| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK10 | MK10_HUMAN | 2R9SA | P53779 | 46 | 401 | 464.0 | 255:502 | Type1 | Inactive | DFGin | 3.9409 | 13.4254 | ABAminus | -77.42, -30.98 | -148.5, -179.18 | -116.23, 5.52 | 300.46, 90.99 | 75.53, -150.76 | in-in | in | 8.7129 | Saltbr-in | 2.8395 | HRD-in | -76.22, -69.01 | 82.11, -12.83 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -61.42, -24.81 | 999.0, 139.49 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | OCY154,OCY175,OCY201 | XRAY | 2.4 | 0.209 | 0.29 | A | 356.0 | 328.0 | 15 | 27 | 12 | 15 | [[64, 359]] | 1.0 | 2r9s | CMGC_MAPK10_HUMAN | CMGC | 1.3e-85 | 293.2 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 2R9SB | P53779 | 46 | 401 | 464.0 | 255:501 | Type1 | Inactive | DFGin | 3.9858 | 13.5505 | ABAminus | -79.38, -32.11 | -143.61, -178.83 | -118.88, 2.05 | 295.67, 88.66 | 84.96, -147.54 | in-in | in | 8.8067 | Saltbr-in | 2.9723 | HRD-in | -81.84, -63.74 | 74.18, -13.93 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -56.16, -23.99 | 999.0, -56.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | OCY154,OCY175,OCY201 | XRAY | 2.4 | 0.209 | 0.29 | B | 356.0 | 328.0 | 15 | 27 | 12 | 15 | [[64, 359]] | 1.0 | 2r9s | CMGC_MAPK10_HUMAN | CMGC | 1.3e-85 | 293.2 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK10 | MK10_HUMAN | 2R9SA | P53779 | 46 | 401 | 464.0 | 255:502 | Type1 | Inactive | DFGin | 3.9409 | 13.4254 | ABAminus | -77.42, -30.98 | -148.5, -179.18 | -116.23, 5.52 | 300.46, 90.99 | 75.53, -150.76 | in-in | in | 8.7129 | Saltbr-in | 2.8395 | HRD-in | -76.22, -69.01 | 82.11, -12.83 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -61.42, -24.81 | 999.0, 139.49 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | OCY154,OCY175,OCY201 | XRAY | 2.4 | 0.209 | 0.29 | A | 356.0 | 328.0 | 15 | 27 | 12 | 15 | [[64, 359]] | 1.0 | 2r9s | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.3e-85 | 293.2 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 2R9SB | P53779 | 46 | 401 | 464.0 | 255:501 | Type1 | Inactive | DFGin | 3.9858 | 13.5505 | ABAminus | -79.38, -32.11 | -143.61, -178.83 | -118.88, 2.05 | 295.67, 88.66 | 84.96, -147.54 | in-in | in | 8.8067 | Saltbr-in | 2.9723 | HRD-in | -81.84, -63.74 | 74.18, -13.93 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -56.16, -23.99 | 999.0, -56.19 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | OCY154,OCY175,OCY201 | XRAY | 2.4 | 0.209 | 0.29 | B | 356.0 | 328.0 | 15 | 27 | 12 | 15 | [[64, 359]] | 1.0 | 2r9s | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.3e-85 | 293.2 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|