| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 6DUKA | P00533 | 701 | 1006 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.4162 | 14.8008 | BLBplus | -133.89, 165.03 | 66.94, 37.08 | -93.36, 166.29 | 58.42, 86.37 | 91.91, 6.11 | out-out | out | 13.9176 | Saltbr-out | 14.1793 | HRD-in | -76.73, -64.87 | 85.37, -18.97 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.4382 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.39, -10.84 | APE9-dihe-in | -125.5, 116.79 | APE8-dihe-in | -80.16, 76.04 | APE8-rot-na | 31.69 | APE67-dihe-in | -76.14, -1.34 | -58.18, -44.83 | APE12-dist-na | 17.3641 | APE11-dist-na | 15.2023 | APE10-dist-na | 11.7763 | APE9-dist-in | 7.3106 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | A | 331.0 | 306.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6duk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKB | P00533 | 699 | 1007 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6806 | 14.6502 | BLBplus | -136.44, 165.42 | 61.83, 36.22 | -89.54, 161.73 | 53.44, 89.67 | 90.48, 19.39 | out-out | out | 13.8125 | Saltbr-out | 14.7331 | HRD-in | -68.48, -61.78 | 82.94, -15.18 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.2922 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 128.53 | APE8-dihe-in | -76.17, 63.91 | APE8-rot-na | 26.99 | APE67-dihe-in | -79.83, -2.27 | -51.77, -41.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.9222 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | B | 331.0 | 296.0 | 13 | 30 | 17 | 13 | [[712, 970]] | 1.0 | 6duk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKC | P00533 | 699 | 1007 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6614 | 14.3909 | BLBplus | -137.36, 170.05 | 61.14, 32.95 | -87.42, 165.36 | 52.89, 84.68 | 86.51, 15.0 | out-out | out | 13.7494 | Saltbr-out | 12.3873 | HRD-in | -66.04, -61.2 | 80.35, -9.27 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.2862 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.92 | APE8-dihe-in | -77.64, 67.39 | APE8-rot-na | 32.93 | APE67-dihe-in | -71.69, -8.16 | -55.72, -42.95 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.8229 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | C | 331.0 | 295.0 | 14 | 30 | 16 | 14 | [[712, 970]] | 1.0 | 6duk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKD | P00533 | 701 | 1007 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6052 | 14.6344 | BLBplus | -137.83, 165.45 | 65.63, 29.61 | -82.3, 167.28 | 56.12, 84.13 | 94.16, 13.47 | out-out | out | 14.053 | Saltbr-out | 14.8858 | HRD-in | -74.03, -57.71 | 81.46, -18.53 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.3207 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -76.03, 11.31 | APE9-dihe-in | -134.89, 121.24 | APE8-dihe-in | -86.59, 77.19 | APE8-rot-na | 34.21 | APE67-dihe-in | -72.84, -7.51 | -59.65, -43.13 | APE12-dist-na | 17.7472 | APE11-dist-na | 15.5553 | APE10-dist-na | 11.9033 | APE9-dist-in | 7.5388 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | D | 331.0 | 307.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6duk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKE | P00533 | 698 | 1007 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.7057 | 14.387 | BLBplus | -132.31, 167.27 | 63.11, 42.82 | -102.17, 159.55 | 52.62, 85.09 | 88.84, 16.78 | out-out | out | 13.7684 | Saltbr-out | 14.3613 | HRD-in | -70.33, -59.21 | 85.76, -23.74 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.6865 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 1.83 | APE9-dihe-in | -127.74, 112.92 | APE8-dihe-in | -68.38, 64.27 | APE8-rot-na | 21.48 | APE67-dihe-in | -73.72, -8.33 | -52.7, -41.98 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.2913 | APE9-dist-in | 7.9406 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | E | 331.0 | 298.0 | 12 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 6duk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKF | P00533 | 701 | 1009 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6528 | 14.6121 | BLBplus | -133.82, 164.75 | 63.96, 32.85 | -83.32, 163.7 | 53.83, 93.49 | 88.31, 19.42 | out-out | out | 14.1084 | Saltbr-out | 15.1439 | HRD-in | -67.38, -62.37 | 88.35, -19.9 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.3188 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 115.72 | APE8-dihe-in | -80.72, 70.63 | APE8-rot-na | 32.98 | APE67-dihe-in | -75.6, -2.87 | -62.49, -36.24 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.8407 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | F | 331.0 | 298.0 | 11 | 30 | 19 | 11 | [[712, 970]] | 1.0 | 6duk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKD | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.8614 | 14.45 | BLBplus | -134.29, 170.65 | 60.11, 37.92 | -95.07, 160.21 | 48.8, 86.41 | 74.63, 26.88 | out-out | out | 13.4574 | Saltbr-out | 11.7626 | HRD-in | -66.46, -59.56 | 80.54, -6.1 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.9029 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.41 | APE8-dihe-in | -81.29, 71.57 | APE8-rot-na | 30.4 | APE67-dihe-in | -73.66, -4.05 | -53.54, -44.77 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4718 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | D | 331.0 | 294.0 | 14 | 30 | 16 | 14 | [[712, 970]] | 1.0 | 7jxk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPA | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.7467 | 14.6167 | BLBplus | -136.18, 166.76 | 64.66, 34.04 | -92.53, 168.9 | 56.02, 85.41 | 85.63, 11.86 | out-out | out | 13.9879 | Saltbr-out | 14.3068 | HRD-in | -74.54, -64.28 | 89.28, -17.63 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.5088 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -97.63, -15.8 | APE9-dihe-in | -113.05, 126.54 | APE8-dihe-in | -83.29, 68.9 | APE8-rot-na | 33.94 | APE67-dihe-in | -74.36, -3.96 | -52.3, -47.62 | APE12-dist-na | 17.0956 | APE11-dist-na | 14.9557 | APE10-dist-na | 11.6928 | APE9-dist-in | 7.4058 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | A | 331.0 | 308.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 7jxp | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPB | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6706 | 14.5109 | BLBplus | -135.21, 165.17 | 64.35, 37.85 | -90.15, 169.17 | 53.82, 91.67 | 84.59, 7.68 | out-out | out | 13.7558 | Saltbr-out | 13.8881 | HRD-in | -70.65, -63.17 | 87.36, -17.28 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.5923 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -97.44, -17.16 | APE9-dihe-in | -126.66, 129.43 | APE8-dihe-in | -78.52, 67.74 | APE8-rot-na | 34.72 | APE67-dihe-in | -76.32, -3.64 | -51.52, -45.13 | APE12-dist-na | 17.4376 | APE11-dist-na | 15.2142 | APE10-dist-na | 12.2746 | APE9-dist-in | 7.6166 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | B | 331.0 | 308.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 7jxp | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPD | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.766 | 14.6606 | BLBplus | -135.69, 167.35 | 65.6, 33.96 | -89.97, 168.72 | 55.6, 87.2 | 84.96, 9.82 | out-out | out | 13.5259 | Saltbr-out | 11.2829 | HRD-in | -71.06, -65.03 | 87.13, -14.24 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.0039 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.01 | APE8-dihe-in | -77.89, 69.26 | APE8-rot-na | 33.29 | APE67-dihe-in | -74.9, -2.69 | -52.27, -42.76 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.7443 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | D | 331.0 | 294.0 | 14 | 30 | 16 | 14 | [[712, 970]] | 1.0 | 7jxp | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPF | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.9745 | 14.7024 | BLBplus | -136.82, 166.82 | 61.14, 36.57 | -93.57, 171.83 | 53.4, 92.66 | 83.03, -0.51 | out-out | out | 13.6744 | Saltbr-out | 11.5698 | HRD-in | -71.01, -63.71 | 87.17, -13.68 | out-out-none | SNCoon | out-none | ActLoopNT-out | 9.118 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 127.33 | APE8-dihe-in | -78.62, 69.48 | APE8-rot-na | 32.72 | APE67-dihe-in | -72.69, -4.28 | -52.16, -45.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.6211 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | F | 331.0 | 294.0 | 14 | 30 | 16 | 14 | [[712, 970]] | 1.0 | 7jxp | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKA | P00533 | 700 | 1007 | 1210.0 | 8BS:1101,JBJ:1102 | Type1,Type3 | Inactive | DFGin | 4.8625 | 14.8244 | BLBplus | -134.12, 169.24 | 58.43, 39.5 | -93.7, 161.51 | 49.25, 87.25 | 75.0, 16.23 | out-out | out | 13.7778 | Saltbr-out | 10.4611 | HRD-in | -66.55, -57.53 | 81.35, -6.11 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.8163 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.68 | APE8-dihe-in | -81.09, 70.58 | APE8-rot-na | 30.58 | APE67-dihe-in | -73.21, -4.24 | -54.1, -46.78 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4886 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | A | 331.0 | 293.0 | 15 | 30 | 15 | 15 | [[712, 970]] | 1.0 | 7jxk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKC | P00533 | 701 | 1007 | 1210.0 | 8BS:1101,JBJ:1102 | Type1,Type3 | Inactive | DFGin | 4.5028 | 14.594 | BLBplus | -134.13, 170.52 | 59.34, 39.88 | -92.58, 159.61 | 51.08, 87.14 | 75.55, 20.71 | out-out | out | 13.6078 | Saltbr-out | 11.9254 | HRD-in | -66.31, -58.5 | 79.98, -6.68 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.4402 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.55 | APE8-dihe-in | -81.28, 70.99 | APE8-rot-na | 30.58 | APE67-dihe-in | -73.05, -5.14 | -53.98, -44.81 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4444 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | C | 331.0 | 292.0 | 15 | 30 | 15 | 15 | [[712, 970]] | 1.0 | 7jxk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKE | P00533 | 700 | 1007 | 1210.0 | 8BS:1101,JBJ:1102 | Type1,Type3 | Inactive | DFGin | 4.8927 | 14.4875 | BLBplus | -134.7, 170.02 | 59.73, 38.84 | -95.72, 161.23 | 49.85, 87.39 | 75.41, 21.47 | out-out | out | 13.5094 | Saltbr-out | 11.7833 | HRD-in | -66.69, -59.11 | 80.54, -6.15 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.43 | APE8-dihe-in | -79.83, 71.88 | APE8-rot-na | 29.74 | APE67-dihe-in | -73.96, -4.52 | -53.36, -45.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.5344 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | E | 331.0 | 287.0 | 16 | 30 | 14 | 16 | [[712, 970]] | 1.0 | 7jxk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKF | P00533 | 700 | 1007 | 1210.0 | 8BS:1101,JBJ:1102 | Type1,Type3 | Inactive | DFGin | 4.8717 | 14.3868 | BLBplus | -134.77, 169.91 | 59.08, 39.36 | -94.94, 160.87 | 49.89, 87.34 | 75.14, 17.06 | out-out | out | 13.5278 | Saltbr-out | 12.787 | HRD-in | -66.88, -58.5 | 80.33, -5.79 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 137.79 | APE8-dihe-in | -81.39, 71.1 | APE8-rot-na | 29.52 | APE67-dihe-in | -73.84, -5.2 | -54.64, -45.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4784 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | F | 331.0 | 292.0 | 16 | 30 | 14 | 16 | [[712, 970]] | 1.0 | 7jxk | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPC | P00533 | 700 | 1007 | 1210.0 | JBJ:1101,YY3:1102 | Type3,Type1 | Inactive | DFGin | 4.791 | 14.4893 | BLBplus | -135.14, 166.93 | 58.75, 39.54 | -88.72, 165.62 | 50.16, 82.07 | 80.91, 11.4 | out-out | out | 13.2148 | Saltbr-out | 10.0097 | HRD-in | -71.03, -65.61 | 90.59, -16.24 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 133.4 | APE8-dihe-in | -78.08, 71.31 | APE8-rot-na | 31.49 | APE67-dihe-in | -74.31, -4.1 | -55.2, -45.03 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.7338 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | C | 331.0 | 292.0 | 16 | 30 | 14 | 16 | [[712, 970]] | 1.0 | 7jxp | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPE | P00533 | 700 | 1007 | 1210.0 | JBJ:1101,YY3:1102 | Type3,Type1 | Inactive | DFGin | 5.0169 | 14.7096 | BLBplus | -135.91, 163.38 | 57.21, 38.2 | -87.34, 167.11 | 54.31, 95.16 | 79.16, 16.43 | out-out | out | 13.5808 | Saltbr-out | 11.0085 | HRD-in | -68.91, -62.25 | 86.58, -12.8 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 129.81 | APE8-dihe-in | -81.71, 69.65 | APE8-rot-na | 31.8 | APE67-dihe-in | -77.02, -5.14 | -52.47, -41.73 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4598 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | E | 331.0 | 287.0 | 16 | 30 | 14 | 16 | [[712, 970]] | 1.0 | 7jxp | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 6DUKA | P00533 | 701 | 1006 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.4162 | 14.8008 | BLBplus | -133.89, 165.03 | 66.94, 37.08 | -93.36, 166.29 | 58.42, 86.37 | 91.91, 6.11 | out-out | out | 13.9176 | Saltbr-out | 14.1793 | HRD-in | -76.73, -64.87 | 85.37, -18.97 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.4382 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.39, -10.84 | APE9-dihe-in | -125.5, 116.79 | APE8-dihe-in | -80.16, 76.04 | APE8-rot-na | 31.69 | APE67-dihe-in | -76.14, -1.34 | -58.18, -44.83 | APE12-dist-na | 17.3641 | APE11-dist-na | 15.2023 | APE10-dist-na | 11.7763 | APE9-dist-in | 7.3106 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | A | 331.0 | 306.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6duk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKB | P00533 | 699 | 1007 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6806 | 14.6502 | BLBplus | -136.44, 165.42 | 61.83, 36.22 | -89.54, 161.73 | 53.44, 89.67 | 90.48, 19.39 | out-out | out | 13.8125 | Saltbr-out | 14.7331 | HRD-in | -68.48, -61.78 | 82.94, -15.18 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.2922 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 128.53 | APE8-dihe-in | -76.17, 63.91 | APE8-rot-na | 26.99 | APE67-dihe-in | -79.83, -2.27 | -51.77, -41.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.9222 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | B | 331.0 | 296.0 | 13 | 30 | 17 | 13 | [[712, 970]] | 1.0 | 6duk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKC | P00533 | 699 | 1007 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6614 | 14.3909 | BLBplus | -137.36, 170.05 | 61.14, 32.95 | -87.42, 165.36 | 52.89, 84.68 | 86.51, 15.0 | out-out | out | 13.7494 | Saltbr-out | 12.3873 | HRD-in | -66.04, -61.2 | 80.35, -9.27 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.2862 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.92 | APE8-dihe-in | -77.64, 67.39 | APE8-rot-na | 32.93 | APE67-dihe-in | -71.69, -8.16 | -55.72, -42.95 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.8229 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | C | 331.0 | 295.0 | 14 | 30 | 16 | 14 | [[712, 970]] | 1.0 | 6duk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKD | P00533 | 701 | 1007 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6052 | 14.6344 | BLBplus | -137.83, 165.45 | 65.63, 29.61 | -82.3, 167.28 | 56.12, 84.13 | 94.16, 13.47 | out-out | out | 14.053 | Saltbr-out | 14.8858 | HRD-in | -74.03, -57.71 | 81.46, -18.53 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.3207 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -76.03, 11.31 | APE9-dihe-in | -134.89, 121.24 | APE8-dihe-in | -86.59, 77.19 | APE8-rot-na | 34.21 | APE67-dihe-in | -72.84, -7.51 | -59.65, -43.13 | APE12-dist-na | 17.7472 | APE11-dist-na | 15.5553 | APE10-dist-na | 11.9033 | APE9-dist-in | 7.5388 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | D | 331.0 | 307.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 6duk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKE | P00533 | 698 | 1007 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.7057 | 14.387 | BLBplus | -132.31, 167.27 | 63.11, 42.82 | -102.17, 159.55 | 52.62, 85.09 | 88.84, 16.78 | out-out | out | 13.7684 | Saltbr-out | 14.3613 | HRD-in | -70.33, -59.21 | 85.76, -23.74 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.6865 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 1.83 | APE9-dihe-in | -127.74, 112.92 | APE8-dihe-in | -68.38, 64.27 | APE8-rot-na | 21.48 | APE67-dihe-in | -73.72, -8.33 | -52.7, -41.98 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.2913 | APE9-dist-in | 7.9406 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | E | 331.0 | 298.0 | 12 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 6duk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 6DUKF | P00533 | 701 | 1009 | 1210.0 | ANP:1102,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6528 | 14.6121 | BLBplus | -133.82, 164.75 | 63.96, 32.85 | -83.32, 163.7 | 53.83, 93.49 | 88.31, 19.42 | out-out | out | 14.1084 | Saltbr-out | 15.1439 | HRD-in | -67.38, -62.37 | 88.35, -19.9 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.3188 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 115.72 | APE8-dihe-in | -80.72, 70.63 | APE8-rot-na | 32.98 | APE67-dihe-in | -75.6, -2.87 | -62.49, -36.24 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.8407 | T790M,V948R | None | None | XRAY | 2.2 | 0.191 | 0.223 | F | 331.0 | 298.0 | 11 | 30 | 19 | 11 | [[712, 970]] | 1.0 | 6duk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKD | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.8614 | 14.45 | BLBplus | -134.29, 170.65 | 60.11, 37.92 | -95.07, 160.21 | 48.8, 86.41 | 74.63, 26.88 | out-out | out | 13.4574 | Saltbr-out | 11.7626 | HRD-in | -66.46, -59.56 | 80.54, -6.1 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.9029 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.41 | APE8-dihe-in | -81.29, 71.57 | APE8-rot-na | 30.4 | APE67-dihe-in | -73.66, -4.05 | -53.54, -44.77 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4718 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | D | 331.0 | 294.0 | 14 | 30 | 16 | 14 | [[712, 970]] | 1.0 | 7jxk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPA | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.7467 | 14.6167 | BLBplus | -136.18, 166.76 | 64.66, 34.04 | -92.53, 168.9 | 56.02, 85.41 | 85.63, 11.86 | out-out | out | 13.9879 | Saltbr-out | 14.3068 | HRD-in | -74.54, -64.28 | 89.28, -17.63 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.5088 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -97.63, -15.8 | APE9-dihe-in | -113.05, 126.54 | APE8-dihe-in | -83.29, 68.9 | APE8-rot-na | 33.94 | APE67-dihe-in | -74.36, -3.96 | -52.3, -47.62 | APE12-dist-na | 17.0956 | APE11-dist-na | 14.9557 | APE10-dist-na | 11.6928 | APE9-dist-in | 7.4058 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | A | 331.0 | 308.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 7jxp | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPB | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.6706 | 14.5109 | BLBplus | -135.21, 165.17 | 64.35, 37.85 | -90.15, 169.17 | 53.82, 91.67 | 84.59, 7.68 | out-out | out | 13.7558 | Saltbr-out | 13.8881 | HRD-in | -70.65, -63.17 | 87.36, -17.28 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.5923 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -97.44, -17.16 | APE9-dihe-in | -126.66, 129.43 | APE8-dihe-in | -78.52, 67.74 | APE8-rot-na | 34.72 | APE67-dihe-in | -76.32, -3.64 | -51.52, -45.13 | APE12-dist-na | 17.4376 | APE11-dist-na | 15.2142 | APE10-dist-na | 12.2746 | APE9-dist-in | 7.6166 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | B | 331.0 | 308.0 | 0 | 30 | 30 | 0 | [[712, 970]] | 1.0 | 7jxp | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPD | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.766 | 14.6606 | BLBplus | -135.69, 167.35 | 65.6, 33.96 | -89.97, 168.72 | 55.6, 87.2 | 84.96, 9.82 | out-out | out | 13.5259 | Saltbr-out | 11.2829 | HRD-in | -71.06, -65.03 | 87.13, -14.24 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.0039 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 134.01 | APE8-dihe-in | -77.89, 69.26 | APE8-rot-na | 33.29 | APE67-dihe-in | -74.9, -2.69 | -52.27, -42.76 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.7443 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | D | 331.0 | 294.0 | 14 | 30 | 16 | 14 | [[712, 970]] | 1.0 | 7jxp | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPF | P00533 | 700 | 1007 | 1210.0 | ANP:1101,JBJ:1103 | ATPlike,Type3 | Inactive | DFGin | 4.9745 | 14.7024 | BLBplus | -136.82, 166.82 | 61.14, 36.57 | -93.57, 171.83 | 53.4, 92.66 | 83.03, -0.51 | out-out | out | 13.6744 | Saltbr-out | 11.5698 | HRD-in | -71.01, -63.71 | 87.17, -13.68 | out-out-none | SNCoon | out-none | ActLoopNT-out | 9.118 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 127.33 | APE8-dihe-in | -78.62, 69.48 | APE8-rot-na | 32.72 | APE67-dihe-in | -72.69, -4.28 | -52.16, -45.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.6211 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | F | 331.0 | 294.0 | 14 | 30 | 16 | 14 | [[712, 970]] | 1.0 | 7jxp | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKA | P00533 | 700 | 1007 | 1210.0 | 8BS:1101,JBJ:1102 | Type1,Type3 | Inactive | DFGin | 4.8625 | 14.8244 | BLBplus | -134.12, 169.24 | 58.43, 39.5 | -93.7, 161.51 | 49.25, 87.25 | 75.0, 16.23 | out-out | out | 13.7778 | Saltbr-out | 10.4611 | HRD-in | -66.55, -57.53 | 81.35, -6.11 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.8163 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.68 | APE8-dihe-in | -81.09, 70.58 | APE8-rot-na | 30.58 | APE67-dihe-in | -73.21, -4.24 | -54.1, -46.78 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4886 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | A | 331.0 | 293.0 | 15 | 30 | 15 | 15 | [[712, 970]] | 1.0 | 7jxk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKC | P00533 | 701 | 1007 | 1210.0 | 8BS:1101,JBJ:1102 | Type1,Type3 | Inactive | DFGin | 4.5028 | 14.594 | BLBplus | -134.13, 170.52 | 59.34, 39.88 | -92.58, 159.61 | 51.08, 87.14 | 75.55, 20.71 | out-out | out | 13.6078 | Saltbr-out | 11.9254 | HRD-in | -66.31, -58.5 | 79.98, -6.68 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.4402 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.55 | APE8-dihe-in | -81.28, 70.99 | APE8-rot-na | 30.58 | APE67-dihe-in | -73.05, -5.14 | -53.98, -44.81 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4444 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | C | 331.0 | 292.0 | 15 | 30 | 15 | 15 | [[712, 970]] | 1.0 | 7jxk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKE | P00533 | 700 | 1007 | 1210.0 | 8BS:1101,JBJ:1102 | Type1,Type3 | Inactive | DFGin | 4.8927 | 14.4875 | BLBplus | -134.7, 170.02 | 59.73, 38.84 | -95.72, 161.23 | 49.85, 87.39 | 75.41, 21.47 | out-out | out | 13.5094 | Saltbr-out | 11.7833 | HRD-in | -66.69, -59.11 | 80.54, -6.15 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.43 | APE8-dihe-in | -79.83, 71.88 | APE8-rot-na | 29.74 | APE67-dihe-in | -73.96, -4.52 | -53.36, -45.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.5344 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | E | 331.0 | 287.0 | 16 | 30 | 14 | 16 | [[712, 970]] | 1.0 | 7jxk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXKF | P00533 | 700 | 1007 | 1210.0 | 8BS:1101,JBJ:1102 | Type1,Type3 | Inactive | DFGin | 4.8717 | 14.3868 | BLBplus | -134.77, 169.91 | 59.08, 39.36 | -94.94, 160.87 | 49.89, 87.34 | 75.14, 17.06 | out-out | out | 13.5278 | Saltbr-out | 12.787 | HRD-in | -66.88, -58.5 | 80.33, -5.79 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 137.79 | APE8-dihe-in | -81.39, 71.1 | APE8-rot-na | 29.52 | APE67-dihe-in | -73.84, -5.2 | -54.64, -45.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4784 | T790M,V948R | None | None | XRAY | 3.1 | 0.223 | 0.261 | F | 331.0 | 292.0 | 16 | 30 | 14 | 16 | [[712, 970]] | 1.0 | 7jxk | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPC | P00533 | 700 | 1007 | 1210.0 | JBJ:1101,YY3:1102 | Type3,Type1 | Inactive | DFGin | 4.791 | 14.4893 | BLBplus | -135.14, 166.93 | 58.75, 39.54 | -88.72, 165.62 | 50.16, 82.07 | 80.91, 11.4 | out-out | out | 13.2148 | Saltbr-out | 10.0097 | HRD-in | -71.03, -65.61 | 90.59, -16.24 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 133.4 | APE8-dihe-in | -78.08, 71.31 | APE8-rot-na | 31.49 | APE67-dihe-in | -74.31, -4.1 | -55.2, -45.03 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.7338 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | C | 331.0 | 292.0 | 16 | 30 | 14 | 16 | [[712, 970]] | 1.0 | 7jxp | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7JXPE | P00533 | 700 | 1007 | 1210.0 | JBJ:1101,YY3:1102 | Type3,Type1 | Inactive | DFGin | 5.0169 | 14.7096 | BLBplus | -135.91, 163.38 | 57.21, 38.2 | -87.34, 167.11 | 54.31, 95.16 | 79.16, 16.43 | out-out | out | 13.5808 | Saltbr-out | 11.0085 | HRD-in | -68.91, -62.25 | 86.58, -12.8 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 129.81 | APE8-dihe-in | -81.71, 69.65 | APE8-rot-na | 31.8 | APE67-dihe-in | -77.02, -5.14 | -52.47, -41.73 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4598 | T790M,V948R | None | None | XRAY | 2.16 | 0.214 | 0.247 | E | 331.0 | 287.0 | 16 | 30 | 14 | 16 | [[712, 970]] | 1.0 | 7jxp | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.3e-88 | 300.5 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|