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| PDB | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 6C7YA | 869 | 1153 | 1154.0 | ADP:61201 | ATPlike | Active | DFGin | 6.032 | 13.967 | BLAminus | -134.15, -164.18 | 58.49, 84.96 | -109.28, 28.04 | 298.78, 97.45 | -66.39, -27.05 | in-in | in | 8.311 | Saltbr-in | 2.732 | HRD-in | -67.59, -46.53 | 68.25, 12.43 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -72.91, 151.36 | APE9-dihe-in | -137.76, 143.32 | APE8-dihe-in | -74.71, 81.76 | APE8-rot-na | 30.49 | APE67-dihe-in | -79.4, -2.38 | -65.2, -24.66 | APE12-dist-na | 12.972 | APE11-dist-na | 8.02 | APE10-dist-na | 10.344 | APE9-dist-in | 6.316 | None | PTR1035 | PTR1035 | XRAY | 2.499 | 0.21 | 0.241 | A | 286 | 273 | 12 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6c7y | TYR_JAK1-2_HUMAN | TYR | 1.8e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| AF-P23458-K2A | 867 | 1154 | 1154.0 | No_ligand | No_ligand | Active | DFGin | 6.307 | 13.773 | BLAminus | -130.0, -171.31 | 51.92, 79.2 | -91.39, 17.47 | 288.09, 81.21 | -63.19, -25.32 | in-in | in | 8.086 | Saltbr-in | 2.719 | HRD-in | -67.76, -41.14 | 64.22, -10.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.94 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -50.83, 123.48 | APE9-dihe-in | -125.8, 136.55 | APE8-dihe-in | -75.77, 67.19 | APE8-rot-na | 34.45 | APE67-dihe-in | -77.12, -11.68 | -54.83, -26.9 | APE12-dist-na | 13.91 | APE11-dist-na | 8.532 | APE10-dist-na | 10.659 | APE9-dist-in | 7.063 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 288 | 288 | 0 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | AF-P23458-K2 | TYR_JAK1-2_HUMAN | TYR | 1.8e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| AF-P23458-K4A | 867 | 1154 | 1154.0 | No_ligand | No_ligand | Active | DFGin | 6.034 | 13.552 | BLAminus | -127.94, -176.44 | 52.21, 91.21 | -99.55, 15.91 | 293.58, 76.0 | -63.9, -24.71 | in-in | in | 7.81 | Saltbr-in | 2.715 | HRD-in | -69.66, -43.24 | 62.91, -1.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.92 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -47.59, 114.14 | APE9-dihe-in | -120.02, 146.94 | APE8-dihe-in | -73.57, 63.93 | APE8-rot-na | 37.51 | APE67-dihe-in | -76.35, -14.96 | -54.26, -27.82 | APE12-dist-na | 13.697 | APE11-dist-na | 8.114 | APE10-dist-na | 10.916 | APE9-dist-in | 6.735 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 288 | 288 | 0 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | AF-P23458-K4 | TYR_JAK1-2_HUMAN | TYR | 1.8e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5KHWA | 867 | 1153 | 1154.0 | ADP:1201 | ATPlike | Inactive | DFGin | 6.293 | 13.595 | ABAminus | -113.62, -36.19 | -113.51, 112.49 | -104.48, 28.51 | 302.05, 98.46 | -68.45, -35.55 | in-in | in | 8.017 | Saltbr-in | 2.811 | HRD-in | -53.69, -54.55 | 74.32, 4.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.817 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.25, 151.86 | APE9-dihe-in | -139.19, 145.92 | APE8-dihe-in | -78.07, 75.73 | APE8-rot-na | 29.65 | APE67-dihe-in | -77.72, -3.4 | -55.44, -31.5 | APE12-dist-na | 13.014 | APE11-dist-na | 7.332 | APE10-dist-na | 9.905 | APE9-dist-in | 6.022 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.47 | 0.188 | 0.231 | A | 316 | 278 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5khw | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4E4LE | 864 | 1154 | 1154.0 | No_ligand | No_ligand | Inactive | DFGin | 6.463 | 13.613 | ABAminus | -114.05, 7.25 | -155.92, 142.83 | -135.92, 30.26 | 296.52, 85.61 | -59.94, -28.28 | in-in | in | 7.87 | Saltbr-in | 2.625 | HRD-in | -76.43, -49.33 | 70.91, 5.03 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.809 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.8, 27.83 | APE9-dihe-in | -58.48, 132.7 | APE8-dihe-in | -75.95, 78.2 | APE8-rot-na | 25.62 | APE67-dihe-in | -75.39, -5.67 | -60.62, -30.34 | APE12-dist-na | 11.404 | APE11-dist-na | 12.865 | APE10-dist-na | 10.335 | APE9-dist-in | 6.766 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.19 | 0.228 | E | 302 | 282 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4l | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 3EYGA | 865 | 1154 | 1154.0 | MI1:1 | Type1 | Inactive | DFGin | 6.484 | 13.585 | ABAminus | -124.32, 8.36 | -155.42, 148.92 | -141.71, 28.09 | 295.61, 92.98 | -69.61, -22.8 | in-in | in | 7.772 | Saltbr-in | 2.871 | HRD-in | -73.25, -48.81 | 76.52, 2.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.829 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -99.1, 4.52 | APE9-dihe-in | -69.5, 129.84 | APE8-dihe-in | -77.86, 81.49 | APE8-rot-na | 30.22 | APE67-dihe-in | -79.56, -5.41 | -59.51, -27.49 | APE12-dist-na | 10.755 | APE11-dist-na | 11.055 | APE10-dist-na | 6.707 | APE9-dist-in | 5.595 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.171 | 0.214 | A | 290 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 3eyg | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 3EYHA | 865 | 1154 | 1154.0 | IZA:2001 | Type1 | Inactive | DFGin | 6.711 | 13.778 | ABAminus | -123.79, 5.59 | -151.26, 147.61 | -137.78, 30.19 | 296.78, 89.6 | -63.64, -28.15 | in-in | in | 7.741 | Saltbr-in | 2.88 | HRD-in | -74.82, -42.99 | 68.23, 5.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.799 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -136.22, 60.46 | APE9-dihe-in | -76.43, 138.22 | APE8-dihe-in | -79.32, 79.81 | APE8-rot-na | 29.32 | APE67-dihe-in | -73.68, -7.92 | -57.92, -30.28 | APE12-dist-na | 10.347 | APE11-dist-na | 10.995 | APE10-dist-na | 9.051 | APE9-dist-in | 5.572 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.178 | 0.237 | A | 290 | 287 | 3 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 3eyh | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5E1EB | 865 | 1154 | 1154.0 | 5JG:1201 | Type1 | Inactive | DFGin | 6.615 | 13.703 | ABAminus | -133.31, 28.19 | -149.71, 114.81 | -114.53, 26.1 | 291.32, 84.42 | -63.72, -24.05 | in-in | in | 7.765 | Saltbr-in | 2.784 | HRD-in | -74.91, -42.75 | 64.28, 0.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.801 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.64, 38.4 | APE9-dihe-in | -74.25, 132.21 | APE8-dihe-in | -79.08, 75.2 | APE8-rot-na | 22.34 | APE67-dihe-in | -75.56, -2.49 | -52.66, -36.06 | APE12-dist-na | 10.857 | APE11-dist-na | 13.311 | APE10-dist-na | 10.039 | APE9-dist-in | 6.874 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.3 | 0.227 | 0.268 | B | 290 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5e1e | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6AAHA | 865 | 1154 | 1154.0 | 9T6:1201 | Type1 | Inactive | DFGin | 6.319 | 13.457 | ABAminus | -111.86, -1.07 | -147.59, 142.74 | -130.77, 31.7 | 296.21, 81.89 | -59.29, -31.87 | in-in | in | 7.837 | Saltbr-in | 2.785 | HRD-in | -79.04, -51.9 | 74.79, 8.24 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.804 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.78, 24.87 | APE9-dihe-in | -65.36, 146.43 | APE8-dihe-in | -84.69, 80.23 | APE8-rot-na | 32.65 | APE67-dihe-in | -73.6, -4.54 | -60.24, -33.63 | APE12-dist-na | 10.501 | APE11-dist-na | 13.066 | APE10-dist-na | 9.901 | APE9-dist-in | 6.422 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.83 | 0.225 | 0.255 | A | 290 | 285 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6aah | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6AAHB | 865 | 1154 | 1154.0 | 9T6:1201 | Type1 | Inactive | DFGin | 6.462 | 13.588 | ABAminus | -114.68, 9.66 | -151.81, 133.96 | -131.35, 23.59 | 291.95, 87.28 | -61.54, -23.21 | in-in | in | 8.041 | Saltbr-in | 2.614 | HRD-in | -74.7, -48.84 | 74.08, 5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.783 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -85.14, 67.65 | APE9-dihe-in | -109.05, 132.69 | APE8-dihe-in | -79.19, 76.3 | APE8-rot-na | 35.14 | APE67-dihe-in | -76.24, -3.1 | -57.7, -33.14 | APE12-dist-na | 10.191 | APE11-dist-na | 12.461 | APE10-dist-na | 9.141 | APE9-dist-in | 6.543 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.83 | 0.225 | 0.255 | B | 290 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6aah | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6TPEA | 864 | 1153 | 1154.0 | NTW:1201 | Type1 | Inactive | DFGin | 6.452 | 13.452 | ABAminus | -113.52, 27.97 | -159.85, 137.75 | -139.89, 37.69 | 300.95, 90.85 | -70.73, -32.53 | in-in | in | 7.984 | Saltbr-in | 2.898 | HRD-in | -77.39, -48.43 | 67.11, 20.0 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.721 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.39, 82.51 | APE9-dihe-in | -109.84, 138.7 | APE8-dihe-in | -71.54, 85.2 | APE8-rot-na | 346.93 | APE67-dihe-in | -79.64, -10.25 | -64.68, -30.27 | APE12-dist-na | 10.125 | APE11-dist-na | 12.13 | APE10-dist-na | 10.498 | APE9-dist-in | 6.452 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.87 | 0.249 | 0.298 | A | 291 | 283 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6tpe | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6TPEB | 864 | 1154 | 1154.0 | NTW:1201 | Type1 | Inactive | DFGin | 6.449 | 13.462 | ABAminus | -113.4, 27.83 | -159.97, 137.64 | -139.8, 37.79 | 300.87, 90.88 | -70.61, -32.51 | in-in | in | 7.994 | Saltbr-in | 2.893 | HRD-in | -77.28, -48.49 | 67.12, 19.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.723 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.48, 82.82 | APE9-dihe-in | -109.8, 138.58 | APE8-dihe-in | -71.3, 85.03 | APE8-rot-na | 346.96 | APE67-dihe-in | -79.6, -10.33 | -64.53, -30.29 | APE12-dist-na | 10.133 | APE11-dist-na | 12.13 | APE10-dist-na | 10.513 | APE9-dist-in | 6.453 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.87 | 0.249 | 0.298 | B | 291 | 283 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6tpe | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6TPFA | 864 | 1153 | 1154.0 | NTQ:1201 | Type1 | Inactive | DFGin | 6.549 | 13.566 | ABAminus | -112.13, 4.42 | -147.17, 134.74 | -132.51, 36.57 | 297.52, 87.9 | -61.56, -38.59 | in-in | in | 7.907 | Saltbr-in | 2.723 | HRD-in | -81.26, -43.5 | 66.58, 8.45 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.755 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.97, 47.61 | APE9-dihe-in | -75.75, 153.17 | APE8-dihe-in | -82.59, 85.83 | APE8-rot-na | 32.54 | APE67-dihe-in | -74.51, -8.6 | -66.85, -35.11 | APE12-dist-na | 10.951 | APE11-dist-na | 12.702 | APE10-dist-na | 10.945 | APE9-dist-in | 6.702 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.31 | 0.266 | 0.327 | A | 291 | 288 | 2 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6tpf | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6TPFB | 865 | 1153 | 1154.0 | NTQ:1201 | Type1 | Inactive | DFGin | 6.516 | 13.607 | ABAminus | -112.38, 6.69 | -146.72, 134.6 | -130.81, 35.94 | 297.58, 85.61 | -65.62, -37.25 | in-in | in | 7.843 | Saltbr-in | 2.72 | HRD-in | -83.36, -42.45 | 66.49, 9.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.762 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 46.13, 45.8 | APE9-dihe-in | -71.68, 152.43 | APE8-dihe-in | -82.66, 85.94 | APE8-rot-na | 32.5 | APE67-dihe-in | -74.85, -9.43 | -66.05, -35.76 | APE12-dist-na | 10.968 | APE11-dist-na | 12.342 | APE10-dist-na | 11.419 | APE9-dist-in | 6.666 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.31 | 0.266 | 0.327 | B | 291 | 278 | 11 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6tpf | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6GGHA | 865 | 1154 | 1154.0 | EYQ:1201 | Type1 | Inactive | DFGin | 6.474 | 13.708 | ABAminus | -120.02, -5.29 | -148.47, 136.5 | -125.28, 25.35 | 294.61, 85.16 | -56.12, -34.28 | in-in | in | 7.718 | Saltbr-in | 2.591 | HRD-in | -74.74, -47.68 | 65.51, 13.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.766 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 52.1, 57.9 | APE9-dihe-in | -80.13, 145.81 | APE8-dihe-in | -79.99, 78.75 | APE8-rot-na | 31.21 | APE67-dihe-in | -74.16, -4.73 | -59.55, -32.45 | APE12-dist-na | 10.105 | APE11-dist-na | 9.884 | APE10-dist-na | 9.981 | APE9-dist-in | 6.106 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.7 | 0.192 | 0.262 | A | 292 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6ggh | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6GGHB | 863 | 1154 | 1154.0 | EYQ:1201 | Type1 | Inactive | DFGin | 6.393 | 13.885 | ABAminus | -111.86, -4.02 | -150.16, 140.27 | -128.87, 25.84 | 291.88, 86.63 | -62.88, -36.22 | in-in | in | 7.795 | Saltbr-in | 2.592 | HRD-in | -72.53, -48.04 | 68.9, 11.02 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.789 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 72.16, 30.7 | APE9-dihe-in | -88.91, 131.65 | APE8-dihe-in | -78.72, 80.52 | APE8-rot-na | 31.53 | APE67-dihe-in | -73.31, -5.76 | -61.33, -30.45 | APE12-dist-na | 10.287 | APE11-dist-na | 10.652 | APE10-dist-na | 8.339 | APE9-dist-in | 5.994 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.7 | 0.192 | 0.262 | B | 292 | 282 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6ggh | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6ELRA | 854 | 1154 | 1154.0 | BFK:1201 | Type1 | Inactive | DFGin | 6.597 | 13.599 | ABAminus | -108.66, 4.92 | -152.97, 140.13 | -131.61, 26.62 | 294.97, 83.84 | -57.45, -30.06 | in-in | in | 7.779 | Saltbr-in | 2.741 | HRD-in | -71.99, -47.83 | 69.61, 1.99 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.831 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.35, 32.0 | APE9-dihe-in | -64.21, 131.29 | APE8-dihe-in | -79.64, 72.85 | APE8-rot-na | 28.8 | APE67-dihe-in | -76.69, -6.06 | -50.77, -33.65 | APE12-dist-na | 10.934 | APE11-dist-na | 12.929 | APE10-dist-na | 9.919 | APE9-dist-in | 6.838 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.182 | 0.205 | A | 301 | 289 | 12 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6elr | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6ELRB | 865 | 1154 | 1154.0 | BFK:1201 | Type1 | Inactive | DFGin | 6.601 | 13.531 | ABAminus | -109.26, 5.99 | -154.04, 139.83 | -131.25, 27.64 | 294.03, 83.78 | -58.7, -28.76 | in-in | in | 7.739 | Saltbr-in | 2.752 | HRD-in | -72.31, -47.94 | 70.47, 1.78 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.838 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.07, 32.45 | APE9-dihe-in | -65.92, 131.99 | APE8-dihe-in | -78.37, 73.16 | APE8-rot-na | 28.72 | APE67-dihe-in | -77.26, -5.72 | -51.85, -33.17 | APE12-dist-na | 11.057 | APE11-dist-na | 13.148 | APE10-dist-na | 10.069 | APE9-dist-in | 6.853 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.182 | 0.205 | B | 301 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6elr | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6SM8B | 865 | 1154 | 1154.0 | LKT:61201 | Type1 | Inactive | DFGin | 6.806 | 13.668 | ABAminus | -102.82, -5.52 | -148.54, 142.3 | -131.39, 24.74 | 291.91, 87.01 | -56.81, -29.39 | in-in | in | 7.801 | Saltbr-in | 2.711 | HRD-in | -72.52, -51.3 | 71.87, 8.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.832 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.32, 29.21 | APE9-dihe-in | -64.29, 137.39 | APE8-dihe-in | -82.59, 73.84 | APE8-rot-na | 28.56 | APE67-dihe-in | -76.5, -2.32 | -51.19, -31.92 | APE12-dist-na | 11.521 | APE11-dist-na | 13.343 | APE10-dist-na | 10.329 | APE9-dist-in | 6.67 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.85 | 0.213 | 0.241 | B | 301 | 284 | 6 | 0 | 0 | 2 | [[583, 847], [875, 1151]] | 2.0 | 6sm8 | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6SMBA | 863 | 1153 | 1154.0 | LKQ:1201 | Type1 | Inactive | DFGin | 6.607 | 13.731 | ABAminus | -104.09, 12.38 | -161.47, 134.46 | -125.84, 26.47 | 298.3, 80.99 | -58.62, -24.17 | in-in | in | 7.831 | Saltbr-in | 2.643 | HRD-in | -73.47, -45.53 | 65.45, 5.36 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.749 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -94.53, 41.14 | APE9-dihe-in | -70.01, 131.09 | APE8-dihe-in | -75.02, 72.06 | APE8-rot-na | 25.33 | APE67-dihe-in | -73.28, -2.79 | -51.04, -36.86 | APE12-dist-na | 12.02 | APE11-dist-na | 12.716 | APE10-dist-na | 10.235 | APE9-dist-in | 6.755 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.04 | 0.224 | 0.265 | A | 301 | 288 | 3 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6smb | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6SMBB | 863 | 1153 | 1154.0 | LKQ:1201 | Type1 | Inactive | DFGin | 6.618 | 13.811 | ABAminus | -106.29, 15.46 | -163.61, 135.62 | -126.74, 26.38 | 298.65, 81.43 | -58.83, -23.63 | in-in | in | 7.869 | Saltbr-in | 2.627 | HRD-in | -72.91, -46.19 | 66.2, 3.06 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.745 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 76.78, 22.71 | APE9-dihe-in | -68.31, 133.01 | APE8-dihe-in | -75.13, 72.89 | APE8-rot-na | 25.36 | APE67-dihe-in | -72.9, -3.33 | -50.86, -36.85 | APE12-dist-na | 10.831 | APE11-dist-na | 12.575 | APE10-dist-na | 10.456 | APE9-dist-in | 6.68 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.04 | 0.224 | 0.265 | B | 301 | 282 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6smb | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4E4LA | 865 | 1154 | 1154.0 | 0NH:1201 | Type1 | Inactive | DFGin | 6.506 | 13.593 | ABAminus | -113.26, 1.55 | -155.7, 141.31 | -133.96, 30.85 | 296.7, 84.55 | -61.93, -29.15 | in-in | in | 7.728 | Saltbr-in | 2.366 | HRD-in | -82.62, -51.73 | 77.35, 2.42 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.833 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.62, 29.91 | APE9-dihe-in | -55.83, 134.62 | APE8-dihe-in | -77.55, 77.11 | APE8-rot-na | 23.92 | APE67-dihe-in | -76.85, -4.17 | -58.31, -32.93 | APE12-dist-na | 11.099 | APE11-dist-na | 12.761 | APE10-dist-na | 10.348 | APE9-dist-in | 6.603 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.19 | 0.228 | A | 302 | 279 | 11 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4l | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4E4LB | 864 | 1154 | 1154.0 | 0NH:1201 | Type1 | Inactive | DFGin | 6.468 | 13.69 | ABAminus | -115.34, 5.94 | -154.23, 143.98 | -136.31, 29.8 | 294.89, 85.73 | -63.4, -28.12 | in-in | in | 7.872 | Saltbr-in | 2.625 | HRD-in | -80.23, -45.9 | 70.61, 1.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.75 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -105.56, 32.84 | APE9-dihe-in | -59.39, 139.65 | APE8-dihe-in | -81.36, 75.53 | APE8-rot-na | 28.93 | APE67-dihe-in | -77.55, -4.05 | -62.31, -27.51 | APE12-dist-na | 10.995 | APE11-dist-na | 12.667 | APE10-dist-na | 10.069 | APE9-dist-in | 6.632 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.19 | 0.228 | B | 302 | 281 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4l | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4E4LD | 864 | 1154 | 1154.0 | 0NH:1201 | Type1 | Inactive | DFGin | 6.536 | 13.748 | ABAminus | -114.27, -0.81 | -153.61, 143.22 | -135.12, 28.03 | 293.73, 85.38 | -57.66, -27.04 | in-in | in | 7.741 | Saltbr-in | 2.555 | HRD-in | -77.01, -53.08 | 75.86, 4.71 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.823 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -115.68, 33.68 | APE9-dihe-in | -65.48, 130.64 | APE8-dihe-in | -74.63, 79.76 | APE8-rot-na | 26.43 | APE67-dihe-in | -75.57, -2.67 | -62.18, -32.34 | APE12-dist-na | 11.513 | APE11-dist-na | 12.875 | APE10-dist-na | 10.415 | APE9-dist-in | 6.7 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.19 | 0.228 | D | 302 | 283 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4l | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4E4NA | 854 | 1154 | 1154.0 | 0NL:61201 | Type1 | Inactive | DFGin | 6.384 | 13.56 | ABAminus | -120.02, 11.21 | -158.48, 139.99 | -136.43, 26.78 | 297.09, 85.57 | -63.39, -21.4 | in-in | in | 7.79 | Saltbr-in | 2.555 | HRD-in | -80.31, -49.85 | 72.5, 4.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.848 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -96.76, 48.8 | APE9-dihe-in | -75.99, 139.57 | APE8-dihe-in | -78.93, 73.17 | APE8-rot-na | 33.7 | APE67-dihe-in | -74.47, -3.41 | -60.94, -30.72 | APE12-dist-na | 11.071 | APE11-dist-na | 12.756 | APE10-dist-na | 10.411 | APE9-dist-in | 6.832 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.183 | 0.226 | A | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4n | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4E4NB | 865 | 1154 | 1154.0 | 0NL:61201 | Type1 | Inactive | DFGin | 6.346 | 13.502 | ABAminus | -119.9, 9.63 | -155.68, 139.61 | -133.8, 28.11 | 297.19, 80.43 | -62.66, -24.74 | in-in | in | 7.737 | Saltbr-in | 2.603 | HRD-in | -78.32, -48.47 | 74.25, 0.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.874 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.54, 49.17 | APE9-dihe-in | -76.21, 142.06 | APE8-dihe-in | -79.22, 71.62 | APE8-rot-na | 25.59 | APE67-dihe-in | -77.0, -5.97 | -60.76, -27.4 | APE12-dist-na | 11.162 | APE11-dist-na | 12.793 | APE10-dist-na | 10.433 | APE9-dist-in | 6.939 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.183 | 0.226 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4n | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4E5WA | 854 | 1154 | 1154.0 | 0NT:61201 | Type1 | Inactive | DFGin | 6.562 | 13.397 | ABAminus | -118.14, 5.18 | -153.89, 137.32 | -129.51, 26.76 | 295.21, 88.69 | -58.94, -26.21 | in-in | in | 7.704 | Saltbr-in | 2.687 | HRD-in | -73.36, -50.75 | 70.96, 2.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.834 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.84, 26.34 | APE9-dihe-in | -57.31, 135.68 | APE8-dihe-in | -78.98, 72.49 | APE8-rot-na | 27.03 | APE67-dihe-in | -72.09, -3.1 | -47.71, -39.24 | APE12-dist-na | 11.088 | APE11-dist-na | 13.57 | APE10-dist-na | 10.45 | APE9-dist-in | 6.738 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.86 | 0.184 | 0.21 | A | 302 | 293 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e5w | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4E5WB | 865 | 1153 | 1154.0 | 0NT:61202 | Type1 | Inactive | DFGin | 6.53 | 13.35 | ABAminus | -114.8, 7.46 | -153.87, 137.96 | -129.8, 26.64 | 296.41, 93.24 | -58.91, -27.51 | in-in | in | 7.691 | Saltbr-in | 2.687 | HRD-in | -74.04, -50.94 | 71.65, 3.46 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.833 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.41, 26.14 | APE9-dihe-in | -57.59, 134.48 | APE8-dihe-in | -78.71, 72.64 | APE8-rot-na | 26.79 | APE67-dihe-in | -72.94, -2.19 | -48.23, -38.49 | APE12-dist-na | 11.113 | APE11-dist-na | 13.557 | APE10-dist-na | 10.431 | APE9-dist-in | 6.758 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.86 | 0.184 | 0.21 | B | 302 | 280 | 9 | 0 | 0 | 2 | [[583, 847], [875, 1151]] | 2.0 | 4e5w | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4EHZA | 858 | 1154 | 1154.0 | JAK:1201 | Type1 | Inactive | DFGin | 6.295 | 13.63 | ABAminus | -122.46, 12.74 | -158.91, 149.59 | -139.33, 23.83 | 295.89, 89.08 | -61.4, -20.25 | in-in | in | 7.795 | Saltbr-in | 2.936 | HRD-in | -79.41, -51.26 | 80.05, -0.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.866 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -94.49, 24.25 | APE9-dihe-in | -61.79, 133.39 | APE8-dihe-in | -76.86, 73.91 | APE8-rot-na | 30.52 | APE67-dihe-in | -75.94, -6.94 | -60.76, -27.83 | APE12-dist-na | 11.438 | APE11-dist-na | 13.16 | APE10-dist-na | 9.871 | APE9-dist-in | 7.032 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.174 | 0.174 | 0.229 | A | 302 | 292 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ehz | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4EHZB | 865 | 1154 | 1154.0 | JAK:1201 | Type1 | Inactive | DFGin | 6.317 | 13.73 | ABAminus | -116.35, 3.51 | -150.61, 148.16 | -138.87, 32.34 | 292.95, 86.02 | -67.41, -23.21 | in-in | in | 7.869 | Saltbr-in | 2.763 | HRD-in | -83.57, -44.01 | 70.15, -1.08 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.733 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.9, 29.19 | APE9-dihe-in | -67.89, 136.88 | APE8-dihe-in | -75.68, 68.81 | APE8-rot-na | 33.04 | APE67-dihe-in | -71.9, -6.58 | -49.99, -36.99 | APE12-dist-na | 11.419 | APE11-dist-na | 13.393 | APE10-dist-na | 10.125 | APE9-dist-in | 6.991 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.174 | 0.174 | 0.229 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ehz | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4EHZC | 866 | 1154 | 1154.0 | JAK:1201 | Type1 | Inactive | DFGin | 6.317 | 13.621 | ABAminus | -118.15, 8.14 | -148.22, 154.09 | -141.74, 25.14 | 292.74, 84.54 | -60.05, -18.24 | in-in | in | 7.859 | Saltbr-in | 2.84 | HRD-in | -77.85, -48.09 | 78.3, 3.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.724 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.81, 30.11 | APE9-dihe-in | -57.01, 145.43 | APE8-dihe-in | -85.32, 74.95 | APE8-rot-na | 31.15 | APE67-dihe-in | -74.27, -3.28 | -56.74, -31.49 | APE12-dist-na | 10.975 | APE11-dist-na | 13.004 | APE10-dist-na | 10.18 | APE9-dist-in | 6.676 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.174 | 0.174 | 0.229 | C | 302 | 280 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ehz | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4EHZD | 865 | 1154 | 1154.0 | JAK:1201 | Type1 | Inactive | DFGin | 6.428 | 13.533 | ABAminus | -123.86, 16.47 | -158.34, 146.22 | -137.38, 32.15 | 296.06, 77.8 | -67.83, -20.15 | in-in | in | 7.679 | Saltbr-in | 3.0 | HRD-in | -85.88, -43.73 | 70.18, 7.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.38, 26.48 | APE9-dihe-in | -59.77, 138.32 | APE8-dihe-in | -81.72, 74.58 | APE8-rot-na | 32.67 | APE67-dihe-in | -77.67, -4.82 | -52.47, -31.56 | APE12-dist-na | 11.043 | APE11-dist-na | 12.962 | APE10-dist-na | 10.009 | APE9-dist-in | 6.688 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.174 | 0.174 | 0.229 | D | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ehz | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4EI4A | 854 | 1154 | 1154.0 | 0Q2:61201 | Type1 | Inactive | DFGin | 6.362 | 13.452 | ABAminus | -125.08, 21.55 | -162.93, 136.7 | -132.47, 29.54 | 298.16, 82.51 | -65.62, -22.07 | in-in | in | 7.843 | Saltbr-in | 2.612 | HRD-in | -82.16, -48.37 | 72.58, 5.29 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.744 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -105.53, 42.94 | APE9-dihe-in | -71.49, 136.49 | APE8-dihe-in | -77.62, 74.63 | APE8-rot-na | 31.88 | APE67-dihe-in | -76.69, -5.39 | -62.91, -28.92 | APE12-dist-na | 10.983 | APE11-dist-na | 12.753 | APE10-dist-na | 10.259 | APE9-dist-in | 6.784 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.22 | 0.202 | 0.239 | A | 302 | 290 | 11 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ei4 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4EI4B | 865 | 1154 | 1154.0 | 0Q2:61201 | Type1 | Inactive | DFGin | 6.382 | 13.518 | ABAminus | -120.19, 16.13 | -160.02, 140.78 | -136.52, 31.88 | 292.39, 84.5 | -65.63, -28.61 | in-in | in | 7.853 | Saltbr-in | 2.827 | HRD-in | -84.06, -46.22 | 68.02, 6.16 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.752 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.4, 38.28 | APE9-dihe-in | -67.47, 135.5 | APE8-dihe-in | -75.19, 75.25 | APE8-rot-na | 28.78 | APE67-dihe-in | -75.9, -4.89 | -57.78, -34.83 | APE12-dist-na | 11.055 | APE11-dist-na | 12.687 | APE10-dist-na | 10.236 | APE9-dist-in | 6.789 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.22 | 0.202 | 0.239 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ei4 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4FK6A | 863 | 1154 | 1154.0 | 0UJ:1201 | Type1 | Inactive | DFGin | 6.577 | 13.413 | ABAminus | -112.19, 2.74 | -147.97, 135.94 | -128.79, 22.38 | 293.74, 90.76 | -52.95, -29.36 | in-in | in | 7.654 | Saltbr-in | 2.674 | HRD-in | -73.71, -49.95 | 70.6, -2.02 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.81 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.7, 28.56 | APE9-dihe-in | -63.18, 134.95 | APE8-dihe-in | -78.74, 77.08 | APE8-rot-na | 27.11 | APE67-dihe-in | -76.1, -2.34 | -51.26, -33.75 | APE12-dist-na | 11.32 | APE11-dist-na | 12.856 | APE10-dist-na | 10.101 | APE9-dist-in | 6.646 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.211 | 0.251 | A | 302 | 287 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4fk6 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4FK6B | 864 | 1154 | 1154.0 | 0UJ:1201 | Type1 | Inactive | DFGin | 6.594 | 13.406 | ABAminus | -112.12, 2.82 | -147.85, 135.79 | -128.94, 22.08 | 293.63, 90.77 | -52.49, -30.06 | in-in | in | 7.638 | Saltbr-in | 2.679 | HRD-in | -73.35, -50.23 | 70.8, -1.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.817 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.94, 28.16 | APE9-dihe-in | -62.61, 135.05 | APE8-dihe-in | -78.72, 77.07 | APE8-rot-na | 27.01 | APE67-dihe-in | -76.01, -2.17 | -51.54, -33.82 | APE12-dist-na | 11.313 | APE11-dist-na | 12.766 | APE10-dist-na | 10.141 | APE9-dist-in | 6.647 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.211 | 0.251 | B | 302 | 286 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4fk6 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4I5CA | 865 | 1154 | 1154.0 | C5I:61201 | Type1 | Inactive | DFGin | 6.372 | 13.098 | ABAminus | -114.74, 13.12 | -159.95, 138.51 | -132.46, 27.57 | 300.19, 86.09 | -57.95, -29.46 | in-in | in | 7.648 | Saltbr-in | 2.663 | HRD-in | -72.51, -44.79 | 66.5, 0.54 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.903 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -124.02, 33.91 | APE9-dihe-in | -66.46, 131.24 | APE8-dihe-in | -75.55, 75.28 | APE8-rot-na | 31.15 | APE67-dihe-in | -75.41, -9.49 | -50.0, -34.68 | APE12-dist-na | 11.26 | APE11-dist-na | 13.341 | APE10-dist-na | 10.194 | APE9-dist-in | 6.774 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.1 | 0.193 | 0.245 | A | 302 | 281 | 9 | 0 | 0 | 1 | [[583, 847], [875, 1151]] | 2.0 | 4i5c | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4I5CB | 854 | 1154 | 1154.0 | C5I:61205 | Type1 | Inactive | DFGin | 6.288 | 13.062 | ABAminus | -117.66, 20.22 | -158.68, 137.22 | -131.37, 22.03 | 299.16, 87.56 | -52.78, -31.38 | in-in | in | 7.784 | Saltbr-in | 2.586 | HRD-in | -74.37, -52.31 | 71.43, 0.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.948 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -101.41, 21.23 | APE9-dihe-in | -58.7, 133.33 | APE8-dihe-in | -78.45, 70.87 | APE8-rot-na | 28.87 | APE67-dihe-in | -73.75, -3.17 | -47.7, -37.18 | APE12-dist-na | 11.146 | APE11-dist-na | 13.194 | APE10-dist-na | 10.032 | APE9-dist-in | 6.84 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.1 | 0.193 | 0.245 | B | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4i5c | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4IVBA | 854 | 1154 | 1154.0 | 1J5:61201 | Type1 | Inactive | DFGin | 6.446 | 13.398 | ABAminus | -120.37, 8.79 | -154.43, 145.03 | -134.59, 25.95 | 296.41, 85.72 | -59.41, -26.27 | in-in | in | 7.777 | Saltbr-in | 2.607 | HRD-in | -81.27, -49.76 | 73.46, 5.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.901 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.65, 36.69 | APE9-dihe-in | -67.09, 139.5 | APE8-dihe-in | -78.95, 74.88 | APE8-rot-na | 31.26 | APE67-dihe-in | -75.42, -5.51 | -58.71, -32.55 | APE12-dist-na | 11.215 | APE11-dist-na | 12.935 | APE10-dist-na | 10.311 | APE9-dist-in | 6.781 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.183 | 0.221 | A | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivb | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4IVBB | 865 | 1154 | 1154.0 | 1J5:61201 | Type1 | Inactive | DFGin | 6.429 | 13.415 | ABAminus | -116.62, 7.74 | -154.57, 143.33 | -132.65, 26.65 | 294.75, 85.72 | -57.0, -32.17 | in-in | in | 7.713 | Saltbr-in | 2.651 | HRD-in | -82.29, -46.68 | 69.34, 6.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.895 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.2, 32.35 | APE9-dihe-in | -63.44, 138.0 | APE8-dihe-in | -78.25, 77.26 | APE8-rot-na | 32.13 | APE67-dihe-in | -75.77, -2.93 | -62.98, -29.79 | APE12-dist-na | 11.263 | APE11-dist-na | 12.983 | APE10-dist-na | 10.306 | APE9-dist-in | 6.769 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.183 | 0.221 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivb | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4IVCA | 854 | 1154 | 1154.0 | 1J6:61201 | Type1 | Inactive | DFGin | 6.249 | 13.251 | ABAminus | -114.51, 9.81 | -157.21, 145.73 | -138.3, 37.36 | 304.45, 81.48 | -64.22, -30.51 | in-in | in | 7.826 | Saltbr-in | 2.692 | HRD-in | -91.76, -42.16 | 67.22, -0.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.842 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.76, 45.97 | APE9-dihe-in | -72.9, 142.32 | APE8-dihe-in | -77.97, 76.61 | APE8-rot-na | 30.79 | APE67-dihe-in | -73.52, -3.32 | -54.87, -39.45 | APE12-dist-na | 11.192 | APE11-dist-na | 12.652 | APE10-dist-na | 10.171 | APE9-dist-in | 6.549 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.35 | 0.2 | 0.263 | A | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivc | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4IVCB | 865 | 1154 | 1154.0 | 1J6:61201 | Type1 | Inactive | DFGin | 6.313 | 13.347 | ABAminus | -119.67, 6.43 | -149.04, 145.44 | -134.49, 29.55 | 297.17, 82.22 | -60.5, -32.79 | in-in | in | 7.525 | Saltbr-in | 2.277 | HRD-in | -89.31, -45.09 | 71.21, 3.65 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.717 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -101.71, 20.54 | APE9-dihe-in | -65.21, 135.06 | APE8-dihe-in | -79.05, 83.59 | APE8-rot-na | 28.99 | APE67-dihe-in | -78.13, -7.38 | -62.67, -27.87 | APE12-dist-na | 11.123 | APE11-dist-na | 12.804 | APE10-dist-na | 9.574 | APE9-dist-in | 6.607 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.35 | 0.2 | 0.263 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivc | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4IVDA | 854 | 1154 | 1154.0 | 15T:61201 | Type1 | Inactive | DFGin | 6.309 | 13.304 | ABAminus | -118.43, 8.35 | -154.11, 148.17 | -137.65, 24.48 | 298.46, 83.68 | -55.12, -27.34 | in-in | in | 7.749 | Saltbr-in | 2.729 | HRD-in | -85.26, -46.42 | 71.64, 5.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.903 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -118.71, 33.92 | APE9-dihe-in | -63.4, 140.18 | APE8-dihe-in | -80.26, 75.71 | APE8-rot-na | 32.55 | APE67-dihe-in | -74.69, -4.74 | -58.39, -31.37 | APE12-dist-na | 11.247 | APE11-dist-na | 12.97 | APE10-dist-na | 10.268 | APE9-dist-in | 6.655 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.93 | 0.204 | 0.247 | A | 302 | 291 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivd | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4IVDB | 865 | 1154 | 1154.0 | 15T:61201 | Type1 | Inactive | DFGin | 6.411 | 13.37 | ABAminus | -112.55, 2.72 | -159.22, 144.81 | -135.21, 28.45 | 296.48, 84.97 | -57.15, -29.77 | in-in | in | 7.676 | Saltbr-in | 2.745 | HRD-in | -84.66, -44.43 | 68.53, 7.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.922 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.94, 35.04 | APE9-dihe-in | -66.46, 139.38 | APE8-dihe-in | -79.29, 77.36 | APE8-rot-na | 30.63 | APE67-dihe-in | -76.81, -5.82 | -62.53, -27.62 | APE12-dist-na | 11.221 | APE11-dist-na | 12.974 | APE10-dist-na | 10.244 | APE9-dist-in | 6.666 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.93 | 0.204 | 0.247 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivd | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4K6ZA | 865 | 1154 | 1154.0 | 1Q3:1201 | Type1 | Inactive | DFGin | 6.368 | 13.629 | ABAminus | -111.25, 5.81 | -148.16, 138.39 | -130.89, 30.06 | 299.5, 88.49 | -54.29, -32.58 | in-in | in | 8.161 | Saltbr-in | 2.913 | HRD-in | -64.09, -54.55 | 67.8, 5.15 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.82 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.94, 36.35 | APE9-dihe-in | -67.0, 125.07 | APE8-dihe-in | -75.83, 85.59 | APE8-rot-na | 25.89 | APE67-dihe-in | -67.06, -19.07 | -53.74, -42.35 | APE12-dist-na | 10.425 | APE11-dist-na | 12.583 | APE10-dist-na | 10.007 | APE9-dist-in | 6.016 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.73 | 0.244 | 0.297 | A | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4k6z | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4K77A | 864 | 1154 | 1154.0 | 1Q4:1201 | Type1 | Inactive | DFGin | 6.256 | 13.464 | ABAminus | -120.21, 6.98 | -152.33, 140.1 | -135.8, 29.32 | 300.23, 84.02 | -66.83, -17.3 | in-in | in | 8.042 | Saltbr-in | 2.62 | HRD-in | -83.59, -46.77 | 75.55, -1.36 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.807 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.78, 30.95 | APE9-dihe-in | -65.86, 137.27 | APE8-dihe-in | -79.1, 74.56 | APE8-rot-na | 31.39 | APE67-dihe-in | -73.63, -7.17 | -57.69, -30.82 | APE12-dist-na | 11.18 | APE11-dist-na | 12.795 | APE10-dist-na | 9.921 | APE9-dist-in | 6.75 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.4 | 0.193 | 0.251 | A | 302 | 284 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4k77 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 4K77B | 865 | 1154 | 1154.0 | 1Q4:1201 | Type1 | Inactive | DFGin | 6.282 | 13.504 | ABAminus | -120.68, 0.99 | -147.42, 142.05 | -133.88, 36.74 | 297.84, 83.5 | -67.02, -18.72 | in-in | in | 7.948 | Saltbr-in | 2.922 | HRD-in | -85.03, -50.83 | 74.8, -3.74 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.726 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.68, 47.05 | APE9-dihe-in | -77.0, 143.68 | APE8-dihe-in | -79.91, 78.18 | APE8-rot-na | 30.27 | APE67-dihe-in | -77.76, -4.87 | -65.15, -27.78 | APE12-dist-na | 11.137 | APE11-dist-na | 12.726 | APE10-dist-na | 10.167 | APE9-dist-in | 6.81 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.4 | 0.193 | 0.251 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4k77 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5HX8A | 855 | 1154 | 1154.0 | 66P:1201 | Type1 | Inactive | DFGin | 6.449 | 13.688 | ABAminus | -102.8, 8.3 | -149.54, 137.76 | -131.57, 23.74 | 295.19, 87.44 | -55.43, -25.96 | in-in | in | 7.925 | Saltbr-in | 2.761 | HRD-in | -74.69, -48.9 | 64.93, 4.52 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.727 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -103.85, 104.76 | APE9-dihe-in | -72.26, 138.18 | APE8-dihe-in | -80.27, 76.7 | APE8-rot-na | 26.46 | APE67-dihe-in | -75.94, -4.44 | -51.82, -37.01 | APE12-dist-na | 11.12 | APE11-dist-na | 12.285 | APE10-dist-na | 11.393 | APE9-dist-in | 6.611 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.199 | 0.24 | A | 302 | 293 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5hx8 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5HX8B | 865 | 1154 | 1154.0 | 66P:1201 | Type1 | Inactive | DFGin | 6.42 | 13.631 | ABAminus | -110.45, 9.62 | -150.03, 136.28 | -131.01, 24.66 | 294.53, 92.56 | -57.47, -31.3 | in-in | in | 7.769 | Saltbr-in | 2.758 | HRD-in | -74.49, -50.24 | 68.18, -1.59 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.774 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -121.57, 40.76 | APE9-dihe-in | -71.94, 141.78 | APE8-dihe-in | -79.55, 77.3 | APE8-rot-na | 24.89 | APE67-dihe-in | -77.48, 1.58 | -49.69, -36.95 | APE12-dist-na | 10.838 | APE11-dist-na | 12.693 | APE10-dist-na | 10.86 | APE9-dist-in | 6.55 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.199 | 0.24 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5hx8 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5WO4A | 854 | 1154 | 1154.0 | B7V:2001 | Type1 | Inactive | DFGin | 6.559 | 13.475 | ABAminus | -113.4, 5.79 | -147.65, 137.71 | -131.93, 25.73 | 295.23, 90.95 | -54.73, -30.34 | in-in | in | 7.676 | Saltbr-in | 2.754 | HRD-in | -72.7, -46.52 | 67.85, -2.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.821 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.62, 42.17 | APE9-dihe-in | -67.76, 140.08 | APE8-dihe-in | -81.09, 72.14 | APE8-rot-na | 29.77 | APE67-dihe-in | -75.22, -1.83 | -52.55, -34.79 | APE12-dist-na | 10.797 | APE11-dist-na | 12.901 | APE10-dist-na | 10.466 | APE9-dist-in | 6.823 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.84 | 0.188 | 0.211 | A | 302 | 294 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5wo4 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5WO4B | 865 | 1154 | 1154.0 | B7V:2001 | Type1 | Inactive | DFGin | 6.55 | 13.411 | ABAminus | -111.8, 3.6 | -145.5, 139.23 | -132.92, 27.81 | 292.27, 90.98 | -57.76, -28.76 | in-in | in | 7.615 | Saltbr-in | 2.781 | HRD-in | -72.82, -49.06 | 69.56, 1.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.838 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.71, 39.74 | APE9-dihe-in | -66.32, 138.27 | APE8-dihe-in | -78.58, 73.11 | APE8-rot-na | 28.91 | APE67-dihe-in | -75.88, -0.88 | -52.5, -34.22 | APE12-dist-na | 10.866 | APE11-dist-na | 12.93 | APE10-dist-na | 10.505 | APE9-dist-in | 6.743 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.84 | 0.188 | 0.211 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5wo4 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6HZUA | 854 | 1154 | 1154.0 | GYQ:61201 | Type1 | Inactive | DFGin | 6.458 | 13.248 | ABAminus | -115.79, 10.1 | -155.61, 143.2 | -135.89, 34.69 | 298.64, 85.33 | -68.92, -23.66 | in-in | in | 7.891 | Saltbr-in | 2.605 | HRD-in | -70.11, -45.53 | 64.37, 7.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.768 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -94.73, 34.76 | APE9-dihe-in | -73.48, 139.36 | APE8-dihe-in | -81.86, 74.79 | APE8-rot-na | 30.37 | APE67-dihe-in | -72.43, -9.67 | -55.59, -34.31 | APE12-dist-na | 10.967 | APE11-dist-na | 13.174 | APE10-dist-na | 9.887 | APE9-dist-in | 6.803 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.204 | 0.265 | A | 302 | 293 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6hzu | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6HZUB | 865 | 1154 | 1154.0 | GYQ:61201 | Type1 | Inactive | DFGin | 6.443 | 13.247 | ABAminus | -119.96, 0.48 | -155.13, 140.72 | -132.65, 33.96 | 299.27, 84.27 | -60.17, -34.27 | in-in | in | 8.023 | Saltbr-in | 2.702 | HRD-in | -82.42, -47.78 | 71.93, 4.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.923 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -93.89, 29.59 | APE9-dihe-in | -63.03, 138.85 | APE8-dihe-in | -81.19, 78.97 | APE8-rot-na | 31.69 | APE67-dihe-in | -73.96, -7.04 | -62.12, -30.09 | APE12-dist-na | 11.006 | APE11-dist-na | 13.225 | APE10-dist-na | 9.885 | APE9-dist-in | 6.657 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.204 | 0.265 | B | 302 | 285 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6hzu | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N77A | 866 | 1154 | 1154.0 | KEJ:1201 | Type1 | Inactive | DFGin | 6.391 | 13.654 | ABAminus | -111.17, 5.93 | -155.03, 145.91 | -137.7, 32.01 | 295.16, 86.03 | -58.79, -28.87 | in-in | in | 8.239 | Saltbr-in | 2.758 | HRD-in | -67.03, -46.69 | 67.69, -1.58 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.924 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 52.82, 53.92 | APE9-dihe-in | -90.09, 140.83 | APE8-dihe-in | -78.25, 71.6 | APE8-rot-na | 26.8 | APE67-dihe-in | -76.7, -1.13 | -52.74, -34.15 | APE12-dist-na | 11.079 | APE11-dist-na | 12.09 | APE10-dist-na | 10.994 | APE9-dist-in | 7.019 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.64 | 0.253 | 0.282 | A | 302 | 280 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n77 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N77B | 865 | 1154 | 1154.0 | KEJ:1202 | Type1 | Inactive | DFGin | 6.447 | 13.754 | ABAminus | -112.96, 6.51 | -156.54, 142.84 | -135.02, 28.22 | 296.71, 89.38 | -58.72, -26.41 | in-in | in | 8.213 | Saltbr-in | 2.737 | HRD-in | -67.03, -48.62 | 72.63, -6.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.844 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.58, 44.0 | APE9-dihe-in | -74.12, 131.71 | APE8-dihe-in | -79.78, 70.31 | APE8-rot-na | 28.35 | APE67-dihe-in | -75.35, -3.65 | -48.14, -35.74 | APE12-dist-na | 10.934 | APE11-dist-na | 12.689 | APE10-dist-na | 9.987 | APE9-dist-in | 6.954 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.64 | 0.253 | 0.282 | B | 302 | 279 | 11 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n77 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N78A | 866 | 1154 | 1154.0 | KEP:1201 | Type1 | Inactive | DFGin | 6.425 | 13.562 | ABAminus | -105.81, -4.17 | -146.0, 143.93 | -133.35, 28.47 | 298.42, 87.41 | -54.49, -32.74 | in-in | in | 8.377 | Saltbr-in | 2.73 | HRD-in | -68.76, -52.63 | 70.44, -3.87 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.811 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -114.29, 50.22 | APE9-dihe-in | -86.39, 131.12 | APE8-dihe-in | -82.28, 79.47 | APE8-rot-na | 24.58 | APE67-dihe-in | -76.5, -2.33 | -53.51, -34.22 | APE12-dist-na | 11.515 | APE11-dist-na | 12.037 | APE10-dist-na | 9.052 | APE9-dist-in | 6.377 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.83 | 0.236 | 0.261 | A | 302 | 277 | 12 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n78 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N79A | 866 | 1154 | 1154.0 | KES:1201 | Type1 | Inactive | DFGin | 6.403 | 13.525 | ABAminus | -99.38, -15.25 | -133.8, 148.14 | -138.23, 25.13 | 295.77, 92.1 | -55.46, -31.57 | in-in | in | 8.295 | Saltbr-in | 2.767 | HRD-in | -74.33, -53.6 | 68.25, 4.98 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.781 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.11, 40.21 | APE9-dihe-in | -76.58, 124.37 | APE8-dihe-in | -77.77, 81.63 | APE8-rot-na | 28.13 | APE67-dihe-in | -77.42, -2.89 | -55.56, -32.1 | APE12-dist-na | 11.219 | APE11-dist-na | 11.887 | APE10-dist-na | 9.075 | APE9-dist-in | 5.964 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.27 | 0.227 | 0.27 | A | 302 | 279 | 10 | 0 | 0 | 2 | [[583, 847], [875, 1151]] | 2.0 | 6n79 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N7BA | 865 | 1154 | 1154.0 | KEY:1201 | Type1 | Inactive | DFGin | 6.45 | 13.456 | ABAminus | -106.32, -1.48 | -152.36, 145.64 | -135.47, 28.3 | 291.96, 86.78 | -55.73, -29.48 | in-in | in | 7.736 | Saltbr-in | 2.768 | HRD-in | -71.34, -49.85 | 67.55, 5.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.806 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.89, 58.14 | APE9-dihe-in | -96.67, 129.96 | APE8-dihe-in | -81.34, 78.4 | APE8-rot-na | 26.42 | APE67-dihe-in | -77.54, 0.39 | -57.77, -29.15 | APE12-dist-na | 11.059 | APE11-dist-na | 11.728 | APE10-dist-na | 8.79 | APE9-dist-in | 6.369 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.81 | 0.222 | 0.264 | A | 302 | 280 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n7b | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N7CA | 865 | 1154 | 1154.0 | KF1:1201 | Type1 | Inactive | DFGin | 6.513 | 13.509 | ABAminus | -110.36, 6.26 | -156.68, 145.17 | -136.24, 27.53 | 295.08, 89.21 | -55.95, -29.39 | in-in | in | 8.096 | Saltbr-in | 2.735 | HRD-in | -68.7, -46.37 | 70.89, -7.05 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.902 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 95.97 | APE9-dihe-in | -107.06, 147.5 | APE8-dihe-in | -79.03, 70.75 | APE8-rot-na | 27.77 | APE67-dihe-in | -74.72, -3.56 | -53.55, -33.63 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.457 | APE9-dist-in | 7.085 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.69 | 0.254 | 0.288 | A | 302 | 275 | 15 | 0 | 0 | 2 | [[583, 847], [875, 1151]] | 2.0 | 6n7c | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N7CB | 865 | 1154 | 1154.0 | KF1:1202 | Type1 | Inactive | DFGin | 6.51 | 13.589 | ABAminus | -115.1, 6.45 | -153.47, 142.93 | -133.09, 25.34 | 294.67, 85.94 | -52.61, -29.28 | in-in | in | 8.155 | Saltbr-in | 2.753 | HRD-in | -67.82, -44.9 | 68.03, -6.1 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.861 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.81 | APE8-dihe-in | -80.52, 71.8 | APE8-rot-na | 28.74 | APE67-dihe-in | -72.99, -4.02 | -55.65, -32.27 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.115 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.69 | 0.254 | 0.288 | B | 302 | 273 | 17 | 0 | 0 | 4 | [[583, 847], [875, 1151]] | 2.0 | 6n7c | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N7DA | 865 | 1154 | 1154.0 | KF4:1201 | Type1 | Inactive | DFGin | 6.476 | 13.402 | ABAminus | -110.67, 4.22 | -155.59, 141.48 | -134.23, 27.49 | 295.25, 85.51 | -53.77, -30.29 | in-in | in | 8.285 | Saltbr-in | 2.637 | HRD-in | -73.25, -49.17 | 70.77, 0.44 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.822 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.59, 31.0 | APE9-dihe-in | -83.57, 124.64 | APE8-dihe-in | -81.68, 83.11 | APE8-rot-na | 27.61 | APE67-dihe-in | -75.33, -0.8 | -58.46, -31.26 | APE12-dist-na | 11.561 | APE11-dist-na | 11.737 | APE10-dist-na | 7.584 | APE9-dist-in | 5.976 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.78 | 0.198 | 0.234 | A | 302 | 280 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n7d | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSBA | 865 | 1154 | 1154.0 | KGZ:1201 | Type1 | Inactive | DFGin | 6.59 | 13.509 | ABAminus | -116.74, 1.69 | -150.38, 137.57 | -126.94, 22.04 | 292.38, 82.89 | -70.44, -11.55 | in-in | in | 8.107 | Saltbr-in | 2.615 | HRD-in | -82.35, -48.96 | 71.74, 9.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.845 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.58, 28.79 | APE9-dihe-in | -52.22, 132.79 | APE8-dihe-in | -77.89, 76.1 | APE8-rot-na | 36.11 | APE67-dihe-in | -73.96, -4.25 | -64.89, -26.96 | APE12-dist-na | 12.037 | APE11-dist-na | 12.29 | APE10-dist-na | 10.327 | APE9-dist-in | 6.885 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.311 | 0.354 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsb | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSBB | 865 | 1154 | 1154.0 | KGZ:1201 | Type1 | Inactive | DFGin | 6.647 | 13.904 | ABAminus | -118.58, -5.18 | -147.32, 138.8 | -128.6, 27.58 | 293.53, 77.97 | -68.36, -16.41 | in-in | in | 8.049 | Saltbr-in | 2.707 | HRD-in | -76.09, -52.98 | 75.83, 4.99 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.959 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.45, 33.45 | APE9-dihe-in | -55.89, 141.48 | APE8-dihe-in | -80.12, 75.54 | APE8-rot-na | 36.76 | APE67-dihe-in | -74.19, -3.49 | -57.35, -33.46 | APE12-dist-na | 11.792 | APE11-dist-na | 12.943 | APE10-dist-na | 10.141 | APE9-dist-in | 6.851 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.311 | 0.354 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsb | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSCA | 865 | 1154 | 1154.0 | KH5:1201 | Type1 | Inactive | DFGin | 6.554 | 13.409 | ABAminus | -117.31, 8.47 | -153.39, 137.28 | -129.48, 30.56 | 297.53, 83.92 | -65.76, -23.88 | in-in | in | 7.663 | Saltbr-in | 2.689 | HRD-in | -79.6, -49.32 | 70.06, 11.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.717 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -98.9, 27.5 | APE9-dihe-in | -67.04, 137.63 | APE8-dihe-in | -80.21, 78.36 | APE8-rot-na | 37.08 | APE67-dihe-in | -76.89, -0.21 | -62.94, -28.86 | APE12-dist-na | 11.004 | APE11-dist-na | 13.576 | APE10-dist-na | 10.231 | APE9-dist-in | 6.858 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.85 | 0.249 | 0.28 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsc | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSCB | 865 | 1154 | 1154.0 | KH5:1201 | Type1 | Inactive | DFGin | 6.556 | 13.712 | ABAminus | -118.51, -2.16 | -150.35, 139.43 | -132.07, 31.9 | 298.68, 77.43 | -57.63, -28.0 | in-in | in | 7.902 | Saltbr-in | 2.662 | HRD-in | -78.87, -51.69 | 73.77, 10.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.917 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.91, 33.47 | APE9-dihe-in | -66.35, 135.05 | APE8-dihe-in | -77.66, 75.63 | APE8-rot-na | 31.23 | APE67-dihe-in | -74.4, -5.72 | -63.02, -28.16 | APE12-dist-na | 11.142 | APE11-dist-na | 13.511 | APE10-dist-na | 10.263 | APE9-dist-in | 6.918 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.85 | 0.249 | 0.28 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsc | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSDA | 865 | 1154 | 1154.0 | KH8:1201 | Type1 | Inactive | DFGin | 6.563 | 13.29 | ABAminus | -121.03, 3.28 | -150.09, 139.62 | -132.15, 26.01 | 293.71, 87.42 | -59.82, -26.08 | in-in | in | 7.641 | Saltbr-in | 2.673 | HRD-in | -81.56, -47.83 | 71.88, 7.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.925 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -96.0, 23.61 | APE9-dihe-in | -58.47, 136.99 | APE8-dihe-in | -79.35, 76.48 | APE8-rot-na | 35.13 | APE67-dihe-in | -77.95, -0.82 | -64.48, -27.09 | APE12-dist-na | 11.03 | APE11-dist-na | 13.568 | APE10-dist-na | 10.219 | APE9-dist-in | 6.806 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.76 | 0.202 | 0.238 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsd | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSDB | 865 | 1154 | 1154.0 | KH8:1201 | Type1 | Inactive | DFGin | 6.567 | 13.42 | ABAminus | -123.92, 1.98 | -149.52, 139.04 | -133.17, 29.94 | 296.8, 84.79 | -64.12, -24.87 | in-in | in | 7.828 | Saltbr-in | 2.619 | HRD-in | -81.48, -52.31 | 73.66, 6.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.886 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 78.39, 5.73 | APE9-dihe-in | -59.21, 132.36 | APE8-dihe-in | -78.28, 75.83 | APE8-rot-na | 31.46 | APE67-dihe-in | -72.63, -5.35 | -64.01, -28.2 | APE12-dist-na | 11.21 | APE11-dist-na | 13.528 | APE10-dist-na | 10.362 | APE9-dist-in | 6.887 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.76 | 0.202 | 0.238 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsd | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSEA | 865 | 1154 | 1154.0 | KHH:1201 | Type1 | Inactive | DFGin | 6.537 | 13.348 | ABAminus | -113.91, 1.27 | -156.33, 137.23 | -131.71, 27.09 | 299.32, 82.9 | -56.09, -32.48 | in-in | in | 7.864 | Saltbr-in | 2.638 | HRD-in | -79.69, -48.26 | 69.1, 11.16 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.716 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -68.92, 43.15 | APE9-dihe-in | -70.68, 135.44 | APE8-dihe-in | -74.14, 74.71 | APE8-rot-na | 28.88 | APE67-dihe-in | -82.04, -6.18 | -60.6, -28.4 | APE12-dist-na | 9.328 | APE11-dist-na | 11.782 | APE10-dist-na | 10.466 | APE9-dist-in | 6.774 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.265 | 0.303 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rse | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSEB | 865 | 1154 | 1154.0 | KHH:1201 | Type1 | Inactive | DFGin | 6.461 | 13.569 | ABAminus | -119.02, 6.25 | -155.18, 136.02 | -130.8, 28.87 | 296.2, 78.44 | -57.74, -31.19 | in-in | in | 8.034 | Saltbr-in | 2.579 | HRD-in | -78.09, -47.4 | 66.03, 12.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.903 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -77.34, 48.11 | APE9-dihe-in | -88.98, 140.2 | APE8-dihe-in | -76.8, 76.65 | APE8-rot-na | 33.64 | APE67-dihe-in | -80.09, -3.14 | -61.43, -26.93 | APE12-dist-na | 13.325 | APE11-dist-na | 11.833 | APE10-dist-na | 10.755 | APE9-dist-in | 6.856 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.265 | 0.303 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rse | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSHA | 865 | 1154 | 1154.0 | KHE:1201 | Type1 | Inactive | DFGin | 6.635 | 13.486 | ABAminus | -113.16, 6.59 | -151.95, 137.99 | -130.33, 27.13 | 294.82, 88.08 | -65.9, -20.74 | in-in | in | 7.441 | Saltbr-in | 2.532 | HRD-in | -77.26, -48.19 | 64.78, 14.62 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.694 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 87.06, 32.22 | APE9-dihe-in | -74.25, 135.13 | APE8-dihe-in | -77.78, 76.14 | APE8-rot-na | 33.2 | APE67-dihe-in | -80.47, -5.2 | -61.66, -26.89 | APE12-dist-na | 11.167 | APE11-dist-na | 12.639 | APE10-dist-na | 10.235 | APE9-dist-in | 6.904 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.71 | 0.271 | 0.311 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsh | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6RSHB | 865 | 1154 | 1154.0 | KHE:1201 | Type1 | Inactive | DFGin | 6.627 | 13.852 | ABAminus | -116.98, -3.62 | -146.38, 138.52 | -131.28, 30.89 | 293.47, 79.95 | -64.48, -19.44 | in-in | in | 7.784 | Saltbr-in | 2.375 | HRD-in | -81.26, -46.13 | 68.12, 10.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.878 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 90.62, 16.91 | APE9-dihe-in | -58.11, 134.31 | APE8-dihe-in | -78.21, 75.43 | APE8-rot-na | 34.5 | APE67-dihe-in | -75.52, -2.49 | -58.55, -33.71 | APE12-dist-na | 11.219 | APE11-dist-na | 13.047 | APE10-dist-na | 10.449 | APE9-dist-in | 6.96 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.71 | 0.271 | 0.311 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsh | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6SM8A | 854 | 1154 | 1154.0 | LKT:61201 | Type1 | Inactive | DFGin | 6.813 | 13.706 | ABAminus | -101.63, -7.1 | -147.81, 142.33 | -131.41, 24.39 | 292.89, 86.49 | -54.23, -31.63 | in-in | in | 7.807 | Saltbr-in | 2.732 | HRD-in | -72.9, -49.47 | 70.53, 3.61 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.836 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.89, 30.48 | APE9-dihe-in | -64.02, 138.21 | APE8-dihe-in | -82.49, 73.83 | APE8-rot-na | 29.16 | APE67-dihe-in | -76.27, -2.8 | -50.53, -32.36 | APE12-dist-na | 11.438 | APE11-dist-na | 13.22 | APE10-dist-na | 10.246 | APE9-dist-in | 6.724 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.85 | 0.213 | 0.241 | A | 302 | 296 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6sm8 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 8S85A | 854 | 1154 | 1154.0 | A1H5R:61201 | Type1 | Inactive | DFGin | 6.63 | 13.345 | ABAminus | -112.23, -7.17 | -149.03, 146.72 | -132.22, 30.5 | 297.85, 84.4 | -54.75, -31.9 | in-in | in | 7.852 | Saltbr-in | 2.618 | HRD-in | -76.09, -48.85 | 71.09, 5.36 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.837 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 58.53, 30.92 | APE9-dihe-in | -76.65, 137.48 | APE8-dihe-in | -75.77, 75.79 | APE8-rot-na | 30.15 | APE67-dihe-in | -76.06, -7.29 | -58.07, -32.61 | APE12-dist-na | 11.266 | APE11-dist-na | 12.679 | APE10-dist-na | 10.467 | APE9-dist-in | 6.878 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.75 | 0.21 | 0.25 | A | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 8s85 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 8S85B | 865 | 1154 | 1154.0 | A1H5R:61201 | Type1 | Inactive | DFGin | 6.696 | 13.355 | ABAminus | -114.2, -1.94 | -152.98, 142.26 | -130.74, 31.83 | 294.81, 85.33 | -58.52, -32.2 | in-in | in | 7.745 | Saltbr-in | 2.614 | HRD-in | -77.39, -48.2 | 72.5, 8.27 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.891 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -105.67, 37.06 | APE9-dihe-in | -66.96, 136.92 | APE8-dihe-in | -79.85, 74.06 | APE8-rot-na | 34.04 | APE67-dihe-in | -73.04, -6.17 | -58.28, -33.1 | APE12-dist-na | 11.159 | APE11-dist-na | 13.098 | APE10-dist-na | 10.453 | APE9-dist-in | 6.796 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.75 | 0.21 | 0.25 | B | 302 | 283 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 8s85 | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N7AA | 865 | 1154 | 1154.0 | KEV:61203 | Type1 | Inactive | DFGin | 6.453 | 13.367 | ABAminus | -116.98, 9.47 | -160.4, 147.32 | -135.39, 27.13 | 297.85, 83.25 | -58.95, -23.42 | in-in | in | 7.745 | Saltbr-in | 2.756 | HRD-in | -75.17, -44.67 | 72.8, -4.01 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.858 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -73.07, 124.84 | APE9-dihe-in | -104.44, 150.91 | APE8-dihe-in | -83.53, 72.06 | APE8-rot-na | 34.1 | APE67-dihe-in | -76.43, -2.54 | -56.05, -29.88 | APE12-dist-na | 14.659 | APE11-dist-na | 9.278 | APE10-dist-na | 12.111 | APE9-dist-in | 7.138 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.33 | 0.192 | 0.207 | A | 304 | 278 | 12 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n7a | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6N7AB | 854 | 1154 | 1154.0 | KEV:61202 | Type1 | Inactive | DFGin | 6.47 | 13.498 | ABAminus | -116.23, 10.2 | -162.11, 148.53 | -137.01, 27.49 | 296.62, 85.6 | -60.22, -22.88 | in-in | in | 7.776 | Saltbr-in | 2.755 | HRD-in | -73.34, -48.05 | 70.64, 1.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.804 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.78, 65.84 | APE9-dihe-in | -92.65, 132.46 | APE8-dihe-in | -84.19, 73.36 | APE8-rot-na | 33.1 | APE67-dihe-in | -76.82, -1.21 | -55.1, -31.23 | APE12-dist-na | 10.789 | APE11-dist-na | 11.689 | APE10-dist-na | 9.266 | APE9-dist-in | 6.819 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.33 | 0.192 | 0.207 | B | 304 | 291 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n7a | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5KHXA | 867 | 1154 | 1154.0 | 6TE:4000 | Type1 | Inactive | DFGin | 6.631 | 13.54 | ABAminus | -113.66, 8.44 | -153.85, 134.53 | -126.55, 25.21 | 296.38, 85.41 | -59.93, -18.33 | in-in | in | 7.565 | Saltbr-in | 2.778 | HRD-in | -73.12, -47.99 | 66.65, 10.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.794 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.92, 156.56 | APE9-dihe-in | -137.25, 140.8 | APE8-dihe-in | -82.8, 71.88 | APE8-rot-na | 32.82 | APE67-dihe-in | -77.93, -4.04 | -54.17, -30.94 | APE12-dist-na | 14.254 | APE11-dist-na | 8.466 | APE10-dist-na | 10.435 | APE9-dist-in | 6.376 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.4 | 0.173 | 0.242 | A | 316 | 278 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5khx | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6BBUA | 867 | 1154 | 1154.0 | D7D:4000 | Type1 | Inactive | DFGin | 6.419 | 13.3 | ABAminus | -116.63, 12.94 | -152.79, 140.28 | -132.74, 24.58 | 296.65, 83.13 | -57.55, -25.0 | in-in | in | 7.644 | Saltbr-in | 2.781 | HRD-in | -73.12, -50.44 | 71.69, 3.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.861 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -135.84, 101.53 | APE9-dihe-in | -119.31, 160.09 | APE8-dihe-in | -78.32, 76.15 | APE8-rot-na | 30.95 | APE67-dihe-in | -74.07, -7.36 | -55.8, -32.39 | APE12-dist-na | 9.748 | APE11-dist-na | 11.183 | APE10-dist-na | 11.299 | APE9-dist-in | 6.263 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.08 | 0.185 | 0.213 | A | 316 | 281 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6bbu | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6DBNA | 867 | 1154 | 1154.0 | G4J:4000 | Type1 | Inactive | DFGin | 6.339 | 13.27 | ABAminus | -106.28, 2.12 | -151.4, 144.25 | -137.1, 32.6 | 295.8, 96.91 | -66.86, -18.69 | in-in | in | 7.596 | Saltbr-in | 2.792 | HRD-in | -66.34, -50.63 | 70.35, -1.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.81 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -142.87, 84.26 | APE9-dihe-in | -94.42, 151.25 | APE8-dihe-in | -77.55, 83.04 | APE8-rot-na | 28.37 | APE67-dihe-in | -75.2, -10.39 | -60.86, -28.98 | APE12-dist-na | 9.302 | APE11-dist-na | 11.031 | APE10-dist-na | 10.809 | APE9-dist-in | 6.01 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.48 | 0.19 | 0.262 | A | 316 | 281 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6dbn | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 6W8LA | 867 | 1154 | 1154.0 | R4S:1201 | Type1 | Inactive | DFGin | 6.52 | 13.639 | ABAminus | -117.57, 7.4 | -146.11, 138.04 | -131.96, 25.84 | 294.24, 93.82 | -58.79, -29.12 | in-in | in | 7.699 | Saltbr-in | 2.747 | HRD-in | -65.59, -50.27 | 70.66, 4.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.796 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -75.31, 154.48 | APE9-dihe-in | -145.69, 148.21 | APE8-dihe-in | -75.35, 73.33 | APE8-rot-na | 31.68 | APE67-dihe-in | -71.12, -8.39 | -52.84, -34.47 | APE12-dist-na | 13.73 | APE11-dist-na | 8.042 | APE10-dist-na | 10.481 | APE9-dist-in | 6.401 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.11 | 0.197 | 0.226 | A | 316 | 280 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6w8l | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5KHWB | 867 | 1153 | 1154.0 | ADP:1201 | ATPlike | Inactive | DFGin | 6.188 | 13.787 | BLAminus | -126.62, -174.05 | 50.66, 92.23 | -105.71, 28.99 | 301.42, 97.18 | -62.73, -33.32 | in-in | in | 7.991 | Saltbr-in | 2.817 | HRD-in | -54.38, -55.02 | 75.74, 4.0 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.811 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -83.14, 18.97 | APE9-dihe-in | -58.32, 113.18 | APE8-dihe-in | -82.04, 77.86 | APE8-rot-na | 28.29 | APE67-dihe-in | -76.85, -3.42 | -56.14, -32.61 | APE12-dist-na | 7.879 | APE11-dist-na | 9.695 | APE10-dist-na | 6.605 | APE9-dist-in | 5.912 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.47 | 0.188 | 0.231 | B | 316 | 278 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5khw | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| 5E1EA | 865 | 1154 | 1154.0 | 5JG:1202 | Type1 | Inactive | DFGin | 6.644 | 13.932 | BLAminus | -119.33, -177.28 | 50.16, 87.79 | -101.77, 31.05 | 290.94, 82.42 | -65.82, -24.94 | in-in | in | 7.872 | Saltbr-in | 2.794 | HRD-in | -75.04, -43.37 | 64.83, -0.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.816 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.99, 41.3 | APE9-dihe-in | -73.96, 132.79 | APE8-dihe-in | -79.05, 75.13 | APE8-rot-na | 22.09 | APE67-dihe-in | -75.65, -2.64 | -52.7, -35.87 | APE12-dist-na | 10.981 | APE11-dist-na | 12.948 | APE10-dist-na | 10.168 | APE9-dist-in | 6.908 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.3 | 0.227 | 0.268 | A | 290 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5e1e | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| JAK1_HUMAN | 6C7YA | P23458 | 869 | 1153 | 1154.0 | ADP:61201 | ATPlike | Active | DFGin | 6.032 | 13.967 | BLAminus | -134.15, -164.18 | 58.49, 84.96 | -109.28, 28.04 | 298.78, 97.45 | -66.39, -27.05 | in-in | in | 8.311 | Saltbr-in | 2.732 | HRD-in | -67.59, -46.53 | 68.25, 12.43 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -72.91, 151.36 | APE9-dihe-in | -137.76, 143.32 | APE8-dihe-in | -74.71, 81.76 | APE8-rot-na | 30.49 | APE67-dihe-in | -79.4, -2.38 | -65.2, -24.66 | APE12-dist-na | 12.972 | APE11-dist-na | 8.02 | APE10-dist-na | 10.344 | APE9-dist-in | 6.316 | None | PTR1035 | PTR1035 | XRAY | 2.499 | 0.21 | 0.241 | A | 286 | 273 | 12 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6c7y | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.8e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | AF-P23458-K2A | P23458 | 867 | 1154 | 1154.0 | No_ligand | No_ligand | Active | DFGin | 6.307 | 13.773 | BLAminus | -130.0, -171.31 | 51.92, 79.2 | -91.39, 17.47 | 288.09, 81.21 | -63.19, -25.32 | in-in | in | 8.086 | Saltbr-in | 2.719 | HRD-in | -67.76, -41.14 | 64.22, -10.98 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.94 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -50.83, 123.48 | APE9-dihe-in | -125.8, 136.55 | APE8-dihe-in | -75.77, 67.19 | APE8-rot-na | 34.45 | APE67-dihe-in | -77.12, -11.68 | -54.83, -26.9 | APE12-dist-na | 13.91 | APE11-dist-na | 8.532 | APE10-dist-na | 10.659 | APE9-dist-in | 7.063 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 288 | 288 | 0 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | AF-P23458-K2 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.8e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | AF-P23458-K4A | P23458 | 867 | 1154 | 1154.0 | No_ligand | No_ligand | Active | DFGin | 6.034 | 13.552 | BLAminus | -127.94, -176.44 | 52.21, 91.21 | -99.55, 15.91 | 293.58, 76.0 | -63.9, -24.71 | in-in | in | 7.81 | Saltbr-in | 2.715 | HRD-in | -69.66, -43.24 | 62.91, -1.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.92 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -47.59, 114.14 | APE9-dihe-in | -120.02, 146.94 | APE8-dihe-in | -73.57, 63.93 | APE8-rot-na | 37.51 | APE67-dihe-in | -76.35, -14.96 | -54.26, -27.82 | APE12-dist-na | 13.697 | APE11-dist-na | 8.114 | APE10-dist-na | 10.916 | APE9-dist-in | 6.735 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 288 | 288 | 0 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | AF-P23458-K4 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.8e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5KHWA | P23458 | 867 | 1153 | 1154.0 | ADP:1201 | ATPlike | Inactive | DFGin | 6.293 | 13.595 | ABAminus | -113.62, -36.19 | -113.51, 112.49 | -104.48, 28.51 | 302.05, 98.46 | -68.45, -35.55 | in-in | in | 8.017 | Saltbr-in | 2.811 | HRD-in | -53.69, -54.55 | 74.32, 4.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.817 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.25, 151.86 | APE9-dihe-in | -139.19, 145.92 | APE8-dihe-in | -78.07, 75.73 | APE8-rot-na | 29.65 | APE67-dihe-in | -77.72, -3.4 | -55.44, -31.5 | APE12-dist-na | 13.014 | APE11-dist-na | 7.332 | APE10-dist-na | 9.905 | APE9-dist-in | 6.022 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.47 | 0.188 | 0.231 | A | 316 | 278 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5khw | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4E4LE | P23458 | 864 | 1154 | 1154.0 | No_ligand | No_ligand | Inactive | DFGin | 6.463 | 13.613 | ABAminus | -114.05, 7.25 | -155.92, 142.83 | -135.92, 30.26 | 296.52, 85.61 | -59.94, -28.28 | in-in | in | 7.87 | Saltbr-in | 2.625 | HRD-in | -76.43, -49.33 | 70.91, 5.03 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.809 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.8, 27.83 | APE9-dihe-in | -58.48, 132.7 | APE8-dihe-in | -75.95, 78.2 | APE8-rot-na | 25.62 | APE67-dihe-in | -75.39, -5.67 | -60.62, -30.34 | APE12-dist-na | 11.404 | APE11-dist-na | 12.865 | APE10-dist-na | 10.335 | APE9-dist-in | 6.766 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.19 | 0.228 | E | 302 | 282 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4l | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 3EYGA | P23458 | 865 | 1154 | 1154.0 | MI1:1 | Type1 | Inactive | DFGin | 6.484 | 13.585 | ABAminus | -124.32, 8.36 | -155.42, 148.92 | -141.71, 28.09 | 295.61, 92.98 | -69.61, -22.8 | in-in | in | 7.772 | Saltbr-in | 2.871 | HRD-in | -73.25, -48.81 | 76.52, 2.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.829 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -99.1, 4.52 | APE9-dihe-in | -69.5, 129.84 | APE8-dihe-in | -77.86, 81.49 | APE8-rot-na | 30.22 | APE67-dihe-in | -79.56, -5.41 | -59.51, -27.49 | APE12-dist-na | 10.755 | APE11-dist-na | 11.055 | APE10-dist-na | 6.707 | APE9-dist-in | 5.595 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.171 | 0.214 | A | 290 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 3eyg | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 3EYHA | P23458 | 865 | 1154 | 1154.0 | IZA:2001 | Type1 | Inactive | DFGin | 6.711 | 13.778 | ABAminus | -123.79, 5.59 | -151.26, 147.61 | -137.78, 30.19 | 296.78, 89.6 | -63.64, -28.15 | in-in | in | 7.741 | Saltbr-in | 2.88 | HRD-in | -74.82, -42.99 | 68.23, 5.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.799 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -136.22, 60.46 | APE9-dihe-in | -76.43, 138.22 | APE8-dihe-in | -79.32, 79.81 | APE8-rot-na | 29.32 | APE67-dihe-in | -73.68, -7.92 | -57.92, -30.28 | APE12-dist-na | 10.347 | APE11-dist-na | 10.995 | APE10-dist-na | 9.051 | APE9-dist-in | 5.572 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.178 | 0.237 | A | 290 | 287 | 3 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 3eyh | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5E1EB | P23458 | 865 | 1154 | 1154.0 | 5JG:1201 | Type1 | Inactive | DFGin | 6.615 | 13.703 | ABAminus | -133.31, 28.19 | -149.71, 114.81 | -114.53, 26.1 | 291.32, 84.42 | -63.72, -24.05 | in-in | in | 7.765 | Saltbr-in | 2.784 | HRD-in | -74.91, -42.75 | 64.28, 0.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.801 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.64, 38.4 | APE9-dihe-in | -74.25, 132.21 | APE8-dihe-in | -79.08, 75.2 | APE8-rot-na | 22.34 | APE67-dihe-in | -75.56, -2.49 | -52.66, -36.06 | APE12-dist-na | 10.857 | APE11-dist-na | 13.311 | APE10-dist-na | 10.039 | APE9-dist-in | 6.874 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.3 | 0.227 | 0.268 | B | 290 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5e1e | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6AAHA | P23458 | 865 | 1154 | 1154.0 | 9T6:1201 | Type1 | Inactive | DFGin | 6.319 | 13.457 | ABAminus | -111.86, -1.07 | -147.59, 142.74 | -130.77, 31.7 | 296.21, 81.89 | -59.29, -31.87 | in-in | in | 7.837 | Saltbr-in | 2.785 | HRD-in | -79.04, -51.9 | 74.79, 8.24 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.804 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.78, 24.87 | APE9-dihe-in | -65.36, 146.43 | APE8-dihe-in | -84.69, 80.23 | APE8-rot-na | 32.65 | APE67-dihe-in | -73.6, -4.54 | -60.24, -33.63 | APE12-dist-na | 10.501 | APE11-dist-na | 13.066 | APE10-dist-na | 9.901 | APE9-dist-in | 6.422 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.83 | 0.225 | 0.255 | A | 290 | 285 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6aah | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6AAHB | P23458 | 865 | 1154 | 1154.0 | 9T6:1201 | Type1 | Inactive | DFGin | 6.462 | 13.588 | ABAminus | -114.68, 9.66 | -151.81, 133.96 | -131.35, 23.59 | 291.95, 87.28 | -61.54, -23.21 | in-in | in | 8.041 | Saltbr-in | 2.614 | HRD-in | -74.7, -48.84 | 74.08, 5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.783 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -85.14, 67.65 | APE9-dihe-in | -109.05, 132.69 | APE8-dihe-in | -79.19, 76.3 | APE8-rot-na | 35.14 | APE67-dihe-in | -76.24, -3.1 | -57.7, -33.14 | APE12-dist-na | 10.191 | APE11-dist-na | 12.461 | APE10-dist-na | 9.141 | APE9-dist-in | 6.543 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.83 | 0.225 | 0.255 | B | 290 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6aah | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6TPEA | P23458 | 864 | 1153 | 1154.0 | NTW:1201 | Type1 | Inactive | DFGin | 6.452 | 13.452 | ABAminus | -113.52, 27.97 | -159.85, 137.75 | -139.89, 37.69 | 300.95, 90.85 | -70.73, -32.53 | in-in | in | 7.984 | Saltbr-in | 2.898 | HRD-in | -77.39, -48.43 | 67.11, 20.0 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.721 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.39, 82.51 | APE9-dihe-in | -109.84, 138.7 | APE8-dihe-in | -71.54, 85.2 | APE8-rot-na | 346.93 | APE67-dihe-in | -79.64, -10.25 | -64.68, -30.27 | APE12-dist-na | 10.125 | APE11-dist-na | 12.13 | APE10-dist-na | 10.498 | APE9-dist-in | 6.452 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.87 | 0.249 | 0.298 | A | 291 | 283 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6tpe | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6TPEB | P23458 | 864 | 1154 | 1154.0 | NTW:1201 | Type1 | Inactive | DFGin | 6.449 | 13.462 | ABAminus | -113.4, 27.83 | -159.97, 137.64 | -139.8, 37.79 | 300.87, 90.88 | -70.61, -32.51 | in-in | in | 7.994 | Saltbr-in | 2.893 | HRD-in | -77.28, -48.49 | 67.12, 19.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.723 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -109.48, 82.82 | APE9-dihe-in | -109.8, 138.58 | APE8-dihe-in | -71.3, 85.03 | APE8-rot-na | 346.96 | APE67-dihe-in | -79.6, -10.33 | -64.53, -30.29 | APE12-dist-na | 10.133 | APE11-dist-na | 12.13 | APE10-dist-na | 10.513 | APE9-dist-in | 6.453 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.87 | 0.249 | 0.298 | B | 291 | 283 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6tpe | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6TPFA | P23458 | 864 | 1153 | 1154.0 | NTQ:1201 | Type1 | Inactive | DFGin | 6.549 | 13.566 | ABAminus | -112.13, 4.42 | -147.17, 134.74 | -132.51, 36.57 | 297.52, 87.9 | -61.56, -38.59 | in-in | in | 7.907 | Saltbr-in | 2.723 | HRD-in | -81.26, -43.5 | 66.58, 8.45 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.755 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.97, 47.61 | APE9-dihe-in | -75.75, 153.17 | APE8-dihe-in | -82.59, 85.83 | APE8-rot-na | 32.54 | APE67-dihe-in | -74.51, -8.6 | -66.85, -35.11 | APE12-dist-na | 10.951 | APE11-dist-na | 12.702 | APE10-dist-na | 10.945 | APE9-dist-in | 6.702 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.31 | 0.266 | 0.327 | A | 291 | 288 | 2 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6tpf | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6TPFB | P23458 | 865 | 1153 | 1154.0 | NTQ:1201 | Type1 | Inactive | DFGin | 6.516 | 13.607 | ABAminus | -112.38, 6.69 | -146.72, 134.6 | -130.81, 35.94 | 297.58, 85.61 | -65.62, -37.25 | in-in | in | 7.843 | Saltbr-in | 2.72 | HRD-in | -83.36, -42.45 | 66.49, 9.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.762 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 46.13, 45.8 | APE9-dihe-in | -71.68, 152.43 | APE8-dihe-in | -82.66, 85.94 | APE8-rot-na | 32.5 | APE67-dihe-in | -74.85, -9.43 | -66.05, -35.76 | APE12-dist-na | 10.968 | APE11-dist-na | 12.342 | APE10-dist-na | 11.419 | APE9-dist-in | 6.666 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.31 | 0.266 | 0.327 | B | 291 | 278 | 11 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6tpf | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6GGHA | P23458 | 865 | 1154 | 1154.0 | EYQ:1201 | Type1 | Inactive | DFGin | 6.474 | 13.708 | ABAminus | -120.02, -5.29 | -148.47, 136.5 | -125.28, 25.35 | 294.61, 85.16 | -56.12, -34.28 | in-in | in | 7.718 | Saltbr-in | 2.591 | HRD-in | -74.74, -47.68 | 65.51, 13.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.766 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 52.1, 57.9 | APE9-dihe-in | -80.13, 145.81 | APE8-dihe-in | -79.99, 78.75 | APE8-rot-na | 31.21 | APE67-dihe-in | -74.16, -4.73 | -59.55, -32.45 | APE12-dist-na | 10.105 | APE11-dist-na | 9.884 | APE10-dist-na | 9.981 | APE9-dist-in | 6.106 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.7 | 0.192 | 0.262 | A | 292 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6ggh | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6GGHB | P23458 | 863 | 1154 | 1154.0 | EYQ:1201 | Type1 | Inactive | DFGin | 6.393 | 13.885 | ABAminus | -111.86, -4.02 | -150.16, 140.27 | -128.87, 25.84 | 291.88, 86.63 | -62.88, -36.22 | in-in | in | 7.795 | Saltbr-in | 2.592 | HRD-in | -72.53, -48.04 | 68.9, 11.02 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.789 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 72.16, 30.7 | APE9-dihe-in | -88.91, 131.65 | APE8-dihe-in | -78.72, 80.52 | APE8-rot-na | 31.53 | APE67-dihe-in | -73.31, -5.76 | -61.33, -30.45 | APE12-dist-na | 10.287 | APE11-dist-na | 10.652 | APE10-dist-na | 8.339 | APE9-dist-in | 5.994 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.7 | 0.192 | 0.262 | B | 292 | 282 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6ggh | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.8 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6ELRA | P23458 | 854 | 1154 | 1154.0 | BFK:1201 | Type1 | Inactive | DFGin | 6.597 | 13.599 | ABAminus | -108.66, 4.92 | -152.97, 140.13 | -131.61, 26.62 | 294.97, 83.84 | -57.45, -30.06 | in-in | in | 7.779 | Saltbr-in | 2.741 | HRD-in | -71.99, -47.83 | 69.61, 1.99 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.831 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.35, 32.0 | APE9-dihe-in | -64.21, 131.29 | APE8-dihe-in | -79.64, 72.85 | APE8-rot-na | 28.8 | APE67-dihe-in | -76.69, -6.06 | -50.77, -33.65 | APE12-dist-na | 10.934 | APE11-dist-na | 12.929 | APE10-dist-na | 9.919 | APE9-dist-in | 6.838 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.182 | 0.205 | A | 301 | 289 | 12 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6elr | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6ELRB | P23458 | 865 | 1154 | 1154.0 | BFK:1201 | Type1 | Inactive | DFGin | 6.601 | 13.531 | ABAminus | -109.26, 5.99 | -154.04, 139.83 | -131.25, 27.64 | 294.03, 83.78 | -58.7, -28.76 | in-in | in | 7.739 | Saltbr-in | 2.752 | HRD-in | -72.31, -47.94 | 70.47, 1.78 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.838 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.07, 32.45 | APE9-dihe-in | -65.92, 131.99 | APE8-dihe-in | -78.37, 73.16 | APE8-rot-na | 28.72 | APE67-dihe-in | -77.26, -5.72 | -51.85, -33.17 | APE12-dist-na | 11.057 | APE11-dist-na | 13.148 | APE10-dist-na | 10.069 | APE9-dist-in | 6.853 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.182 | 0.205 | B | 301 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6elr | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6SM8B | P23458 | 865 | 1154 | 1154.0 | LKT:61201 | Type1 | Inactive | DFGin | 6.806 | 13.668 | ABAminus | -102.82, -5.52 | -148.54, 142.3 | -131.39, 24.74 | 291.91, 87.01 | -56.81, -29.39 | in-in | in | 7.801 | Saltbr-in | 2.711 | HRD-in | -72.52, -51.3 | 71.87, 8.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.832 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.32, 29.21 | APE9-dihe-in | -64.29, 137.39 | APE8-dihe-in | -82.59, 73.84 | APE8-rot-na | 28.56 | APE67-dihe-in | -76.5, -2.32 | -51.19, -31.92 | APE12-dist-na | 11.521 | APE11-dist-na | 13.343 | APE10-dist-na | 10.329 | APE9-dist-in | 6.67 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.85 | 0.213 | 0.241 | B | 301 | 284 | 6 | 0 | 0 | 2 | [[583, 847], [875, 1151]] | 2.0 | 6sm8 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6SMBA | P23458 | 863 | 1153 | 1154.0 | LKQ:1201 | Type1 | Inactive | DFGin | 6.607 | 13.731 | ABAminus | -104.09, 12.38 | -161.47, 134.46 | -125.84, 26.47 | 298.3, 80.99 | -58.62, -24.17 | in-in | in | 7.831 | Saltbr-in | 2.643 | HRD-in | -73.47, -45.53 | 65.45, 5.36 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.749 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -94.53, 41.14 | APE9-dihe-in | -70.01, 131.09 | APE8-dihe-in | -75.02, 72.06 | APE8-rot-na | 25.33 | APE67-dihe-in | -73.28, -2.79 | -51.04, -36.86 | APE12-dist-na | 12.02 | APE11-dist-na | 12.716 | APE10-dist-na | 10.235 | APE9-dist-in | 6.755 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.04 | 0.224 | 0.265 | A | 301 | 288 | 3 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6smb | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6SMBB | P23458 | 863 | 1153 | 1154.0 | LKQ:1201 | Type1 | Inactive | DFGin | 6.618 | 13.811 | ABAminus | -106.29, 15.46 | -163.61, 135.62 | -126.74, 26.38 | 298.65, 81.43 | -58.83, -23.63 | in-in | in | 7.869 | Saltbr-in | 2.627 | HRD-in | -72.91, -46.19 | 66.2, 3.06 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.745 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 76.78, 22.71 | APE9-dihe-in | -68.31, 133.01 | APE8-dihe-in | -75.13, 72.89 | APE8-rot-na | 25.36 | APE67-dihe-in | -72.9, -3.33 | -50.86, -36.85 | APE12-dist-na | 10.831 | APE11-dist-na | 12.575 | APE10-dist-na | 10.456 | APE9-dist-in | 6.68 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.04 | 0.224 | 0.265 | B | 301 | 282 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6smb | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.1e-87 | 298.7 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4E4LA | P23458 | 865 | 1154 | 1154.0 | 0NH:1201 | Type1 | Inactive | DFGin | 6.506 | 13.593 | ABAminus | -113.26, 1.55 | -155.7, 141.31 | -133.96, 30.85 | 296.7, 84.55 | -61.93, -29.15 | in-in | in | 7.728 | Saltbr-in | 2.366 | HRD-in | -82.62, -51.73 | 77.35, 2.42 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.833 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.62, 29.91 | APE9-dihe-in | -55.83, 134.62 | APE8-dihe-in | -77.55, 77.11 | APE8-rot-na | 23.92 | APE67-dihe-in | -76.85, -4.17 | -58.31, -32.93 | APE12-dist-na | 11.099 | APE11-dist-na | 12.761 | APE10-dist-na | 10.348 | APE9-dist-in | 6.603 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.19 | 0.228 | A | 302 | 279 | 11 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4l | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4E4LB | P23458 | 864 | 1154 | 1154.0 | 0NH:1201 | Type1 | Inactive | DFGin | 6.468 | 13.69 | ABAminus | -115.34, 5.94 | -154.23, 143.98 | -136.31, 29.8 | 294.89, 85.73 | -63.4, -28.12 | in-in | in | 7.872 | Saltbr-in | 2.625 | HRD-in | -80.23, -45.9 | 70.61, 1.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.75 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -105.56, 32.84 | APE9-dihe-in | -59.39, 139.65 | APE8-dihe-in | -81.36, 75.53 | APE8-rot-na | 28.93 | APE67-dihe-in | -77.55, -4.05 | -62.31, -27.51 | APE12-dist-na | 10.995 | APE11-dist-na | 12.667 | APE10-dist-na | 10.069 | APE9-dist-in | 6.632 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.19 | 0.228 | B | 302 | 281 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4l | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4E4LD | P23458 | 864 | 1154 | 1154.0 | 0NH:1201 | Type1 | Inactive | DFGin | 6.536 | 13.748 | ABAminus | -114.27, -0.81 | -153.61, 143.22 | -135.12, 28.03 | 293.73, 85.38 | -57.66, -27.04 | in-in | in | 7.741 | Saltbr-in | 2.555 | HRD-in | -77.01, -53.08 | 75.86, 4.71 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.823 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -115.68, 33.68 | APE9-dihe-in | -65.48, 130.64 | APE8-dihe-in | -74.63, 79.76 | APE8-rot-na | 26.43 | APE67-dihe-in | -75.57, -2.67 | -62.18, -32.34 | APE12-dist-na | 11.513 | APE11-dist-na | 12.875 | APE10-dist-na | 10.415 | APE9-dist-in | 6.7 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.0 | 0.19 | 0.228 | D | 302 | 283 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4l | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4E4NA | P23458 | 854 | 1154 | 1154.0 | 0NL:61201 | Type1 | Inactive | DFGin | 6.384 | 13.56 | ABAminus | -120.02, 11.21 | -158.48, 139.99 | -136.43, 26.78 | 297.09, 85.57 | -63.39, -21.4 | in-in | in | 7.79 | Saltbr-in | 2.555 | HRD-in | -80.31, -49.85 | 72.5, 4.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.848 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -96.76, 48.8 | APE9-dihe-in | -75.99, 139.57 | APE8-dihe-in | -78.93, 73.17 | APE8-rot-na | 33.7 | APE67-dihe-in | -74.47, -3.41 | -60.94, -30.72 | APE12-dist-na | 11.071 | APE11-dist-na | 12.756 | APE10-dist-na | 10.411 | APE9-dist-in | 6.832 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.183 | 0.226 | A | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4n | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4E4NB | P23458 | 865 | 1154 | 1154.0 | 0NL:61201 | Type1 | Inactive | DFGin | 6.346 | 13.502 | ABAminus | -119.9, 9.63 | -155.68, 139.61 | -133.8, 28.11 | 297.19, 80.43 | -62.66, -24.74 | in-in | in | 7.737 | Saltbr-in | 2.603 | HRD-in | -78.32, -48.47 | 74.25, 0.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.874 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.54, 49.17 | APE9-dihe-in | -76.21, 142.06 | APE8-dihe-in | -79.22, 71.62 | APE8-rot-na | 25.59 | APE67-dihe-in | -77.0, -5.97 | -60.76, -27.4 | APE12-dist-na | 11.162 | APE11-dist-na | 12.793 | APE10-dist-na | 10.433 | APE9-dist-in | 6.939 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.183 | 0.226 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e4n | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4E5WA | P23458 | 854 | 1154 | 1154.0 | 0NT:61201 | Type1 | Inactive | DFGin | 6.562 | 13.397 | ABAminus | -118.14, 5.18 | -153.89, 137.32 | -129.51, 26.76 | 295.21, 88.69 | -58.94, -26.21 | in-in | in | 7.704 | Saltbr-in | 2.687 | HRD-in | -73.36, -50.75 | 70.96, 2.6 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.834 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.84, 26.34 | APE9-dihe-in | -57.31, 135.68 | APE8-dihe-in | -78.98, 72.49 | APE8-rot-na | 27.03 | APE67-dihe-in | -72.09, -3.1 | -47.71, -39.24 | APE12-dist-na | 11.088 | APE11-dist-na | 13.57 | APE10-dist-na | 10.45 | APE9-dist-in | 6.738 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.86 | 0.184 | 0.21 | A | 302 | 293 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4e5w | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4E5WB | P23458 | 865 | 1153 | 1154.0 | 0NT:61202 | Type1 | Inactive | DFGin | 6.53 | 13.35 | ABAminus | -114.8, 7.46 | -153.87, 137.96 | -129.8, 26.64 | 296.41, 93.24 | -58.91, -27.51 | in-in | in | 7.691 | Saltbr-in | 2.687 | HRD-in | -74.04, -50.94 | 71.65, 3.46 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.833 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.41, 26.14 | APE9-dihe-in | -57.59, 134.48 | APE8-dihe-in | -78.71, 72.64 | APE8-rot-na | 26.79 | APE67-dihe-in | -72.94, -2.19 | -48.23, -38.49 | APE12-dist-na | 11.113 | APE11-dist-na | 13.557 | APE10-dist-na | 10.431 | APE9-dist-in | 6.758 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.86 | 0.184 | 0.21 | B | 302 | 280 | 9 | 0 | 0 | 2 | [[583, 847], [875, 1151]] | 2.0 | 4e5w | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4EHZA | P23458 | 858 | 1154 | 1154.0 | JAK:1201 | Type1 | Inactive | DFGin | 6.295 | 13.63 | ABAminus | -122.46, 12.74 | -158.91, 149.59 | -139.33, 23.83 | 295.89, 89.08 | -61.4, -20.25 | in-in | in | 7.795 | Saltbr-in | 2.936 | HRD-in | -79.41, -51.26 | 80.05, -0.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.866 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -94.49, 24.25 | APE9-dihe-in | -61.79, 133.39 | APE8-dihe-in | -76.86, 73.91 | APE8-rot-na | 30.52 | APE67-dihe-in | -75.94, -6.94 | -60.76, -27.83 | APE12-dist-na | 11.438 | APE11-dist-na | 13.16 | APE10-dist-na | 9.871 | APE9-dist-in | 7.032 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.174 | 0.174 | 0.229 | A | 302 | 292 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ehz | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4EHZB | P23458 | 865 | 1154 | 1154.0 | JAK:1201 | Type1 | Inactive | DFGin | 6.317 | 13.73 | ABAminus | -116.35, 3.51 | -150.61, 148.16 | -138.87, 32.34 | 292.95, 86.02 | -67.41, -23.21 | in-in | in | 7.869 | Saltbr-in | 2.763 | HRD-in | -83.57, -44.01 | 70.15, -1.08 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.733 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.9, 29.19 | APE9-dihe-in | -67.89, 136.88 | APE8-dihe-in | -75.68, 68.81 | APE8-rot-na | 33.04 | APE67-dihe-in | -71.9, -6.58 | -49.99, -36.99 | APE12-dist-na | 11.419 | APE11-dist-na | 13.393 | APE10-dist-na | 10.125 | APE9-dist-in | 6.991 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.174 | 0.174 | 0.229 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ehz | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4EHZC | P23458 | 866 | 1154 | 1154.0 | JAK:1201 | Type1 | Inactive | DFGin | 6.317 | 13.621 | ABAminus | -118.15, 8.14 | -148.22, 154.09 | -141.74, 25.14 | 292.74, 84.54 | -60.05, -18.24 | in-in | in | 7.859 | Saltbr-in | 2.84 | HRD-in | -77.85, -48.09 | 78.3, 3.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.724 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.81, 30.11 | APE9-dihe-in | -57.01, 145.43 | APE8-dihe-in | -85.32, 74.95 | APE8-rot-na | 31.15 | APE67-dihe-in | -74.27, -3.28 | -56.74, -31.49 | APE12-dist-na | 10.975 | APE11-dist-na | 13.004 | APE10-dist-na | 10.18 | APE9-dist-in | 6.676 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.174 | 0.174 | 0.229 | C | 302 | 280 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ehz | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4EHZD | P23458 | 865 | 1154 | 1154.0 | JAK:1201 | Type1 | Inactive | DFGin | 6.428 | 13.533 | ABAminus | -123.86, 16.47 | -158.34, 146.22 | -137.38, 32.15 | 296.06, 77.8 | -67.83, -20.15 | in-in | in | 7.679 | Saltbr-in | 3.0 | HRD-in | -85.88, -43.73 | 70.18, 7.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.38, 26.48 | APE9-dihe-in | -59.77, 138.32 | APE8-dihe-in | -81.72, 74.58 | APE8-rot-na | 32.67 | APE67-dihe-in | -77.67, -4.82 | -52.47, -31.56 | APE12-dist-na | 11.043 | APE11-dist-na | 12.962 | APE10-dist-na | 10.009 | APE9-dist-in | 6.688 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.174 | 0.174 | 0.229 | D | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ehz | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4EI4A | P23458 | 854 | 1154 | 1154.0 | 0Q2:61201 | Type1 | Inactive | DFGin | 6.362 | 13.452 | ABAminus | -125.08, 21.55 | -162.93, 136.7 | -132.47, 29.54 | 298.16, 82.51 | -65.62, -22.07 | in-in | in | 7.843 | Saltbr-in | 2.612 | HRD-in | -82.16, -48.37 | 72.58, 5.29 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.744 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -105.53, 42.94 | APE9-dihe-in | -71.49, 136.49 | APE8-dihe-in | -77.62, 74.63 | APE8-rot-na | 31.88 | APE67-dihe-in | -76.69, -5.39 | -62.91, -28.92 | APE12-dist-na | 10.983 | APE11-dist-na | 12.753 | APE10-dist-na | 10.259 | APE9-dist-in | 6.784 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.22 | 0.202 | 0.239 | A | 302 | 290 | 11 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ei4 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4EI4B | P23458 | 865 | 1154 | 1154.0 | 0Q2:61201 | Type1 | Inactive | DFGin | 6.382 | 13.518 | ABAminus | -120.19, 16.13 | -160.02, 140.78 | -136.52, 31.88 | 292.39, 84.5 | -65.63, -28.61 | in-in | in | 7.853 | Saltbr-in | 2.827 | HRD-in | -84.06, -46.22 | 68.02, 6.16 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.752 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.4, 38.28 | APE9-dihe-in | -67.47, 135.5 | APE8-dihe-in | -75.19, 75.25 | APE8-rot-na | 28.78 | APE67-dihe-in | -75.9, -4.89 | -57.78, -34.83 | APE12-dist-na | 11.055 | APE11-dist-na | 12.687 | APE10-dist-na | 10.236 | APE9-dist-in | 6.789 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.22 | 0.202 | 0.239 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ei4 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4FK6A | P23458 | 863 | 1154 | 1154.0 | 0UJ:1201 | Type1 | Inactive | DFGin | 6.577 | 13.413 | ABAminus | -112.19, 2.74 | -147.97, 135.94 | -128.79, 22.38 | 293.74, 90.76 | -52.95, -29.36 | in-in | in | 7.654 | Saltbr-in | 2.674 | HRD-in | -73.71, -49.95 | 70.6, -2.02 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.81 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.7, 28.56 | APE9-dihe-in | -63.18, 134.95 | APE8-dihe-in | -78.74, 77.08 | APE8-rot-na | 27.11 | APE67-dihe-in | -76.1, -2.34 | -51.26, -33.75 | APE12-dist-na | 11.32 | APE11-dist-na | 12.856 | APE10-dist-na | 10.101 | APE9-dist-in | 6.646 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.211 | 0.251 | A | 302 | 287 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4fk6 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4FK6B | P23458 | 864 | 1154 | 1154.0 | 0UJ:1201 | Type1 | Inactive | DFGin | 6.594 | 13.406 | ABAminus | -112.12, 2.82 | -147.85, 135.79 | -128.94, 22.08 | 293.63, 90.77 | -52.49, -30.06 | in-in | in | 7.638 | Saltbr-in | 2.679 | HRD-in | -73.35, -50.23 | 70.8, -1.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.817 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.94, 28.16 | APE9-dihe-in | -62.61, 135.05 | APE8-dihe-in | -78.72, 77.07 | APE8-rot-na | 27.01 | APE67-dihe-in | -76.01, -2.17 | -51.54, -33.82 | APE12-dist-na | 11.313 | APE11-dist-na | 12.766 | APE10-dist-na | 10.141 | APE9-dist-in | 6.647 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.211 | 0.251 | B | 302 | 286 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4fk6 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4I5CA | P23458 | 865 | 1154 | 1154.0 | C5I:61201 | Type1 | Inactive | DFGin | 6.372 | 13.098 | ABAminus | -114.74, 13.12 | -159.95, 138.51 | -132.46, 27.57 | 300.19, 86.09 | -57.95, -29.46 | in-in | in | 7.648 | Saltbr-in | 2.663 | HRD-in | -72.51, -44.79 | 66.5, 0.54 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.903 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -124.02, 33.91 | APE9-dihe-in | -66.46, 131.24 | APE8-dihe-in | -75.55, 75.28 | APE8-rot-na | 31.15 | APE67-dihe-in | -75.41, -9.49 | -50.0, -34.68 | APE12-dist-na | 11.26 | APE11-dist-na | 13.341 | APE10-dist-na | 10.194 | APE9-dist-in | 6.774 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.1 | 0.193 | 0.245 | A | 302 | 281 | 9 | 0 | 0 | 1 | [[583, 847], [875, 1151]] | 2.0 | 4i5c | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4I5CB | P23458 | 854 | 1154 | 1154.0 | C5I:61205 | Type1 | Inactive | DFGin | 6.288 | 13.062 | ABAminus | -117.66, 20.22 | -158.68, 137.22 | -131.37, 22.03 | 299.16, 87.56 | -52.78, -31.38 | in-in | in | 7.784 | Saltbr-in | 2.586 | HRD-in | -74.37, -52.31 | 71.43, 0.95 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.948 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -101.41, 21.23 | APE9-dihe-in | -58.7, 133.33 | APE8-dihe-in | -78.45, 70.87 | APE8-rot-na | 28.87 | APE67-dihe-in | -73.75, -3.17 | -47.7, -37.18 | APE12-dist-na | 11.146 | APE11-dist-na | 13.194 | APE10-dist-na | 10.032 | APE9-dist-in | 6.84 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.1 | 0.193 | 0.245 | B | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4i5c | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4IVBA | P23458 | 854 | 1154 | 1154.0 | 1J5:61201 | Type1 | Inactive | DFGin | 6.446 | 13.398 | ABAminus | -120.37, 8.79 | -154.43, 145.03 | -134.59, 25.95 | 296.41, 85.72 | -59.41, -26.27 | in-in | in | 7.777 | Saltbr-in | 2.607 | HRD-in | -81.27, -49.76 | 73.46, 5.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.901 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.65, 36.69 | APE9-dihe-in | -67.09, 139.5 | APE8-dihe-in | -78.95, 74.88 | APE8-rot-na | 31.26 | APE67-dihe-in | -75.42, -5.51 | -58.71, -32.55 | APE12-dist-na | 11.215 | APE11-dist-na | 12.935 | APE10-dist-na | 10.311 | APE9-dist-in | 6.781 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.183 | 0.221 | A | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivb | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4IVBB | P23458 | 865 | 1154 | 1154.0 | 1J5:61201 | Type1 | Inactive | DFGin | 6.429 | 13.415 | ABAminus | -116.62, 7.74 | -154.57, 143.33 | -132.65, 26.65 | 294.75, 85.72 | -57.0, -32.17 | in-in | in | 7.713 | Saltbr-in | 2.651 | HRD-in | -82.29, -46.68 | 69.34, 6.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.895 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.2, 32.35 | APE9-dihe-in | -63.44, 138.0 | APE8-dihe-in | -78.25, 77.26 | APE8-rot-na | 32.13 | APE67-dihe-in | -75.77, -2.93 | -62.98, -29.79 | APE12-dist-na | 11.263 | APE11-dist-na | 12.983 | APE10-dist-na | 10.306 | APE9-dist-in | 6.769 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.9 | 0.183 | 0.221 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivb | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4IVCA | P23458 | 854 | 1154 | 1154.0 | 1J6:61201 | Type1 | Inactive | DFGin | 6.249 | 13.251 | ABAminus | -114.51, 9.81 | -157.21, 145.73 | -138.3, 37.36 | 304.45, 81.48 | -64.22, -30.51 | in-in | in | 7.826 | Saltbr-in | 2.692 | HRD-in | -91.76, -42.16 | 67.22, -0.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.842 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.76, 45.97 | APE9-dihe-in | -72.9, 142.32 | APE8-dihe-in | -77.97, 76.61 | APE8-rot-na | 30.79 | APE67-dihe-in | -73.52, -3.32 | -54.87, -39.45 | APE12-dist-na | 11.192 | APE11-dist-na | 12.652 | APE10-dist-na | 10.171 | APE9-dist-in | 6.549 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.35 | 0.2 | 0.263 | A | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivc | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4IVCB | P23458 | 865 | 1154 | 1154.0 | 1J6:61201 | Type1 | Inactive | DFGin | 6.313 | 13.347 | ABAminus | -119.67, 6.43 | -149.04, 145.44 | -134.49, 29.55 | 297.17, 82.22 | -60.5, -32.79 | in-in | in | 7.525 | Saltbr-in | 2.277 | HRD-in | -89.31, -45.09 | 71.21, 3.65 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.717 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -101.71, 20.54 | APE9-dihe-in | -65.21, 135.06 | APE8-dihe-in | -79.05, 83.59 | APE8-rot-na | 28.99 | APE67-dihe-in | -78.13, -7.38 | -62.67, -27.87 | APE12-dist-na | 11.123 | APE11-dist-na | 12.804 | APE10-dist-na | 9.574 | APE9-dist-in | 6.607 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.35 | 0.2 | 0.263 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivc | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4IVDA | P23458 | 854 | 1154 | 1154.0 | 15T:61201 | Type1 | Inactive | DFGin | 6.309 | 13.304 | ABAminus | -118.43, 8.35 | -154.11, 148.17 | -137.65, 24.48 | 298.46, 83.68 | -55.12, -27.34 | in-in | in | 7.749 | Saltbr-in | 2.729 | HRD-in | -85.26, -46.42 | 71.64, 5.83 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.903 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -118.71, 33.92 | APE9-dihe-in | -63.4, 140.18 | APE8-dihe-in | -80.26, 75.71 | APE8-rot-na | 32.55 | APE67-dihe-in | -74.69, -4.74 | -58.39, -31.37 | APE12-dist-na | 11.247 | APE11-dist-na | 12.97 | APE10-dist-na | 10.268 | APE9-dist-in | 6.655 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.93 | 0.204 | 0.247 | A | 302 | 291 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivd | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4IVDB | P23458 | 865 | 1154 | 1154.0 | 15T:61201 | Type1 | Inactive | DFGin | 6.411 | 13.37 | ABAminus | -112.55, 2.72 | -159.22, 144.81 | -135.21, 28.45 | 296.48, 84.97 | -57.15, -29.77 | in-in | in | 7.676 | Saltbr-in | 2.745 | HRD-in | -84.66, -44.43 | 68.53, 7.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.922 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.94, 35.04 | APE9-dihe-in | -66.46, 139.38 | APE8-dihe-in | -79.29, 77.36 | APE8-rot-na | 30.63 | APE67-dihe-in | -76.81, -5.82 | -62.53, -27.62 | APE12-dist-na | 11.221 | APE11-dist-na | 12.974 | APE10-dist-na | 10.244 | APE9-dist-in | 6.666 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.93 | 0.204 | 0.247 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4ivd | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4K6ZA | P23458 | 865 | 1154 | 1154.0 | 1Q3:1201 | Type1 | Inactive | DFGin | 6.368 | 13.629 | ABAminus | -111.25, 5.81 | -148.16, 138.39 | -130.89, 30.06 | 299.5, 88.49 | -54.29, -32.58 | in-in | in | 8.161 | Saltbr-in | 2.913 | HRD-in | -64.09, -54.55 | 67.8, 5.15 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.82 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.94, 36.35 | APE9-dihe-in | -67.0, 125.07 | APE8-dihe-in | -75.83, 85.59 | APE8-rot-na | 25.89 | APE67-dihe-in | -67.06, -19.07 | -53.74, -42.35 | APE12-dist-na | 10.425 | APE11-dist-na | 12.583 | APE10-dist-na | 10.007 | APE9-dist-in | 6.016 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.73 | 0.244 | 0.297 | A | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4k6z | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4K77A | P23458 | 864 | 1154 | 1154.0 | 1Q4:1201 | Type1 | Inactive | DFGin | 6.256 | 13.464 | ABAminus | -120.21, 6.98 | -152.33, 140.1 | -135.8, 29.32 | 300.23, 84.02 | -66.83, -17.3 | in-in | in | 8.042 | Saltbr-in | 2.62 | HRD-in | -83.59, -46.77 | 75.55, -1.36 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.807 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.78, 30.95 | APE9-dihe-in | -65.86, 137.27 | APE8-dihe-in | -79.1, 74.56 | APE8-rot-na | 31.39 | APE67-dihe-in | -73.63, -7.17 | -57.69, -30.82 | APE12-dist-na | 11.18 | APE11-dist-na | 12.795 | APE10-dist-na | 9.921 | APE9-dist-in | 6.75 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.4 | 0.193 | 0.251 | A | 302 | 284 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4k77 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 4K77B | P23458 | 865 | 1154 | 1154.0 | 1Q4:1201 | Type1 | Inactive | DFGin | 6.282 | 13.504 | ABAminus | -120.68, 0.99 | -147.42, 142.05 | -133.88, 36.74 | 297.84, 83.5 | -67.02, -18.72 | in-in | in | 7.948 | Saltbr-in | 2.922 | HRD-in | -85.03, -50.83 | 74.8, -3.74 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.726 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -112.68, 47.05 | APE9-dihe-in | -77.0, 143.68 | APE8-dihe-in | -79.91, 78.18 | APE8-rot-na | 30.27 | APE67-dihe-in | -77.76, -4.87 | -65.15, -27.78 | APE12-dist-na | 11.137 | APE11-dist-na | 12.726 | APE10-dist-na | 10.167 | APE9-dist-in | 6.81 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.4 | 0.193 | 0.251 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 4k77 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5HX8A | P23458 | 855 | 1154 | 1154.0 | 66P:1201 | Type1 | Inactive | DFGin | 6.449 | 13.688 | ABAminus | -102.8, 8.3 | -149.54, 137.76 | -131.57, 23.74 | 295.19, 87.44 | -55.43, -25.96 | in-in | in | 7.925 | Saltbr-in | 2.761 | HRD-in | -74.69, -48.9 | 64.93, 4.52 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.727 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -103.85, 104.76 | APE9-dihe-in | -72.26, 138.18 | APE8-dihe-in | -80.27, 76.7 | APE8-rot-na | 26.46 | APE67-dihe-in | -75.94, -4.44 | -51.82, -37.01 | APE12-dist-na | 11.12 | APE11-dist-na | 12.285 | APE10-dist-na | 11.393 | APE9-dist-in | 6.611 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.199 | 0.24 | A | 302 | 293 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5hx8 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5HX8B | P23458 | 865 | 1154 | 1154.0 | 66P:1201 | Type1 | Inactive | DFGin | 6.42 | 13.631 | ABAminus | -110.45, 9.62 | -150.03, 136.28 | -131.01, 24.66 | 294.53, 92.56 | -57.47, -31.3 | in-in | in | 7.769 | Saltbr-in | 2.758 | HRD-in | -74.49, -50.24 | 68.18, -1.59 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.774 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -121.57, 40.76 | APE9-dihe-in | -71.94, 141.78 | APE8-dihe-in | -79.55, 77.3 | APE8-rot-na | 24.89 | APE67-dihe-in | -77.48, 1.58 | -49.69, -36.95 | APE12-dist-na | 10.838 | APE11-dist-na | 12.693 | APE10-dist-na | 10.86 | APE9-dist-in | 6.55 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.199 | 0.24 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5hx8 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5WO4A | P23458 | 854 | 1154 | 1154.0 | B7V:2001 | Type1 | Inactive | DFGin | 6.559 | 13.475 | ABAminus | -113.4, 5.79 | -147.65, 137.71 | -131.93, 25.73 | 295.23, 90.95 | -54.73, -30.34 | in-in | in | 7.676 | Saltbr-in | 2.754 | HRD-in | -72.7, -46.52 | 67.85, -2.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.821 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.62, 42.17 | APE9-dihe-in | -67.76, 140.08 | APE8-dihe-in | -81.09, 72.14 | APE8-rot-na | 29.77 | APE67-dihe-in | -75.22, -1.83 | -52.55, -34.79 | APE12-dist-na | 10.797 | APE11-dist-na | 12.901 | APE10-dist-na | 10.466 | APE9-dist-in | 6.823 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.84 | 0.188 | 0.211 | A | 302 | 294 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5wo4 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5WO4B | P23458 | 865 | 1154 | 1154.0 | B7V:2001 | Type1 | Inactive | DFGin | 6.55 | 13.411 | ABAminus | -111.8, 3.6 | -145.5, 139.23 | -132.92, 27.81 | 292.27, 90.98 | -57.76, -28.76 | in-in | in | 7.615 | Saltbr-in | 2.781 | HRD-in | -72.82, -49.06 | 69.56, 1.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.838 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.71, 39.74 | APE9-dihe-in | -66.32, 138.27 | APE8-dihe-in | -78.58, 73.11 | APE8-rot-na | 28.91 | APE67-dihe-in | -75.88, -0.88 | -52.5, -34.22 | APE12-dist-na | 10.866 | APE11-dist-na | 12.93 | APE10-dist-na | 10.505 | APE9-dist-in | 6.743 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.84 | 0.188 | 0.211 | B | 302 | 282 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5wo4 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6HZUA | P23458 | 854 | 1154 | 1154.0 | GYQ:61201 | Type1 | Inactive | DFGin | 6.458 | 13.248 | ABAminus | -115.79, 10.1 | -155.61, 143.2 | -135.89, 34.69 | 298.64, 85.33 | -68.92, -23.66 | in-in | in | 7.891 | Saltbr-in | 2.605 | HRD-in | -70.11, -45.53 | 64.37, 7.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.768 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -94.73, 34.76 | APE9-dihe-in | -73.48, 139.36 | APE8-dihe-in | -81.86, 74.79 | APE8-rot-na | 30.37 | APE67-dihe-in | -72.43, -9.67 | -55.59, -34.31 | APE12-dist-na | 10.967 | APE11-dist-na | 13.174 | APE10-dist-na | 9.887 | APE9-dist-in | 6.803 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.204 | 0.265 | A | 302 | 293 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6hzu | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6HZUB | P23458 | 865 | 1154 | 1154.0 | GYQ:61201 | Type1 | Inactive | DFGin | 6.443 | 13.247 | ABAminus | -119.96, 0.48 | -155.13, 140.72 | -132.65, 33.96 | 299.27, 84.27 | -60.17, -34.27 | in-in | in | 8.023 | Saltbr-in | 2.702 | HRD-in | -82.42, -47.78 | 71.93, 4.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.923 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -93.89, 29.59 | APE9-dihe-in | -63.03, 138.85 | APE8-dihe-in | -81.19, 78.97 | APE8-rot-na | 31.69 | APE67-dihe-in | -73.96, -7.04 | -62.12, -30.09 | APE12-dist-na | 11.006 | APE11-dist-na | 13.225 | APE10-dist-na | 9.885 | APE9-dist-in | 6.657 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.2 | 0.204 | 0.265 | B | 302 | 285 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6hzu | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N77A | P23458 | 866 | 1154 | 1154.0 | KEJ:1201 | Type1 | Inactive | DFGin | 6.391 | 13.654 | ABAminus | -111.17, 5.93 | -155.03, 145.91 | -137.7, 32.01 | 295.16, 86.03 | -58.79, -28.87 | in-in | in | 8.239 | Saltbr-in | 2.758 | HRD-in | -67.03, -46.69 | 67.69, -1.58 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.924 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 52.82, 53.92 | APE9-dihe-in | -90.09, 140.83 | APE8-dihe-in | -78.25, 71.6 | APE8-rot-na | 26.8 | APE67-dihe-in | -76.7, -1.13 | -52.74, -34.15 | APE12-dist-na | 11.079 | APE11-dist-na | 12.09 | APE10-dist-na | 10.994 | APE9-dist-in | 7.019 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.64 | 0.253 | 0.282 | A | 302 | 280 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n77 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N77B | P23458 | 865 | 1154 | 1154.0 | KEJ:1202 | Type1 | Inactive | DFGin | 6.447 | 13.754 | ABAminus | -112.96, 6.51 | -156.54, 142.84 | -135.02, 28.22 | 296.71, 89.38 | -58.72, -26.41 | in-in | in | 8.213 | Saltbr-in | 2.737 | HRD-in | -67.03, -48.62 | 72.63, -6.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.844 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.58, 44.0 | APE9-dihe-in | -74.12, 131.71 | APE8-dihe-in | -79.78, 70.31 | APE8-rot-na | 28.35 | APE67-dihe-in | -75.35, -3.65 | -48.14, -35.74 | APE12-dist-na | 10.934 | APE11-dist-na | 12.689 | APE10-dist-na | 9.987 | APE9-dist-in | 6.954 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.64 | 0.253 | 0.282 | B | 302 | 279 | 11 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n77 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N78A | P23458 | 866 | 1154 | 1154.0 | KEP:1201 | Type1 | Inactive | DFGin | 6.425 | 13.562 | ABAminus | -105.81, -4.17 | -146.0, 143.93 | -133.35, 28.47 | 298.42, 87.41 | -54.49, -32.74 | in-in | in | 8.377 | Saltbr-in | 2.73 | HRD-in | -68.76, -52.63 | 70.44, -3.87 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.811 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -114.29, 50.22 | APE9-dihe-in | -86.39, 131.12 | APE8-dihe-in | -82.28, 79.47 | APE8-rot-na | 24.58 | APE67-dihe-in | -76.5, -2.33 | -53.51, -34.22 | APE12-dist-na | 11.515 | APE11-dist-na | 12.037 | APE10-dist-na | 9.052 | APE9-dist-in | 6.377 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.83 | 0.236 | 0.261 | A | 302 | 277 | 12 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n78 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N79A | P23458 | 866 | 1154 | 1154.0 | KES:1201 | Type1 | Inactive | DFGin | 6.403 | 13.525 | ABAminus | -99.38, -15.25 | -133.8, 148.14 | -138.23, 25.13 | 295.77, 92.1 | -55.46, -31.57 | in-in | in | 8.295 | Saltbr-in | 2.767 | HRD-in | -74.33, -53.6 | 68.25, 4.98 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.781 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.11, 40.21 | APE9-dihe-in | -76.58, 124.37 | APE8-dihe-in | -77.77, 81.63 | APE8-rot-na | 28.13 | APE67-dihe-in | -77.42, -2.89 | -55.56, -32.1 | APE12-dist-na | 11.219 | APE11-dist-na | 11.887 | APE10-dist-na | 9.075 | APE9-dist-in | 5.964 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.27 | 0.227 | 0.27 | A | 302 | 279 | 10 | 0 | 0 | 2 | [[583, 847], [875, 1151]] | 2.0 | 6n79 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N7BA | P23458 | 865 | 1154 | 1154.0 | KEY:1201 | Type1 | Inactive | DFGin | 6.45 | 13.456 | ABAminus | -106.32, -1.48 | -152.36, 145.64 | -135.47, 28.3 | 291.96, 86.78 | -55.73, -29.48 | in-in | in | 7.736 | Saltbr-in | 2.768 | HRD-in | -71.34, -49.85 | 67.55, 5.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.806 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -113.89, 58.14 | APE9-dihe-in | -96.67, 129.96 | APE8-dihe-in | -81.34, 78.4 | APE8-rot-na | 26.42 | APE67-dihe-in | -77.54, 0.39 | -57.77, -29.15 | APE12-dist-na | 11.059 | APE11-dist-na | 11.728 | APE10-dist-na | 8.79 | APE9-dist-in | 6.369 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.81 | 0.222 | 0.264 | A | 302 | 280 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n7b | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N7CA | P23458 | 865 | 1154 | 1154.0 | KF1:1201 | Type1 | Inactive | DFGin | 6.513 | 13.509 | ABAminus | -110.36, 6.26 | -156.68, 145.17 | -136.24, 27.53 | 295.08, 89.21 | -55.95, -29.39 | in-in | in | 8.096 | Saltbr-in | 2.735 | HRD-in | -68.7, -46.37 | 70.89, -7.05 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.902 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 95.97 | APE9-dihe-in | -107.06, 147.5 | APE8-dihe-in | -79.03, 70.75 | APE8-rot-na | 27.77 | APE67-dihe-in | -74.72, -3.56 | -53.55, -33.63 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.457 | APE9-dist-in | 7.085 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.69 | 0.254 | 0.288 | A | 302 | 275 | 15 | 0 | 0 | 2 | [[583, 847], [875, 1151]] | 2.0 | 6n7c | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N7CB | P23458 | 865 | 1154 | 1154.0 | KF1:1202 | Type1 | Inactive | DFGin | 6.51 | 13.589 | ABAminus | -115.1, 6.45 | -153.47, 142.93 | -133.09, 25.34 | 294.67, 85.94 | -52.61, -29.28 | in-in | in | 8.155 | Saltbr-in | 2.753 | HRD-in | -67.82, -44.9 | 68.03, -6.1 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.861 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 138.81 | APE8-dihe-in | -80.52, 71.8 | APE8-rot-na | 28.74 | APE67-dihe-in | -72.99, -4.02 | -55.65, -32.27 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.115 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.69 | 0.254 | 0.288 | B | 302 | 273 | 17 | 0 | 0 | 4 | [[583, 847], [875, 1151]] | 2.0 | 6n7c | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N7DA | P23458 | 865 | 1154 | 1154.0 | KF4:1201 | Type1 | Inactive | DFGin | 6.476 | 13.402 | ABAminus | -110.67, 4.22 | -155.59, 141.48 | -134.23, 27.49 | 295.25, 85.51 | -53.77, -30.29 | in-in | in | 8.285 | Saltbr-in | 2.637 | HRD-in | -73.25, -49.17 | 70.77, 0.44 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.822 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.59, 31.0 | APE9-dihe-in | -83.57, 124.64 | APE8-dihe-in | -81.68, 83.11 | APE8-rot-na | 27.61 | APE67-dihe-in | -75.33, -0.8 | -58.46, -31.26 | APE12-dist-na | 11.561 | APE11-dist-na | 11.737 | APE10-dist-na | 7.584 | APE9-dist-in | 5.976 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.78 | 0.198 | 0.234 | A | 302 | 280 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n7d | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSBA | P23458 | 865 | 1154 | 1154.0 | KGZ:1201 | Type1 | Inactive | DFGin | 6.59 | 13.509 | ABAminus | -116.74, 1.69 | -150.38, 137.57 | -126.94, 22.04 | 292.38, 82.89 | -70.44, -11.55 | in-in | in | 8.107 | Saltbr-in | 2.615 | HRD-in | -82.35, -48.96 | 71.74, 9.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.845 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.58, 28.79 | APE9-dihe-in | -52.22, 132.79 | APE8-dihe-in | -77.89, 76.1 | APE8-rot-na | 36.11 | APE67-dihe-in | -73.96, -4.25 | -64.89, -26.96 | APE12-dist-na | 12.037 | APE11-dist-na | 12.29 | APE10-dist-na | 10.327 | APE9-dist-in | 6.885 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.311 | 0.354 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsb | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSBB | P23458 | 865 | 1154 | 1154.0 | KGZ:1201 | Type1 | Inactive | DFGin | 6.647 | 13.904 | ABAminus | -118.58, -5.18 | -147.32, 138.8 | -128.6, 27.58 | 293.53, 77.97 | -68.36, -16.41 | in-in | in | 8.049 | Saltbr-in | 2.707 | HRD-in | -76.09, -52.98 | 75.83, 4.99 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.959 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -104.45, 33.45 | APE9-dihe-in | -55.89, 141.48 | APE8-dihe-in | -80.12, 75.54 | APE8-rot-na | 36.76 | APE67-dihe-in | -74.19, -3.49 | -57.35, -33.46 | APE12-dist-na | 11.792 | APE11-dist-na | 12.943 | APE10-dist-na | 10.141 | APE9-dist-in | 6.851 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.311 | 0.354 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsb | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSCA | P23458 | 865 | 1154 | 1154.0 | KH5:1201 | Type1 | Inactive | DFGin | 6.554 | 13.409 | ABAminus | -117.31, 8.47 | -153.39, 137.28 | -129.48, 30.56 | 297.53, 83.92 | -65.76, -23.88 | in-in | in | 7.663 | Saltbr-in | 2.689 | HRD-in | -79.6, -49.32 | 70.06, 11.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.717 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -98.9, 27.5 | APE9-dihe-in | -67.04, 137.63 | APE8-dihe-in | -80.21, 78.36 | APE8-rot-na | 37.08 | APE67-dihe-in | -76.89, -0.21 | -62.94, -28.86 | APE12-dist-na | 11.004 | APE11-dist-na | 13.576 | APE10-dist-na | 10.231 | APE9-dist-in | 6.858 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.85 | 0.249 | 0.28 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsc | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSCB | P23458 | 865 | 1154 | 1154.0 | KH5:1201 | Type1 | Inactive | DFGin | 6.556 | 13.712 | ABAminus | -118.51, -2.16 | -150.35, 139.43 | -132.07, 31.9 | 298.68, 77.43 | -57.63, -28.0 | in-in | in | 7.902 | Saltbr-in | 2.662 | HRD-in | -78.87, -51.69 | 73.77, 10.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.917 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.91, 33.47 | APE9-dihe-in | -66.35, 135.05 | APE8-dihe-in | -77.66, 75.63 | APE8-rot-na | 31.23 | APE67-dihe-in | -74.4, -5.72 | -63.02, -28.16 | APE12-dist-na | 11.142 | APE11-dist-na | 13.511 | APE10-dist-na | 10.263 | APE9-dist-in | 6.918 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.85 | 0.249 | 0.28 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsc | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSDA | P23458 | 865 | 1154 | 1154.0 | KH8:1201 | Type1 | Inactive | DFGin | 6.563 | 13.29 | ABAminus | -121.03, 3.28 | -150.09, 139.62 | -132.15, 26.01 | 293.71, 87.42 | -59.82, -26.08 | in-in | in | 7.641 | Saltbr-in | 2.673 | HRD-in | -81.56, -47.83 | 71.88, 7.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.925 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -96.0, 23.61 | APE9-dihe-in | -58.47, 136.99 | APE8-dihe-in | -79.35, 76.48 | APE8-rot-na | 35.13 | APE67-dihe-in | -77.95, -0.82 | -64.48, -27.09 | APE12-dist-na | 11.03 | APE11-dist-na | 13.568 | APE10-dist-na | 10.219 | APE9-dist-in | 6.806 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.76 | 0.202 | 0.238 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsd | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSDB | P23458 | 865 | 1154 | 1154.0 | KH8:1201 | Type1 | Inactive | DFGin | 6.567 | 13.42 | ABAminus | -123.92, 1.98 | -149.52, 139.04 | -133.17, 29.94 | 296.8, 84.79 | -64.12, -24.87 | in-in | in | 7.828 | Saltbr-in | 2.619 | HRD-in | -81.48, -52.31 | 73.66, 6.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.886 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 78.39, 5.73 | APE9-dihe-in | -59.21, 132.36 | APE8-dihe-in | -78.28, 75.83 | APE8-rot-na | 31.46 | APE67-dihe-in | -72.63, -5.35 | -64.01, -28.2 | APE12-dist-na | 11.21 | APE11-dist-na | 13.528 | APE10-dist-na | 10.362 | APE9-dist-in | 6.887 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.76 | 0.202 | 0.238 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsd | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSEA | P23458 | 865 | 1154 | 1154.0 | KHH:1201 | Type1 | Inactive | DFGin | 6.537 | 13.348 | ABAminus | -113.91, 1.27 | -156.33, 137.23 | -131.71, 27.09 | 299.32, 82.9 | -56.09, -32.48 | in-in | in | 7.864 | Saltbr-in | 2.638 | HRD-in | -79.69, -48.26 | 69.1, 11.16 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.716 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -68.92, 43.15 | APE9-dihe-in | -70.68, 135.44 | APE8-dihe-in | -74.14, 74.71 | APE8-rot-na | 28.88 | APE67-dihe-in | -82.04, -6.18 | -60.6, -28.4 | APE12-dist-na | 9.328 | APE11-dist-na | 11.782 | APE10-dist-na | 10.466 | APE9-dist-in | 6.774 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.265 | 0.303 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rse | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSEB | P23458 | 865 | 1154 | 1154.0 | KHH:1201 | Type1 | Inactive | DFGin | 6.461 | 13.569 | ABAminus | -119.02, 6.25 | -155.18, 136.02 | -130.8, 28.87 | 296.2, 78.44 | -57.74, -31.19 | in-in | in | 8.034 | Saltbr-in | 2.579 | HRD-in | -78.09, -47.4 | 66.03, 12.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.903 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -77.34, 48.11 | APE9-dihe-in | -88.98, 140.2 | APE8-dihe-in | -76.8, 76.65 | APE8-rot-na | 33.64 | APE67-dihe-in | -80.09, -3.14 | -61.43, -26.93 | APE12-dist-na | 13.325 | APE11-dist-na | 11.833 | APE10-dist-na | 10.755 | APE9-dist-in | 6.856 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.8 | 0.265 | 0.303 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rse | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSHA | P23458 | 865 | 1154 | 1154.0 | KHE:1201 | Type1 | Inactive | DFGin | 6.635 | 13.486 | ABAminus | -113.16, 6.59 | -151.95, 137.99 | -130.33, 27.13 | 294.82, 88.08 | -65.9, -20.74 | in-in | in | 7.441 | Saltbr-in | 2.532 | HRD-in | -77.26, -48.19 | 64.78, 14.62 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.694 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 87.06, 32.22 | APE9-dihe-in | -74.25, 135.13 | APE8-dihe-in | -77.78, 76.14 | APE8-rot-na | 33.2 | APE67-dihe-in | -80.47, -5.2 | -61.66, -26.89 | APE12-dist-na | 11.167 | APE11-dist-na | 12.639 | APE10-dist-na | 10.235 | APE9-dist-in | 6.904 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.71 | 0.271 | 0.311 | A | 302 | 286 | 4 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsh | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6RSHB | P23458 | 865 | 1154 | 1154.0 | KHE:1201 | Type1 | Inactive | DFGin | 6.627 | 13.852 | ABAminus | -116.98, -3.62 | -146.38, 138.52 | -131.28, 30.89 | 293.47, 79.95 | -64.48, -19.44 | in-in | in | 7.784 | Saltbr-in | 2.375 | HRD-in | -81.26, -46.13 | 68.12, 10.14 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.878 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 90.62, 16.91 | APE9-dihe-in | -58.11, 134.31 | APE8-dihe-in | -78.21, 75.43 | APE8-rot-na | 34.5 | APE67-dihe-in | -75.52, -2.49 | -58.55, -33.71 | APE12-dist-na | 11.219 | APE11-dist-na | 13.047 | APE10-dist-na | 10.449 | APE9-dist-in | 6.96 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.71 | 0.271 | 0.311 | B | 302 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6rsh | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6SM8A | P23458 | 854 | 1154 | 1154.0 | LKT:61201 | Type1 | Inactive | DFGin | 6.813 | 13.706 | ABAminus | -101.63, -7.1 | -147.81, 142.33 | -131.41, 24.39 | 292.89, 86.49 | -54.23, -31.63 | in-in | in | 7.807 | Saltbr-in | 2.732 | HRD-in | -72.9, -49.47 | 70.53, 3.61 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.836 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.89, 30.48 | APE9-dihe-in | -64.02, 138.21 | APE8-dihe-in | -82.49, 73.83 | APE8-rot-na | 29.16 | APE67-dihe-in | -76.27, -2.8 | -50.53, -32.36 | APE12-dist-na | 11.438 | APE11-dist-na | 13.22 | APE10-dist-na | 10.246 | APE9-dist-in | 6.724 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.85 | 0.213 | 0.241 | A | 302 | 296 | 5 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6sm8 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 8S85A | P23458 | 854 | 1154 | 1154.0 | A1H5R:61201 | Type1 | Inactive | DFGin | 6.63 | 13.345 | ABAminus | -112.23, -7.17 | -149.03, 146.72 | -132.22, 30.5 | 297.85, 84.4 | -54.75, -31.9 | in-in | in | 7.852 | Saltbr-in | 2.618 | HRD-in | -76.09, -48.85 | 71.09, 5.36 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.837 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 58.53, 30.92 | APE9-dihe-in | -76.65, 137.48 | APE8-dihe-in | -75.77, 75.79 | APE8-rot-na | 30.15 | APE67-dihe-in | -76.06, -7.29 | -58.07, -32.61 | APE12-dist-na | 11.266 | APE11-dist-na | 12.679 | APE10-dist-na | 10.467 | APE9-dist-in | 6.878 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.75 | 0.21 | 0.25 | A | 302 | 292 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 8s85 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 8S85B | P23458 | 865 | 1154 | 1154.0 | A1H5R:61201 | Type1 | Inactive | DFGin | 6.696 | 13.355 | ABAminus | -114.2, -1.94 | -152.98, 142.26 | -130.74, 31.83 | 294.81, 85.33 | -58.52, -32.2 | in-in | in | 7.745 | Saltbr-in | 2.614 | HRD-in | -77.39, -48.2 | 72.5, 8.27 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.891 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -105.67, 37.06 | APE9-dihe-in | -66.96, 136.92 | APE8-dihe-in | -79.85, 74.06 | APE8-rot-na | 34.04 | APE67-dihe-in | -73.04, -6.17 | -58.28, -33.1 | APE12-dist-na | 11.159 | APE11-dist-na | 13.098 | APE10-dist-na | 10.453 | APE9-dist-in | 6.796 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.75 | 0.21 | 0.25 | B | 302 | 283 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 8s85 | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N7AA | P23458 | 865 | 1154 | 1154.0 | KEV:61203 | Type1 | Inactive | DFGin | 6.453 | 13.367 | ABAminus | -116.98, 9.47 | -160.4, 147.32 | -135.39, 27.13 | 297.85, 83.25 | -58.95, -23.42 | in-in | in | 7.745 | Saltbr-in | 2.756 | HRD-in | -75.17, -44.67 | 72.8, -4.01 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.858 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -73.07, 124.84 | APE9-dihe-in | -104.44, 150.91 | APE8-dihe-in | -83.53, 72.06 | APE8-rot-na | 34.1 | APE67-dihe-in | -76.43, -2.54 | -56.05, -29.88 | APE12-dist-na | 14.659 | APE11-dist-na | 9.278 | APE10-dist-na | 12.111 | APE9-dist-in | 7.138 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.33 | 0.192 | 0.207 | A | 304 | 278 | 12 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n7a | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6N7AB | P23458 | 854 | 1154 | 1154.0 | KEV:61202 | Type1 | Inactive | DFGin | 6.47 | 13.498 | ABAminus | -116.23, 10.2 | -162.11, 148.53 | -137.01, 27.49 | 296.62, 85.6 | -60.22, -22.88 | in-in | in | 7.776 | Saltbr-in | 2.755 | HRD-in | -73.34, -48.05 | 70.64, 1.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.804 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -94.78, 65.84 | APE9-dihe-in | -92.65, 132.46 | APE8-dihe-in | -84.19, 73.36 | APE8-rot-na | 33.1 | APE67-dihe-in | -76.82, -1.21 | -55.1, -31.23 | APE12-dist-na | 10.789 | APE11-dist-na | 11.689 | APE10-dist-na | 9.266 | APE9-dist-in | 6.819 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 1.33 | 0.192 | 0.207 | B | 304 | 291 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6n7a | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.2e-87 | 298.6 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5KHXA | P23458 | 867 | 1154 | 1154.0 | 6TE:4000 | Type1 | Inactive | DFGin | 6.631 | 13.54 | ABAminus | -113.66, 8.44 | -153.85, 134.53 | -126.55, 25.21 | 296.38, 85.41 | -59.93, -18.33 | in-in | in | 7.565 | Saltbr-in | 2.778 | HRD-in | -73.12, -47.99 | 66.65, 10.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.794 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.92, 156.56 | APE9-dihe-in | -137.25, 140.8 | APE8-dihe-in | -82.8, 71.88 | APE8-rot-na | 32.82 | APE67-dihe-in | -77.93, -4.04 | -54.17, -30.94 | APE12-dist-na | 14.254 | APE11-dist-na | 8.466 | APE10-dist-na | 10.435 | APE9-dist-in | 6.376 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.4 | 0.173 | 0.242 | A | 316 | 278 | 10 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5khx | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6BBUA | P23458 | 867 | 1154 | 1154.0 | D7D:4000 | Type1 | Inactive | DFGin | 6.419 | 13.3 | ABAminus | -116.63, 12.94 | -152.79, 140.28 | -132.74, 24.58 | 296.65, 83.13 | -57.55, -25.0 | in-in | in | 7.644 | Saltbr-in | 2.781 | HRD-in | -73.12, -50.44 | 71.69, 3.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.861 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -135.84, 101.53 | APE9-dihe-in | -119.31, 160.09 | APE8-dihe-in | -78.32, 76.15 | APE8-rot-na | 30.95 | APE67-dihe-in | -74.07, -7.36 | -55.8, -32.39 | APE12-dist-na | 9.748 | APE11-dist-na | 11.183 | APE10-dist-na | 11.299 | APE9-dist-in | 6.263 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.08 | 0.185 | 0.213 | A | 316 | 281 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6bbu | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6DBNA | P23458 | 867 | 1154 | 1154.0 | G4J:4000 | Type1 | Inactive | DFGin | 6.339 | 13.27 | ABAminus | -106.28, 2.12 | -151.4, 144.25 | -137.1, 32.6 | 295.8, 96.91 | -66.86, -18.69 | in-in | in | 7.596 | Saltbr-in | 2.792 | HRD-in | -66.34, -50.63 | 70.35, -1.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.81 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -142.87, 84.26 | APE9-dihe-in | -94.42, 151.25 | APE8-dihe-in | -77.55, 83.04 | APE8-rot-na | 28.37 | APE67-dihe-in | -75.2, -10.39 | -60.86, -28.98 | APE12-dist-na | 9.302 | APE11-dist-na | 11.031 | APE10-dist-na | 10.809 | APE9-dist-in | 6.01 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.48 | 0.19 | 0.262 | A | 316 | 281 | 7 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6dbn | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 6W8LA | P23458 | 867 | 1154 | 1154.0 | R4S:1201 | Type1 | Inactive | DFGin | 6.52 | 13.639 | ABAminus | -117.57, 7.4 | -146.11, 138.04 | -131.96, 25.84 | 294.24, 93.82 | -58.79, -29.12 | in-in | in | 7.699 | Saltbr-in | 2.747 | HRD-in | -65.59, -50.27 | 70.66, 4.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.796 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -75.31, 154.48 | APE9-dihe-in | -145.69, 148.21 | APE8-dihe-in | -75.35, 73.33 | APE8-rot-na | 31.68 | APE67-dihe-in | -71.12, -8.39 | -52.84, -34.47 | APE12-dist-na | 13.73 | APE11-dist-na | 8.042 | APE10-dist-na | 10.481 | APE9-dist-in | 6.401 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.11 | 0.197 | 0.226 | A | 316 | 280 | 8 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 6w8l | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5KHWB | P23458 | 867 | 1153 | 1154.0 | ADP:1201 | ATPlike | Inactive | DFGin | 6.188 | 13.787 | BLAminus | -126.62, -174.05 | 50.66, 92.23 | -105.71, 28.99 | 301.42, 97.18 | -62.73, -33.32 | in-in | in | 7.991 | Saltbr-in | 2.817 | HRD-in | -54.38, -55.02 | 75.74, 4.0 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.811 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -83.14, 18.97 | APE9-dihe-in | -58.32, 113.18 | APE8-dihe-in | -82.04, 77.86 | APE8-rot-na | 28.29 | APE67-dihe-in | -76.85, -3.42 | -56.14, -32.61 | APE12-dist-na | 7.879 | APE11-dist-na | 9.695 | APE10-dist-na | 6.605 | APE9-dist-in | 5.912 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.47 | 0.188 | 0.231 | B | 316 | 278 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5khw | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 2.6e-87 | 298.4 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| JAK1_HUMAN | 5E1EA | P23458 | 865 | 1154 | 1154.0 | 5JG:1202 | Type1 | Inactive | DFGin | 6.644 | 13.932 | BLAminus | -119.33, -177.28 | 50.16, 87.79 | -101.77, 31.05 | 290.94, 82.42 | -65.82, -24.94 | in-in | in | 7.872 | Saltbr-in | 2.794 | HRD-in | -75.04, -43.37 | 64.83, -0.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.816 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.99, 41.3 | APE9-dihe-in | -73.96, 132.79 | APE8-dihe-in | -79.05, 75.13 | APE8-rot-na | 22.09 | APE67-dihe-in | -75.65, -2.64 | -52.7, -35.87 | APE12-dist-na | 10.981 | APE11-dist-na | 12.948 | APE10-dist-na | 10.168 | APE9-dist-in | 6.908 | None | PTR1034,PTR1035 | PTR1034,PTR1035 | XRAY | 2.3 | 0.227 | 0.268 | A | 290 | 281 | 9 | 0 | 0 | 0 | [[583, 847], [875, 1151]] | 2.0 | 5e1e | Homo sapiens | TYR_JAK1-2_HUMAN | TYR | 1.9e-87 | 298.9 | 2 | 259 | 258 | 1020 | 1021 | 1022 | 1024 | 1026 | 908 | 925 | 929 | 1000 | 1002 | 1001 | 1003 | 1063 | 1051 | 1046 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 957 | Tyrosine-protein kinase JAK1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
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