AGC_CDC42BPA (Serine/threonine-protein kinase MRCK alpha)

Total number of chains: 2
Active chains: 2
Uniprot: MRCKA_HUMAN
Kinase Domain Residues: 77 - 343
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 2 100.0% AF-Q5VT25-K1A

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PDB Resolution Activity_label Spatial_Dihedral_labels ChelixSaltbr_label ActLoopNT-ActLoopCT APEtype APEdihe_label APEdist_label Ligand Ligand_type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
AF-Q5VT25-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 69 - 351 0 None None Serine/threonine-protein kinase MRCK alpha
AF-Q5VT25-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 69 - 351 0 None None Serine/threonine-protein kinase MRCK alpha

AGC_CDC42BPA (Serine/threonine-protein kinase MRCK alpha)

Total number of chains: 3
Active chains: 3
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 3 100.0% AF-Q5VT25-K1A

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UniprotID PDB Resolution Activity_label Spatial_Dihedral_labels ChelixSaltbr_label ActLoopNT-ActLoopCT APEtype APEdihe_label APEdist_label Ligand Ligand_type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
MRCKA_HUMAN AF-Q5VT25-K1A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 69 - 351 0 None None Serine/threonine-protein kinase MRCK alpha Homo sapiens
MRCKA_HUMAN AF-Q5VT25-K3A -1.0 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii No_ligand No_ligand 69 - 351 0 None None Serine/threonine-protein kinase MRCK alpha Homo sapiens
MRCKA_RAT 4AW2A 1.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 22E Allosteric 2 - 417 0 None D254G Serine/threonine-protein kinase MRCK alpha Rattus norvegicus

AGC_CDC42BPA (Serine/threonine-protein kinase MRCK alpha)

Total number of chains: 1
Active chains: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 1 100.0% 4AW2A

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UniprotID PDB Resolution Activity_label Spatial_Dihedral_labels ChelixSaltbr_label ActLoopNT-ActLoopCT APEtype APEdihe_label APEdist_label Ligand Ligand_type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
MRCKA_RAT 4AW2A 1.7 Active DFGin‑BLAminus in-in in-in nonTYR APEdihe_aaiii APEdist_iiii 22E Allosteric 2 - 417 0 None D254G Serine/threonine-protein kinase MRCK alpha Rattus norvegicus