Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 8GB4A | P00533 | 700 | 1007 | 1210.0 | ANP:1102,YW5:1103 | ATPlike,Type3 | Inactive | DFGin | 4.738 | 14.778 | BLBplus | -140.96, 174.92 | 57.37, 44.23 | -99.53, 158.98 | 50.67, 86.24 | 74.62, 16.37 | out-out | out | 13.355 | Saltbr-out | 11.698 | HRD-in | -69.91, -59.18 | 79.33, -9.52 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 127.01 | APE8-dihe-in | -76.27, 67.14 | APE8-rot-na | 30.24 | APE67-dihe-in | -75.65, -5.48 | -58.37, -41.11 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.058 | T790M,V948R | None | None | XRAY | 2.59 | 0.23 | 0.254 | A | 331 | 292 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 8gb4 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GB4B | P00533 | 700 | 1007 | 1210.0 | ANP:1102,YW5:1103 | ATPlike,Type3 | Inactive | DFGin | 4.858 | 14.681 | BLBplus | -140.61, 174.15 | 57.09, 43.59 | -100.33, 162.57 | 51.99, 86.76 | 77.41, 18.84 | out-out | out | 13.39 | Saltbr-out | 10.531 | HRD-in | -69.24, -58.17 | 79.24, -10.08 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 66.16 | APE8-rot-na | 30.06 | APE67-dihe-in | -75.09, -5.85 | -58.81, -39.96 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | T790M,V948R | None | None | XRAY | 2.59 | 0.23 | 0.254 | B | 331 | 290 | 18 | 0 | 0 | 18 | [[712, 970]] | 1.0 | 8gb4 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GB4C | P00533 | 700 | 1012 | 1210.0 | ANP:1102,YW5:1103 | ATPlike,Type3 | Inactive | DFGin | 4.732 | 14.602 | BLBplus | -141.16, 174.43 | 57.44, 44.8 | -99.46, 158.79 | 49.11, 85.48 | 74.36, 22.53 | out-out | out | 13.185 | Saltbr-out | 11.537 | HRD-in | -70.07, -59.0 | 77.64, -8.57 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 127.65 | APE8-dihe-in | -76.99, 66.94 | APE8-rot-na | 30.24 | APE67-dihe-in | -75.42, -5.6 | -59.05, -41.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.014 | T790M,V948R | None | None | XRAY | 2.59 | 0.23 | 0.254 | C | 331 | 297 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 8gb4 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GB4D | P00533 | 700 | 1007 | 1210.0 | ANP:1102,YW5:1103 | ATPlike,Type3 | Inactive | DFGin | 4.686 | 14.698 | BLBplus | -141.21, 175.0 | 57.29, 43.49 | -99.79, 159.92 | 51.61, 87.18 | 76.57, 22.15 | out-out | out | 13.561 | Saltbr-out | 10.91 | HRD-in | -69.19, -58.43 | 79.07, -10.45 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 65.97 | APE8-rot-na | 30.21 | APE67-dihe-in | -74.96, -5.48 | -59.31, -40.09 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | T790M,V948R | None | None | XRAY | 2.59 | 0.23 | 0.254 | D | 331 | 291 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gb4 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5A | P00533 | 701 | 1011 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.808 | 14.912 | BLBplus | -132.77, 163.28 | 59.53, 50.36 | -94.02, 166.24 | 50.17, 88.29 | 66.49, 24.24 | out-out | out | 13.127 | Saltbr-out | 9.96 | HRD-in | -72.38, -54.99 | 79.4, -8.54 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 131.66 | APE8-dihe-in | -80.77, 69.75 | APE8-rot-na | 32.13 | APE67-dihe-in | -76.82, -3.31 | -58.55, -37.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.087 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | A | 331 | 294 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gk5 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5B | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.513 | 14.722 | BLBplus | -133.17, 164.36 | 59.73, 51.31 | -91.4, 162.53 | 47.93, 87.21 | 64.33, 22.83 | out-out | out | 13.093 | Saltbr-out | 12.438 | HRD-in | -72.73, -55.9 | 79.15, -8.43 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 131.91 | APE8-dihe-in | -79.02, 69.83 | APE8-rot-na | 32.01 | APE67-dihe-in | -76.26, -3.86 | -58.1, -38.17 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.867 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | B | 331 | 292 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gk5 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5C | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.465 | 14.758 | BLBplus | -134.6, 164.78 | 60.76, 50.7 | -93.92, 162.62 | 46.93, 87.83 | 64.54, 21.99 | out-out | out | 13.135 | Saltbr-out | 11.494 | HRD-in | -72.37, -55.98 | 79.27, -6.85 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.09 | APE8-dihe-in | -76.74, 68.64 | APE8-rot-na | 31.76 | APE67-dihe-in | -75.53, -4.34 | -59.95, -38.1 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.102 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | C | 331 | 293 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 8gk5 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5D | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.407 | 14.729 | BLBplus | -134.17, 163.98 | 61.67, 51.99 | -93.03, 163.58 | 47.55, 87.87 | 65.01, 22.54 | out-out | out | 13.091 | Saltbr-out | 12.29 | HRD-in | -70.88, -54.33 | 77.76, -8.04 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -1.54 | APE9-dihe-in | -75.57, 134.88 | APE8-dihe-in | -77.01, 71.98 | APE8-rot-na | 32.06 | APE67-dihe-in | -76.98, -3.79 | -58.78, -38.58 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.721 | APE9-dist-in | 7.558 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | D | 331 | 294 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 8gk5 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 8GB4A | P00533 | 700 | 1007 | 1210.0 | ANP:1102,YW5:1103 | ATPlike,Type3 | Inactive | DFGin | 4.738 | 14.778 | BLBplus | -140.96, 174.92 | 57.37, 44.23 | -99.53, 158.98 | 50.67, 86.24 | 74.62, 16.37 | out-out | out | 13.355 | Saltbr-out | 11.698 | HRD-in | -69.91, -59.18 | 79.33, -9.52 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 127.01 | APE8-dihe-in | -76.27, 67.14 | APE8-rot-na | 30.24 | APE67-dihe-in | -75.65, -5.48 | -58.37, -41.11 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.058 | T790M,V948R | None | None | XRAY | 2.59 | 0.23 | 0.254 | A | 331 | 292 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 8gb4 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GB4B | P00533 | 700 | 1007 | 1210.0 | ANP:1102,YW5:1103 | ATPlike,Type3 | Inactive | DFGin | 4.858 | 14.681 | BLBplus | -140.61, 174.15 | 57.09, 43.59 | -100.33, 162.57 | 51.99, 86.76 | 77.41, 18.84 | out-out | out | 13.39 | Saltbr-out | 10.531 | HRD-in | -69.24, -58.17 | 79.24, -10.08 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 66.16 | APE8-rot-na | 30.06 | APE67-dihe-in | -75.09, -5.85 | -58.81, -39.96 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | T790M,V948R | None | None | XRAY | 2.59 | 0.23 | 0.254 | B | 331 | 290 | 18 | 0 | 0 | 18 | [[712, 970]] | 1.0 | 8gb4 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GB4C | P00533 | 700 | 1012 | 1210.0 | ANP:1102,YW5:1103 | ATPlike,Type3 | Inactive | DFGin | 4.732 | 14.602 | BLBplus | -141.16, 174.43 | 57.44, 44.8 | -99.46, 158.79 | 49.11, 85.48 | 74.36, 22.53 | out-out | out | 13.185 | Saltbr-out | 11.537 | HRD-in | -70.07, -59.0 | 77.64, -8.57 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 127.65 | APE8-dihe-in | -76.99, 66.94 | APE8-rot-na | 30.24 | APE67-dihe-in | -75.42, -5.6 | -59.05, -41.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.014 | T790M,V948R | None | None | XRAY | 2.59 | 0.23 | 0.254 | C | 331 | 297 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 8gb4 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GB4D | P00533 | 700 | 1007 | 1210.0 | ANP:1102,YW5:1103 | ATPlike,Type3 | Inactive | DFGin | 4.686 | 14.698 | BLBplus | -141.21, 175.0 | 57.29, 43.49 | -99.79, 159.92 | 51.61, 87.18 | 76.57, 22.15 | out-out | out | 13.561 | Saltbr-out | 10.91 | HRD-in | -69.19, -58.43 | 79.07, -10.45 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 65.97 | APE8-rot-na | 30.21 | APE67-dihe-in | -74.96, -5.48 | -59.31, -40.09 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | T790M,V948R | None | None | XRAY | 2.59 | 0.23 | 0.254 | D | 331 | 291 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gb4 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5A | P00533 | 701 | 1011 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.808 | 14.912 | BLBplus | -132.77, 163.28 | 59.53, 50.36 | -94.02, 166.24 | 50.17, 88.29 | 66.49, 24.24 | out-out | out | 13.127 | Saltbr-out | 9.96 | HRD-in | -72.38, -54.99 | 79.4, -8.54 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 131.66 | APE8-dihe-in | -80.77, 69.75 | APE8-rot-na | 32.13 | APE67-dihe-in | -76.82, -3.31 | -58.55, -37.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.087 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | A | 331 | 294 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gk5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5B | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.513 | 14.722 | BLBplus | -133.17, 164.36 | 59.73, 51.31 | -91.4, 162.53 | 47.93, 87.21 | 64.33, 22.83 | out-out | out | 13.093 | Saltbr-out | 12.438 | HRD-in | -72.73, -55.9 | 79.15, -8.43 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 131.91 | APE8-dihe-in | -79.02, 69.83 | APE8-rot-na | 32.01 | APE67-dihe-in | -76.26, -3.86 | -58.1, -38.17 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.867 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | B | 331 | 292 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gk5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5C | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.465 | 14.758 | BLBplus | -134.6, 164.78 | 60.76, 50.7 | -93.92, 162.62 | 46.93, 87.83 | 64.54, 21.99 | out-out | out | 13.135 | Saltbr-out | 11.494 | HRD-in | -72.37, -55.98 | 79.27, -6.85 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.09 | APE8-dihe-in | -76.74, 68.64 | APE8-rot-na | 31.76 | APE67-dihe-in | -75.53, -4.34 | -59.95, -38.1 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.102 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | C | 331 | 293 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 8gk5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5D | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.407 | 14.729 | BLBplus | -134.17, 163.98 | 61.67, 51.99 | -93.03, 163.58 | 47.55, 87.87 | 65.01, 22.54 | out-out | out | 13.091 | Saltbr-out | 12.29 | HRD-in | -70.88, -54.33 | 77.76, -8.04 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -1.54 | APE9-dihe-in | -75.57, 134.88 | APE8-dihe-in | -77.01, 71.98 | APE8-rot-na | 32.06 | APE67-dihe-in | -76.98, -3.79 | -58.78, -38.58 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.721 | APE9-dist-in | 7.558 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | D | 331 | 294 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 8gk5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|