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| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 7JXQB | P00533 | 701 | 1007 | 1210.0 | ANP:1102,VNS:1103 | ATPlike,Type3 | Inactive | DFGin | 4.915 | 14.438 | BLBplus | -136.8, 171.78 | 58.87, 35.86 | -91.33, 162.29 | 51.51, 87.21 | 80.67, 16.0 | out-out | out | 13.335 | Saltbr-out | 12.698 | HRD-in | -67.21, -58.71 | 77.88, -12.51 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.896 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -177.71 | APE9-dihe-in | -105.47, 135.84 | APE8-dihe-in | -83.2, 67.78 | APE8-rot-na | 33.37 | APE67-dihe-in | -74.22, -7.65 | -49.73, -41.79 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.734 | APE9-dist-in | 7.645 | T790M,V948R | None | None | XRAY | 1.83 | 0.185 | 0.218 | B | 331 | 297 | 10 | 0 | 0 | 10 | [[712, 970]] | 1.0 | 7jxq | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXQD | P00533 | 700 | 1007 | 1210.0 | ANP:1102,VNS:1103 | ATPlike,Type3 | Inactive | DFGin | 4.844 | 14.328 | BLBplus | -136.14, 172.56 | 58.98, 36.18 | -92.84, 162.13 | 51.55, 88.05 | 79.36, 17.26 | out-out | out | 13.42 | Saltbr-out | 11.89 | HRD-in | -65.12, -58.0 | 78.92, -12.53 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.94 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.09 | APE8-dihe-in | -80.19, 68.24 | APE8-rot-na | 33.29 | APE67-dihe-in | -74.77, -5.19 | -50.69, -44.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.579 | T790M,V948R | None | None | XRAY | 1.83 | 0.185 | 0.218 | D | 331 | 298 | 10 | 0 | 0 | 10 | [[712, 970]] | 1.0 | 7jxq | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1IA | P00533 | 700 | 1007 | 1210.0 | ANP:1102,VNS:1103 | ATPlike,Type3 | Inactive | DFGin | 4.837 | 14.412 | BLBplus | -124.92, 173.52 | 55.34, 38.4 | -93.27, 168.4 | 51.69, 86.03 | 70.99, 11.24 | out-out | out | 13.596 | Saltbr-out | 12.212 | HRD-in | -68.02, -55.76 | 76.66, -7.58 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 142.86 | APE8-dihe-in | -84.0, 73.03 | APE8-rot-na | 29.2 | APE67-dihe-in | -72.27, -9.54 | -58.41, -42.03 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.42 | L858R,V948R | None | None | XRAY | 3.202 | 0.266 | 0.311 | A | 331 | 288 | 20 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7k1i | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXWA | P00533 | 700 | 1007 | 1210.0 | YY3:1301,VNS:1302 | Type1,Type3 | Inactive | DFGin | 4.579 | 14.666 | BLBplus | -138.64, 168.46 | 50.29, 44.7 | -88.71, 170.77 | 52.75, 84.47 | 69.65, 17.94 | out-out | out | 13.177 | Saltbr-out | 9.933 | HRD-in | -64.27, -62.7 | 83.56, -10.71 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -29.5 | APE8-dihe-in | -90.52, 58.97 | APE8-rot-na | 25.71 | APE67-dihe-in | -73.18, -5.87 | -63.78, -37.62 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.655 | T790M,V948R | None | None | XRAY | 2.5 | 0.276 | 0.319 | A | 331 | 288 | 20 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 7jxw | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXWB | P00533 | 700 | 1007 | 1210.0 | YY3:1301,VNS:1302 | Type1,Type3 | Inactive | DFGin | 4.889 | 14.548 | BLBplus | -137.39, 167.04 | 52.05, 48.78 | -89.33, 172.11 | 49.0, 84.75 | 70.86, 14.53 | out-out | out | 12.88 | Saltbr-out | 9.64 | HRD-in | -63.98, -61.04 | 82.53, -9.45 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.58 | APE8-rot-na | 26.38 | APE67-dihe-in | -75.13, -4.52 | -61.59, -34.64 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | T790M,V948R | None | None | XRAY | 2.5 | 0.276 | 0.319 | B | 331 | 291 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7jxw | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXWC | P00533 | 700 | 1007 | 1210.0 | YY3:1301,VNS:1302 | Type1,Type3 | Inactive | DFGin | 4.644 | 14.309 | BLBplus | -142.67, 169.6 | 56.07, 43.83 | -87.93, 169.01 | 48.26, 81.62 | 68.95, 14.82 | out-out | out | 13.394 | Saltbr-out | 10.06 | HRD-in | -68.52, -63.21 | 83.53, -10.12 | out-out-none | SNCoon | out-none | ActLoopNT-out | 9.372 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 123.99 | APE8-dihe-in | -72.85, 69.17 | APE8-rot-na | 25.57 | APE67-dihe-in | -79.13, -5.07 | -61.58, -38.99 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.741 | T790M,V948R | None | None | XRAY | 2.5 | 0.276 | 0.319 | C | 331 | 293 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7jxw | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXWD | P00533 | 700 | 1007 | 1210.0 | YY3:1301,VNS:1302 | Type1,Type3 | Inactive | DFGin | 4.474 | 14.215 | BLBplus | -140.27, 167.25 | 54.64, 43.57 | -89.93, 170.58 | 53.09, 83.38 | 70.73, 14.16 | out-out | out | 13.287 | Saltbr-out | 10.176 | HRD-in | -66.78, -61.63 | 83.28, -9.7 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.01 | APE8-dihe-in | -78.05, 71.87 | APE8-rot-na | 25.04 | APE67-dihe-in | -75.98, -6.06 | -65.38, -38.44 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.012 | T790M,V948R | None | None | XRAY | 2.5 | 0.276 | 0.319 | D | 331 | 287 | 21 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7jxw | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LG8B | P00533 | 702 | 1002 | 1210.0 | VNS:1101,8RC:1102 | Type1.5_Front,Type1 | Inactive | DFGin | 4.918 | 14.797 | BLBplus | -141.19, 170.16 | 49.38, 57.43 | -105.85, 156.28 | 47.74, 86.43 | 72.05, 29.16 | out-out | out | 13.829 | Saltbr-out | 11.399 | HRD-in | -68.62, -56.52 | 80.22, -7.8 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 72.88 | APE9-dihe-in | -61.52, 127.34 | APE8-dihe-in | -70.71, 68.41 | APE8-rot-na | 28.03 | APE67-dihe-in | -75.05, -4.72 | -60.67, -37.03 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 14.938 | APE9-dist-out | 8.676 | T790M,V948R | None | None | XRAY | 2.93 | 0.237 | 0.27 | B | 331 | 275 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7lg8 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXQA | P00533 | 700 | 1007 | 1210.0 | VNS:1102,ANP:1103 | Type3,ATPlike | Inactive | DFGin | 4.86 | 14.542 | BLBplus | -136.59, 171.99 | 58.78, 36.07 | -93.08, 163.3 | 53.5, 85.99 | 81.0, 16.2 | out-out | out | 13.6 | Saltbr-out | 11.402 | HRD-in | -66.89, -59.97 | 80.26, -12.87 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.834 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 0.37 | APE9-dihe-in | -62.95, 136.95 | APE8-dihe-in | -80.94, 64.03 | APE8-rot-na | 32.82 | APE67-dihe-in | -75.31, -4.79 | -52.17, -43.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.411 | APE9-dist-out | 8.21 | T790M,V948R | None | None | XRAY | 1.83 | 0.185 | 0.218 | A | 331 | 296 | 12 | 0 | 0 | 12 | [[712, 970]] | 1.0 | 7jxq | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXQC | P00533 | 700 | 1007 | 1210.0 | VNS:1102,ANP:1103 | Type3,ATPlike | Inactive | DFGin | 4.785 | 14.453 | BLBplus | -135.56, 173.47 | 59.34, 36.33 | -94.04, 161.61 | 52.57, 85.94 | 80.36, 16.26 | out-out | out | 13.527 | Saltbr-out | 12.033 | HRD-in | -65.88, -57.49 | 78.82, -12.32 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.819 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.15 | APE8-dihe-in | -80.46, 67.52 | APE8-rot-na | 31.26 | APE67-dihe-in | -73.66, -6.11 | -51.25, -43.4 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.434 | T790M,V948R | None | None | XRAY | 1.83 | 0.185 | 0.218 | C | 331 | 298 | 10 | 0 | 0 | 10 | [[712, 970]] | 1.0 | 7jxq | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LG8A | P00533 | 702 | 1006 | 1210.0 | VNS:1101,8RC:1102 | Type3,Type1 | Inactive | DFGin | 4.633 | 14.844 | BLBplus | -140.27, 173.45 | 52.29, 60.01 | -103.04, 154.16 | 45.73, 86.09 | 71.19, 28.15 | out-out | out | 14.014 | Saltbr-out | 11.713 | HRD-in | -68.53, -55.23 | 80.07, -8.53 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.249 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 124.7 | APE8-dihe-in | -73.13, 67.89 | APE8-rot-na | 28.49 | APE67-dihe-in | -77.47, -4.15 | -60.09, -40.28 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.274 | T790M,V948R | None | None | XRAY | 2.93 | 0.237 | 0.27 | A | 331 | 280 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7lg8 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LG8C | P00533 | 703 | 1004 | 1210.0 | VNS:1101,8RC:1102 | Type3,Type1 | Inactive | DFGin | 4.832 | 14.737 | BLBplus | -140.02, 171.29 | 50.44, 57.58 | -106.29, 155.85 | 48.29, 87.01 | 71.42, 29.21 | out-out | out | 13.235 | Saltbr-out | 10.883 | HRD-in | -68.15, -55.55 | 79.56, -8.95 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.216 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 125.11 | APE8-dihe-in | -71.99, 68.12 | APE8-rot-na | 28.1 | APE67-dihe-in | -76.72, -3.4 | -59.75, -39.52 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.305 | T790M,V948R | None | None | XRAY | 2.93 | 0.237 | 0.27 | C | 331 | 274 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7lg8 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LG8D | P00533 | 702 | 1003 | 1210.0 | VNS:1101,8RC:1102 | Type3,Type1 | Inactive | DFGin | 4.926 | 15.183 | BLBplus | -140.41, 172.1 | 51.47, 58.23 | -106.49, 156.3 | 49.03, 86.93 | 72.22, 33.01 | out-out | out | 13.784 | Saltbr-out | 11.231 | HRD-in | -67.28, -53.4 | 81.73, -11.75 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 125.55 | APE8-dihe-in | -71.42, 69.12 | APE8-rot-na | 28.09 | APE67-dihe-in | -78.92, -4.05 | -59.63, -41.22 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.446 | T790M,V948R | None | None | XRAY | 2.93 | 0.237 | 0.27 | D | 331 | 271 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7lg8 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HA | P00533 | 701 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 4.897 | 14.502 | BLBplus | -130.97, 170.62 | 58.17, 48.68 | -100.05, 161.6 | 49.16, 78.42 | 69.2, 1.23 | out-out | out | 13.749 | Saltbr-out | 11.264 | HRD-in | -77.07, -52.87 | 73.56, -9.67 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 120.57 | APE8-dihe-in | -79.59, 69.97 | APE8-rot-na | 32.69 | APE67-dihe-in | -73.02, -4.47 | -58.4, -43.53 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.87 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | A | 331 | 291 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 7k1h | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HB | P00533 | 701 | 1008 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 5.245 | 14.539 | BLBplus | -131.19, 172.0 | 58.43, 45.25 | -101.59, 170.23 | 51.81, 92.29 | 77.64, 116.53 | out-out | out | 13.419 | Saltbr-out | 9.137 | HRD-in | -79.53, -53.07 | 76.7, -9.03 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 117.65 | APE8-dihe-in | -81.29, 70.54 | APE8-rot-na | 31.4 | APE67-dihe-in | -72.0, -4.51 | -57.97, -43.84 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.952 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | B | 331 | 291 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7k1h | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HC | P00533 | 701 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 4.744 | 14.74 | BLBplus | -129.93, 170.49 | 56.69, 44.1 | -96.18, 166.59 | 55.18, 77.55 | 73.78, 46.77 | out-out | out | 13.454 | Saltbr-out | 8.834 | HRD-in | -79.27, -50.75 | 74.55, -8.77 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 118.24 | APE8-dihe-in | -82.15, 68.56 | APE8-rot-na | 31.93 | APE67-dihe-in | -74.95, -6.33 | -58.99, -43.36 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.006 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | C | 331 | 290 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7k1h | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HD | P00533 | 701 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 5.019 | 14.819 | BLBplus | -131.91, 172.88 | 57.19, 43.91 | -99.27, 163.9 | 51.77, 84.58 | 74.04, -2.08 | out-out | out | 13.649 | Saltbr-out | 10.156 | HRD-in | -78.62, -53.76 | 74.56, -9.86 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.68 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 117.98 | APE8-dihe-in | -78.93, 62.04 | APE8-rot-na | 29.95 | APE67-dihe-in | -73.79, -3.52 | -56.56, -42.2 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.07 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | D | 331 | 292 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7k1h | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HE | P00533 | 703 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 5.157 | 14.635 | BLBplus | -131.84, 173.0 | 58.55, 47.55 | -102.27, 167.87 | 51.85, 86.34 | 79.14, -85.43 | out-out | out | 13.629 | Saltbr-out | 10.317 | HRD-in | -78.55, -50.1 | 74.47, -8.94 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 114.83 | APE8-dihe-in | -83.11, 68.71 | APE8-rot-na | 30.98 | APE67-dihe-in | -72.18, -4.84 | -60.68, -43.88 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.99 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | E | 331 | 289 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 7k1h | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HF | P00533 | 701 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 4.905 | 14.421 | BLBplus | -132.01, 174.64 | 57.0, 46.09 | -100.49, 170.69 | 50.88, 85.85 | 82.59, -107.03 | out-out | out | 13.717 | Saltbr-out | 10.964 | HRD-in | -78.66, -52.82 | 76.59, -9.2 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 119.26 | APE8-dihe-in | -81.53, 68.79 | APE8-rot-na | 32.04 | APE67-dihe-in | -72.57, -5.45 | -59.56, -43.26 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.067 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | F | 331 | 290 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7k1h | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 7JXQB | P00533 | 701 | 1007 | 1210.0 | ANP:1102,VNS:1103 | ATPlike,Type3 | Inactive | DFGin | 4.915 | 14.438 | BLBplus | -136.8, 171.78 | 58.87, 35.86 | -91.33, 162.29 | 51.51, 87.21 | 80.67, 16.0 | out-out | out | 13.335 | Saltbr-out | 12.698 | HRD-in | -67.21, -58.71 | 77.88, -12.51 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.896 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -177.71 | APE9-dihe-in | -105.47, 135.84 | APE8-dihe-in | -83.2, 67.78 | APE8-rot-na | 33.37 | APE67-dihe-in | -74.22, -7.65 | -49.73, -41.79 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.734 | APE9-dist-in | 7.645 | T790M,V948R | None | None | XRAY | 1.83 | 0.185 | 0.218 | B | 331 | 297 | 10 | 0 | 0 | 10 | [[712, 970]] | 1.0 | 7jxq | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXQD | P00533 | 700 | 1007 | 1210.0 | ANP:1102,VNS:1103 | ATPlike,Type3 | Inactive | DFGin | 4.844 | 14.328 | BLBplus | -136.14, 172.56 | 58.98, 36.18 | -92.84, 162.13 | 51.55, 88.05 | 79.36, 17.26 | out-out | out | 13.42 | Saltbr-out | 11.89 | HRD-in | -65.12, -58.0 | 78.92, -12.53 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.94 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.09 | APE8-dihe-in | -80.19, 68.24 | APE8-rot-na | 33.29 | APE67-dihe-in | -74.77, -5.19 | -50.69, -44.59 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.579 | T790M,V948R | None | None | XRAY | 1.83 | 0.185 | 0.218 | D | 331 | 298 | 10 | 0 | 0 | 10 | [[712, 970]] | 1.0 | 7jxq | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1IA | P00533 | 700 | 1007 | 1210.0 | ANP:1102,VNS:1103 | ATPlike,Type3 | Inactive | DFGin | 4.837 | 14.412 | BLBplus | -124.92, 173.52 | 55.34, 38.4 | -93.27, 168.4 | 51.69, 86.03 | 70.99, 11.24 | out-out | out | 13.596 | Saltbr-out | 12.212 | HRD-in | -68.02, -55.76 | 76.66, -7.58 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 142.86 | APE8-dihe-in | -84.0, 73.03 | APE8-rot-na | 29.2 | APE67-dihe-in | -72.27, -9.54 | -58.41, -42.03 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.42 | L858R,V948R | None | None | XRAY | 3.202 | 0.266 | 0.311 | A | 331 | 288 | 20 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7k1i | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXWA | P00533 | 700 | 1007 | 1210.0 | YY3:1301,VNS:1302 | Type1,Type3 | Inactive | DFGin | 4.579 | 14.666 | BLBplus | -138.64, 168.46 | 50.29, 44.7 | -88.71, 170.77 | 52.75, 84.47 | 69.65, 17.94 | out-out | out | 13.177 | Saltbr-out | 9.933 | HRD-in | -64.27, -62.7 | 83.56, -10.71 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -29.5 | APE8-dihe-in | -90.52, 58.97 | APE8-rot-na | 25.71 | APE67-dihe-in | -73.18, -5.87 | -63.78, -37.62 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.655 | T790M,V948R | None | None | XRAY | 2.5 | 0.276 | 0.319 | A | 331 | 288 | 20 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 7jxw | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXWB | P00533 | 700 | 1007 | 1210.0 | YY3:1301,VNS:1302 | Type1,Type3 | Inactive | DFGin | 4.889 | 14.548 | BLBplus | -137.39, 167.04 | 52.05, 48.78 | -89.33, 172.11 | 49.0, 84.75 | 70.86, 14.53 | out-out | out | 12.88 | Saltbr-out | 9.64 | HRD-in | -63.98, -61.04 | 82.53, -9.45 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 67.58 | APE8-rot-na | 26.38 | APE67-dihe-in | -75.13, -4.52 | -61.59, -34.64 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | T790M,V948R | None | None | XRAY | 2.5 | 0.276 | 0.319 | B | 331 | 291 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7jxw | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXWC | P00533 | 700 | 1007 | 1210.0 | YY3:1301,VNS:1302 | Type1,Type3 | Inactive | DFGin | 4.644 | 14.309 | BLBplus | -142.67, 169.6 | 56.07, 43.83 | -87.93, 169.01 | 48.26, 81.62 | 68.95, 14.82 | out-out | out | 13.394 | Saltbr-out | 10.06 | HRD-in | -68.52, -63.21 | 83.53, -10.12 | out-out-none | SNCoon | out-none | ActLoopNT-out | 9.372 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 123.99 | APE8-dihe-in | -72.85, 69.17 | APE8-rot-na | 25.57 | APE67-dihe-in | -79.13, -5.07 | -61.58, -38.99 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.741 | T790M,V948R | None | None | XRAY | 2.5 | 0.276 | 0.319 | C | 331 | 293 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7jxw | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXWD | P00533 | 700 | 1007 | 1210.0 | YY3:1301,VNS:1302 | Type1,Type3 | Inactive | DFGin | 4.474 | 14.215 | BLBplus | -140.27, 167.25 | 54.64, 43.57 | -89.93, 170.58 | 53.09, 83.38 | 70.73, 14.16 | out-out | out | 13.287 | Saltbr-out | 10.176 | HRD-in | -66.78, -61.63 | 83.28, -9.7 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.01 | APE8-dihe-in | -78.05, 71.87 | APE8-rot-na | 25.04 | APE67-dihe-in | -75.98, -6.06 | -65.38, -38.44 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.012 | T790M,V948R | None | None | XRAY | 2.5 | 0.276 | 0.319 | D | 331 | 287 | 21 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7jxw | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LG8B | P00533 | 702 | 1002 | 1210.0 | VNS:1101,8RC:1102 | Type1.5_Front,Type1 | Inactive | DFGin | 4.918 | 14.797 | BLBplus | -141.19, 170.16 | 49.38, 57.43 | -105.85, 156.28 | 47.74, 86.43 | 72.05, 29.16 | out-out | out | 13.829 | Saltbr-out | 11.399 | HRD-in | -68.62, -56.52 | 80.22, -7.8 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 72.88 | APE9-dihe-in | -61.52, 127.34 | APE8-dihe-in | -70.71, 68.41 | APE8-rot-na | 28.03 | APE67-dihe-in | -75.05, -4.72 | -60.67, -37.03 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 14.938 | APE9-dist-out | 8.676 | T790M,V948R | None | None | XRAY | 2.93 | 0.237 | 0.27 | B | 331 | 275 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7lg8 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXQA | P00533 | 700 | 1007 | 1210.0 | VNS:1102,ANP:1103 | Type3,ATPlike | Inactive | DFGin | 4.86 | 14.542 | BLBplus | -136.59, 171.99 | 58.78, 36.07 | -93.08, 163.3 | 53.5, 85.99 | 81.0, 16.2 | out-out | out | 13.6 | Saltbr-out | 11.402 | HRD-in | -66.89, -59.97 | 80.26, -12.87 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.834 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 0.37 | APE9-dihe-in | -62.95, 136.95 | APE8-dihe-in | -80.94, 64.03 | APE8-rot-na | 32.82 | APE67-dihe-in | -75.31, -4.79 | -52.17, -43.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.411 | APE9-dist-out | 8.21 | T790M,V948R | None | None | XRAY | 1.83 | 0.185 | 0.218 | A | 331 | 296 | 12 | 0 | 0 | 12 | [[712, 970]] | 1.0 | 7jxq | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXQC | P00533 | 700 | 1007 | 1210.0 | VNS:1102,ANP:1103 | Type3,ATPlike | Inactive | DFGin | 4.785 | 14.453 | BLBplus | -135.56, 173.47 | 59.34, 36.33 | -94.04, 161.61 | 52.57, 85.94 | 80.36, 16.26 | out-out | out | 13.527 | Saltbr-out | 12.033 | HRD-in | -65.88, -57.49 | 78.82, -12.32 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.819 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.15 | APE8-dihe-in | -80.46, 67.52 | APE8-rot-na | 31.26 | APE67-dihe-in | -73.66, -6.11 | -51.25, -43.4 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.434 | T790M,V948R | None | None | XRAY | 1.83 | 0.185 | 0.218 | C | 331 | 298 | 10 | 0 | 0 | 10 | [[712, 970]] | 1.0 | 7jxq | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LG8A | P00533 | 702 | 1006 | 1210.0 | VNS:1101,8RC:1102 | Type3,Type1 | Inactive | DFGin | 4.633 | 14.844 | BLBplus | -140.27, 173.45 | 52.29, 60.01 | -103.04, 154.16 | 45.73, 86.09 | 71.19, 28.15 | out-out | out | 14.014 | Saltbr-out | 11.713 | HRD-in | -68.53, -55.23 | 80.07, -8.53 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.249 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 124.7 | APE8-dihe-in | -73.13, 67.89 | APE8-rot-na | 28.49 | APE67-dihe-in | -77.47, -4.15 | -60.09, -40.28 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.274 | T790M,V948R | None | None | XRAY | 2.93 | 0.237 | 0.27 | A | 331 | 280 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7lg8 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LG8C | P00533 | 703 | 1004 | 1210.0 | VNS:1101,8RC:1102 | Type3,Type1 | Inactive | DFGin | 4.832 | 14.737 | BLBplus | -140.02, 171.29 | 50.44, 57.58 | -106.29, 155.85 | 48.29, 87.01 | 71.42, 29.21 | out-out | out | 13.235 | Saltbr-out | 10.883 | HRD-in | -68.15, -55.55 | 79.56, -8.95 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.216 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 125.11 | APE8-dihe-in | -71.99, 68.12 | APE8-rot-na | 28.1 | APE67-dihe-in | -76.72, -3.4 | -59.75, -39.52 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.305 | T790M,V948R | None | None | XRAY | 2.93 | 0.237 | 0.27 | C | 331 | 274 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7lg8 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LG8D | P00533 | 702 | 1003 | 1210.0 | VNS:1101,8RC:1102 | Type3,Type1 | Inactive | DFGin | 4.926 | 15.183 | BLBplus | -140.41, 172.1 | 51.47, 58.23 | -106.49, 156.3 | 49.03, 86.93 | 72.22, 33.01 | out-out | out | 13.784 | Saltbr-out | 11.231 | HRD-in | -67.28, -53.4 | 81.73, -11.75 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 125.55 | APE8-dihe-in | -71.42, 69.12 | APE8-rot-na | 28.09 | APE67-dihe-in | -78.92, -4.05 | -59.63, -41.22 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.446 | T790M,V948R | None | None | XRAY | 2.93 | 0.237 | 0.27 | D | 331 | 271 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7lg8 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HA | P00533 | 701 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 4.897 | 14.502 | BLBplus | -130.97, 170.62 | 58.17, 48.68 | -100.05, 161.6 | 49.16, 78.42 | 69.2, 1.23 | out-out | out | 13.749 | Saltbr-out | 11.264 | HRD-in | -77.07, -52.87 | 73.56, -9.67 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 120.57 | APE8-dihe-in | -79.59, 69.97 | APE8-rot-na | 32.69 | APE67-dihe-in | -73.02, -4.47 | -58.4, -43.53 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.87 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | A | 331 | 291 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 7k1h | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HB | P00533 | 701 | 1008 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 5.245 | 14.539 | BLBplus | -131.19, 172.0 | 58.43, 45.25 | -101.59, 170.23 | 51.81, 92.29 | 77.64, 116.53 | out-out | out | 13.419 | Saltbr-out | 9.137 | HRD-in | -79.53, -53.07 | 76.7, -9.03 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 117.65 | APE8-dihe-in | -81.29, 70.54 | APE8-rot-na | 31.4 | APE67-dihe-in | -72.0, -4.51 | -57.97, -43.84 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.952 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | B | 331 | 291 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7k1h | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HC | P00533 | 701 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 4.744 | 14.74 | BLBplus | -129.93, 170.49 | 56.69, 44.1 | -96.18, 166.59 | 55.18, 77.55 | 73.78, 46.77 | out-out | out | 13.454 | Saltbr-out | 8.834 | HRD-in | -79.27, -50.75 | 74.55, -8.77 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 118.24 | APE8-dihe-in | -82.15, 68.56 | APE8-rot-na | 31.93 | APE67-dihe-in | -74.95, -6.33 | -58.99, -43.36 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.006 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | C | 331 | 290 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7k1h | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HD | P00533 | 701 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 5.019 | 14.819 | BLBplus | -131.91, 172.88 | 57.19, 43.91 | -99.27, 163.9 | 51.77, 84.58 | 74.04, -2.08 | out-out | out | 13.649 | Saltbr-out | 10.156 | HRD-in | -78.62, -53.76 | 74.56, -9.86 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.68 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 117.98 | APE8-dihe-in | -78.93, 62.04 | APE8-rot-na | 29.95 | APE67-dihe-in | -73.79, -3.52 | -56.56, -42.2 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.07 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | D | 331 | 292 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 7k1h | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HE | P00533 | 703 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 5.157 | 14.635 | BLBplus | -131.84, 173.0 | 58.55, 47.55 | -102.27, 167.87 | 51.85, 86.34 | 79.14, -85.43 | out-out | out | 13.629 | Saltbr-out | 10.317 | HRD-in | -78.55, -50.1 | 74.47, -8.94 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 114.83 | APE8-dihe-in | -83.11, 68.71 | APE8-rot-na | 30.98 | APE67-dihe-in | -72.18, -4.84 | -60.68, -43.88 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.99 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | E | 331 | 289 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 7k1h | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7K1HF | P00533 | 701 | 1007 | 1210.0 | VNS:1301,YY3:1302 | Type3,Type1 | Inactive | DFGin | 4.905 | 14.421 | BLBplus | -132.01, 174.64 | 57.0, 46.09 | -100.49, 170.69 | 50.88, 85.85 | 82.59, -107.03 | out-out | out | 13.717 | Saltbr-out | 10.964 | HRD-in | -78.66, -52.82 | 76.59, -9.2 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 119.26 | APE8-dihe-in | -81.53, 68.79 | APE8-rot-na | 32.04 | APE67-dihe-in | -72.57, -5.45 | -59.56, -43.26 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.067 | L858R,V948R | None | None | XRAY | 2.602 | 0.233 | 0.275 | F | 331 | 290 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7k1h | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.5e-87 | 296.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|