CAMK_PLK1 (Serine/threonine-protein kinase PLK1)

Total number of chains: 30
Active chains: 2
Uniprot: PLK1_HUMAN
Kinase Domain Residues: 53 - 305
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 30 100.0% AF-P53350-K1A

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PLK1 AF-P53350-K1A P53350 45 313 603.0 No_ligand No_ligand Active DFGin 5.5497 14.0178 BLAminus -138.81, -176.13 59.79, 75.65 -83.94, 15.34 292.62, 90.11 -62.81, -20.58 in-in in 9.0389 Saltbr-in 2.5765 HRD-in -77.19, -43.8 61.96, 8.95 in-in-in SNCiii in-in ActLoopNT-in 2.8977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.58, 167.37 APE9-dihe-na 111.84, 169.16 APE8-dihe-in -85.0, 135.3 APE8-rot-in 298.31 APE67-dihe-in -79.3, -5.41 -49.93, -42.14 APE12-dist-in 8.6475 APE11-dist-in 11.4873 APE10-dist-in 5.7926 APE9-dist-in 3.5019 None None None AF2 -1.0 1.0 1.0 A 269.0 269.0 0 28 28 0 [[53, 305]] 1.0 AF-P53350-K1 CAMK_PLK1_HUMAN CAMK 1.5e-79 272.9 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 AF-P53350-K3A P53350 45 313 603.0 No_ligand No_ligand Active DFGin 5.3419 13.9791 BLAminus -140.81, -172.37 56.25, 72.33 -75.86, 12.77 292.93, 94.61 -62.92, -13.77 in-in in 9.3285 Saltbr-in 2.5773 HRD-in -78.81, -41.77 63.16, 8.34 in-in-in SNCiii in-in ActLoopNT-in 2.9297 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.05, 166.42 APE9-dihe-na 111.25, 170.64 APE8-dihe-in -84.99, 137.05 APE8-rot-in 295.25 APE67-dihe-in -75.5, -4.86 -51.24, -44.46 APE12-dist-in 8.6323 APE11-dist-in 11.5523 APE10-dist-in 5.8724 APE9-dist-in 3.3228 None None None AF2 -1.0 1.0 1.0 A 269.0 269.0 0 28 28 0 [[53, 305]] 1.0 AF-P53350-K3 CAMK_PLK1_HUMAN CAMK 1.5e-79 272.9 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 8X72A P53350 37 330 603.0 ANP:401 ATPlike Inactive DFGin 5.6741 14.5619 BLAminus -124.66, -175.79 56.01, 84.34 -93.5, 28.11 290.48, 83.55 -67.08, -22.62 out-in out 10.0362 Saltbr-in 3.3691 HRD-in -69.02, -52.36 73.21, 2.03 in-in-out SNCiio in-out ActLoopNT-in 2.9948 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -79.36, 95.87 APE9-dihe-na 140.51, 168.33 APE8-dihe-in -120.38, 96.0 APE8-rot-in 313.63 APE67-dihe-out -71.46, -55.88 -64.61, 149.56 APE12-dist-in 10.8497 APE11-dist-out 7.4546 APE10-dist-in 7.6527 APE9-dist-out 8.0434 None None None XRAY 2.2 0.198 0.25 A 333.0 294.0 0 28 28 0 [[53, 305]] 1.0 8x72 CAMK_PLK1_HUMAN CAMK 1.7e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 2OU7A P53350 37 328 603.0 ANP:500 ATPlike Inactive DFGin 5.511 14.6261 BLAminus -126.46, 177.9 64.03, 83.89 -94.43, 31.27 293.9, 81.92 -69.65, -29.63 out-in out 10.0179 Saltbr-in 3.5992 HRD-in -73.43, -50.53 79.22, -6.25 in-in-out SNCiio in-out ActLoopNT-in 2.9589 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.17, 94.2 APE9-dihe-na 146.34, 174.25 APE8-dihe-in -131.14, 97.57 APE8-rot-in 299.54 APE67-dihe-out -68.04, -58.6 -56.03, 146.92 APE12-dist-in 10.3811 APE11-dist-out 7.1861 APE10-dist-in 7.4365 APE9-dist-out 8.2407 T210V None None XRAY 2.4 0.205 0.235 A 335.0 292.0 0 28 28 0 [[53, 305]] 1.0 2ou7 CAMK_PLK1_HUMAN CAMK 1.8e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 2V5QA P53350 39 323 603.0 No_ligand No_ligand Inactive DFGin 5.6857 14.7178 BLAminus -129.1, -167.08 62.93, 75.17 -93.89, 21.76 291.51, 90.84 -61.9, -28.72 out-in out 10.0226 Saltbr-in 3.0555 HRD-in -67.98, -52.02 73.91, 7.34 in-in-out SNCiio in-out ActLoopNT-in 2.8292 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -88.56, 3.75 APE9-dihe-na -179.48, -164.77 APE8-dihe-in -107.94, 115.2 APE8-rot-in 298.84 APE67-dihe-out -71.25, -55.87 -61.61, 160.98 APE12-dist-in 10.4375 APE11-dist-out 6.2368 APE10-dist-in 5.1223 APE9-dist-out 8.3334 None None None XRAY 2.3 0.184 0.224 A 315.0 285.0 0 28 28 0 [[53, 305]] 1.0 2v5q CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 2V5QB P53350 39 323 603.0 No_ligand No_ligand Inactive DFGin 5.6851 14.9246 BLAminus -131.35, -166.96 60.96, 77.54 -92.83, 32.21 286.27, 87.97 -68.24, -26.27 in-out in 9.9987 Saltbr-out 3.8415 HRD-in -74.56, -53.71 79.97, 1.03 out-in-out SNCoio in-out ActLoopNT-in 2.8674 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -91.44, 9.2 APE9-dihe-na -170.42, 178.21 APE8-dihe-in -101.74, 116.95 APE8-rot-in 316.2 APE67-dihe-out -61.71, -54.24 -52.66, 144.9 APE12-dist-in 9.9909 APE11-dist-out 6.7742 APE10-dist-in 6.4067 APE9-dist-out 8.4067 None None None XRAY 2.3 0.184 0.224 B 315.0 285.0 0 28 28 0 [[53, 305]] 1.0 2v5q CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 2YACA P53350 39 329 603.0 937:501 Type1 Inactive DFGin 5.7158 14.3054 BLAminus -136.25, -176.52 54.6, 87.71 -92.92, 28.24 289.9, 84.23 -75.6, -9.88 in-in in 9.4138 Saltbr-in 2.8323 HRD-in -79.87, -54.28 83.91, -4.3 in-in-out SNCiio in-out ActLoopNT-in 2.9371 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -90.18, 95.11 APE9-dihe-na 155.4, 174.07 APE8-dihe-in -130.99, 84.18 APE8-rot-out 67.16 APE67-dihe-out -74.05, -70.88 -62.65, 161.23 APE12-dist-in 11.0681 APE11-dist-out 7.3206 APE10-dist-in 7.6251 APE9-dist-out 8.1362 None None None XRAY 2.2 0.213 0.255 A 311.0 291.0 0 28 28 0 [[53, 305]] 1.0 2yac CAMK_PLK1_HUMAN CAMK 2.5e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 3KB7A P53350 39 328 603.0 071:1 Type1 Inactive DFGin 5.7088 14.0424 BLAminus -133.88, 179.17 62.15, 88.77 -94.79, 24.7 288.92, 88.27 -73.01, -6.62 in-in in 8.8871 Saltbr-in 2.6738 HRD-in -67.89, -55.24 69.06, -3.76 in-in-out SNCiio in-out ActLoopNT-in 2.9089 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_iooo APE10-dihe-na -99.22, 86.88 APE9-dihe-na 165.83, 172.24 APE8-dihe-in -120.96, 91.28 APE8-rot-out 68.09 APE67-dihe-out -76.36, -59.91 -62.3, 158.23 APE12-dist-in 11.1305 APE11-dist-out 7.3774 APE10-dist-out 8.0773 APE9-dist-out 8.1697 None None NMM324 XRAY 2.5 0.212 0.303 A 311.0 290.0 0 28 28 0 [[53, 305]] 1.0 3kb7 CAMK_PLK1_HUMAN CAMK 2.5e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 4A4LA P53350 39 329 603.0 939:1331 Type1 Inactive DFGin 5.7799 14.1347 BLAminus -141.7, -176.08 58.67, 82.87 -91.4, 34.14 289.94, 83.08 -71.42, -15.93 in-in in 9.4203 Saltbr-in 2.9397 HRD-in -74.58, -53.49 81.34, -4.51 in-in-out SNCiio in-out ActLoopNT-in 2.9169 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -83.54, 86.55 APE9-dihe-na 154.14, -178.12 APE8-dihe-in -129.31, 90.58 APE8-rot-out 60.31 APE67-dihe-out -60.53, -82.61 -62.07, 154.01 APE12-dist-in 11.0591 APE11-dist-out 7.3243 APE10-dist-in 7.6164 APE9-dist-out 8.4265 None None None XRAY 2.35 0.224 0.274 A 311.0 291.0 0 28 28 0 [[53, 305]] 1.0 4a4l CAMK_PLK1_HUMAN CAMK 2.5e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 4A4OA P53350 39 329 603.0 664:1332 Type1 Inactive DFGin 5.6431 14.005 BLAminus -140.91, 173.61 55.04, 90.94 -98.45, 26.61 287.86, 85.19 -77.07, -1.22 in-in in 9.3392 Saltbr-in 3.3484 HRD-in -69.08, -52.1 82.91, 0.02 in-in-out SNCiio in-out ActLoopNT-in 3.0053 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -84.2, 81.23 APE9-dihe-na 164.33, -176.93 APE8-dihe-in -120.87, 80.43 APE8-rot-in 310.59 APE67-dihe-out -59.02, -78.88 -57.5, 148.27 APE12-dist-in 11.1607 APE11-dist-out 7.22 APE10-dist-in 7.7616 APE9-dist-out 8.2051 None None None XRAY 2.7 0.23 0.282 A 311.0 291.0 0 28 28 0 [[53, 305]] 1.0 4a4o CAMK_PLK1_HUMAN CAMK 2.5e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R8BA P53350 37 326 603.0 A1JCP:1001 Type1 Inactive DFGin 5.7645 14.4195 BLAminus -135.37, -173.77 58.86, 75.37 -91.12, 20.8 284.65, 94.62 -63.52, -25.59 in-in in 8.4904 Saltbr-in 2.7158 HRD-in -71.84, -53.97 76.03, -0.52 in-in-out SNCiio in-out ActLoopNT-in 3.0153 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -85.35, 5.7 APE9-dihe-na -171.65, -172.53 APE8-dihe-in -108.35, 119.77 APE8-rot-in 298.21 APE67-dihe-out -65.23, -55.38 -66.82, 157.06 APE12-dist-in 10.6191 APE11-dist-out 6.9373 APE10-dist-in 5.948 APE9-dist-out 8.3177 None None None XRAY 2.2 0.191 0.238 A 315.0 290.0 0 28 28 0 [[53, 305]] 1.0 9r8b CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R8BB P53350 37 323 603.0 A1JCP:402 Type1 Inactive DFGin 5.8352 14.2917 BLAminus -131.75, -174.5 64.87, 76.68 -96.77, 19.5 288.39, 99.04 -77.27, -4.94 in-in in 8.1199 Saltbr-in 2.7542 HRD-out -68.92, 136.67 -118.63, -11.46 in-in-out SNCiio in-out ActLoopNT-in 3.0307 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiio APE10-dihe-na 86.04, 0.68 APE9-dihe-na 169.71, -156.66 APE8-dihe-in -118.48, 123.54 APE8-rot-in 319.34 APE67-dihe-out -62.56, -51.97 -66.18, 154.73 APE12-dist-in 10.4716 APE11-dist-in 8.1897 APE10-dist-in 5.7403 APE9-dist-out 9.562 None None None XRAY 2.2 0.191 0.238 B 315.0 287.0 0 28 28 0 [[53, 305]] 1.0 9r8b CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R8CA P53350 38 326 603.0 R78:1001 Type1 Inactive DFGin 5.5848 14.99 BLAminus -126.1, -176.63 65.4, 78.62 -95.8, 30.2 285.88, 88.19 -70.16, -23.86 in-in in 9.0969 Saltbr-in 2.8706 HRD-in -73.52, -53.38 78.38, -0.66 in-in-out SNCiio in-out ActLoopNT-in 2.9616 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.03, 32.02 APE9-dihe-na 163.26, -177.26 APE8-dihe-in -109.84, 116.09 APE8-rot-in 291.16 APE67-dihe-out -62.02, -59.2 -61.3, 153.09 APE12-dist-in 10.4112 APE11-dist-out 6.2561 APE10-dist-in 5.7623 APE9-dist-out 8.6225 None None None XRAY 2.243 0.191 0.236 A 315.0 289.0 0 28 28 0 [[53, 305]] 1.0 9r8c CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R8CB P53350 38 323 603.0 R78:1001 Type1 Inactive DFGin 5.5457 14.9956 BLAminus -130.55, -176.06 59.62, 83.99 -94.79, 30.62 285.83, 86.69 -68.45, -26.03 in-in in 9.1508 Saltbr-in 2.7676 HRD-in -75.84, -53.52 77.99, 2.7 in-in-out SNCiio in-out ActLoopNT-in 2.9529 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -89.08, 50.7 APE9-dihe-na 152.38, 176.7 APE8-dihe-in -113.61, 115.98 APE8-rot-in 316.69 APE67-dihe-out -67.47, -56.35 -62.32, 152.06 APE12-dist-in 9.9595 APE11-dist-out 7.059 APE10-dist-in 6.6227 APE9-dist-out 8.5077 None None None XRAY 2.243 0.191 0.236 B 315.0 286.0 0 28 28 0 [[53, 305]] 1.0 9r8c CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 4J52A P53350 38 330 603.0 1J3:400 Type1 Inactive DFGin 5.6732 14.405 BLAminus -132.19, -178.32 57.1, 88.41 -99.88, 23.54 290.9, 84.86 -66.29, -8.43 in-in in 9.3919 Saltbr-in 2.7014 HRD-in -83.32, -51.41 78.14, -8.7 in-in-out SNCiio in-out ActLoopNT-in 2.8667 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -92.24, 97.88 APE9-dihe-na 154.03, 172.56 APE8-dihe-in -123.15, 84.89 APE8-rot-in 302.52 APE67-dihe-out -69.1, -50.77 -69.03, 151.29 APE12-dist-in 10.9789 APE11-dist-out 7.3536 APE10-dist-in 7.8183 APE9-dist-out 7.821 T210V None None XRAY 2.3 0.198 0.241 A 293.0 293.0 0 28 28 0 [[53, 305]] 1.0 4j52 CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 4J53A P53350 38 330 603.0 1J4:403 Type1 Inactive DFGin 5.6397 14.5788 BLAminus -129.35, -169.37 44.41, 85.29 -91.22, 24.89 291.84, 82.06 -64.71, -23.25 in-in in 9.981 Saltbr-in 3.0097 HRD-in -75.81, -49.76 74.88, 0.23 in-in-out SNCiio in-out ActLoopNT-in 2.933 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -78.39, 101.76 APE9-dihe-na 146.02, 166.78 APE8-dihe-in -121.83, 82.96 APE8-rot-in 302.16 APE67-dihe-out -75.51, -62.04 -60.01, 151.77 APE12-dist-in 10.9528 APE11-dist-out 7.4006 APE10-dist-in 7.7633 APE9-dist-out 7.8563 T210V None None XRAY 2.5 0.183 0.24 A 293.0 293.0 0 28 28 0 [[53, 305]] 1.0 4j53 CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 2RKUA P53350 37 330 603.0 R78:500 Type1 Inactive DFGin 5.6778 15.0171 BLAminus -134.22, -169.5 54.06, 79.11 -86.67, 25.63 283.82, 88.21 -64.51, -26.07 in-in in 9.7168 Saltbr-in 3.0799 HRD-in -74.95, -48.26 75.93, -2.57 in-in-out SNCiio in-out ActLoopNT-in 2.9425 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -90.21, 90.69 APE9-dihe-na 162.46, 178.28 APE8-dihe-in -124.7, 88.6 APE8-rot-in 309.54 APE67-dihe-out -73.41, -64.04 -71.02, 160.05 APE12-dist-in 10.9294 APE11-dist-out 7.2828 APE10-dist-in 7.9206 APE9-dist-out 8.1342 T210V None None XRAY 1.95 0.192 0.241 A 294.0 294.0 0 28 28 0 [[53, 305]] 1.0 2rku CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 8BJTA P53350 39 330 603.0 8X7:402 Type1 Inactive DFGin 5.7433 14.3115 BLAminus -146.49, -170.45 55.69, 70.04 -90.08, 22.34 281.62, 90.95 -60.02, -37.94 in-in in 9.2218 Saltbr-in 2.728 HRD-in -68.54, -47.7 72.42, -10.0 in-in-out SNCiio in-out ActLoopNT-in 2.9242 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_iooo APE10-dihe-na -90.89, 99.31 APE9-dihe-na 143.06, 169.47 APE8-dihe-in -120.75, 101.21 APE8-rot-out 199.98 APE67-dihe-out -76.79, -55.69 -65.4, 158.12 APE12-dist-in 11.1597 APE11-dist-out 7.4033 APE10-dist-out 8.2363 APE9-dist-out 8.5627 None None None XRAY 2.188 0.203 0.255 A 294.0 292.0 0 28 28 0 [[53, 305]] 1.0 8bjt CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 3THBA P53350 42 328 603.0 3TA:1 Type1 Inactive DFGin 5.7628 14.2461 BLAminus -135.92, -170.43 55.15, 75.45 -87.11, 14.2 290.23, 88.06 -65.07, -8.71 in-in in 9.1247 Saltbr-in 3.5491 HRD-in -66.85, -49.24 73.84, -10.07 in-in-out SNCiio in-out ActLoopNT-in 2.9833 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -91.42, 101.79 APE9-dihe-na 126.02, 172.43 APE8-dihe-in -121.57, 103.22 APE8-rot-out 68.36 APE67-dihe-out -75.15, -60.09 -61.3, 157.38 APE12-dist-in 11.5794 APE11-dist-out 7.5519 APE10-dist-in 7.7464 APE9-dist-out 8.6498 T210V None None XRAY 2.5 0.253 0.286 A 333.0 287.0 0 28 28 0 [[53, 305]] 1.0 3thb CAMK_PLK1_HUMAN CAMK 1.7e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 2OWBA P53350 37 330 603.0 626:500 Type1 Inactive DFGin 5.7411 14.2734 BLAminus -131.62, -172.7 55.05, 82.45 -94.97, 27.99 289.46, 84.52 -70.38, -17.86 in-in in 9.5051 Saltbr-in 2.6351 HRD-in -72.25, -49.78 72.96, -0.12 in-in-out SNCiio in-out ActLoopNT-in 3.0056 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -85.58, 102.01 APE9-dihe-na 139.92, 169.2 APE8-dihe-in -127.98, 85.88 APE8-rot-in 302.45 APE67-dihe-out -70.16, -61.75 -57.83, 150.59 APE12-dist-in 10.9432 APE11-dist-out 7.4221 APE10-dist-in 7.6185 APE9-dist-out 7.9791 T210V None None XRAY 2.1 0.205 0.243 A 335.0 294.0 0 28 28 0 [[53, 305]] 1.0 2owb CAMK_PLK1_HUMAN CAMK 1.8e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 3FC2A P53350 37 329 603.0 IBI:10 Type1 Inactive DFGin 5.6869 14.8439 BLAminus -136.2, -169.15 47.8, 83.29 -92.73, 30.51 290.96, 88.11 -72.2, -20.77 in-in in 9.8452 Saltbr-in 2.7866 HRD-in -72.68, -50.74 75.03, 6.56 in-in-out SNCiio in-out ActLoopNT-in 2.9723 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -91.8, 110.95 APE9-dihe-na 128.06, 168.28 APE8-dihe-in -129.49, 88.48 APE8-rot-in 292.3 APE67-dihe-out -76.49, -62.11 -61.16, 163.08 APE12-dist-in 11.0036 APE11-dist-out 7.3642 APE10-dist-in 7.5319 APE9-dist-out 7.8848 T210V None None XRAY 2.45 0.184 0.226 A 335.0 293.0 0 28 28 0 [[53, 305]] 1.0 3fc2 CAMK_PLK1_HUMAN CAMK 1.8e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9D0PA P53350 37 330 603.0 8X7:401 Type1 Inactive DFGin 5.9321 14.4667 BLAminus -127.97, -167.66 73.35, 57.17 -81.61, 36.59 285.64, 88.68 -94.22, -12.32 in-in in 9.0933 Saltbr-in 2.7584 HRD-in -81.82, -53.71 82.64, -7.07 in-in-out SNCiio in-out ActLoopNT-in 2.9118 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -92.87, 112.89 APE9-dihe-na 127.84, 173.17 APE8-dihe-in -124.26, 98.89 APE8-rot-in 301.22 APE67-dihe-out -72.74, -55.92 -71.3, 155.26 APE12-dist-in 11.2956 APE11-dist-out 7.351 APE10-dist-in 7.4828 APE9-dist-out 8.252 T210V None None XRAY 2.65 0.247 0.29 A 335.0 294.0 0 28 28 0 [[53, 305]] 1.0 9d0p CAMK_PLK1_HUMAN CAMK 1.8e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R1WAAA P53350 38 334 603.0 A1JCP:401 Type1 Inactive DFGin 5.6292 14.3068 BLAminus -134.11, -168.09 56.45, 78.1 -90.07, 23.96 287.47, 94.05 -61.0, -27.64 in-in in 9.0559 Saltbr-in 2.8172 HRD-in -73.41, -49.99 71.11, 3.55 in-in-out SNCiio in-out ActLoopNT-in 2.9617 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -89.16, 9.34 APE9-dihe-na -169.47, 176.32 APE8-dihe-in -98.59, 112.0 APE8-rot-in 302.37 APE67-dihe-out -62.18, -51.19 -58.71, 150.32 APE12-dist-in 10.1834 APE11-dist-out 6.5586 APE10-dist-in 6.2363 APE9-dist-out 8.5025 K225D,K226A None None XRAY 2.2 0.18 0.216 AAA 325.0 297.0 0 28 28 0 [[53, 305]] 1.0 9r1w CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R1WBBB P53350 38 325 603.0 A1JCP:401 Type1 Inactive DFGin 5.6297 14.3508 BLAminus -133.86, -166.71 56.12, 78.59 -90.53, 23.21 288.19, 92.88 -61.02, -27.23 in-in in 9.2288 Saltbr-in 2.7447 HRD-in -73.38, -50.78 71.42, 4.57 in-in-out SNCiio in-out ActLoopNT-in 2.9696 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -89.57, 8.7 APE9-dihe-na -168.16, 173.41 APE8-dihe-in -98.08, 111.85 APE8-rot-in 305.79 APE67-dihe-out -62.5, -50.96 -59.11, 151.11 APE12-dist-in 10.0722 APE11-dist-out 6.5984 APE10-dist-in 6.1802 APE9-dist-out 8.4386 K225D,K226A None None XRAY 2.2 0.18 0.216 BBB 325.0 288.0 0 28 28 0 [[53, 305]] 1.0 9r1w CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R1XA P53350 39 334 603.0 R78:401 Type1 Inactive DFGin 5.4509 14.7459 BLAminus -129.34, -169.27 61.33, 81.84 -99.46, 30.78 291.65, 94.79 -60.61, -43.02 in-in in 9.6846 Saltbr-in 2.7211 HRD-in -71.39, -48.31 73.02, 3.83 in-in-out SNCiio in-out ActLoopNT-in 2.9715 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.63, 46.88 APE9-dihe-na 161.22, 163.69 APE8-dihe-in -103.28, 108.1 APE8-rot-in 301.35 APE67-dihe-out -58.97, -56.16 -54.1, 148.74 APE12-dist-in 10.3877 APE11-dist-out 6.5599 APE10-dist-in 6.7414 APE9-dist-out 8.5087 K225D,K226A None None XRAY 2.84 0.222 0.277 A 325.0 296.0 0 28 28 0 [[53, 305]] 1.0 9r1x CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R1XB P53350 39 326 603.0 R78:401 Type1 Inactive DFGin 5.4448 14.7258 BLAminus -129.89, -169.09 62.76, 81.42 -99.44, 28.81 292.45, 94.66 -58.03, -43.63 in-in in 9.6661 Saltbr-in 2.714 HRD-in -71.6, -47.96 72.32, 5.61 in-in-out SNCiio in-out ActLoopNT-in 2.9664 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -82.43, 34.44 APE9-dihe-na 160.48, 165.73 APE8-dihe-in -102.91, 108.17 APE8-rot-in 301.26 APE67-dihe-out -58.46, -55.69 -54.97, 148.64 APE12-dist-in 10.4044 APE11-dist-out 6.5324 APE10-dist-in 5.999 APE9-dist-out 8.4468 K225D,K226A None None XRAY 2.84 0.222 0.277 B 325.0 288.0 0 28 28 0 [[53, 305]] 1.0 9r1x CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R1YAAA P53350 38 334 603.0 A1JCQ:401 Type1 Inactive DFGin 5.4927 14.2673 BLAminus -126.75, -172.44 65.19, 77.92 -95.78, 35.59 294.04, 83.7 -66.64, -28.98 in-in in 9.4644 Saltbr-in 2.7444 HRD-in -71.96, -50.24 71.88, 5.14 in-in-out SNCiio in-out ActLoopNT-in 3.1029 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -88.57, 8.2 APE9-dihe-na -166.23, -178.27 APE8-dihe-in -105.79, 106.71 APE8-rot-in 300.95 APE67-dihe-out -66.32, -52.43 -54.05, 151.38 APE12-dist-in 10.2803 APE11-dist-out 6.4939 APE10-dist-in 6.1368 APE9-dist-out 8.3805 K225D,K226A None None XRAY 2.602 0.187 0.218 AAA 325.0 297.0 0 28 28 0 [[53, 305]] 1.0 9r1y CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 9R1YBBB P53350 38 325 603.0 A1JCQ:401 Type1 Inactive DFGin 5.5166 14.3492 BLAminus -126.84, -171.95 66.19, 77.61 -96.17, 35.42 294.69, 83.98 -66.59, -29.54 in-in in 9.5027 Saltbr-in 2.7444 HRD-in -72.69, -50.41 71.98, 5.19 in-in-out SNCiio in-out ActLoopNT-in 3.1096 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -88.39, 7.64 APE9-dihe-na -166.1, -178.49 APE8-dihe-in -105.58, 106.71 APE8-rot-in 302.14 APE67-dihe-out -65.99, -51.73 -54.43, 151.5 APE12-dist-in 10.3012 APE11-dist-out 6.4798 APE10-dist-in 5.9907 APE9-dist-out 8.3631 K225D,K226A None None XRAY 2.602 0.187 0.218 BBB 325.0 288.0 0 28 28 0 [[53, 305]] 1.0 9r1y CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 5TA6A P53350 37 330 603.0 79D:1000 Type1 Inactive DFGin 5.7677 14.6912 BLAminus -129.81, 178.93 63.79, 86.6 -95.82, 28.6 292.13, 79.82 -68.79, -23.38 in-in in 9.776 Saltbr-in 3.0598 HRD-in -68.63, -52.95 71.96, 8.35 in-in-out SNCiio in-out ActLoopNT-in 2.8889 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -85.92, 111.12 APE9-dihe-na 138.09, 164.23 APE8-dihe-in -126.56, 95.9 APE8-rot-out 85.27 APE67-dihe-out -71.06, -59.19 -57.19, 156.45 APE12-dist-in 10.9082 APE11-dist-out 7.3284 APE10-dist-in 7.6939 APE9-dist-out 7.5992 None None None XRAY 2.5 0.183 0.26 A 358.0 294.0 0 28 28 0 [[53, 305]] 1.0 5ta6 CAMK_PLK1_HUMAN CAMK 2.2e-78 269.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 5TA8A P53350 37 330 603.0 79C:402 Type1 Inactive DFGin 5.5977 14.3108 BLAminus -141.08, -172.7 51.52, 90.37 -96.67, 41.3 290.69, 89.43 -72.33, -19.61 in-in in 9.1072 Saltbr-in 2.7273 HRD-in -66.37, -49.24 72.53, -11.97 in-in-out SNCiio in-out ActLoopNT-in 2.8816 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -88.19, 81.36 APE9-dihe-na 134.61, 175.47 APE8-dihe-in -125.29, 109.1 APE8-rot-out 49.04 APE67-dihe-out -73.09, -62.08 -71.65, 169.34 APE12-dist-in 10.8099 APE11-dist-out 7.4727 APE10-dist-in 7.1878 APE9-dist-out 8.6926 None None None XRAY 2.6 0.185 0.247 A 358.0 294.0 0 28 28 0 [[53, 305]] 1.0 5ta8 CAMK_PLK1_HUMAN CAMK 2.2e-78 269.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1

CAMK_PLK1 (Serine/threonine-protein kinase PLK1)

Total number of chains: 42
Active chains: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 41 97.6% AF-P53350-K1A
DFGin ABAminus 1 2.4% 4J7BD

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PLK1 Q6DRK7_DANRE 4J7BD Q6DRK7 20 311 595.0 No_ligand No_ligand Inactive DFGin 5.4866 14.5549 ABAminus -129.81, -7.43 -133.83, 113.48 -107.04, 20.33 291.52, 92.27 -51.62, -38.38 out-in out 10.214 Saltbr-in 2.9657 HRD-in -68.9, -50.24 76.71, 4.14 in-in-out SNCiio in-out ActLoopNT-in 2.7455 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -126.82 APE8-dihe-in -131.87, 100.17 APE8-rot-in 301.55 APE67-dihe-out -78.82, -54.23 -64.35, 166.22 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 7.9466 D162N,E192F None None XRAY 2.3 0.208 0.264 D 297.0 281.0 11 28 17 11 [[39, 291]] 1.0 4j7b Danio rerio CAMK_PLK1_DANRE CAMK 8.1e-76 260.6 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3D5WA Q4KMI8 24 310 595.0 ADP:313 ATPlike Inactive DFGin 5.8398 15.103 BLAminus -136.31, -173.3 52.58, 90.43 -100.9, 29.72 290.61, 88.81 -67.31, -18.54 out-out out 10.538 Saltbr-out 4.5698 HRD-in -72.81, -47.33 67.56, -5.93 out-in-in SNCoii in-in ActLoopNT-in 2.9013 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.0, 153.74 APE9-dihe-na 145.11, -167.91 APE8-dihe-in -110.25, 127.19 APE8-rot-in 299.86 APE67-dihe-in -70.02, -15.96 -37.98, -47.89 APE12-dist-in 8.2509 APE11-dist-in 11.2747 APE10-dist-in 5.6458 APE9-dist-in 3.9124 None TPO196 TPO196 XRAY 2.6 0.244 0.271 A 317.0 285.0 2 28 28 0 [[39, 291]] 1.0 3d5w Danio rerio CAMK_PLK1_DANRE CAMK 4.6e-77 264.7 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q6DRK7_DANRE 3D5UA Q6DRK7 23 310 595.0 No_ligand No_ligand Inactive DFGin 5.6927 14.8088 BLAminus -132.0, -170.66 53.21, 91.71 -105.63, 34.97 291.53, 90.32 -70.7, -17.69 out-out out 10.6997 Saltbr-out 4.3498 HRD-in -73.43, -47.86 66.94, -9.91 out-in-out SNCoio in-out ActLoopNT-in 2.8874 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -83.53, 77.69 APE9-dihe-na 160.43, 176.55 APE8-dihe-in -120.81, 90.57 APE8-rot-in 316.96 APE67-dihe-out -68.11, -72.46 -73.03, 158.49 APE12-dist-in 10.6665 APE11-dist-out 7.4011 APE10-dist-in 7.5221 APE9-dist-out 8.4661 None None None XRAY 2.8 0.231 0.281 A 317.0 288.0 0 28 28 0 [[39, 291]] 1.0 3d5u Danio rerio CAMK_PLK1_DANRE CAMK 4.6e-77 264.7 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q6DRK7_DANRE 4J7BA Q6DRK7 18 311 595.0 No_ligand No_ligand Inactive DFGin 5.9575 14.8219 BLAminus -127.79, -166.66 63.28, 73.86 -94.07, 24.02 287.22, 93.09 -58.39, -32.32 in-in in 9.948 Saltbr-in 2.5261 HRD-in -69.09, -53.7 77.98, -8.47 in-in-out SNCiio in-out ActLoopNT-in 2.8139 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_nnio APE10-dihe-na 999.0, 170.84 APE9-dihe-na -82.59, -164.35 APE8-dihe-in -106.73, 113.42 APE8-rot-out 172.88 APE67-dihe-out -56.23, -64.85 -68.6, 152.66 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 5.9329 APE9-dist-out 8.4727 D162N,E192F None None XRAY 2.3 0.208 0.264 A 297.0 284.0 10 28 18 10 [[39, 291]] 1.0 4j7b Danio rerio CAMK_PLK1_DANRE CAMK 8.1e-76 260.6 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3D5XA Q4KMI8 24 309 595.0 KWT:1 Type1 Inactive DFGin 5.7483 14.936 BLAminus -139.39, -170.01 59.65, 84.09 -100.6, 25.02 290.64, 93.65 -64.4, -14.86 out-out out 10.666 Saltbr-out 4.3942 HRD-in -69.94, -48.19 73.11, -11.18 out-in-none SNCoin in-none ActLoopNT-in 3.0678 ActLoopCT-none nonTYR APEdihe_aannn APEdist_innn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-in 10.2963 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 2.8 0.263 0.299 A 301.0 279.0 7 28 21 7 [[39, 291]] 1.0 3d5x Danio rerio CAMK_PLK1_DANRE CAMK 8.9e-77 263.8 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DBEA Q4KMI8 24 310 595.0 4FR:1 Type1 Inactive DFGin 5.3305 14.2611 BLAminus -130.08, -172.43 53.96, 104.63 -115.22, 13.87 295.84, 91.17 -49.61, -15.58 out-out out 10.0731 Saltbr-out 4.3667 HRD-in -75.7, -52.21 77.46, -22.23 out-in-out SNCoio in-out ActLoopNT-in 2.9691 ActLoopCT-out nonTYR APEdihe_aannn APEdist_ionn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -89.97, -74.84 999.0, 157.6 APE12-dist-in 10.4051 APE11-dist-out 7.7345 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.32 0.237 0.27 A 301.0 284.0 3 28 25 3 [[39, 291]] 1.0 3dbe Danio rerio CAMK_PLK1_DANRE CAMK 8.9e-77 263.8 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DBFA Q4KMI8 24 310 595.0 5FR:1 Type1 Inactive DFGin 5.5692 14.5066 BLAminus -126.48, -167.26 59.45, 92.34 -110.0, 25.26 297.55, 90.95 -54.7, -27.45 in-out in 9.8779 Saltbr-out 4.027 HRD-in -77.45, -40.3 68.16, -16.48 out-in-none SNCoin in-none ActLoopNT-in 2.9286 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.2 0.234 0.275 A 301.0 261.0 26 28 8 20 [[39, 291]] 1.0 3dbf Danio rerio CAMK_PLK1_DANRE CAMK 8.9e-77 263.8 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DB8A Q4KMI8 24 310 595.0 1FR:313 Type1 Inactive DFGin 5.7592 14.6569 BLAminus -132.17, -175.89 60.33, 81.89 -97.25, 28.2 286.75, 81.14 -57.5, -31.84 in-out in 9.9095 Saltbr-out 3.8295 HRD-in -71.72, -45.68 69.14, -18.96 out-in-none SNCoin in-none ActLoopNT-in 2.8276 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.15 0.232 0.274 A 317.0 261.0 26 28 8 20 [[39, 291]] 1.0 3db8 Danio rerio CAMK_PLK1_DANRE CAMK 1.1e-76 263.5 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DBCA Q4KMI8 24 310 595.0 2FR:313 Type1 Inactive DFGin 5.7335 14.6643 BLAminus -136.39, -168.79 53.28, 74.51 -89.66, 27.23 289.49, 88.8 -63.71, -13.19 in-out in 9.6385 Saltbr-out 4.0559 HRD-in -85.71, -43.45 67.47, -24.22 out-in-none SNCoin in-none ActLoopNT-in 3.0181 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.35 0.245 0.288 A 317.0 261.0 26 28 8 20 [[39, 291]] 1.0 3dbc Danio rerio CAMK_PLK1_DANRE CAMK 1.1e-76 263.5 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DBDA Q4KMI8 24 310 595.0 3FR:313 Type1 Inactive DFGin 5.9088 14.9414 BLAminus -134.29, -167.77 57.39, 80.83 -100.95, 31.61 290.61, 85.71 -63.54, -20.94 out-out out 10.0443 Saltbr-out 4.2986 HRD-in -65.46, -53.96 81.32, -10.52 out-in-none SNCoin in-none ActLoopNT-in 2.8671 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.05 0.252 0.276 A 317.0 261.0 26 28 8 20 [[39, 291]] 1.0 3dbd Danio rerio CAMK_PLK1_DANRE CAMK 1.1e-76 263.5 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DB6A Q4KMI8 24 310 595.0 FRS:1 Type1.5_Front Inactive DFGin 5.8169 15.9541 BLAminus -142.4, -169.51 60.61, 84.89 -102.5, 26.5 287.92, 83.73 -63.45, -15.75 out-out out 11.6427 Saltbr-out 7.2053 HRD-in -75.01, -40.51 67.41, -16.08 out-in-out SNCoio in-out ActLoopNT-in 3.0249 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -91.76, 87.23 APE9-dihe-na 133.88, 161.1 APE8-dihe-in -107.95, 116.2 APE8-rot-in 306.39 APE67-dihe-out -75.67, -58.88 -71.76, 164.15 APE12-dist-in 11.272 APE11-dist-out 7.4839 APE10-dist-in 7.5109 APE9-dist-out 8.7756 T196D None None XRAY 2.85 0.225 0.257 A 301.0 287.0 0 28 28 0 [[39, 291]] 1.0 3db6 Danio rerio CAMK_PLK1_DANRE CAMK 8.9e-77 263.8 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q6DRK7_DANRE 3D5VA Q6DRK7 25 312 595.0 No_ligand No_ligand None DFGin 5.892 14.8682 BLAminus -136.77, -170.94 58.3, 78.56 -96.91, 24.94 292.69, 93.45 -65.35, -19.51 out-in out 10.4049 Saltbr-in 3.4081 HRD-in -70.1, -47.78 72.09, -9.5 in-in-none SNCiin in-none ActLoopNT-in 2.8844 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 2.4 0.237 0.269 A 317.0 260.0 28 28 9 19 [[39, 291]] 1.0 3d5v Danio rerio CAMK_PLK1_DANRE CAMK 1.1e-76 263.5 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 PLK1_HUMAN AF-P53350-K1A P53350 45 313 603.0 No_ligand No_ligand Active DFGin 5.5497 14.0178 BLAminus -138.81, -176.13 59.79, 75.65 -83.94, 15.34 292.62, 90.11 -62.81, -20.58 in-in in 9.0389 Saltbr-in 2.5765 HRD-in -77.19, -43.8 61.96, 8.95 in-in-in SNCiii in-in ActLoopNT-in 2.8977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.58, 167.37 APE9-dihe-na 111.84, 169.16 APE8-dihe-in -85.0, 135.3 APE8-rot-in 298.31 APE67-dihe-in -79.3, -5.41 -49.93, -42.14 APE12-dist-in 8.6475 APE11-dist-in 11.4873 APE10-dist-in 5.7926 APE9-dist-in 3.5019 None None None AF2 -1.0 1.0 1.0 A 269.0 269.0 0 28 28 0 [[53, 305]] 1.0 AF-P53350-K1 Homo sapiens CAMK_PLK1_HUMAN CAMK 1.5e-79 272.9 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN AF-P53350-K3A P53350 45 313 603.0 No_ligand No_ligand Active DFGin 5.3419 13.9791 BLAminus -140.81, -172.37 56.25, 72.33 -75.86, 12.77 292.93, 94.61 -62.92, -13.77 in-in in 9.3285 Saltbr-in 2.5773 HRD-in -78.81, -41.77 63.16, 8.34 in-in-in SNCiii in-in ActLoopNT-in 2.9297 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.05, 166.42 APE9-dihe-na 111.25, 170.64 APE8-dihe-in -84.99, 137.05 APE8-rot-in 295.25 APE67-dihe-in -75.5, -4.86 -51.24, -44.46 APE12-dist-in 8.6323 APE11-dist-in 11.5523 APE10-dist-in 5.8724 APE9-dist-in 3.3228 None None None AF2 -1.0 1.0 1.0 A 269.0 269.0 0 28 28 0 [[53, 305]] 1.0 AF-P53350-K3 Homo sapiens CAMK_PLK1_HUMAN CAMK 1.5e-79 272.9 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 8X72A P53350 37 330 603.0 ANP:401 ATPlike Inactive DFGin 5.6741 14.5619 BLAminus -124.66, -175.79 56.01, 84.34 -93.5, 28.11 290.48, 83.55 -67.08, -22.62 out-in out 10.0362 Saltbr-in 3.3691 HRD-in -69.02, -52.36 73.21, 2.03 in-in-out SNCiio in-out ActLoopNT-in 2.9948 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -79.36, 95.87 APE9-dihe-na 140.51, 168.33 APE8-dihe-in -120.38, 96.0 APE8-rot-in 313.63 APE67-dihe-out -71.46, -55.88 -64.61, 149.56 APE12-dist-in 10.8497 APE11-dist-out 7.4546 APE10-dist-in 7.6527 APE9-dist-out 8.0434 None None None XRAY 2.2 0.198 0.25 A 333.0 294.0 0 28 28 0 [[53, 305]] 1.0 8x72 Homo sapiens CAMK_PLK1_HUMAN CAMK 1.7e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 2OU7A P53350 37 328 603.0 ANP:500 ATPlike Inactive DFGin 5.511 14.6261 BLAminus -126.46, 177.9 64.03, 83.89 -94.43, 31.27 293.9, 81.92 -69.65, -29.63 out-in out 10.0179 Saltbr-in 3.5992 HRD-in -73.43, -50.53 79.22, -6.25 in-in-out SNCiio in-out ActLoopNT-in 2.9589 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.17, 94.2 APE9-dihe-na 146.34, 174.25 APE8-dihe-in -131.14, 97.57 APE8-rot-in 299.54 APE67-dihe-out -68.04, -58.6 -56.03, 146.92 APE12-dist-in 10.3811 APE11-dist-out 7.1861 APE10-dist-in 7.4365 APE9-dist-out 8.2407 T210V None None XRAY 2.4 0.205 0.235 A 335.0 292.0 0 28 28 0 [[53, 305]] 1.0 2ou7 Homo sapiens CAMK_PLK1_HUMAN CAMK 1.8e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 2V5QA P53350 39 323 603.0 No_ligand No_ligand Inactive DFGin 5.6857 14.7178 BLAminus -129.1, -167.08 62.93, 75.17 -93.89, 21.76 291.51, 90.84 -61.9, -28.72 out-in out 10.0226 Saltbr-in 3.0555 HRD-in -67.98, -52.02 73.91, 7.34 in-in-out SNCiio in-out ActLoopNT-in 2.8292 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -88.56, 3.75 APE9-dihe-na -179.48, -164.77 APE8-dihe-in -107.94, 115.2 APE8-rot-in 298.84 APE67-dihe-out -71.25, -55.87 -61.61, 160.98 APE12-dist-in 10.4375 APE11-dist-out 6.2368 APE10-dist-in 5.1223 APE9-dist-out 8.3334 None None None XRAY 2.3 0.184 0.224 A 315.0 285.0 0 28 28 0 [[53, 305]] 1.0 2v5q Homo sapiens CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 2V5QB P53350 39 323 603.0 No_ligand No_ligand Inactive DFGin 5.6851 14.9246 BLAminus -131.35, -166.96 60.96, 77.54 -92.83, 32.21 286.27, 87.97 -68.24, -26.27 in-out in 9.9987 Saltbr-out 3.8415 HRD-in -74.56, -53.71 79.97, 1.03 out-in-out SNCoio in-out ActLoopNT-in 2.8674 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -91.44, 9.2 APE9-dihe-na -170.42, 178.21 APE8-dihe-in -101.74, 116.95 APE8-rot-in 316.2 APE67-dihe-out -61.71, -54.24 -52.66, 144.9 APE12-dist-in 9.9909 APE11-dist-out 6.7742 APE10-dist-in 6.4067 APE9-dist-out 8.4067 None None None XRAY 2.3 0.184 0.224 B 315.0 285.0 0 28 28 0 [[53, 305]] 1.0 2v5q Homo sapiens CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 2YACA P53350 39 329 603.0 937:501 Type1 Inactive DFGin 5.7158 14.3054 BLAminus -136.25, -176.52 54.6, 87.71 -92.92, 28.24 289.9, 84.23 -75.6, -9.88 in-in in 9.4138 Saltbr-in 2.8323 HRD-in -79.87, -54.28 83.91, -4.3 in-in-out SNCiio in-out ActLoopNT-in 2.9371 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -90.18, 95.11 APE9-dihe-na 155.4, 174.07 APE8-dihe-in -130.99, 84.18 APE8-rot-out 67.16 APE67-dihe-out -74.05, -70.88 -62.65, 161.23 APE12-dist-in 11.0681 APE11-dist-out 7.3206 APE10-dist-in 7.6251 APE9-dist-out 8.1362 None None None XRAY 2.2 0.213 0.255 A 311.0 291.0 0 28 28 0 [[53, 305]] 1.0 2yac Homo sapiens CAMK_PLK1_HUMAN CAMK 2.5e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 3KB7A P53350 39 328 603.0 071:1 Type1 Inactive DFGin 5.7088 14.0424 BLAminus -133.88, 179.17 62.15, 88.77 -94.79, 24.7 288.92, 88.27 -73.01, -6.62 in-in in 8.8871 Saltbr-in 2.6738 HRD-in -67.89, -55.24 69.06, -3.76 in-in-out SNCiio in-out ActLoopNT-in 2.9089 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_iooo APE10-dihe-na -99.22, 86.88 APE9-dihe-na 165.83, 172.24 APE8-dihe-in -120.96, 91.28 APE8-rot-out 68.09 APE67-dihe-out -76.36, -59.91 -62.3, 158.23 APE12-dist-in 11.1305 APE11-dist-out 7.3774 APE10-dist-out 8.0773 APE9-dist-out 8.1697 None None NMM324 XRAY 2.5 0.212 0.303 A 311.0 290.0 0 28 28 0 [[53, 305]] 1.0 3kb7 Homo sapiens CAMK_PLK1_HUMAN CAMK 2.5e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 4A4LA P53350 39 329 603.0 939:1331 Type1 Inactive DFGin 5.7799 14.1347 BLAminus -141.7, -176.08 58.67, 82.87 -91.4, 34.14 289.94, 83.08 -71.42, -15.93 in-in in 9.4203 Saltbr-in 2.9397 HRD-in -74.58, -53.49 81.34, -4.51 in-in-out SNCiio in-out ActLoopNT-in 2.9169 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -83.54, 86.55 APE9-dihe-na 154.14, -178.12 APE8-dihe-in -129.31, 90.58 APE8-rot-out 60.31 APE67-dihe-out -60.53, -82.61 -62.07, 154.01 APE12-dist-in 11.0591 APE11-dist-out 7.3243 APE10-dist-in 7.6164 APE9-dist-out 8.4265 None None None XRAY 2.35 0.224 0.274 A 311.0 291.0 0 28 28 0 [[53, 305]] 1.0 4a4l Homo sapiens CAMK_PLK1_HUMAN CAMK 2.5e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 4A4OA P53350 39 329 603.0 664:1332 Type1 Inactive DFGin 5.6431 14.005 BLAminus -140.91, 173.61 55.04, 90.94 -98.45, 26.61 287.86, 85.19 -77.07, -1.22 in-in in 9.3392 Saltbr-in 3.3484 HRD-in -69.08, -52.1 82.91, 0.02 in-in-out SNCiio in-out ActLoopNT-in 3.0053 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -84.2, 81.23 APE9-dihe-na 164.33, -176.93 APE8-dihe-in -120.87, 80.43 APE8-rot-in 310.59 APE67-dihe-out -59.02, -78.88 -57.5, 148.27 APE12-dist-in 11.1607 APE11-dist-out 7.22 APE10-dist-in 7.7616 APE9-dist-out 8.2051 None None None XRAY 2.7 0.23 0.282 A 311.0 291.0 0 28 28 0 [[53, 305]] 1.0 4a4o Homo sapiens CAMK_PLK1_HUMAN CAMK 2.5e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R8BA P53350 37 326 603.0 A1JCP:1001 Type1 Inactive DFGin 5.7645 14.4195 BLAminus -135.37, -173.77 58.86, 75.37 -91.12, 20.8 284.65, 94.62 -63.52, -25.59 in-in in 8.4904 Saltbr-in 2.7158 HRD-in -71.84, -53.97 76.03, -0.52 in-in-out SNCiio in-out ActLoopNT-in 3.0153 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -85.35, 5.7 APE9-dihe-na -171.65, -172.53 APE8-dihe-in -108.35, 119.77 APE8-rot-in 298.21 APE67-dihe-out -65.23, -55.38 -66.82, 157.06 APE12-dist-in 10.6191 APE11-dist-out 6.9373 APE10-dist-in 5.948 APE9-dist-out 8.3177 None None None XRAY 2.2 0.191 0.238 A 315.0 290.0 0 28 28 0 [[53, 305]] 1.0 9r8b Homo sapiens CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R8BB P53350 37 323 603.0 A1JCP:402 Type1 Inactive DFGin 5.8352 14.2917 BLAminus -131.75, -174.5 64.87, 76.68 -96.77, 19.5 288.39, 99.04 -77.27, -4.94 in-in in 8.1199 Saltbr-in 2.7542 HRD-out -68.92, 136.67 -118.63, -11.46 in-in-out SNCiio in-out ActLoopNT-in 3.0307 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiio APE10-dihe-na 86.04, 0.68 APE9-dihe-na 169.71, -156.66 APE8-dihe-in -118.48, 123.54 APE8-rot-in 319.34 APE67-dihe-out -62.56, -51.97 -66.18, 154.73 APE12-dist-in 10.4716 APE11-dist-in 8.1897 APE10-dist-in 5.7403 APE9-dist-out 9.562 None None None XRAY 2.2 0.191 0.238 B 315.0 287.0 0 28 28 0 [[53, 305]] 1.0 9r8b Homo sapiens CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R8CA P53350 38 326 603.0 R78:1001 Type1 Inactive DFGin 5.5848 14.99 BLAminus -126.1, -176.63 65.4, 78.62 -95.8, 30.2 285.88, 88.19 -70.16, -23.86 in-in in 9.0969 Saltbr-in 2.8706 HRD-in -73.52, -53.38 78.38, -0.66 in-in-out SNCiio in-out ActLoopNT-in 2.9616 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.03, 32.02 APE9-dihe-na 163.26, -177.26 APE8-dihe-in -109.84, 116.09 APE8-rot-in 291.16 APE67-dihe-out -62.02, -59.2 -61.3, 153.09 APE12-dist-in 10.4112 APE11-dist-out 6.2561 APE10-dist-in 5.7623 APE9-dist-out 8.6225 None None None XRAY 2.243 0.191 0.236 A 315.0 289.0 0 28 28 0 [[53, 305]] 1.0 9r8c Homo sapiens CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R8CB P53350 38 323 603.0 R78:1001 Type1 Inactive DFGin 5.5457 14.9956 BLAminus -130.55, -176.06 59.62, 83.99 -94.79, 30.62 285.83, 86.69 -68.45, -26.03 in-in in 9.1508 Saltbr-in 2.7676 HRD-in -75.84, -53.52 77.99, 2.7 in-in-out SNCiio in-out ActLoopNT-in 2.9529 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -89.08, 50.7 APE9-dihe-na 152.38, 176.7 APE8-dihe-in -113.61, 115.98 APE8-rot-in 316.69 APE67-dihe-out -67.47, -56.35 -62.32, 152.06 APE12-dist-in 9.9595 APE11-dist-out 7.059 APE10-dist-in 6.6227 APE9-dist-out 8.5077 None None None XRAY 2.243 0.191 0.236 B 315.0 286.0 0 28 28 0 [[53, 305]] 1.0 9r8c Homo sapiens CAMK_PLK1_HUMAN CAMK 2.6e-79 272.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 4J52A P53350 38 330 603.0 1J3:400 Type1 Inactive DFGin 5.6732 14.405 BLAminus -132.19, -178.32 57.1, 88.41 -99.88, 23.54 290.9, 84.86 -66.29, -8.43 in-in in 9.3919 Saltbr-in 2.7014 HRD-in -83.32, -51.41 78.14, -8.7 in-in-out SNCiio in-out ActLoopNT-in 2.8667 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -92.24, 97.88 APE9-dihe-na 154.03, 172.56 APE8-dihe-in -123.15, 84.89 APE8-rot-in 302.52 APE67-dihe-out -69.1, -50.77 -69.03, 151.29 APE12-dist-in 10.9789 APE11-dist-out 7.3536 APE10-dist-in 7.8183 APE9-dist-out 7.821 T210V None None XRAY 2.3 0.198 0.241 A 293.0 293.0 0 28 28 0 [[53, 305]] 1.0 4j52 Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 4J53A P53350 38 330 603.0 1J4:403 Type1 Inactive DFGin 5.6397 14.5788 BLAminus -129.35, -169.37 44.41, 85.29 -91.22, 24.89 291.84, 82.06 -64.71, -23.25 in-in in 9.981 Saltbr-in 3.0097 HRD-in -75.81, -49.76 74.88, 0.23 in-in-out SNCiio in-out ActLoopNT-in 2.933 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -78.39, 101.76 APE9-dihe-na 146.02, 166.78 APE8-dihe-in -121.83, 82.96 APE8-rot-in 302.16 APE67-dihe-out -75.51, -62.04 -60.01, 151.77 APE12-dist-in 10.9528 APE11-dist-out 7.4006 APE10-dist-in 7.7633 APE9-dist-out 7.8563 T210V None None XRAY 2.5 0.183 0.24 A 293.0 293.0 0 28 28 0 [[53, 305]] 1.0 4j53 Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 2RKUA P53350 37 330 603.0 R78:500 Type1 Inactive DFGin 5.6778 15.0171 BLAminus -134.22, -169.5 54.06, 79.11 -86.67, 25.63 283.82, 88.21 -64.51, -26.07 in-in in 9.7168 Saltbr-in 3.0799 HRD-in -74.95, -48.26 75.93, -2.57 in-in-out SNCiio in-out ActLoopNT-in 2.9425 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -90.21, 90.69 APE9-dihe-na 162.46, 178.28 APE8-dihe-in -124.7, 88.6 APE8-rot-in 309.54 APE67-dihe-out -73.41, -64.04 -71.02, 160.05 APE12-dist-in 10.9294 APE11-dist-out 7.2828 APE10-dist-in 7.9206 APE9-dist-out 8.1342 T210V None None XRAY 1.95 0.192 0.241 A 294.0 294.0 0 28 28 0 [[53, 305]] 1.0 2rku Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 8BJTA P53350 39 330 603.0 8X7:402 Type1 Inactive DFGin 5.7433 14.3115 BLAminus -146.49, -170.45 55.69, 70.04 -90.08, 22.34 281.62, 90.95 -60.02, -37.94 in-in in 9.2218 Saltbr-in 2.728 HRD-in -68.54, -47.7 72.42, -10.0 in-in-out SNCiio in-out ActLoopNT-in 2.9242 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_iooo APE10-dihe-na -90.89, 99.31 APE9-dihe-na 143.06, 169.47 APE8-dihe-in -120.75, 101.21 APE8-rot-out 199.98 APE67-dihe-out -76.79, -55.69 -65.4, 158.12 APE12-dist-in 11.1597 APE11-dist-out 7.4033 APE10-dist-out 8.2363 APE9-dist-out 8.5627 None None None XRAY 2.188 0.203 0.255 A 294.0 292.0 0 28 28 0 [[53, 305]] 1.0 8bjt Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 3THBA P53350 42 328 603.0 3TA:1 Type1 Inactive DFGin 5.7628 14.2461 BLAminus -135.92, -170.43 55.15, 75.45 -87.11, 14.2 290.23, 88.06 -65.07, -8.71 in-in in 9.1247 Saltbr-in 3.5491 HRD-in -66.85, -49.24 73.84, -10.07 in-in-out SNCiio in-out ActLoopNT-in 2.9833 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -91.42, 101.79 APE9-dihe-na 126.02, 172.43 APE8-dihe-in -121.57, 103.22 APE8-rot-out 68.36 APE67-dihe-out -75.15, -60.09 -61.3, 157.38 APE12-dist-in 11.5794 APE11-dist-out 7.5519 APE10-dist-in 7.7464 APE9-dist-out 8.6498 T210V None None XRAY 2.5 0.253 0.286 A 333.0 287.0 0 28 28 0 [[53, 305]] 1.0 3thb Homo sapiens CAMK_PLK1_HUMAN CAMK 1.7e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 2OWBA P53350 37 330 603.0 626:500 Type1 Inactive DFGin 5.7411 14.2734 BLAminus -131.62, -172.7 55.05, 82.45 -94.97, 27.99 289.46, 84.52 -70.38, -17.86 in-in in 9.5051 Saltbr-in 2.6351 HRD-in -72.25, -49.78 72.96, -0.12 in-in-out SNCiio in-out ActLoopNT-in 3.0056 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -85.58, 102.01 APE9-dihe-na 139.92, 169.2 APE8-dihe-in -127.98, 85.88 APE8-rot-in 302.45 APE67-dihe-out -70.16, -61.75 -57.83, 150.59 APE12-dist-in 10.9432 APE11-dist-out 7.4221 APE10-dist-in 7.6185 APE9-dist-out 7.9791 T210V None None XRAY 2.1 0.205 0.243 A 335.0 294.0 0 28 28 0 [[53, 305]] 1.0 2owb Homo sapiens CAMK_PLK1_HUMAN CAMK 1.8e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 3FC2A P53350 37 329 603.0 IBI:10 Type1 Inactive DFGin 5.6869 14.8439 BLAminus -136.2, -169.15 47.8, 83.29 -92.73, 30.51 290.96, 88.11 -72.2, -20.77 in-in in 9.8452 Saltbr-in 2.7866 HRD-in -72.68, -50.74 75.03, 6.56 in-in-out SNCiio in-out ActLoopNT-in 2.9723 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -91.8, 110.95 APE9-dihe-na 128.06, 168.28 APE8-dihe-in -129.49, 88.48 APE8-rot-in 292.3 APE67-dihe-out -76.49, -62.11 -61.16, 163.08 APE12-dist-in 11.0036 APE11-dist-out 7.3642 APE10-dist-in 7.5319 APE9-dist-out 7.8848 T210V None None XRAY 2.45 0.184 0.226 A 335.0 293.0 0 28 28 0 [[53, 305]] 1.0 3fc2 Homo sapiens CAMK_PLK1_HUMAN CAMK 1.8e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9D0PA P53350 37 330 603.0 8X7:401 Type1 Inactive DFGin 5.9321 14.4667 BLAminus -127.97, -167.66 73.35, 57.17 -81.61, 36.59 285.64, 88.68 -94.22, -12.32 in-in in 9.0933 Saltbr-in 2.7584 HRD-in -81.82, -53.71 82.64, -7.07 in-in-out SNCiio in-out ActLoopNT-in 2.9118 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -92.87, 112.89 APE9-dihe-na 127.84, 173.17 APE8-dihe-in -124.26, 98.89 APE8-rot-in 301.22 APE67-dihe-out -72.74, -55.92 -71.3, 155.26 APE12-dist-in 11.2956 APE11-dist-out 7.351 APE10-dist-in 7.4828 APE9-dist-out 8.252 T210V None None XRAY 2.65 0.247 0.29 A 335.0 294.0 0 28 28 0 [[53, 305]] 1.0 9d0p Homo sapiens CAMK_PLK1_HUMAN CAMK 1.8e-78 269.4 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R1WAAA P53350 38 334 603.0 A1JCP:401 Type1 Inactive DFGin 5.6292 14.3068 BLAminus -134.11, -168.09 56.45, 78.1 -90.07, 23.96 287.47, 94.05 -61.0, -27.64 in-in in 9.0559 Saltbr-in 2.8172 HRD-in -73.41, -49.99 71.11, 3.55 in-in-out SNCiio in-out ActLoopNT-in 2.9617 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -89.16, 9.34 APE9-dihe-na -169.47, 176.32 APE8-dihe-in -98.59, 112.0 APE8-rot-in 302.37 APE67-dihe-out -62.18, -51.19 -58.71, 150.32 APE12-dist-in 10.1834 APE11-dist-out 6.5586 APE10-dist-in 6.2363 APE9-dist-out 8.5025 K225D,K226A None None XRAY 2.2 0.18 0.216 AAA 325.0 297.0 0 28 28 0 [[53, 305]] 1.0 9r1w Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R1WBBB P53350 38 325 603.0 A1JCP:401 Type1 Inactive DFGin 5.6297 14.3508 BLAminus -133.86, -166.71 56.12, 78.59 -90.53, 23.21 288.19, 92.88 -61.02, -27.23 in-in in 9.2288 Saltbr-in 2.7447 HRD-in -73.38, -50.78 71.42, 4.57 in-in-out SNCiio in-out ActLoopNT-in 2.9696 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -89.57, 8.7 APE9-dihe-na -168.16, 173.41 APE8-dihe-in -98.08, 111.85 APE8-rot-in 305.79 APE67-dihe-out -62.5, -50.96 -59.11, 151.11 APE12-dist-in 10.0722 APE11-dist-out 6.5984 APE10-dist-in 6.1802 APE9-dist-out 8.4386 K225D,K226A None None XRAY 2.2 0.18 0.216 BBB 325.0 288.0 0 28 28 0 [[53, 305]] 1.0 9r1w Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R1XA P53350 39 334 603.0 R78:401 Type1 Inactive DFGin 5.4509 14.7459 BLAminus -129.34, -169.27 61.33, 81.84 -99.46, 30.78 291.65, 94.79 -60.61, -43.02 in-in in 9.6846 Saltbr-in 2.7211 HRD-in -71.39, -48.31 73.02, 3.83 in-in-out SNCiio in-out ActLoopNT-in 2.9715 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -86.63, 46.88 APE9-dihe-na 161.22, 163.69 APE8-dihe-in -103.28, 108.1 APE8-rot-in 301.35 APE67-dihe-out -58.97, -56.16 -54.1, 148.74 APE12-dist-in 10.3877 APE11-dist-out 6.5599 APE10-dist-in 6.7414 APE9-dist-out 8.5087 K225D,K226A None None XRAY 2.84 0.222 0.277 A 325.0 296.0 0 28 28 0 [[53, 305]] 1.0 9r1x Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R1XB P53350 39 326 603.0 R78:401 Type1 Inactive DFGin 5.4448 14.7258 BLAminus -129.89, -169.09 62.76, 81.42 -99.44, 28.81 292.45, 94.66 -58.03, -43.63 in-in in 9.6661 Saltbr-in 2.714 HRD-in -71.6, -47.96 72.32, 5.61 in-in-out SNCiio in-out ActLoopNT-in 2.9664 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -82.43, 34.44 APE9-dihe-na 160.48, 165.73 APE8-dihe-in -102.91, 108.17 APE8-rot-in 301.26 APE67-dihe-out -58.46, -55.69 -54.97, 148.64 APE12-dist-in 10.4044 APE11-dist-out 6.5324 APE10-dist-in 5.999 APE9-dist-out 8.4468 K225D,K226A None None XRAY 2.84 0.222 0.277 B 325.0 288.0 0 28 28 0 [[53, 305]] 1.0 9r1x Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R1YAAA P53350 38 334 603.0 A1JCQ:401 Type1 Inactive DFGin 5.4927 14.2673 BLAminus -126.75, -172.44 65.19, 77.92 -95.78, 35.59 294.04, 83.7 -66.64, -28.98 in-in in 9.4644 Saltbr-in 2.7444 HRD-in -71.96, -50.24 71.88, 5.14 in-in-out SNCiio in-out ActLoopNT-in 3.1029 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -88.57, 8.2 APE9-dihe-na -166.23, -178.27 APE8-dihe-in -105.79, 106.71 APE8-rot-in 300.95 APE67-dihe-out -66.32, -52.43 -54.05, 151.38 APE12-dist-in 10.2803 APE11-dist-out 6.4939 APE10-dist-in 6.1368 APE9-dist-out 8.3805 K225D,K226A None None XRAY 2.602 0.187 0.218 AAA 325.0 297.0 0 28 28 0 [[53, 305]] 1.0 9r1y Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 9R1YBBB P53350 38 325 603.0 A1JCQ:401 Type1 Inactive DFGin 5.5166 14.3492 BLAminus -126.84, -171.95 66.19, 77.61 -96.17, 35.42 294.69, 83.98 -66.59, -29.54 in-in in 9.5027 Saltbr-in 2.7444 HRD-in -72.69, -50.41 71.98, 5.19 in-in-out SNCiio in-out ActLoopNT-in 3.1096 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -88.39, 7.64 APE9-dihe-na -166.1, -178.49 APE8-dihe-in -105.58, 106.71 APE8-rot-in 302.14 APE67-dihe-out -65.99, -51.73 -54.43, 151.5 APE12-dist-in 10.3012 APE11-dist-out 6.4798 APE10-dist-in 5.9907 APE9-dist-out 8.3631 K225D,K226A None None XRAY 2.602 0.187 0.218 BBB 325.0 288.0 0 28 28 0 [[53, 305]] 1.0 9r1y Homo sapiens CAMK_PLK1_HUMAN CAMK 1.1e-78 270.0 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 5TA6A P53350 37 330 603.0 79D:1000 Type1 Inactive DFGin 5.7677 14.6912 BLAminus -129.81, 178.93 63.79, 86.6 -95.82, 28.6 292.13, 79.82 -68.79, -23.38 in-in in 9.776 Saltbr-in 3.0598 HRD-in -68.63, -52.95 71.96, 8.35 in-in-out SNCiio in-out ActLoopNT-in 2.8889 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -85.92, 111.12 APE9-dihe-na 138.09, 164.23 APE8-dihe-in -126.56, 95.9 APE8-rot-out 85.27 APE67-dihe-out -71.06, -59.19 -57.19, 156.45 APE12-dist-in 10.9082 APE11-dist-out 7.3284 APE10-dist-in 7.6939 APE9-dist-out 7.5992 None None None XRAY 2.5 0.183 0.26 A 358.0 294.0 0 28 28 0 [[53, 305]] 1.0 5ta6 Homo sapiens CAMK_PLK1_HUMAN CAMK 2.2e-78 269.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1
PLK1 PLK1_HUMAN 5TA8A P53350 37 330 603.0 79C:402 Type1 Inactive DFGin 5.5977 14.3108 BLAminus -141.08, -172.7 51.52, 90.37 -96.67, 41.3 290.69, 89.43 -72.33, -19.61 in-in in 9.1072 Saltbr-in 2.7273 HRD-in -66.37, -49.24 72.53, -11.97 in-in-out SNCiio in-out ActLoopNT-in 2.8816 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_ioio APE10-dihe-na -88.19, 81.36 APE9-dihe-na 134.61, 175.47 APE8-dihe-in -125.29, 109.1 APE8-rot-out 49.04 APE67-dihe-out -73.09, -62.08 -71.65, 169.34 APE12-dist-in 10.8099 APE11-dist-out 7.4727 APE10-dist-in 7.1878 APE9-dist-out 8.6926 None None None XRAY 2.6 0.185 0.247 A 358.0 294.0 0 28 28 0 [[53, 305]] 1.0 5ta8 Homo sapiens CAMK_PLK1_HUMAN CAMK 2.2e-78 269.1 1.0 256.0 256.0 193 194 195 197 199 82 101 105 173 175 174 176.0 233 221 216 215 214 213 212 211 210 131 Serine/threonine-protein kinase PLK1

CAMK_PLK1 (Serine/threonine-protein kinase PLK1)

Total number of chains: 12
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 11 91.7% 3D5UA
DFGin ABAminus 1 8.3% 4J7BD

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PLK1 Q6DRK7_DANRE 4J7BD Q6DRK7 20 311 595.0 No_ligand No_ligand Inactive DFGin 5.4866 14.5549 ABAminus -129.81, -7.43 -133.83, 113.48 -107.04, 20.33 291.52, 92.27 -51.62, -38.38 out-in out 10.214 Saltbr-in 2.9657 HRD-in -68.9, -50.24 76.71, 4.14 in-in-out SNCiio in-out ActLoopNT-in 2.7455 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -126.82 APE8-dihe-in -131.87, 100.17 APE8-rot-in 301.55 APE67-dihe-out -78.82, -54.23 -64.35, 166.22 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 7.9466 D162N,E192F None None XRAY 2.3 0.208 0.264 D 297.0 281.0 11 28 17 11 [[39, 291]] 1.0 4j7b Danio rerio CAMK_PLK1_DANRE CAMK 8.1e-76 260.6 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3D5WA Q4KMI8 24 310 595.0 ADP:313 ATPlike Inactive DFGin 5.8398 15.103 BLAminus -136.31, -173.3 52.58, 90.43 -100.9, 29.72 290.61, 88.81 -67.31, -18.54 out-out out 10.538 Saltbr-out 4.5698 HRD-in -72.81, -47.33 67.56, -5.93 out-in-in SNCoii in-in ActLoopNT-in 2.9013 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.0, 153.74 APE9-dihe-na 145.11, -167.91 APE8-dihe-in -110.25, 127.19 APE8-rot-in 299.86 APE67-dihe-in -70.02, -15.96 -37.98, -47.89 APE12-dist-in 8.2509 APE11-dist-in 11.2747 APE10-dist-in 5.6458 APE9-dist-in 3.9124 None TPO196 TPO196 XRAY 2.6 0.244 0.271 A 317.0 285.0 2 28 28 0 [[39, 291]] 1.0 3d5w Danio rerio CAMK_PLK1_DANRE CAMK 4.6e-77 264.7 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q6DRK7_DANRE 3D5UA Q6DRK7 23 310 595.0 No_ligand No_ligand Inactive DFGin 5.6927 14.8088 BLAminus -132.0, -170.66 53.21, 91.71 -105.63, 34.97 291.53, 90.32 -70.7, -17.69 out-out out 10.6997 Saltbr-out 4.3498 HRD-in -73.43, -47.86 66.94, -9.91 out-in-out SNCoio in-out ActLoopNT-in 2.8874 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -83.53, 77.69 APE9-dihe-na 160.43, 176.55 APE8-dihe-in -120.81, 90.57 APE8-rot-in 316.96 APE67-dihe-out -68.11, -72.46 -73.03, 158.49 APE12-dist-in 10.6665 APE11-dist-out 7.4011 APE10-dist-in 7.5221 APE9-dist-out 8.4661 None None None XRAY 2.8 0.231 0.281 A 317.0 288.0 0 28 28 0 [[39, 291]] 1.0 3d5u Danio rerio CAMK_PLK1_DANRE CAMK 4.6e-77 264.7 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q6DRK7_DANRE 4J7BA Q6DRK7 18 311 595.0 No_ligand No_ligand Inactive DFGin 5.9575 14.8219 BLAminus -127.79, -166.66 63.28, 73.86 -94.07, 24.02 287.22, 93.09 -58.39, -32.32 in-in in 9.948 Saltbr-in 2.5261 HRD-in -69.09, -53.7 77.98, -8.47 in-in-out SNCiio in-out ActLoopNT-in 2.8139 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_nnio APE10-dihe-na 999.0, 170.84 APE9-dihe-na -82.59, -164.35 APE8-dihe-in -106.73, 113.42 APE8-rot-out 172.88 APE67-dihe-out -56.23, -64.85 -68.6, 152.66 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 5.9329 APE9-dist-out 8.4727 D162N,E192F None None XRAY 2.3 0.208 0.264 A 297.0 284.0 10 28 18 10 [[39, 291]] 1.0 4j7b Danio rerio CAMK_PLK1_DANRE CAMK 8.1e-76 260.6 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3D5XA Q4KMI8 24 309 595.0 KWT:1 Type1 Inactive DFGin 5.7483 14.936 BLAminus -139.39, -170.01 59.65, 84.09 -100.6, 25.02 290.64, 93.65 -64.4, -14.86 out-out out 10.666 Saltbr-out 4.3942 HRD-in -69.94, -48.19 73.11, -11.18 out-in-none SNCoin in-none ActLoopNT-in 3.0678 ActLoopCT-none nonTYR APEdihe_aannn APEdist_innn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-in 10.2963 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 2.8 0.263 0.299 A 301.0 279.0 7 28 21 7 [[39, 291]] 1.0 3d5x Danio rerio CAMK_PLK1_DANRE CAMK 8.9e-77 263.8 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DBEA Q4KMI8 24 310 595.0 4FR:1 Type1 Inactive DFGin 5.3305 14.2611 BLAminus -130.08, -172.43 53.96, 104.63 -115.22, 13.87 295.84, 91.17 -49.61, -15.58 out-out out 10.0731 Saltbr-out 4.3667 HRD-in -75.7, -52.21 77.46, -22.23 out-in-out SNCoio in-out ActLoopNT-in 2.9691 ActLoopCT-out nonTYR APEdihe_aannn APEdist_ionn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -89.97, -74.84 999.0, 157.6 APE12-dist-in 10.4051 APE11-dist-out 7.7345 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.32 0.237 0.27 A 301.0 284.0 3 28 25 3 [[39, 291]] 1.0 3dbe Danio rerio CAMK_PLK1_DANRE CAMK 8.9e-77 263.8 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DBFA Q4KMI8 24 310 595.0 5FR:1 Type1 Inactive DFGin 5.5692 14.5066 BLAminus -126.48, -167.26 59.45, 92.34 -110.0, 25.26 297.55, 90.95 -54.7, -27.45 in-out in 9.8779 Saltbr-out 4.027 HRD-in -77.45, -40.3 68.16, -16.48 out-in-none SNCoin in-none ActLoopNT-in 2.9286 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.2 0.234 0.275 A 301.0 261.0 26 28 8 20 [[39, 291]] 1.0 3dbf Danio rerio CAMK_PLK1_DANRE CAMK 8.9e-77 263.8 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DB8A Q4KMI8 24 310 595.0 1FR:313 Type1 Inactive DFGin 5.7592 14.6569 BLAminus -132.17, -175.89 60.33, 81.89 -97.25, 28.2 286.75, 81.14 -57.5, -31.84 in-out in 9.9095 Saltbr-out 3.8295 HRD-in -71.72, -45.68 69.14, -18.96 out-in-none SNCoin in-none ActLoopNT-in 2.8276 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.15 0.232 0.274 A 317.0 261.0 26 28 8 20 [[39, 291]] 1.0 3db8 Danio rerio CAMK_PLK1_DANRE CAMK 1.1e-76 263.5 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DBCA Q4KMI8 24 310 595.0 2FR:313 Type1 Inactive DFGin 5.7335 14.6643 BLAminus -136.39, -168.79 53.28, 74.51 -89.66, 27.23 289.49, 88.8 -63.71, -13.19 in-out in 9.6385 Saltbr-out 4.0559 HRD-in -85.71, -43.45 67.47, -24.22 out-in-none SNCoin in-none ActLoopNT-in 3.0181 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.35 0.245 0.288 A 317.0 261.0 26 28 8 20 [[39, 291]] 1.0 3dbc Danio rerio CAMK_PLK1_DANRE CAMK 1.1e-76 263.5 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DBDA Q4KMI8 24 310 595.0 3FR:313 Type1 Inactive DFGin 5.9088 14.9414 BLAminus -134.29, -167.77 57.39, 80.83 -100.95, 31.61 290.61, 85.71 -63.54, -20.94 out-out out 10.0443 Saltbr-out 4.2986 HRD-in -65.46, -53.96 81.32, -10.52 out-in-none SNCoin in-none ActLoopNT-in 2.8671 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 3.05 0.252 0.276 A 317.0 261.0 26 28 8 20 [[39, 291]] 1.0 3dbd Danio rerio CAMK_PLK1_DANRE CAMK 1.1e-76 263.5 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q4KMI8_DANRE 3DB6A Q4KMI8 24 310 595.0 FRS:1 Type1.5_Front Inactive DFGin 5.8169 15.9541 BLAminus -142.4, -169.51 60.61, 84.89 -102.5, 26.5 287.92, 83.73 -63.45, -15.75 out-out out 11.6427 Saltbr-out 7.2053 HRD-in -75.01, -40.51 67.41, -16.08 out-in-out SNCoio in-out ActLoopNT-in 3.0249 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_ioio APE10-dihe-na -91.76, 87.23 APE9-dihe-na 133.88, 161.1 APE8-dihe-in -107.95, 116.2 APE8-rot-in 306.39 APE67-dihe-out -75.67, -58.88 -71.76, 164.15 APE12-dist-in 11.272 APE11-dist-out 7.4839 APE10-dist-in 7.5109 APE9-dist-out 8.7756 T196D None None XRAY 2.85 0.225 0.257 A 301.0 287.0 0 28 28 0 [[39, 291]] 1.0 3db6 Danio rerio CAMK_PLK1_DANRE CAMK 8.9e-77 263.8 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK
PLK1 Q6DRK7_DANRE 3D5VA Q6DRK7 25 312 595.0 No_ligand No_ligand None DFGin 5.892 14.8682 BLAminus -136.77, -170.94 58.3, 78.56 -96.91, 24.94 292.69, 93.45 -65.35, -19.51 out-in out 10.4049 Saltbr-in 3.4081 HRD-in -70.1, -47.78 72.09, -9.5 in-in-none SNCiin in-none ActLoopNT-in 2.8844 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 T196D None None XRAY 2.4 0.237 0.269 A 317.0 260.0 28 28 9 19 [[39, 291]] 1.0 3d5v Danio rerio CAMK_PLK1_DANRE CAMK 1.1e-76 263.5 1.0 256.0 256.0 179 180 181 183 185 68 87 91 159 161 160 162.0 219 207 202 201 200 199 198 197 196 117 Serine/threonine-protein kinase PLK