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| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 9BY6A | P00533 | 698 | 1009 | 1210.0 | PDO:1301,Q6K:1302 | Allosteric,Type1 | Active | DFGin | 6.002 | 15.663 | BLAminus | -149.77, -168.8 | 56.86, 79.46 | -96.38, 24.13 | 296.36, 92.05 | -63.66, -24.81 | in-in | in | 9.063 | Saltbr-in | 3.491 | HRD-in | -75.7, -50.64 | 70.26, 5.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.955 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.71, 133.19 | APE9-dihe-in | -133.13, 146.74 | APE8-dihe-in | -72.35, 102.77 | APE8-rot-na | 25.41 | APE67-dihe-in | -79.34, -8.97 | -76.98, -28.96 | APE12-dist-na | 12.695 | APE11-dist-na | 9.472 | APE10-dist-na | 11.091 | APE9-dist-in | 6.657 | None | None | None | XRAY | 2.551 | 0.208 | 0.245 | A | 338 | 311 | 1 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 9by6 | TYR_EGFR_HUMAN | TYR | 1.2e-87 | 299.6 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 9BY4A | P00533 | 696 | 1010 | 1210.0 | PDO:61301,Q6K:61302,PDO:61304,PDO:61305 | Allosteric,Type1,Allosteric,Type1 | Active | DFGin | 6.118 | 15.558 | BLAminus | -131.58, -170.69 | 55.04, 91.41 | -104.93, 32.17 | 291.61, 87.59 | -69.69, -25.35 | in-in | in | 8.748 | Saltbr-in | 2.724 | HRD-in | -74.22, -51.47 | 72.05, 2.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.974 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -66.0, 133.58 | APE9-dihe-in | -140.48, 146.73 | APE8-dihe-in | -77.28, 98.44 | APE8-rot-na | 2.83 | APE67-dihe-in | -69.73, -13.67 | -59.81, -44.15 | APE12-dist-na | 11.983 | APE11-dist-na | 10.159 | APE10-dist-na | 10.796 | APE9-dist-in | 6.63 | None | None | None | XRAY | 2.307 | 0.197 | 0.22 | A | 338 | 315 | 0 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 9by4 | TYR_EGFR_HUMAN | TYR | 1.2e-87 | 299.6 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LGSA | P00533 | 702 | 984 | 1210.0 | Q6K:61101 | Type1 | Active | DFGin | 5.798 | 13.848 | BLAminus | -148.14, -179.86 | 66.83, 93.39 | -109.24, 25.55 | 296.83, 82.02 | -45.71, -51.38 | in-in | in | 8.254 | Saltbr-in | 2.914 | HRD-in | -61.85, -36.93 | 72.75, -6.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.819 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -110.14, 118.29 | APE9-dihe-in | -124.18, 152.07 | APE8-dihe-in | -87.87, 98.71 | APE8-rot-na | 33.29 | APE67-dihe-in | -76.07, 20.02 | -59.01, -47.71 | APE12-dist-na | 10.735 | APE11-dist-na | 9.717 | APE10-dist-na | 10.441 | APE9-dist-in | 6.735 | V948R | None | None | XRAY | 3.1 | 0.241 | 0.305 | A | 331 | 280 | 3 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7lgs | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LGSB | P00533 | 702 | 984 | 1210.0 | Q6K:62703 | Type1 | Active | DFGin | 6.065 | 14.132 | BLAminus | -143.64, 174.55 | 75.07, 86.01 | -103.95, 23.76 | 297.26, 76.2 | -47.19, -46.41 | in-in | in | 8.489 | Saltbr-in | 2.925 | HRD-in | -70.84, -32.42 | 56.54, 26.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.24, 133.4 | APE9-dihe-in | -137.17, 157.48 | APE8-dihe-in | -85.36, 106.29 | APE8-rot-na | 33.1 | APE67-dihe-in | -76.15, 7.94 | -70.75, -39.01 | APE12-dist-na | 11.907 | APE11-dist-na | 9.426 | APE10-dist-na | 10.275 | APE9-dist-in | 6.571 | V948R | None | None | XRAY | 3.1 | 0.241 | 0.305 | B | 331 | 283 | 0 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7lgs | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LGSC | P00533 | 701 | 984 | 1210.0 | Q6K:61101 | Type1 | Active | DFGin | 5.788 | 13.836 | BLAminus | -144.73, 172.67 | 64.73, 92.38 | -102.97, 22.8 | 303.24, 82.51 | -50.29, -34.49 | in-in | in | 8.064 | Saltbr-in | 3.457 | HRD-in | -60.12, -39.38 | 78.78, -23.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.202 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -145.58, 117.71 | APE9-dihe-in | -124.38, 146.08 | APE8-dihe-in | -62.99, 124.66 | APE8-rot-na | 21.56 | APE67-dihe-in | -104.68, 1.44 | -87.08, -8.44 | APE12-dist-na | 11.582 | APE11-dist-na | 9.289 | APE10-dist-na | 9.921 | APE9-dist-in | 6.458 | V948R | None | None | XRAY | 3.1 | 0.241 | 0.305 | C | 331 | 280 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7lgs | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LGSD | P00533 | 701 | 984 | 1210.0 | Q6K:62500 | Type1 | Active | DFGin | 5.717 | 14.024 | BLAminus | -133.47, 170.68 | 74.78, 90.52 | -109.47, 24.05 | 298.1, 77.01 | -64.19, -15.34 | in-in | in | 8.201 | Saltbr-in | 2.786 | HRD-in | -55.31, -49.72 | 74.8, 6.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.837 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -72.9, 130.33 | APE9-dihe-in | -138.85, 149.74 | APE8-dihe-in | -80.14, 110.14 | APE8-rot-na | 30.64 | APE67-dihe-in | -83.2, -1.33 | -71.86, -29.25 | APE12-dist-na | 11.726 | APE11-dist-na | 9.543 | APE10-dist-na | 10.278 | APE9-dist-in | 6.353 | V948R | None | None | XRAY | 3.1 | 0.241 | 0.305 | D | 331 | 276 | 8 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7lgs | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6XL4A | P00533 | 700 | 1007 | 1210.0 | Q6K:1301,NQ1:1302 | Type1,Type3 | Inactive | DFGin | 5.098 | 14.695 | BLBplus | -134.42, 176.69 | 66.92, 16.35 | -78.69, 146.78 | 51.46, 92.89 | 75.99, 3.76 | out-out | out | 13.363 | Saltbr-out | 12.539 | HRD-in | -71.16, -58.13 | 77.59, -5.31 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.386 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 139.31 | APE8-dihe-in | -78.15, 72.0 | APE8-rot-na | 31.9 | APE67-dihe-in | -74.09, -1.62 | -55.44, -42.27 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.703 | T790M,V948R | None | None | XRAY | 2.06 | 0.216 | 0.252 | A | 328 | 293 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 6xl4 | TYR_EGFR_HUMAN | TYR | 6.1e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5A | P00533 | 701 | 1011 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.808 | 14.912 | BLBplus | -132.77, 163.28 | 59.53, 50.36 | -94.02, 166.24 | 50.17, 88.29 | 66.49, 24.24 | out-out | out | 13.127 | Saltbr-out | 9.96 | HRD-in | -72.38, -54.99 | 79.4, -8.54 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 131.66 | APE8-dihe-in | -80.77, 69.75 | APE8-rot-na | 32.13 | APE67-dihe-in | -76.82, -3.31 | -58.55, -37.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.087 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | A | 331 | 294 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gk5 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5B | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.513 | 14.722 | BLBplus | -133.17, 164.36 | 59.73, 51.31 | -91.4, 162.53 | 47.93, 87.21 | 64.33, 22.83 | out-out | out | 13.093 | Saltbr-out | 12.438 | HRD-in | -72.73, -55.9 | 79.15, -8.43 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 131.91 | APE8-dihe-in | -79.02, 69.83 | APE8-rot-na | 32.01 | APE67-dihe-in | -76.26, -3.86 | -58.1, -38.17 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.867 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | B | 331 | 292 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gk5 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5C | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.465 | 14.758 | BLBplus | -134.6, 164.78 | 60.76, 50.7 | -93.92, 162.62 | 46.93, 87.83 | 64.54, 21.99 | out-out | out | 13.135 | Saltbr-out | 11.494 | HRD-in | -72.37, -55.98 | 79.27, -6.85 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.09 | APE8-dihe-in | -76.74, 68.64 | APE8-rot-na | 31.76 | APE67-dihe-in | -75.53, -4.34 | -59.95, -38.1 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.102 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | C | 331 | 293 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 8gk5 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5D | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.407 | 14.729 | BLBplus | -134.17, 163.98 | 61.67, 51.99 | -93.03, 163.58 | 47.55, 87.87 | 65.01, 22.54 | out-out | out | 13.091 | Saltbr-out | 12.29 | HRD-in | -70.88, -54.33 | 77.76, -8.04 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -1.54 | APE9-dihe-in | -75.57, 134.88 | APE8-dihe-in | -77.01, 71.98 | APE8-rot-na | 32.06 | APE67-dihe-in | -76.98, -3.79 | -58.78, -38.58 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.721 | APE9-dist-in | 7.558 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | D | 331 | 294 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 8gk5 | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6Z4BA | P00533 | 700 | 982 | 1210.0 | Q6K:1101,9LL:1102 | Type1,Type3 | Inactive | DFGin | 5.693 | 14.816 | BLBplus | -133.89, 164.94 | 59.43, 51.96 | -98.19, 144.81 | 41.57, 85.88 | 67.58, 19.62 | out-none | out | 14.398 | Saltbr-none | 999.0 | HRD-in | -67.89, -64.09 | 87.77, -27.23 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 7.141 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, -2.64 | APE9-dihe-in | -120.02, 130.13 | APE8-dihe-in | -80.9, 78.34 | APE8-rot-na | 31.39 | APE67-dihe-in | -73.81, -4.61 | -60.28, -41.17 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 12.71 | APE9-dist-out | 8.134 | T790M,V948R | None | None | XRAY | 2.5 | 0.222 | 0.251 | A | 333 | 271 | 12 | 0 | 0 | 12 | [[712, 970]] | 1.0 | 6z4b | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6Z4BB | P00533 | 699 | 984 | 1210.0 | Q6K:1101,9LL:1102 | Type1,Type3 | Inactive | DFGin | 6.233 | 14.529 | BLBplus | -131.04, 166.01 | 60.41, 49.56 | -101.97, 145.48 | 42.99, 86.21 | -89.28, 999.0 | out-out | out | 12.903 | Saltbr-out | 9.732 | HRD-out | -138.19, 95.22 | -83.97, -17.5 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 123.87 | APE8-dihe-in | -88.45, 76.4 | APE8-rot-na | 32.2 | APE67-dihe-in | -72.84, -5.09 | -59.16, -39.52 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.257 | T790M,V948R | None | None | XRAY | 2.5 | 0.222 | 0.251 | B | 333 | 263 | 23 | 0 | 0 | 18 | [[712, 970]] | 1.0 | 6z4b | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6XL4B | P00533 | 700 | 1007 | 1210.0 | NQ1:1201,Q6K:1202 | Type3,Type1 | Inactive | DFGin | 4.808 | 14.497 | BLBplus | -133.43, 176.08 | 66.75, 17.79 | -78.7, 146.83 | 53.41, 93.69 | 78.85, 14.72 | out-out | out | 13.809 | Saltbr-out | 14.224 | HRD-in | -71.6, -57.82 | 77.95, -5.56 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 139.66 | APE8-dihe-in | -77.94, 72.67 | APE8-rot-na | 31.42 | APE67-dihe-in | -72.46, -3.15 | -55.35, -40.72 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.932 | T790M,V948R | None | None | XRAY | 2.06 | 0.216 | 0.252 | B | 328 | 292 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 6xl4 | TYR_EGFR_HUMAN | TYR | 6.1e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 9GDVA | P00533 | 702 | 985 | 1210.0 | Q6K:1101 | Type1 | Inactive | DFGin | 5.61 | 15.829 | BLBtrans | -107.73, 177.69 | 65.5, 33.1 | -82.9, 128.34 | 164.87, 70.16 | 94.26, -7.41 | out-none | out | 12.642 | Saltbr-none | 999.0 | HRD-in | -75.43, -53.65 | 76.33, -6.74 | none-out-none | SNCnon | out-none | ActLoopNT-out | 7.915 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 143.05 | APE8-dihe-in | -77.71, 68.12 | APE8-rot-na | 28.54 | APE67-dihe-in | -70.85, -6.5 | -47.64, -45.7 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.734 | V948R | None | None | XRAY | 2.218 | 0.235 | 0.293 | A | 330 | 262 | 22 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 9gdv | TYR_EGFR_HUMAN | TYR | 8.1e-88 | 300.1 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 9GDVB | P00533 | 702 | 985 | 1210.0 | Q6K:1101 | Type1 | Inactive | DFGin | 4.579 | 15.491 | BLBtrans | -111.43, 179.21 | 66.37, 26.18 | -74.59, 129.04 | 147.85, 63.03 | 60.16, 37.36 | out-none | out | 12.538 | Saltbr-none | 999.0 | HRD-out | -124.5, 90.89 | -69.11, -17.02 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.32 | APE8-dihe-in | -80.3, 68.77 | APE8-rot-na | 2.98 | APE67-dihe-in | -69.33, -16.36 | -50.05, -40.21 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.271 | V948R | None | None | XRAY | 2.218 | 0.235 | 0.293 | B | 330 | 267 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 9gdv | TYR_EGFR_HUMAN | TYR | 8.1e-88 | 300.1 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 9BY6A | P00533 | 698 | 1009 | 1210.0 | PDO:1301,Q6K:1302 | Allosteric,Type1 | Active | DFGin | 6.002 | 15.663 | BLAminus | -149.77, -168.8 | 56.86, 79.46 | -96.38, 24.13 | 296.36, 92.05 | -63.66, -24.81 | in-in | in | 9.063 | Saltbr-in | 3.491 | HRD-in | -75.7, -50.64 | 70.26, 5.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.955 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.71, 133.19 | APE9-dihe-in | -133.13, 146.74 | APE8-dihe-in | -72.35, 102.77 | APE8-rot-na | 25.41 | APE67-dihe-in | -79.34, -8.97 | -76.98, -28.96 | APE12-dist-na | 12.695 | APE11-dist-na | 9.472 | APE10-dist-na | 11.091 | APE9-dist-in | 6.657 | None | None | None | XRAY | 2.551 | 0.208 | 0.245 | A | 338 | 311 | 1 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 9by6 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.2e-87 | 299.6 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 9BY4A | P00533 | 696 | 1010 | 1210.0 | PDO:61301,Q6K:61302,PDO:61304,PDO:61305 | Allosteric,Type1,Allosteric,Type1 | Active | DFGin | 6.118 | 15.558 | BLAminus | -131.58, -170.69 | 55.04, 91.41 | -104.93, 32.17 | 291.61, 87.59 | -69.69, -25.35 | in-in | in | 8.748 | Saltbr-in | 2.724 | HRD-in | -74.22, -51.47 | 72.05, 2.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.974 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -66.0, 133.58 | APE9-dihe-in | -140.48, 146.73 | APE8-dihe-in | -77.28, 98.44 | APE8-rot-na | 2.83 | APE67-dihe-in | -69.73, -13.67 | -59.81, -44.15 | APE12-dist-na | 11.983 | APE11-dist-na | 10.159 | APE10-dist-na | 10.796 | APE9-dist-in | 6.63 | None | None | None | XRAY | 2.307 | 0.197 | 0.22 | A | 338 | 315 | 0 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 9by4 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.2e-87 | 299.6 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LGSA | P00533 | 702 | 984 | 1210.0 | Q6K:61101 | Type1 | Active | DFGin | 5.798 | 13.848 | BLAminus | -148.14, -179.86 | 66.83, 93.39 | -109.24, 25.55 | 296.83, 82.02 | -45.71, -51.38 | in-in | in | 8.254 | Saltbr-in | 2.914 | HRD-in | -61.85, -36.93 | 72.75, -6.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.819 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -110.14, 118.29 | APE9-dihe-in | -124.18, 152.07 | APE8-dihe-in | -87.87, 98.71 | APE8-rot-na | 33.29 | APE67-dihe-in | -76.07, 20.02 | -59.01, -47.71 | APE12-dist-na | 10.735 | APE11-dist-na | 9.717 | APE10-dist-na | 10.441 | APE9-dist-in | 6.735 | V948R | None | None | XRAY | 3.1 | 0.241 | 0.305 | A | 331 | 280 | 3 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7lgs | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LGSB | P00533 | 702 | 984 | 1210.0 | Q6K:62703 | Type1 | Active | DFGin | 6.065 | 14.132 | BLAminus | -143.64, 174.55 | 75.07, 86.01 | -103.95, 23.76 | 297.26, 76.2 | -47.19, -46.41 | in-in | in | 8.489 | Saltbr-in | 2.925 | HRD-in | -70.84, -32.42 | 56.54, 26.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.803 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.24, 133.4 | APE9-dihe-in | -137.17, 157.48 | APE8-dihe-in | -85.36, 106.29 | APE8-rot-na | 33.1 | APE67-dihe-in | -76.15, 7.94 | -70.75, -39.01 | APE12-dist-na | 11.907 | APE11-dist-na | 9.426 | APE10-dist-na | 10.275 | APE9-dist-in | 6.571 | V948R | None | None | XRAY | 3.1 | 0.241 | 0.305 | B | 331 | 283 | 0 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7lgs | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LGSC | P00533 | 701 | 984 | 1210.0 | Q6K:61101 | Type1 | Active | DFGin | 5.788 | 13.836 | BLAminus | -144.73, 172.67 | 64.73, 92.38 | -102.97, 22.8 | 303.24, 82.51 | -50.29, -34.49 | in-in | in | 8.064 | Saltbr-in | 3.457 | HRD-in | -60.12, -39.38 | 78.78, -23.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.202 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -145.58, 117.71 | APE9-dihe-in | -124.38, 146.08 | APE8-dihe-in | -62.99, 124.66 | APE8-rot-na | 21.56 | APE67-dihe-in | -104.68, 1.44 | -87.08, -8.44 | APE12-dist-na | 11.582 | APE11-dist-na | 9.289 | APE10-dist-na | 9.921 | APE9-dist-in | 6.458 | V948R | None | None | XRAY | 3.1 | 0.241 | 0.305 | C | 331 | 280 | 4 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7lgs | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7LGSD | P00533 | 701 | 984 | 1210.0 | Q6K:62500 | Type1 | Active | DFGin | 5.717 | 14.024 | BLAminus | -133.47, 170.68 | 74.78, 90.52 | -109.47, 24.05 | 298.1, 77.01 | -64.19, -15.34 | in-in | in | 8.201 | Saltbr-in | 2.786 | HRD-in | -55.31, -49.72 | 74.8, 6.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.837 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -72.9, 130.33 | APE9-dihe-in | -138.85, 149.74 | APE8-dihe-in | -80.14, 110.14 | APE8-rot-na | 30.64 | APE67-dihe-in | -83.2, -1.33 | -71.86, -29.25 | APE12-dist-na | 11.726 | APE11-dist-na | 9.543 | APE10-dist-na | 10.278 | APE9-dist-in | 6.353 | V948R | None | None | XRAY | 3.1 | 0.241 | 0.305 | D | 331 | 276 | 8 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7lgs | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6XL4A | P00533 | 700 | 1007 | 1210.0 | Q6K:1301,NQ1:1302 | Type1,Type3 | Inactive | DFGin | 5.098 | 14.695 | BLBplus | -134.42, 176.69 | 66.92, 16.35 | -78.69, 146.78 | 51.46, 92.89 | 75.99, 3.76 | out-out | out | 13.363 | Saltbr-out | 12.539 | HRD-in | -71.16, -58.13 | 77.59, -5.31 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.386 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 139.31 | APE8-dihe-in | -78.15, 72.0 | APE8-rot-na | 31.9 | APE67-dihe-in | -74.09, -1.62 | -55.44, -42.27 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.703 | T790M,V948R | None | None | XRAY | 2.06 | 0.216 | 0.252 | A | 328 | 293 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 6xl4 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.1e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5A | P00533 | 701 | 1011 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.808 | 14.912 | BLBplus | -132.77, 163.28 | 59.53, 50.36 | -94.02, 166.24 | 50.17, 88.29 | 66.49, 24.24 | out-out | out | 13.127 | Saltbr-out | 9.96 | HRD-in | -72.38, -54.99 | 79.4, -8.54 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 131.66 | APE8-dihe-in | -80.77, 69.75 | APE8-rot-na | 32.13 | APE67-dihe-in | -76.82, -3.31 | -58.55, -37.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.087 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | A | 331 | 294 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gk5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5B | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.513 | 14.722 | BLBplus | -133.17, 164.36 | 59.73, 51.31 | -91.4, 162.53 | 47.93, 87.21 | 64.33, 22.83 | out-out | out | 13.093 | Saltbr-out | 12.438 | HRD-in | -72.73, -55.9 | 79.15, -8.43 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 131.91 | APE8-dihe-in | -79.02, 69.83 | APE8-rot-na | 32.01 | APE67-dihe-in | -76.26, -3.86 | -58.1, -38.17 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.867 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | B | 331 | 292 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 8gk5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5C | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.465 | 14.758 | BLBplus | -134.6, 164.78 | 60.76, 50.7 | -93.92, 162.62 | 46.93, 87.83 | 64.54, 21.99 | out-out | out | 13.135 | Saltbr-out | 11.494 | HRD-in | -72.37, -55.98 | 79.27, -6.85 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.09 | APE8-dihe-in | -76.74, 68.64 | APE8-rot-na | 31.76 | APE67-dihe-in | -75.53, -4.34 | -59.95, -38.1 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.102 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | C | 331 | 293 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 8gk5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8GK5D | P00533 | 700 | 1008 | 1210.0 | Q6K:1101,YW5:1102 | Type1,Type3 | Inactive | DFGin | 4.407 | 14.729 | BLBplus | -134.17, 163.98 | 61.67, 51.99 | -93.03, 163.58 | 47.55, 87.87 | 65.01, 22.54 | out-out | out | 13.091 | Saltbr-out | 12.29 | HRD-in | -70.88, -54.33 | 77.76, -8.04 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -1.54 | APE9-dihe-in | -75.57, 134.88 | APE8-dihe-in | -77.01, 71.98 | APE8-rot-na | 32.06 | APE67-dihe-in | -76.98, -3.79 | -58.78, -38.58 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.721 | APE9-dist-in | 7.558 | T790M,V948R | None | None | XRAY | 2.3 | 0.224 | 0.252 | D | 331 | 294 | 15 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 8gk5 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6Z4BA | P00533 | 700 | 982 | 1210.0 | Q6K:1101,9LL:1102 | Type1,Type3 | Inactive | DFGin | 5.693 | 14.816 | BLBplus | -133.89, 164.94 | 59.43, 51.96 | -98.19, 144.81 | 41.57, 85.88 | 67.58, 19.62 | out-none | out | 14.398 | Saltbr-none | 999.0 | HRD-in | -67.89, -64.09 | 87.77, -27.23 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 7.141 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, -2.64 | APE9-dihe-in | -120.02, 130.13 | APE8-dihe-in | -80.9, 78.34 | APE8-rot-na | 31.39 | APE67-dihe-in | -73.81, -4.61 | -60.28, -41.17 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 12.71 | APE9-dist-out | 8.134 | T790M,V948R | None | None | XRAY | 2.5 | 0.222 | 0.251 | A | 333 | 271 | 12 | 0 | 0 | 12 | [[712, 970]] | 1.0 | 6z4b | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6Z4BB | P00533 | 699 | 984 | 1210.0 | Q6K:1101,9LL:1102 | Type1,Type3 | Inactive | DFGin | 6.233 | 14.529 | BLBplus | -131.04, 166.01 | 60.41, 49.56 | -101.97, 145.48 | 42.99, 86.21 | -89.28, 999.0 | out-out | out | 12.903 | Saltbr-out | 9.732 | HRD-out | -138.19, 95.22 | -83.97, -17.5 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 123.87 | APE8-dihe-in | -88.45, 76.4 | APE8-rot-na | 32.2 | APE67-dihe-in | -72.84, -5.09 | -59.16, -39.52 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.257 | T790M,V948R | None | None | XRAY | 2.5 | 0.222 | 0.251 | B | 333 | 263 | 23 | 0 | 0 | 18 | [[712, 970]] | 1.0 | 6z4b | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6XL4B | P00533 | 700 | 1007 | 1210.0 | NQ1:1201,Q6K:1202 | Type3,Type1 | Inactive | DFGin | 4.808 | 14.497 | BLBplus | -133.43, 176.08 | 66.75, 17.79 | -78.7, 146.83 | 53.41, 93.69 | 78.85, 14.72 | out-out | out | 13.809 | Saltbr-out | 14.224 | HRD-in | -71.6, -57.82 | 77.95, -5.56 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 139.66 | APE8-dihe-in | -77.94, 72.67 | APE8-rot-na | 31.42 | APE67-dihe-in | -72.46, -3.15 | -55.35, -40.72 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.932 | T790M,V948R | None | None | XRAY | 2.06 | 0.216 | 0.252 | B | 328 | 292 | 16 | 0 | 0 | 16 | [[712, 970]] | 1.0 | 6xl4 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.1e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 9GDVA | P00533 | 702 | 985 | 1210.0 | Q6K:1101 | Type1 | Inactive | DFGin | 5.61 | 15.829 | BLBtrans | -107.73, 177.69 | 65.5, 33.1 | -82.9, 128.34 | 164.87, 70.16 | 94.26, -7.41 | out-none | out | 12.642 | Saltbr-none | 999.0 | HRD-in | -75.43, -53.65 | 76.33, -6.74 | none-out-none | SNCnon | out-none | ActLoopNT-out | 7.915 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 143.05 | APE8-dihe-in | -77.71, 68.12 | APE8-rot-na | 28.54 | APE67-dihe-in | -70.85, -6.5 | -47.64, -45.7 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.734 | V948R | None | None | XRAY | 2.218 | 0.235 | 0.293 | A | 330 | 262 | 22 | 0 | 0 | 15 | [[712, 970]] | 1.0 | 9gdv | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.1e-88 | 300.1 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 9GDVB | P00533 | 702 | 985 | 1210.0 | Q6K:1101 | Type1 | Inactive | DFGin | 4.579 | 15.491 | BLBtrans | -111.43, 179.21 | 66.37, 26.18 | -74.59, 129.04 | 147.85, 63.03 | 60.16, 37.36 | out-none | out | 12.538 | Saltbr-none | 999.0 | HRD-out | -124.5, 90.89 | -69.11, -17.02 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 149.32 | APE8-dihe-in | -80.3, 68.77 | APE8-rot-na | 2.98 | APE67-dihe-in | -69.33, -16.36 | -50.05, -40.21 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.271 | V948R | None | None | XRAY | 2.218 | 0.235 | 0.293 | B | 330 | 267 | 17 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 9gdv | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.1e-88 | 300.1 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|