| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | INSR | INSR_HUMAN | 3ETAA | P06213 | 1017 | 1310 | 1382.0 | 351:62001 | Type2 | Inactive | DFGout | 15.7961 | 11.0134 | BBAminus | -132.13, -174.21 | -157.85, 103.42 | -76.03, -16.02 | 293.96, 86.44 | 92.76, -168.27 | in-in | in | 8.3215 | Saltbr-in | 2.7567 | HRD-in | -66.68, -47.32 | 76.44, -15.87 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8262 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -58.11, 133.17 | APE9-dihe-in | -138.51, 142.25 | APE8-dihe-in | -82.26, 68.13 | APE8-rot-na | 29.26 | APE67-dihe-in | -71.63, -9.4 | -61.34, -31.95 | APE12-dist-na | 14.3031 | APE11-dist-na | 10.2115 | APE10-dist-na | 6.0412 | APE9-dist-in | 7.1449 | None | None | None | XRAY | 2.6 | 0.203 | 0.232 | A | 317.0 | 293.0 | 1 | 30 | 29 | 1 | [[1023, 1292]] | 1.0 | 3eta | TYR_INSR_HUMAN | TYR | 1.6e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| TYR | INSR | INSR_HUMAN | 3ETAB | P06213 | 1017 | 1310 | 1382.0 | 351:62001 | Type2 | Inactive | DFGout | 15.9171 | 11.1754 | BBAminus | -133.15, -176.66 | -152.04, 106.96 | -74.04, -41.1 | 283.79, 91.95 | 126.4, -175.96 | in-in | in | 8.351 | Saltbr-in | 3.1113 | HRD-in | -71.49, -47.77 | 78.43, -20.3 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8821 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.8, 131.91 | APE9-dihe-in | -139.37, 136.91 | APE8-dihe-in | -77.51, 68.63 | APE8-rot-na | 28.59 | APE67-dihe-in | -74.17, -10.01 | -54.55, -36.82 | APE12-dist-na | 14.3265 | APE11-dist-na | 10.1734 | APE10-dist-na | 5.8956 | APE9-dist-in | 7.247 | None | None | None | XRAY | 2.6 | 0.203 | 0.232 | B | 317.0 | 292.0 | 2 | 30 | 28 | 2 | [[1023, 1292]] | 1.0 | 3eta | TYR_INSR_HUMAN | TYR | 1.6e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | INSR | INSR_HUMAN | 3ETAA | P06213 | 1017 | 1310 | 1382.0 | 351:62001 | Type2 | Inactive | DFGout | 15.7961 | 11.0134 | BBAminus | -132.13, -174.21 | -157.85, 103.42 | -76.03, -16.02 | 293.96, 86.44 | 92.76, -168.27 | in-in | in | 8.3215 | Saltbr-in | 2.7567 | HRD-in | -66.68, -47.32 | 76.44, -15.87 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8262 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -58.11, 133.17 | APE9-dihe-in | -138.51, 142.25 | APE8-dihe-in | -82.26, 68.13 | APE8-rot-na | 29.26 | APE67-dihe-in | -71.63, -9.4 | -61.34, -31.95 | APE12-dist-na | 14.3031 | APE11-dist-na | 10.2115 | APE10-dist-na | 6.0412 | APE9-dist-in | 7.1449 | None | None | None | XRAY | 2.6 | 0.203 | 0.232 | A | 317.0 | 293.0 | 1 | 30 | 29 | 1 | [[1023, 1292]] | 1.0 | 3eta | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.6e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| TYR | INSR | INSR_HUMAN | 3ETAB | P06213 | 1017 | 1310 | 1382.0 | 351:62001 | Type2 | Inactive | DFGout | 15.9171 | 11.1754 | BBAminus | -133.15, -176.66 | -152.04, 106.96 | -74.04, -41.1 | 283.79, 91.95 | 126.4, -175.96 | in-in | in | 8.351 | Saltbr-in | 3.1113 | HRD-in | -71.49, -47.77 | 78.43, -20.3 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8821 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.8, 131.91 | APE9-dihe-in | -139.37, 136.91 | APE8-dihe-in | -77.51, 68.63 | APE8-rot-na | 28.59 | APE67-dihe-in | -74.17, -10.01 | -54.55, -36.82 | APE12-dist-na | 14.3265 | APE11-dist-na | 10.1734 | APE10-dist-na | 5.8956 | APE9-dist-in | 7.247 | None | None | None | XRAY | 2.6 | 0.203 | 0.232 | B | 317.0 | 292.0 | 2 | 30 | 28 | 2 | [[1023, 1292]] | 1.0 | 3eta | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.6e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|