| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK1 | MK01_HUMAN | 4QTAA | P28482 | 10 | 358 | 360.0 | 38Z:411 | Type1.5_Front | Inactive | DFGin | 6.9014 | 16.419 | BLAminus | -127.54, 173.07 | 71.53, 87.6 | -104.51, 22.85 | 289.22, 73.36 | -66.57, -25.44 | in-in | in | 9.6271 | Saltbr-in | 2.6475 | HRD-in | -72.05, -50.52 | 77.72, -5.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7868 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 141.19 | APE8-rot-out | 186.7 | APE67-dihe-in | -78.23, -10.32 | -106.34, 7.24 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.45 | 0.16 | 0.191 | A | 361.0 | 335.0 | 14 | 31 | 17 | 14 | [[25, 313]] | 1.0 | 4qta | CMGC_MAPK1_HUMAN | CMGC | 9.2e-86 | 293.7 | 1.0 | 301.0 | 301.0 | 166 | 167 | 168 | 170 | 172 | 54 | 71 | 75 | 146 | 148 | 147 | 149.0 | 210 | 197 | 192 | 191 | 190 | 189 | 188 | 187 | 186 | 106 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK3 | MK03_HUMAN | 4QTBA | P27361 | 24 | 374 | 379.0 | 38Z:418 | Type1.5_Front | Inactive | DFGin | 6.9632 | 16.1915 | BLAminus | -128.63, 172.06 | 72.12, 87.31 | -104.64, 23.58 | 286.23, 74.76 | -64.07, -28.14 | in-in | in | 9.6383 | Saltbr-in | 2.6538 | HRD-in | -72.11, -54.76 | 73.09, 8.34 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7675 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -93.95, -29.12 | APE9-dihe-na | -67.78, 160.1 | APE8-dihe-in | -53.91, 125.98 | APE8-rot-in | 310.28 | APE67-dihe-in | -65.26, -17.27 | -52.54, -50.1 | APE12-dist-out | 14.1554 | APE11-dist-in | 10.8041 | APE10-dist-in | 6.8428 | APE9-dist-in | 4.4119 | None | None | None | XRAY | 1.4 | 0.148 | 0.175 | A | 380.0 | 351.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 4qtb | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| CMGC | MAPK3 | MK03_HUMAN | 4QTBB | P27361 | 27 | 374 | 379.0 | 38Z:412 | Type1.5_Front | Inactive | DFGin | 6.9886 | 16.0949 | BLAminus | -131.38, 169.9 | 76.01, 86.99 | -105.18, 21.27 | 288.36, 77.86 | -59.51, -32.2 | in-in | in | 9.5939 | Saltbr-in | 2.7088 | HRD-in | -72.51, -53.5 | 77.51, 5.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8241 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -90.9, -27.9 | APE9-dihe-na | -67.55, 157.04 | APE8-dihe-in | -54.84, 126.95 | APE8-rot-in | 308.82 | APE67-dihe-in | -67.72, -16.58 | -53.94, -47.75 | APE12-dist-out | 14.1875 | APE11-dist-in | 10.8583 | APE10-dist-in | 7.0815 | APE9-dist-in | 4.4109 | None | None | None | XRAY | 1.4 | 0.148 | 0.175 | B | 380.0 | 348.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 4qtb | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| CMGC | MAPK8 | MK08_HUMAN | 4QTDA | P45983 | 6 | 363 | 427.0 | 38Z:424,ANP:425 | Type1,Allosteric | Inactive | DFGin | 4.2787 | 13.95 | ABAminus | -89.69, -21.2 | -135.34, 171.77 | -115.48, 9.24 | 298.02, 89.8 | 87.52, -156.74 | in-out | in | 9.5926 | Saltbr-out | 4.1531 | HRD-in | -75.36, -55.62 | 72.51, -12.26 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.6893 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -117.32, 137.81 | APE9-dihe-na | -80.42, 132.23 | APE8-dihe-in | -83.54, 120.1 | APE8-rot-in | 296.41 | APE67-dihe-in | -61.39, -20.52 | -109.55, -3.05 | APE12-dist-out | 21.1401 | APE11-dist-out | 16.032 | APE10-dist-out | 16.5166 | APE9-dist-out | 11.1471 | None | None | None | XRAY | 1.5 | 0.167 | 0.192 | A | 364.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 4qtd | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| OTHER | HASPIN | HASP_HUMAN | 4QTCA | Q8TF76 | 469 | 798 | 798.0 | 38Z:804 | Type1 | Active | DFGin | 4.7427 | 12.6972 | BLAminus | -128.25, 174.11 | 72.8, 94.29 | -100.86, 22.55 | 311.48, 126.56 | -49.88, -46.32 | in-in | in | 9.2442 | Saltbr-in | 2.7674 | HRD-naN | -70.64, -49.71 | 73.49, 0.07 | in-in-na | SNCiia | in-na | ActLoopNT-in | 2.8616 | ActLoopCT-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | APE10-dihe-na | -118.14, 15.58 | APE9-dihe-na | -74.4, 166.34 | APE8-dihe-na | -155.61, 167.98 | APE8-rot-na | 54.8 | APE67-dihe-na | -159.6, 141.49 | 96.89, -1.32 | APE12-dist-na | 9.3996 | APE11-dist-na | 13.2932 | APE10-dist-na | 16.8897 | APE9-dist-na | 13.1424 | None | None | None | XRAY | 1.4 | 0.15 | 0.164 | A | 357.0 | 330.0 | 0 | 35 | 35 | 0 | [[484, 797]] | 1.0 | 4qtc | OTHER_HASPIN_HUMAN | HASP | 1.4e-226 | 756.6 | 1.0 | 314.0 | 314.0 | 686 | 687 | 688 | 690 | 692 | 511 | 535 | 539 | 646 | 648 | 647 | 649.0 | 741 | 721 | 716 | 715 | 714 | 713 | 712 | 711 | 710 | 604 | Serine/threonine-protein kinase haspin |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK1 | MK01_HUMAN | 4QTAA | P28482 | 10 | 358 | 360.0 | 38Z:411 | Type1.5_Front | Inactive | DFGin | 6.9014 | 16.419 | BLAminus | -127.54, 173.07 | 71.53, 87.6 | -104.51, 22.85 | 289.22, 73.36 | -66.57, -25.44 | in-in | in | 9.6271 | Saltbr-in | 2.6475 | HRD-in | -72.05, -50.52 | 77.72, -5.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7868 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 141.19 | APE8-rot-out | 186.7 | APE67-dihe-in | -78.23, -10.32 | -106.34, 7.24 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.45 | 0.16 | 0.191 | A | 361.0 | 335.0 | 14 | 31 | 17 | 14 | [[25, 313]] | 1.0 | 4qta | Homo sapiens | CMGC_MAPK1_HUMAN | CMGC | 9.2e-86 | 293.7 | 1.0 | 301.0 | 301.0 | 166 | 167 | 168 | 170 | 172 | 54 | 71 | 75 | 146 | 148 | 147 | 149.0 | 210 | 197 | 192 | 191 | 190 | 189 | 188 | 187 | 186 | 106 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK3 | MK03_HUMAN | 4QTBA | P27361 | 24 | 374 | 379.0 | 38Z:418 | Type1.5_Front | Inactive | DFGin | 6.9632 | 16.1915 | BLAminus | -128.63, 172.06 | 72.12, 87.31 | -104.64, 23.58 | 286.23, 74.76 | -64.07, -28.14 | in-in | in | 9.6383 | Saltbr-in | 2.6538 | HRD-in | -72.11, -54.76 | 73.09, 8.34 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7675 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -93.95, -29.12 | APE9-dihe-na | -67.78, 160.1 | APE8-dihe-in | -53.91, 125.98 | APE8-rot-in | 310.28 | APE67-dihe-in | -65.26, -17.27 | -52.54, -50.1 | APE12-dist-out | 14.1554 | APE11-dist-in | 10.8041 | APE10-dist-in | 6.8428 | APE9-dist-in | 4.4119 | None | None | None | XRAY | 1.4 | 0.148 | 0.175 | A | 380.0 | 351.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 4qtb | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| CMGC | MAPK3 | MK03_HUMAN | 4QTBB | P27361 | 27 | 374 | 379.0 | 38Z:412 | Type1.5_Front | Inactive | DFGin | 6.9886 | 16.0949 | BLAminus | -131.38, 169.9 | 76.01, 86.99 | -105.18, 21.27 | 288.36, 77.86 | -59.51, -32.2 | in-in | in | 9.5939 | Saltbr-in | 2.7088 | HRD-in | -72.51, -53.5 | 77.51, 5.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8241 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -90.9, -27.9 | APE9-dihe-na | -67.55, 157.04 | APE8-dihe-in | -54.84, 126.95 | APE8-rot-in | 308.82 | APE67-dihe-in | -67.72, -16.58 | -53.94, -47.75 | APE12-dist-out | 14.1875 | APE11-dist-in | 10.8583 | APE10-dist-in | 7.0815 | APE9-dist-in | 4.4109 | None | None | None | XRAY | 1.4 | 0.148 | 0.175 | B | 380.0 | 348.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | 4qtb | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 3.2e-87 | 298.5 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| CMGC | MAPK8 | MK08_HUMAN | 4QTDA | P45983 | 6 | 363 | 427.0 | 38Z:424,ANP:425 | Type1,Allosteric | Inactive | DFGin | 4.2787 | 13.95 | ABAminus | -89.69, -21.2 | -135.34, 171.77 | -115.48, 9.24 | 298.02, 89.8 | 87.52, -156.74 | in-out | in | 9.5926 | Saltbr-out | 4.1531 | HRD-in | -75.36, -55.62 | 72.51, -12.26 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.6893 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oooo | APE10-dihe-na | -117.32, 137.81 | APE9-dihe-na | -80.42, 132.23 | APE8-dihe-in | -83.54, 120.1 | APE8-rot-in | 296.41 | APE67-dihe-in | -61.39, -20.52 | -109.55, -3.05 | APE12-dist-out | 21.1401 | APE11-dist-out | 16.032 | APE10-dist-out | 16.5166 | APE9-dist-out | 11.1471 | None | None | None | XRAY | 1.5 | 0.167 | 0.192 | A | 364.0 | 355.0 | 3 | 27 | 24 | 3 | [[26, 321]] | 1.0 | 4qtd | Homo sapiens | CMGC_MAPK8_HUMAN | CMGC | 4.3e-84 | 288.2 | 1.0 | 301.0 | 301.0 | 168 | 169 | 170 | 172 | 174 | 55 | 73 | 77 | 148 | 150 | 149 | 151.0 | 207 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 109 | Mitogen-activated protein kinase 8 |
| OTHER | HASPIN | HASP_HUMAN | 4QTCA | Q8TF76 | 469 | 798 | 798.0 | 38Z:804 | Type1 | Active | DFGin | 4.7427 | 12.6972 | BLAminus | -128.25, 174.11 | 72.8, 94.29 | -100.86, 22.55 | 311.48, 126.56 | -49.88, -46.32 | in-in | in | 9.2442 | Saltbr-in | 2.7674 | HRD-naN | -70.64, -49.71 | 73.49, 0.07 | in-in-na | SNCiia | in-na | ActLoopNT-in | 2.8616 | ActLoopCT-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | APE10-dihe-na | -118.14, 15.58 | APE9-dihe-na | -74.4, 166.34 | APE8-dihe-na | -155.61, 167.98 | APE8-rot-na | 54.8 | APE67-dihe-na | -159.6, 141.49 | 96.89, -1.32 | APE12-dist-na | 9.3996 | APE11-dist-na | 13.2932 | APE10-dist-na | 16.8897 | APE9-dist-na | 13.1424 | None | None | None | XRAY | 1.4 | 0.15 | 0.164 | A | 357.0 | 330.0 | 0 | 35 | 35 | 0 | [[484, 797]] | 1.0 | 4qtc | Homo sapiens | OTHER_HASPIN_HUMAN | HASP | 1.4e-226 | 756.6 | 1.0 | 314.0 | 314.0 | 686 | 687 | 688 | 690 | 692 | 511 | 535 | 539 | 646 | 648 | 647 | 649.0 | 741 | 721 | 716 | 715 | 714 | 713 | 712 | 711 | 710 | 604 | Serine/threonine-protein kinase haspin |
| CMGC | MAPK1 | MK01_RAT | 5HD7A | P63086 | 9 | 355 | 358.0 | 38Z:401 | Type1 | Inactive | DFGin | 6.6169 | 16.3974 | BLAminus | -128.09, 178.37 | 68.56, 85.26 | -107.06, 21.62 | 285.69, 78.69 | -70.28, -12.54 | in-in | in | 9.5452 | Saltbr-in | 2.6662 | HRD-in | -71.35, -50.28 | 70.7, 8.65 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7976 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -98.73, -37.18 | APE9-dihe-na | -62.95, 158.16 | APE8-dihe-in | -50.32, 124.93 | APE8-rot-in | 314.5 | APE67-dihe-in | -63.38, -19.4 | -51.82, -51.63 | APE12-dist-out | 14.404 | APE11-dist-in | 11.122 | APE10-dist-in | 7.2822 | APE9-dist-in | 4.4034 | G167D | None | None | XRAY | 1.69 | 0.182 | 0.207 | A | 365.0 | 347.0 | 0 | 31 | 31 | 0 | [[23, 311]] | 1.0 | 5hd7 | Rattus norvegicus | CMGC_MAPK1_RAT | CMGC | 8e-84 | 287.3 | 1.0 | 301.0 | 301.0 | 164 | 165 | 166 | 168 | 170 | 52 | 69 | 73 | 144 | 146 | 145 | 147.0 | 208 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 104 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_RAT | 5HD4A | P63086 | 9 | 355 | 358.0 | 38Z:401 | Type1.5_Front | Inactive | DFGin | 6.7617 | 16.3963 | BLAminus | -132.15, 171.71 | 72.04, 89.95 | -105.49, 25.28 | 288.89, 74.15 | -62.94, -29.6 | in-in | in | 9.6091 | Saltbr-in | 2.6511 | HRD-in | -73.9, -52.49 | 73.6, 6.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7885 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -96.81, -40.96 | APE9-dihe-na | -60.91, 155.22 | APE8-dihe-in | -46.4, 120.98 | APE8-rot-in | 315.89 | APE67-dihe-in | -62.79, -18.63 | -49.8, -50.9 | APE12-dist-out | 14.32 | APE11-dist-in | 11.0677 | APE10-dist-in | 7.1595 | APE9-dist-in | 4.4363 | None | None | None | XRAY | 1.45 | 0.177 | 0.199 | A | 365.0 | 347.0 | 0 | 31 | 31 | 0 | [[23, 311]] | 1.0 | 5hd4 | Rattus norvegicus | CMGC_MAPK1_RAT | CMGC | 1.4e-85 | 293.1 | 1.0 | 301.0 | 301.0 | 164 | 165 | 166 | 168 | 170 | 52 | 69 | 73 | 144 | 146 | 145 | 147.0 | 208 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 104 | Mitogen-activated protein kinase 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK1 | MK01_RAT | 5HD7A | P63086 | 9 | 355 | 358.0 | 38Z:401 | Type1 | Inactive | DFGin | 6.6169 | 16.3974 | BLAminus | -128.09, 178.37 | 68.56, 85.26 | -107.06, 21.62 | 285.69, 78.69 | -70.28, -12.54 | in-in | in | 9.5452 | Saltbr-in | 2.6662 | HRD-in | -71.35, -50.28 | 70.7, 8.65 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7976 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -98.73, -37.18 | APE9-dihe-na | -62.95, 158.16 | APE8-dihe-in | -50.32, 124.93 | APE8-rot-in | 314.5 | APE67-dihe-in | -63.38, -19.4 | -51.82, -51.63 | APE12-dist-out | 14.404 | APE11-dist-in | 11.122 | APE10-dist-in | 7.2822 | APE9-dist-in | 4.4034 | G167D | None | None | XRAY | 1.69 | 0.182 | 0.207 | A | 365.0 | 347.0 | 0 | 31 | 31 | 0 | [[23, 311]] | 1.0 | 5hd7 | Rattus norvegicus | CMGC_MAPK1_RAT | CMGC | 8e-84 | 287.3 | 1.0 | 301.0 | 301.0 | 164 | 165 | 166 | 168 | 170 | 52 | 69 | 73 | 144 | 146 | 145 | 147.0 | 208 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 104 | Mitogen-activated protein kinase 1 |
| CMGC | MAPK1 | MK01_RAT | 5HD4A | P63086 | 9 | 355 | 358.0 | 38Z:401 | Type1.5_Front | Inactive | DFGin | 6.7617 | 16.3963 | BLAminus | -132.15, 171.71 | 72.04, 89.95 | -105.49, 25.28 | 288.89, 74.15 | -62.94, -29.6 | in-in | in | 9.6091 | Saltbr-in | 2.6511 | HRD-in | -73.9, -52.49 | 73.6, 6.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7885 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_oiii | APE10-dihe-na | -96.81, -40.96 | APE9-dihe-na | -60.91, 155.22 | APE8-dihe-in | -46.4, 120.98 | APE8-rot-in | 315.89 | APE67-dihe-in | -62.79, -18.63 | -49.8, -50.9 | APE12-dist-out | 14.32 | APE11-dist-in | 11.0677 | APE10-dist-in | 7.1595 | APE9-dist-in | 4.4363 | None | None | None | XRAY | 1.45 | 0.177 | 0.199 | A | 365.0 | 347.0 | 0 | 31 | 31 | 0 | [[23, 311]] | 1.0 | 5hd4 | Rattus norvegicus | CMGC_MAPK1_RAT | CMGC | 1.4e-85 | 293.1 | 1.0 | 301.0 | 301.0 | 164 | 165 | 166 | 168 | 170 | 52 | 69 | 73 | 144 | 146 | 145 | 147.0 | 208 | 195 | 190 | 189 | 188 | 187 | 186 | 185 | 184 | 104 | Mitogen-activated protein kinase 1 |