| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TGFBR2 | 5E92A | P37173 | 240 | 543 | 567.0 | ANP:601 | ATPlike | Active | DFGin | 7.3963 | 13.3025 | BLAminus | -134.93, 178.1 | 63.07, 87.04 | -105.26, 16.76 | 300.78, 96.96 | -60.58, -26.14 | in-in | in | 7.67 | Saltbr-in | 2.7517 | HRD-in | -64.87, -46.8 | 71.14, -4.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9815 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.21, 144.17 | APE9-dihe-na | 126.96, -149.92 | APE8-dihe-in | -116.55, 119.38 | APE8-rot-in | 300.41 | APE67-dihe-in | -54.91, -33.03 | -42.96, -45.47 | APE12-dist-in | 11.7882 | APE11-dist-in | 12.049 | APE10-dist-in | 6.0891 | APE9-dist-in | 3.4015 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.08 | 0.204 | 0.231 | A | 316.0 | 298.0 | 6 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 5e92 | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | AF-P37173-K1A | P37173 | 236 | 548 | 567.0 | No_ligand | No_ligand | Active | DFGin | 7.0837 | 13.9094 | BLAminus | -138.68, 178.14 | 66.07, 64.88 | -85.47, 16.34 | 299.05, 89.75 | -63.1, -19.55 | in-in | in | 7.9081 | Saltbr-in | 2.7125 | HRD-in | -79.08, -44.48 | 64.09, 6.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9495 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.89, 165.46 | APE9-dihe-na | 108.18, -177.72 | APE8-dihe-in | -90.28, 117.48 | APE8-rot-in | 303.87 | APE67-dihe-in | -56.54, -32.09 | -49.32, -37.74 | APE12-dist-in | 9.805 | APE11-dist-in | 11.6546 | APE10-dist-in | 5.7311 | APE9-dist-in | 3.4147 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 313.0 | 313.0 | 0 | 32 | 32 | 0 | [[244, 540]] | 1.0 | AF-P37173-K1 | TKL_TGFBR2_HUMAN | TKL | 7.6e-79 | 270.9 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | AF-P37173-K3A | P37173 | 236 | 548 | 567.0 | No_ligand | No_ligand | Active | DFGin | 7.0961 | 13.7999 | BLAminus | -145.43, -179.8 | 65.44, 55.08 | -78.17, 15.93 | 302.31, 97.78 | -63.13, -21.78 | in-in | in | 7.8135 | Saltbr-in | 2.6752 | HRD-in | -76.21, -45.24 | 65.87, -7.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9064 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.68, 164.76 | APE9-dihe-na | 101.26, -174.37 | APE8-dihe-in | -91.39, 117.43 | APE8-rot-in | 302.24 | APE67-dihe-in | -56.09, -30.7 | -47.98, -39.29 | APE12-dist-in | 10.0905 | APE11-dist-in | 11.7738 | APE10-dist-in | 5.8324 | APE9-dist-in | 3.3885 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 313.0 | 313.0 | 0 | 32 | 32 | 0 | [[244, 540]] | 1.0 | AF-P37173-K3 | TKL_TGFBR2_HUMAN | TKL | 7.6e-79 | 270.9 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | 8YGZA | P37173 | 240 | 541 | 567.0 | No_ligand | No_ligand | Active | DFGin | 7.1674 | 13.4988 | BLAminus | -147.8, -174.95 | 64.63, 68.72 | -94.18, 14.72 | 296.7, 105.77 | -58.39, -30.7 | in-in | in | 7.556 | Saltbr-in | 2.7124 | HRD-in | -68.27, -53.07 | 76.97, -2.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9275 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -76.56, 144.37 | APE9-dihe-na | 118.33, -168.14 | APE8-dihe-in | -88.89, 116.91 | APE8-rot-in | 306.92 | APE67-dihe-in | -53.81, -35.04 | -53.5, -42.61 | APE12-dist-in | 11.4813 | APE11-dist-in | 11.99 | APE10-dist-in | 6.1235 | APE9-dist-in | 4.0018 | None | None | CSO483 | XRAY | 2.1 | 0.198 | 0.254 | A | 314.0 | 290.0 | 12 | 32 | 28 | 4 | [[244, 540]] | 1.0 | 8ygz | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | 5E8VA | P37173 | 240 | 541 | 567.0 | No_ligand | No_ligand | Active | DFGin | 7.3995 | 13.7547 | BLAminus | -147.31, -173.83 | 59.32, 66.92 | -91.34, 13.8 | 295.18, 100.62 | -56.78, -28.25 | in-in | in | 7.5858 | Saltbr-in | 2.721 | HRD-in | -69.01, -47.09 | 70.71, -0.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9044 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -110.44, 139.23 | APE9-dihe-na | 124.18, -154.69 | APE8-dihe-in | -103.85, 121.46 | APE8-rot-in | 300.53 | APE67-dihe-in | -54.24, -33.71 | -49.52, -44.15 | APE12-dist-in | 12.0242 | APE11-dist-in | 12.0587 | APE10-dist-in | 6.1979 | APE9-dist-in | 3.5162 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 1.69 | 0.194 | 0.219 | A | 316.0 | 296.0 | 6 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 5e8v | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | 5E91A | P37173 | 240 | 543 | 567.0 | 5L4:601 | Type1 | Active | DFGin | 7.3985 | 13.6133 | BLAminus | -147.14, -171.85 | 61.39, 64.81 | -93.01, 17.49 | 298.43, 101.83 | -55.7, -31.33 | in-in | in | 7.6524 | Saltbr-in | 2.7401 | HRD-in | -67.96, -50.27 | 72.9, 0.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9217 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.96, 139.39 | APE9-dihe-na | 125.36, -159.39 | APE8-dihe-in | -101.78, 120.18 | APE8-rot-in | 301.71 | APE67-dihe-in | -56.78, -33.79 | -49.19, -43.11 | APE12-dist-in | 11.4745 | APE11-dist-in | 11.874 | APE10-dist-in | 5.9086 | APE9-dist-in | 3.6604 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.42 | 0.209 | 0.242 | A | 316.0 | 297.0 | 7 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 5e91 | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | 7DV6A | P37173 | 240 | 543 | 567.0 | HJF:9000 | Type1 | Active | DFGin | 7.1311 | 13.4318 | BLAminus | -156.15, -164.95 | 57.9, 60.45 | -93.44, 15.51 | 294.56, 110.64 | -56.6, -36.89 | in-in | in | 7.4443 | Saltbr-in | 2.6595 | HRD-in | -60.78, -51.79 | 74.77, -4.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8603 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.14, 141.57 | APE9-dihe-na | 113.33, -173.4 | APE8-dihe-in | -82.04, 128.94 | APE8-rot-in | 303.35 | APE67-dihe-in | -55.96, -36.36 | -60.86, -38.17 | APE12-dist-in | 11.5078 | APE11-dist-in | 11.8903 | APE10-dist-in | 6.0465 | APE9-dist-in | 3.9117 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.39 | 0.163 | 0.224 | A | 323.0 | 304.0 | 0 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 7dv6 | TKL_TGFBR2_HUMAN | TKL | 2.1e-77 | 266.2 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | 5E8YA | P37173 | 240 | 541 | 567.0 | STU:601 | Type1 | Inactive | DFGin | 7.4313 | 13.6382 | ABAminus | -147.57, -29.88 | -97.01, 88.29 | -98.27, 19.66 | 300.85, 114.87 | -63.28, -27.98 | in-in | in | 7.6628 | Saltbr-in | 2.6836 | HRD-in | -60.19, -53.17 | 75.99, -7.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8159 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -101.67, 141.68 | APE9-dihe-na | 119.62, -164.78 | APE8-dihe-in | -99.54, 120.03 | APE8-rot-in | 310.13 | APE67-dihe-in | -59.04, -35.21 | -51.44, -37.92 | APE12-dist-in | 11.2111 | APE11-dist-in | 12.0735 | APE10-dist-in | 5.9745 | APE9-dist-in | 4.0108 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.05 | 0.198 | 0.227 | A | 316.0 | 298.0 | 4 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 5e8y | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | 5QINA | P37173 | 240 | 541 | 567.0 | J2V:601 | Type1 | None | DFGin | 7.4322 | 13.6924 | BLAminus | -160.38, -171.51 | 70.13, 63.56 | -97.31, 22.31 | 300.17, 115.61 | -64.51, -28.45 | in-in | in | 7.7525 | Saltbr-in | 2.968 | HRD-in | -64.72, -51.48 | 70.07, 3.51 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9449 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -105.98, 157.24 | APE9-dihe-na | 110.69, -170.54 | APE8-dihe-in | -92.43, 119.77 | APE8-rot-in | 303.14 | APE67-dihe-in | -57.21, -32.74 | -53.66, -41.1 | APE12-dist-none | 999.0 | APE11-dist-in | 12.1938 | APE10-dist-in | 6.0999 | APE9-dist-in | 3.9176 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 1.57 | 0.188 | 0.203 | A | 316.0 | 295.0 | 7 | 32 | 30 | 2 | [[244, 540]] | 1.0 | 5qin | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TGFBR2 | TGFR2_HUMAN | 5E92A | P37173 | 240 | 543 | 567.0 | ANP:601 | ATPlike | Active | DFGin | 7.3963 | 13.3025 | BLAminus | -134.93, 178.1 | 63.07, 87.04 | -105.26, 16.76 | 300.78, 96.96 | -60.58, -26.14 | in-in | in | 7.67 | Saltbr-in | 2.7517 | HRD-in | -64.87, -46.8 | 71.14, -4.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9815 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.21, 144.17 | APE9-dihe-na | 126.96, -149.92 | APE8-dihe-in | -116.55, 119.38 | APE8-rot-in | 300.41 | APE67-dihe-in | -54.91, -33.03 | -42.96, -45.47 | APE12-dist-in | 11.7882 | APE11-dist-in | 12.049 | APE10-dist-in | 6.0891 | APE9-dist-in | 3.4015 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.08 | 0.204 | 0.231 | A | 316.0 | 298.0 | 6 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 5e92 | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | TGFR2_HUMAN | AF-P37173-K1A | P37173 | 236 | 548 | 567.0 | No_ligand | No_ligand | Active | DFGin | 7.0837 | 13.9094 | BLAminus | -138.68, 178.14 | 66.07, 64.88 | -85.47, 16.34 | 299.05, 89.75 | -63.1, -19.55 | in-in | in | 7.9081 | Saltbr-in | 2.7125 | HRD-in | -79.08, -44.48 | 64.09, 6.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9495 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.89, 165.46 | APE9-dihe-na | 108.18, -177.72 | APE8-dihe-in | -90.28, 117.48 | APE8-rot-in | 303.87 | APE67-dihe-in | -56.54, -32.09 | -49.32, -37.74 | APE12-dist-in | 9.805 | APE11-dist-in | 11.6546 | APE10-dist-in | 5.7311 | APE9-dist-in | 3.4147 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 313.0 | 313.0 | 0 | 32 | 32 | 0 | [[244, 540]] | 1.0 | AF-P37173-K1 | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 7.6e-79 | 270.9 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | TGFR2_HUMAN | AF-P37173-K3A | P37173 | 236 | 548 | 567.0 | No_ligand | No_ligand | Active | DFGin | 7.0961 | 13.7999 | BLAminus | -145.43, -179.8 | 65.44, 55.08 | -78.17, 15.93 | 302.31, 97.78 | -63.13, -21.78 | in-in | in | 7.8135 | Saltbr-in | 2.6752 | HRD-in | -76.21, -45.24 | 65.87, -7.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9064 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.68, 164.76 | APE9-dihe-na | 101.26, -174.37 | APE8-dihe-in | -91.39, 117.43 | APE8-rot-in | 302.24 | APE67-dihe-in | -56.09, -30.7 | -47.98, -39.29 | APE12-dist-in | 10.0905 | APE11-dist-in | 11.7738 | APE10-dist-in | 5.8324 | APE9-dist-in | 3.3885 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 313.0 | 313.0 | 0 | 32 | 32 | 0 | [[244, 540]] | 1.0 | AF-P37173-K3 | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 7.6e-79 | 270.9 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | TGFR2_HUMAN | 8YGZA | P37173 | 240 | 541 | 567.0 | No_ligand | No_ligand | Active | DFGin | 7.1674 | 13.4988 | BLAminus | -147.8, -174.95 | 64.63, 68.72 | -94.18, 14.72 | 296.7, 105.77 | -58.39, -30.7 | in-in | in | 7.556 | Saltbr-in | 2.7124 | HRD-in | -68.27, -53.07 | 76.97, -2.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9275 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -76.56, 144.37 | APE9-dihe-na | 118.33, -168.14 | APE8-dihe-in | -88.89, 116.91 | APE8-rot-in | 306.92 | APE67-dihe-in | -53.81, -35.04 | -53.5, -42.61 | APE12-dist-in | 11.4813 | APE11-dist-in | 11.99 | APE10-dist-in | 6.1235 | APE9-dist-in | 4.0018 | None | None | CSO483 | XRAY | 2.1 | 0.198 | 0.254 | A | 314.0 | 290.0 | 12 | 32 | 28 | 4 | [[244, 540]] | 1.0 | 8ygz | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | TGFR2_HUMAN | 5E8VA | P37173 | 240 | 541 | 567.0 | No_ligand | No_ligand | Active | DFGin | 7.3995 | 13.7547 | BLAminus | -147.31, -173.83 | 59.32, 66.92 | -91.34, 13.8 | 295.18, 100.62 | -56.78, -28.25 | in-in | in | 7.5858 | Saltbr-in | 2.721 | HRD-in | -69.01, -47.09 | 70.71, -0.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9044 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -110.44, 139.23 | APE9-dihe-na | 124.18, -154.69 | APE8-dihe-in | -103.85, 121.46 | APE8-rot-in | 300.53 | APE67-dihe-in | -54.24, -33.71 | -49.52, -44.15 | APE12-dist-in | 12.0242 | APE11-dist-in | 12.0587 | APE10-dist-in | 6.1979 | APE9-dist-in | 3.5162 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 1.69 | 0.194 | 0.219 | A | 316.0 | 296.0 | 6 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 5e8v | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | TGFR2_HUMAN | 5E91A | P37173 | 240 | 543 | 567.0 | 5L4:601 | Type1 | Active | DFGin | 7.3985 | 13.6133 | BLAminus | -147.14, -171.85 | 61.39, 64.81 | -93.01, 17.49 | 298.43, 101.83 | -55.7, -31.33 | in-in | in | 7.6524 | Saltbr-in | 2.7401 | HRD-in | -67.96, -50.27 | 72.9, 0.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9217 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.96, 139.39 | APE9-dihe-na | 125.36, -159.39 | APE8-dihe-in | -101.78, 120.18 | APE8-rot-in | 301.71 | APE67-dihe-in | -56.78, -33.79 | -49.19, -43.11 | APE12-dist-in | 11.4745 | APE11-dist-in | 11.874 | APE10-dist-in | 5.9086 | APE9-dist-in | 3.6604 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.42 | 0.209 | 0.242 | A | 316.0 | 297.0 | 7 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 5e91 | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | TGFR2_HUMAN | 7DV6A | P37173 | 240 | 543 | 567.0 | HJF:9000 | Type1 | Active | DFGin | 7.1311 | 13.4318 | BLAminus | -156.15, -164.95 | 57.9, 60.45 | -93.44, 15.51 | 294.56, 110.64 | -56.6, -36.89 | in-in | in | 7.4443 | Saltbr-in | 2.6595 | HRD-in | -60.78, -51.79 | 74.77, -4.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8603 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.14, 141.57 | APE9-dihe-na | 113.33, -173.4 | APE8-dihe-in | -82.04, 128.94 | APE8-rot-in | 303.35 | APE67-dihe-in | -55.96, -36.36 | -60.86, -38.17 | APE12-dist-in | 11.5078 | APE11-dist-in | 11.8903 | APE10-dist-in | 6.0465 | APE9-dist-in | 3.9117 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.39 | 0.163 | 0.224 | A | 323.0 | 304.0 | 0 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 7dv6 | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 2.1e-77 | 266.2 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | TGFR2_HUMAN | 5E8YA | P37173 | 240 | 541 | 567.0 | STU:601 | Type1 | Inactive | DFGin | 7.4313 | 13.6382 | ABAminus | -147.57, -29.88 | -97.01, 88.29 | -98.27, 19.66 | 300.85, 114.87 | -63.28, -27.98 | in-in | in | 7.6628 | Saltbr-in | 2.6836 | HRD-in | -60.19, -53.17 | 75.99, -7.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8159 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -101.67, 141.68 | APE9-dihe-na | 119.62, -164.78 | APE8-dihe-in | -99.54, 120.03 | APE8-rot-in | 310.13 | APE67-dihe-in | -59.04, -35.21 | -51.44, -37.92 | APE12-dist-in | 11.2111 | APE11-dist-in | 12.0735 | APE10-dist-in | 5.9745 | APE9-dist-in | 4.0108 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 2.05 | 0.198 | 0.227 | A | 316.0 | 298.0 | 4 | 32 | 32 | 0 | [[244, 540]] | 1.0 | 5e8y | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| TGFBR2 | TGFR2_HUMAN | 5QINA | P37173 | 240 | 541 | 567.0 | J2V:601 | Type1 | None | DFGin | 7.4322 | 13.6924 | BLAminus | -160.38, -171.51 | 70.13, 63.56 | -97.31, 22.31 | 300.17, 115.61 | -64.51, -28.45 | in-in | in | 7.7525 | Saltbr-in | 2.968 | HRD-in | -64.72, -51.48 | 70.07, 3.51 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9449 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_niii | APE10-dihe-na | -105.98, 157.24 | APE9-dihe-na | 110.69, -170.54 | APE8-dihe-in | -92.43, 119.77 | APE8-rot-in | 303.14 | APE67-dihe-in | -57.21, -32.74 | -53.66, -41.1 | APE12-dist-none | 999.0 | APE11-dist-in | 12.1938 | APE10-dist-in | 6.0999 | APE9-dist-in | 3.9176 | E431A,R433A,E485A,K488A,R493A,R495A | None | None | XRAY | 1.57 | 0.188 | 0.203 | A | 316.0 | 295.0 | 7 | 32 | 30 | 2 | [[244, 540]] | 1.0 | 5qin | Homo sapiens | TKL_TGFBR2_HUMAN | TKL | 1.9e-77 | 266.3 | 2.0 | 266.0 | 265.0 | 396 | 397 | 398 | 400 | 402 | 277 | 290 | 294 | 376 | 378 | 377 | 379.0 | 446 | 428 | 423 | 422 | 421 | 420 | 419 | 418 | 417 | 326 | TGF-beta receptor type-2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|