.4731 | APE10-dist-na | 12.1304 | APE9-dist-in | 7.1921 | D816H | None | None | XRAY | 2.6 | 0.212 | 0.255 | B | 336.0 | 293.0 | 16 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 3g0f | TYR_KIT_HUMAN | TYR | 9.5e-102 | 346.0 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 3G0FA | P10721 | 566 | 930 | 976.0 | B49:9001 | Type1 | Inactive | DFGout | 15.9324 | 11.0239 | BBAminus | -133.24, 143.68 | -91.38, 106.1 | -85.13, 9.55 | 260.45, 86.5 | -43.92, 131.31 | in-in | in | 7.3079 | Saltbr-in | 2.8577 | HRD-out | -104.98, 124.53 | -81.9, 0.65 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.723 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -98.6, 122.46 | APE9-dihe-in | -125.81, 152.57 | APE8-dihe-in | -80.31, 82.53 | APE8-rot-na | 33.57 | APE67-dihe-in | -64.38, -18.09 | -77.28, -33.89 | APE12-dist-na | 17.5119 | APE11-dist-na | 13.7561 | APE10-dist-na | 12.6611 | APE9-dist-in | 7.4975 | D816H | None | None | XRAY | 2.6 | 0.212 | 0.255 | A | 336.0 | 291.0 | 16 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 3g0f | Homo sapiens | TYR_KIT_HUMAN | TYR | 9.5e-102 | 346.0 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 3G0FB | P10721 | 564 | 930 | 976.0 | B49:9001 | Type1 | Inactive | DFGout | 16.0247 | 10.6077 | BBAminus | -141.97, 146.96 | -100.97, 117.58 | -98.35, 1.5 | 249.66, 85.76 | -37.59, 131.92 | in-in | in | 7.3721 | Saltbr-in | 2.8397 | HRD-out | -103.28, 116.42 | -91.73, 18.13 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.63 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.56, 113.86 | APE9-dihe-in | -119.17, 158.81 | APE8-dihe-in | -86.16, 69.24 | APE8-rot-na | 31.3 | APE67-dihe-in | -71.68, -15.15 | -66.98, -25.93 | APE12-dist-na | 16.5739 | APE11-dist-na | 13.4731 | APE10-dist-na | 12.1304 | APE9-dist-in | 7.1921 | D816H | None | None | XRAY | 2.6 | 0.212 | 0.255 | B | 336.0 | 293.0 | 16 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 3g0f | Homo sapiens | TYR_KIT_HUMAN | TYR | 9.5e-102 | 346.0 | 1.0 | 260.0 | 260.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|