Ligand: WAK

Total number of chains: 3
Active chains: 2
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 3 100.0% 8P05A

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
CMGC CLK1 CLK1_HUMAN 8P04A 2.6 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaono APEdist_nnni WAK Type1 148 - 481 0 None None Dual specificity protein kinase CLK1
CMGC CSNK2A1 CSK21_HUMAN 8P05A 2.45 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii WAK Type1 2 - 330 0 None None Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 8P05B 2.45 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii WAK Type1 3 - 330 0 None None Casein kinase II subunit alpha

Ligand: WAK

Total number of chains: 3
Active chains: 2
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 3 100.0% 8P05A

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
CMGC CLK1 CLK1_HUMAN 8P04A 2.6 Inactive DFGin‑BLAminus in-in in-out nonTYR APEdihe_aaono APEdist_nnni WAK Type1 148 - 481 0 None None Dual specificity protein kinase CLK1 Homo sapiens
CMGC CSNK2A1 CSK21_HUMAN 8P05A 2.45 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii WAK Type1 2 - 330 0 None None Casein kinase II subunit alpha Homo sapiens
CMGC CSNK2A1 CSK21_HUMAN 8P05B 2.45 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii WAK Type1 3 - 330 0 None None Casein kinase II subunit alpha Homo sapiens

Ligand: WAK

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism