| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 5Z0SA | P11362 | 464 | 762 | 822.0 | 960:801 | Type1 | Inactive | DFGin | 5.1257 | 13.6012 | BLAplus | -107.75, 154.51 | 67.56, 21.06 | -67.0, -16.05 | 58.84, 83.24 | -104.7, 10.76 | in-in | in | 8.0938 | Saltbr-in | 2.7426 | HRD-in | -68.85, -52.46 | 79.64, -4.73 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7089 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -91.28, 165.51 | APE9-dihe-in | -109.21, 113.36 | APE8-dihe-out | -56.28, -24.44 | APE8-rot-na | 329.92 | APE67-dihe-in | -71.21, -1.87 | -54.7, -23.75 | APE12-dist-na | 19.955 | APE11-dist-na | 21.515 | APE10-dist-na | 19.768 | APE9-dist-out | 11.9765 | C488A,C584S | None | None | XRAY | 2.45 | 0.227 | 0.275 | A | 308.0 | 285.0 | 14 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5z0s | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5Z0SB | P11362 | 464 | 761 | 822.0 | 960:801 | Type1 | Inactive | DFGin | 5.1968 | 13.4303 | BLAplus | -118.1, 161.06 | 54.97, 27.99 | -69.34, -31.76 | 53.53, 89.4 | -87.91, 8.99 | in-in | in | 7.9457 | Saltbr-in | 2.9791 | HRD-in | -70.36, -53.32 | 74.41, -8.98 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8736 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.22, 166.31 | APE9-dihe-in | -107.5, 114.63 | APE8-dihe-out | -57.82, -27.73 | APE8-rot-na | 335.53 | APE67-dihe-in | -71.06, -7.47 | -49.72, -27.2 | APE12-dist-na | 19.5916 | APE11-dist-na | 21.3902 | APE10-dist-na | 19.7826 | APE9-dist-out | 11.7613 | C488A,C584S | None | None | XRAY | 2.45 | 0.227 | 0.275 | B | 308.0 | 281.0 | 17 | 30 | 29 | 1 | [[478, 756]] | 1.0 | 5z0s | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 5Z0SA | P11362 | 464 | 762 | 822.0 | 960:801 | Type1 | Inactive | DFGin | 5.1257 | 13.6012 | BLAplus | -107.75, 154.51 | 67.56, 21.06 | -67.0, -16.05 | 58.84, 83.24 | -104.7, 10.76 | in-in | in | 8.0938 | Saltbr-in | 2.7426 | HRD-in | -68.85, -52.46 | 79.64, -4.73 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7089 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -91.28, 165.51 | APE9-dihe-in | -109.21, 113.36 | APE8-dihe-out | -56.28, -24.44 | APE8-rot-na | 329.92 | APE67-dihe-in | -71.21, -1.87 | -54.7, -23.75 | APE12-dist-na | 19.955 | APE11-dist-na | 21.515 | APE10-dist-na | 19.768 | APE9-dist-out | 11.9765 | C488A,C584S | None | None | XRAY | 2.45 | 0.227 | 0.275 | A | 308.0 | 285.0 | 14 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5z0s | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5Z0SB | P11362 | 464 | 761 | 822.0 | 960:801 | Type1 | Inactive | DFGin | 5.1968 | 13.4303 | BLAplus | -118.1, 161.06 | 54.97, 27.99 | -69.34, -31.76 | 53.53, 89.4 | -87.91, 8.99 | in-in | in | 7.9457 | Saltbr-in | 2.9791 | HRD-in | -70.36, -53.32 | 74.41, -8.98 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8736 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.22, 166.31 | APE9-dihe-in | -107.5, 114.63 | APE8-dihe-out | -57.82, -27.73 | APE8-rot-na | 335.53 | APE67-dihe-in | -71.06, -7.47 | -49.72, -27.2 | APE12-dist-na | 19.5916 | APE11-dist-na | 21.3902 | APE10-dist-na | 19.7826 | APE9-dist-out | 11.7613 | C488A,C584S | None | None | XRAY | 2.45 | 0.227 | 0.275 | B | 308.0 | 281.0 | 17 | 30 | 29 | 1 | [[478, 756]] | 1.0 | 5z0s | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|