| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK6 | GRK6_HUMAN | 2ACXA | P43250 | 14 | 532 | 576.0 | ANP:577 | ATPlike | Active | DFGin | 6.2066 | 13.2835 | BLAminus | -133.82, 164.79 | 58.79, 76.03 | -96.19, 24.41 | 281.42, 82.4 | -59.68, -24.05 | in-in | in | 9.3415 | Saltbr-in | 3.2194 | HRD-in | -78.26, -56.85 | 77.2, -1.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9714 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.49, 157.4 | APE9-dihe-na | 123.02, -168.26 | APE8-dihe-in | -95.03, 140.31 | APE8-rot-in | 303.17 | APE67-dihe-in | -86.56, -0.13 | -45.11, -52.69 | APE12-dist-in | 10.4784 | APE11-dist-in | 11.834 | APE10-dist-in | 6.0832 | APE9-dist-in | 3.9058 | C561S,C562S,C565S | None | None | XRAY | 2.6 | 0.204 | 0.243 | A | 576.0 | 495.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 2acx | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| AGC | GRK6 | GRK6_HUMAN | 2ACXB | P43250 | 14 | 535 | 576.0 | ANP:577 | ATPlike | Active | DFGin | 6.0903 | 13.1455 | BLAminus | -128.37, 163.87 | 55.35, 87.14 | -100.56, 21.26 | 285.61, 77.77 | -55.4, -30.56 | in-in | in | 9.2313 | Saltbr-in | 2.4394 | HRD-in | -77.3, -59.12 | 75.78, 1.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9766 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.83, 161.38 | APE9-dihe-na | 125.99, -167.44 | APE8-dihe-in | -95.89, 144.8 | APE8-rot-in | 307.19 | APE67-dihe-in | -70.72, -14.39 | -48.06, -55.51 | APE12-dist-in | 10.4768 | APE11-dist-in | 11.8719 | APE10-dist-in | 6.1674 | APE9-dist-in | 3.7096 | C561S,C562S,C565S | None | None | XRAY | 2.6 | 0.204 | 0.243 | B | 576.0 | 492.0 | 5 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 2acx | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK6 | GRK6_HUMAN | 2ACXA | P43250 | 14 | 532 | 576.0 | ANP:577 | ATPlike | Active | DFGin | 6.2066 | 13.2835 | BLAminus | -133.82, 164.79 | 58.79, 76.03 | -96.19, 24.41 | 281.42, 82.4 | -59.68, -24.05 | in-in | in | 9.3415 | Saltbr-in | 3.2194 | HRD-in | -78.26, -56.85 | 77.2, -1.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9714 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.49, 157.4 | APE9-dihe-na | 123.02, -168.26 | APE8-dihe-in | -95.03, 140.31 | APE8-rot-in | 303.17 | APE67-dihe-in | -86.56, -0.13 | -45.11, -52.69 | APE12-dist-in | 10.4784 | APE11-dist-in | 11.834 | APE10-dist-in | 6.0832 | APE9-dist-in | 3.9058 | C561S,C562S,C565S | None | None | XRAY | 2.6 | 0.204 | 0.243 | A | 576.0 | 495.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 2acx | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| AGC | GRK6 | GRK6_HUMAN | 2ACXB | P43250 | 14 | 535 | 576.0 | ANP:577 | ATPlike | Active | DFGin | 6.0903 | 13.1455 | BLAminus | -128.37, 163.87 | 55.35, 87.14 | -100.56, 21.26 | 285.61, 77.77 | -55.4, -30.56 | in-in | in | 9.2313 | Saltbr-in | 2.4394 | HRD-in | -77.3, -59.12 | 75.78, 1.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9766 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.83, 161.38 | APE9-dihe-na | 125.99, -167.44 | APE8-dihe-in | -95.89, 144.8 | APE8-rot-in | 307.19 | APE67-dihe-in | -70.72, -14.39 | -48.06, -55.51 | APE12-dist-in | 10.4768 | APE11-dist-in | 11.8719 | APE10-dist-in | 6.1674 | APE9-dist-in | 3.7096 | C561S,C562S,C565S | None | None | XRAY | 2.6 | 0.204 | 0.243 | B | 576.0 | 492.0 | 5 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 2acx | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|