| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AAK1 | AF-Q2M2I8-K1A | Q2M2I8 | 38 | 321 | 961.0 | No_ligand | No_ligand | Active | DFGin | 6.0898 | 13.1573 | BLAminus | -130.76, 177.11 | 65.46, 72.88 | -86.17, 13.75 | 306.15, 100.85 | -62.63, -26.92 | in-in | in | 8.6944 | Saltbr-in | 2.6952 | HRD-in | -71.29, -40.47 | 67.96, -14.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7672 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.43, 1.5 | APE9-dihe-na | -133.56, 144.49 | APE8-dihe-in | -85.09, 124.69 | APE8-rot-in | 302.03 | APE67-dihe-in | -65.48, -12.52 | -47.91, -50.11 | APE12-dist-in | 12.1054 | APE11-dist-in | 8.3861 | APE10-dist-in | 4.1768 | APE9-dist-in | 3.7633 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 284.0 | 284.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | AF-Q2M2I8-K1 | OTHER_AAK1_HUMAN | OTHER | 2.4e-41 | 147.8 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AF-Q2M2I8-K3A | Q2M2I8 | 38 | 321 | 961.0 | No_ligand | No_ligand | Active | DFGin | 5.9088 | 13.3704 | BLAminus | -128.17, 175.79 | 57.92, 95.09 | -102.83, 15.36 | 298.99, 95.97 | -62.48, -26.93 | in-in | in | 8.8052 | Saltbr-in | 2.6864 | HRD-in | -73.71, -40.34 | 66.99, -5.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8022 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.85, -5.0 | APE9-dihe-na | -133.21, 117.79 | APE8-dihe-in | -58.72, 127.19 | APE8-rot-in | 304.31 | APE67-dihe-in | -63.7, -12.57 | -50.37, -47.6 | APE12-dist-in | 12.0248 | APE11-dist-in | 8.4592 | APE10-dist-in | 4.1293 | APE9-dist-in | 3.4894 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 284.0 | 284.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | AF-Q2M2I8-K3 | OTHER_AAK1_HUMAN | OTHER | 2.4e-41 | 147.8 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 4WSQA | Q2M2I8 | 29 | 345 | 961.0 | KSA:405 | Type1 | Active | DFGin | 6.307 | 13.7534 | BLAminus | -126.2, -179.67 | 69.61, 90.76 | -108.14, 19.69 | 293.57, 82.96 | -69.52, -19.34 | in-in | in | 9.5238 | Saltbr-in | 3.051 | HRD-in | -67.42, -46.62 | 67.64, 3.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8695 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -110.1, -8.47 | APE9-dihe-na | -120.84, 162.67 | APE8-dihe-in | -101.84, 124.39 | APE8-rot-in | 300.18 | APE67-dihe-in | -59.62, -25.15 | -50.19, -46.52 | APE12-dist-in | 12.3768 | APE11-dist-in | 8.8309 | APE10-dist-in | 4.4743 | APE9-dist-in | 3.6746 | None | None | None | XRAY | 1.95 | 0.182 | 0.208 | A | 317.0 | 317.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 4wsq | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.5 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 4WSQB | Q2M2I8 | 33 | 342 | 961.0 | KSA:404 | Type1 | Active | DFGin | 6.4483 | 13.4911 | BLAminus | -125.14, -178.62 | 72.01, 91.87 | -111.17, 20.84 | 297.62, 84.5 | -70.3, -20.72 | in-in | in | 9.3105 | Saltbr-in | 2.7431 | HRD-in | -70.2, -48.3 | 68.24, 1.29 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8464 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -110.84, -7.92 | APE9-dihe-na | -118.96, 162.19 | APE8-dihe-in | -104.95, 123.2 | APE8-rot-in | 302.88 | APE67-dihe-in | -62.15, -24.37 | -51.37, -45.33 | APE12-dist-in | 12.2082 | APE11-dist-in | 8.5573 | APE10-dist-in | 4.2501 | APE9-dist-in | 3.7443 | None | None | None | XRAY | 1.95 | 0.182 | 0.208 | B | 317.0 | 310.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 4wsq | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.5 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 8GMCA | Q2M2I8 | 34 | 330 | 961.0 | YFV:401 | Type1 | Active | DFGin | 6.2956 | 13.3438 | BLAminus | -132.35, 179.07 | 63.58, 102.47 | -106.53, 19.35 | 292.32, 96.59 | -60.5, -34.69 | in-in | in | 8.5015 | Saltbr-in | 2.7401 | HRD-in | -65.3, -44.13 | 71.44, -0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.984 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -101.27, -5.42 | APE9-dihe-na | -117.59, 149.82 | APE8-dihe-in | -99.03, 116.29 | APE8-rot-in | 299.63 | APE67-dihe-in | -50.9, -25.95 | -44.55, -54.08 | APE12-dist-in | 12.2292 | APE11-dist-in | 8.5323 | APE10-dist-in | 4.1896 | APE9-dist-in | 3.8809 | None | None | None | XRAY | 2.5 | 0.228 | 0.256 | A | 318.0 | 293.0 | 4 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 8gmc | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.6 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 8GMCB | Q2M2I8 | 31 | 330 | 961.0 | YFV:401 | Type1 | Active | DFGin | 6.6132 | 13.4444 | BLAminus | -132.15, -179.67 | 62.85, 102.24 | -105.78, 18.46 | 292.58, 96.33 | -60.62, -34.17 | in-in | in | 8.465 | Saltbr-in | 2.9369 | HRD-in | -65.77, -42.15 | 71.41, -5.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.983 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.13, -3.18 | APE9-dihe-na | -121.52, 151.08 | APE8-dihe-in | -97.1, 121.04 | APE8-rot-in | 308.13 | APE67-dihe-in | -59.64, -26.78 | -53.61, -40.63 | APE12-dist-in | 12.1812 | APE11-dist-in | 8.453 | APE10-dist-in | 4.1545 | APE9-dist-in | 3.9786 | None | None | None | XRAY | 2.5 | 0.228 | 0.256 | B | 318.0 | 294.0 | 5 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 8gmc | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.6 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 8GMDA | Q2M2I8 | 34 | 329 | 961.0 | ZRR:401 | Type1 | Active | DFGin | 6.1668 | 13.3321 | BLAminus | -127.52, 174.84 | 65.86, 97.82 | -104.03, 21.57 | 300.09, 93.49 | -64.42, -30.01 | in-in | in | 8.5756 | Saltbr-in | 2.7839 | HRD-in | -64.68, -46.09 | 71.69, -3.04 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9742 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.71, -15.11 | APE9-dihe-na | -111.33, 160.49 | APE8-dihe-in | -104.37, 121.78 | APE8-rot-in | 304.75 | APE67-dihe-in | -58.75, -28.21 | -47.17, -46.33 | APE12-dist-in | 12.1626 | APE11-dist-in | 8.4335 | APE10-dist-in | 4.1468 | APE9-dist-in | 3.5664 | None | None | None | XRAY | 2.2 | 0.233 | 0.25 | A | 318.0 | 294.0 | 2 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 8gmd | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.6 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 8GMDB | Q2M2I8 | 29 | 330 | 961.0 | ZRR:401 | Type1 | Active | DFGin | 6.3724 | 13.4776 | BLAminus | -123.19, 179.01 | 67.0, 97.52 | -104.44, 17.42 | 296.06, 83.59 | -61.74, -25.96 | in-in | in | 8.4316 | Saltbr-in | 2.7776 | HRD-in | -64.58, -45.6 | 71.56, -2.33 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9573 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -115.95, -11.7 | APE9-dihe-na | -117.06, 155.74 | APE8-dihe-in | -98.45, 121.78 | APE8-rot-in | 305.28 | APE67-dihe-in | -59.45, -28.48 | -46.11, -46.72 | APE12-dist-in | 12.1776 | APE11-dist-in | 8.3744 | APE10-dist-in | 4.1429 | APE9-dist-in | 3.5971 | None | None | None | XRAY | 2.2 | 0.233 | 0.25 | B | 318.0 | 299.0 | 3 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 8gmd | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.6 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 9QB5A | Q2M2I8 | 29 | 343 | 961.0 | F7I:60401 | Type1 | Active | DFGin | 6.406 | 13.358 | BLAminus | -132.26, 177.36 | 64.71, 93.28 | -102.58, 23.65 | 295.99, 87.8 | -68.89, -14.08 | in-in | in | 8.4517 | Saltbr-in | 2.5766 | HRD-in | -65.82, -48.18 | 75.53, -3.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8781 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.0, -10.1 | APE9-dihe-na | -117.28, 159.33 | APE8-dihe-in | -101.85, 125.23 | APE8-rot-in | 303.31 | APE67-dihe-in | -61.58, -23.49 | -52.0, -46.22 | APE12-dist-in | 12.1582 | APE11-dist-in | 8.502 | APE10-dist-in | 4.1257 | APE9-dist-in | 3.6319 | None | None | None | XRAY | 2.0 | 0.199 | 0.227 | A | 318.0 | 313.0 | 2 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 9qb5 | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.5 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 9QB5B | Q2M2I8 | 34 | 342 | 961.0 | F7I:60401 | Type1 | Active | DFGin | 6.4569 | 13.0394 | BLAminus | -136.45, 178.27 | 73.68, 94.2 | -109.77, 25.54 | 300.89, 108.71 | -73.91, -11.3 | in-in | in | 8.0922 | Saltbr-in | 2.4615 | HRD-in | -66.48, -48.55 | 75.65, -3.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9081 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.0, -6.97 | APE9-dihe-na | -121.88, 160.23 | APE8-dihe-in | -103.81, 124.81 | APE8-rot-in | 304.19 | APE67-dihe-in | -60.83, -28.74 | -52.63, -42.77 | APE12-dist-in | 12.174 | APE11-dist-in | 8.5775 | APE10-dist-in | 4.3028 | APE9-dist-in | 3.6645 | None | None | None | XRAY | 2.0 | 0.199 | 0.227 | B | 318.0 | 309.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 9qb5 | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.5 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 5L4QA | Q2M2I8 | 33 | 335 | 961.0 | LKB:401 | Type1 | Active | DFGin | 6.0047 | 13.2273 | BLAminus | -132.85, -177.94 | 63.93, 92.35 | -114.27, 19.37 | 301.1, 98.45 | -80.74, -11.63 | in-in | in | 8.685 | Saltbr-in | 2.708 | HRD-in | -67.77, -48.62 | 71.48, 2.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9221 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.55, -17.02 | APE9-dihe-na | -109.84, 154.17 | APE8-dihe-in | -96.17, 123.72 | APE8-rot-in | 302.79 | APE67-dihe-in | -62.67, -23.02 | -45.97, -51.51 | APE12-dist-in | 11.9991 | APE11-dist-in | 8.3501 | APE10-dist-in | 4.067 | APE9-dist-in | 3.4826 | None | None | None | XRAY | 1.97 | 0.208 | 0.227 | A | 346.0 | 293.0 | 10 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 5l4q | OTHER_AAK1_HUMAN | OTHER | 4.8e-41 | 147.2 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 5L4QB | Q2M2I8 | 33 | 333 | 961.0 | LKB:401 | Type1 | Active | DFGin | 6.0008 | 13.2527 | BLAminus | -132.29, -178.13 | 64.06, 92.67 | -114.66, 18.46 | 300.35, 97.82 | -80.3, -11.3 | in-in | in | 8.5651 | Saltbr-in | 2.7137 | HRD-in | -67.84, -48.94 | 70.89, 2.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8784 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -107.29, -16.57 | APE9-dihe-na | -109.81, 154.98 | APE8-dihe-in | -96.35, 124.27 | APE8-rot-in | 304.05 | APE67-dihe-in | -62.49, -22.16 | -46.27, -52.25 | APE12-dist-in | 11.9555 | APE11-dist-in | 8.4008 | APE10-dist-in | 4.043 | APE9-dist-in | 3.5048 | None | None | None | XRAY | 1.97 | 0.208 | 0.227 | B | 346.0 | 287.0 | 14 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 5l4q | OTHER_AAK1_HUMAN | OTHER | 4.8e-41 | 147.2 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | 5TE0A | Q2M2I8 | 27 | 345 | 961.0 | XIN:60401 | Type1 | Active | DFGin | 6.1767 | 13.7286 | BLAminus | -133.95, 173.97 | 66.46, 103.31 | -110.15, 22.69 | 304.86, 94.85 | -65.74, -20.86 | in-in | in | 9.0545 | Saltbr-in | 3.4906 | HRD-in | -62.42, -46.29 | 70.69, -4.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8421 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -107.12, -11.26 | APE9-dihe-na | -114.88, 156.03 | APE8-dihe-in | -99.05, 119.5 | APE8-rot-in | 300.83 | APE67-dihe-in | -58.27, -25.82 | -45.89, -49.71 | APE12-dist-in | 12.1407 | APE11-dist-in | 8.3978 | APE10-dist-in | 4.1462 | APE9-dist-in | 3.7311 | None | None | None | XRAY | 1.9 | 0.182 | 0.199 | A | 347.0 | 315.0 | 4 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 5te0 | OTHER_AAK1_HUMAN | OTHER | 4.8e-41 | 147.2 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AAK1 | AAK1_HUMAN | AF-Q2M2I8-K1A | Q2M2I8 | 38 | 321 | 961.0 | No_ligand | No_ligand | Active | DFGin | 6.0898 | 13.1573 | BLAminus | -130.76, 177.11 | 65.46, 72.88 | -86.17, 13.75 | 306.15, 100.85 | -62.63, -26.92 | in-in | in | 8.6944 | Saltbr-in | 2.6952 | HRD-in | -71.29, -40.47 | 67.96, -14.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7672 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.43, 1.5 | APE9-dihe-na | -133.56, 144.49 | APE8-dihe-in | -85.09, 124.69 | APE8-rot-in | 302.03 | APE67-dihe-in | -65.48, -12.52 | -47.91, -50.11 | APE12-dist-in | 12.1054 | APE11-dist-in | 8.3861 | APE10-dist-in | 4.1768 | APE9-dist-in | 3.7633 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 284.0 | 284.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | AF-Q2M2I8-K1 | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 2.4e-41 | 147.8 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | AF-Q2M2I8-K3A | Q2M2I8 | 38 | 321 | 961.0 | No_ligand | No_ligand | Active | DFGin | 5.9088 | 13.3704 | BLAminus | -128.17, 175.79 | 57.92, 95.09 | -102.83, 15.36 | 298.99, 95.97 | -62.48, -26.93 | in-in | in | 8.8052 | Saltbr-in | 2.6864 | HRD-in | -73.71, -40.34 | 66.99, -5.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8022 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.85, -5.0 | APE9-dihe-na | -133.21, 117.79 | APE8-dihe-in | -58.72, 127.19 | APE8-rot-in | 304.31 | APE67-dihe-in | -63.7, -12.57 | -50.37, -47.6 | APE12-dist-in | 12.0248 | APE11-dist-in | 8.4592 | APE10-dist-in | 4.1293 | APE9-dist-in | 3.4894 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 284.0 | 284.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | AF-Q2M2I8-K3 | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 2.4e-41 | 147.8 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 4WSQA | Q2M2I8 | 29 | 345 | 961.0 | KSA:405 | Type1 | Active | DFGin | 6.307 | 13.7534 | BLAminus | -126.2, -179.67 | 69.61, 90.76 | -108.14, 19.69 | 293.57, 82.96 | -69.52, -19.34 | in-in | in | 9.5238 | Saltbr-in | 3.051 | HRD-in | -67.42, -46.62 | 67.64, 3.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8695 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -110.1, -8.47 | APE9-dihe-na | -120.84, 162.67 | APE8-dihe-in | -101.84, 124.39 | APE8-rot-in | 300.18 | APE67-dihe-in | -59.62, -25.15 | -50.19, -46.52 | APE12-dist-in | 12.3768 | APE11-dist-in | 8.8309 | APE10-dist-in | 4.4743 | APE9-dist-in | 3.6746 | None | None | None | XRAY | 1.95 | 0.182 | 0.208 | A | 317.0 | 317.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 4wsq | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.5 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 4WSQB | Q2M2I8 | 33 | 342 | 961.0 | KSA:404 | Type1 | Active | DFGin | 6.4483 | 13.4911 | BLAminus | -125.14, -178.62 | 72.01, 91.87 | -111.17, 20.84 | 297.62, 84.5 | -70.3, -20.72 | in-in | in | 9.3105 | Saltbr-in | 2.7431 | HRD-in | -70.2, -48.3 | 68.24, 1.29 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8464 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -110.84, -7.92 | APE9-dihe-na | -118.96, 162.19 | APE8-dihe-in | -104.95, 123.2 | APE8-rot-in | 302.88 | APE67-dihe-in | -62.15, -24.37 | -51.37, -45.33 | APE12-dist-in | 12.2082 | APE11-dist-in | 8.5573 | APE10-dist-in | 4.2501 | APE9-dist-in | 3.7443 | None | None | None | XRAY | 1.95 | 0.182 | 0.208 | B | 317.0 | 310.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 4wsq | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.5 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 8GMCA | Q2M2I8 | 34 | 330 | 961.0 | YFV:401 | Type1 | Active | DFGin | 6.2956 | 13.3438 | BLAminus | -132.35, 179.07 | 63.58, 102.47 | -106.53, 19.35 | 292.32, 96.59 | -60.5, -34.69 | in-in | in | 8.5015 | Saltbr-in | 2.7401 | HRD-in | -65.3, -44.13 | 71.44, -0.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.984 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -101.27, -5.42 | APE9-dihe-na | -117.59, 149.82 | APE8-dihe-in | -99.03, 116.29 | APE8-rot-in | 299.63 | APE67-dihe-in | -50.9, -25.95 | -44.55, -54.08 | APE12-dist-in | 12.2292 | APE11-dist-in | 8.5323 | APE10-dist-in | 4.1896 | APE9-dist-in | 3.8809 | None | None | None | XRAY | 2.5 | 0.228 | 0.256 | A | 318.0 | 293.0 | 4 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 8gmc | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.6 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 8GMCB | Q2M2I8 | 31 | 330 | 961.0 | YFV:401 | Type1 | Active | DFGin | 6.6132 | 13.4444 | BLAminus | -132.15, -179.67 | 62.85, 102.24 | -105.78, 18.46 | 292.58, 96.33 | -60.62, -34.17 | in-in | in | 8.465 | Saltbr-in | 2.9369 | HRD-in | -65.77, -42.15 | 71.41, -5.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.983 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.13, -3.18 | APE9-dihe-na | -121.52, 151.08 | APE8-dihe-in | -97.1, 121.04 | APE8-rot-in | 308.13 | APE67-dihe-in | -59.64, -26.78 | -53.61, -40.63 | APE12-dist-in | 12.1812 | APE11-dist-in | 8.453 | APE10-dist-in | 4.1545 | APE9-dist-in | 3.9786 | None | None | None | XRAY | 2.5 | 0.228 | 0.256 | B | 318.0 | 294.0 | 5 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 8gmc | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.6 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 8GMDA | Q2M2I8 | 34 | 329 | 961.0 | ZRR:401 | Type1 | Active | DFGin | 6.1668 | 13.3321 | BLAminus | -127.52, 174.84 | 65.86, 97.82 | -104.03, 21.57 | 300.09, 93.49 | -64.42, -30.01 | in-in | in | 8.5756 | Saltbr-in | 2.7839 | HRD-in | -64.68, -46.09 | 71.69, -3.04 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9742 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.71, -15.11 | APE9-dihe-na | -111.33, 160.49 | APE8-dihe-in | -104.37, 121.78 | APE8-rot-in | 304.75 | APE67-dihe-in | -58.75, -28.21 | -47.17, -46.33 | APE12-dist-in | 12.1626 | APE11-dist-in | 8.4335 | APE10-dist-in | 4.1468 | APE9-dist-in | 3.5664 | None | None | None | XRAY | 2.2 | 0.233 | 0.25 | A | 318.0 | 294.0 | 2 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 8gmd | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.6 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 8GMDB | Q2M2I8 | 29 | 330 | 961.0 | ZRR:401 | Type1 | Active | DFGin | 6.3724 | 13.4776 | BLAminus | -123.19, 179.01 | 67.0, 97.52 | -104.44, 17.42 | 296.06, 83.59 | -61.74, -25.96 | in-in | in | 8.4316 | Saltbr-in | 2.7776 | HRD-in | -64.58, -45.6 | 71.56, -2.33 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9573 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -115.95, -11.7 | APE9-dihe-na | -117.06, 155.74 | APE8-dihe-in | -98.45, 121.78 | APE8-rot-in | 305.28 | APE67-dihe-in | -59.45, -28.48 | -46.11, -46.72 | APE12-dist-in | 12.1776 | APE11-dist-in | 8.3744 | APE10-dist-in | 4.1429 | APE9-dist-in | 3.5971 | None | None | None | XRAY | 2.2 | 0.233 | 0.25 | B | 318.0 | 299.0 | 3 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 8gmd | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.6 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 9QB5A | Q2M2I8 | 29 | 343 | 961.0 | F7I:60401 | Type1 | Active | DFGin | 6.406 | 13.358 | BLAminus | -132.26, 177.36 | 64.71, 93.28 | -102.58, 23.65 | 295.99, 87.8 | -68.89, -14.08 | in-in | in | 8.4517 | Saltbr-in | 2.5766 | HRD-in | -65.82, -48.18 | 75.53, -3.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8781 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -111.0, -10.1 | APE9-dihe-na | -117.28, 159.33 | APE8-dihe-in | -101.85, 125.23 | APE8-rot-in | 303.31 | APE67-dihe-in | -61.58, -23.49 | -52.0, -46.22 | APE12-dist-in | 12.1582 | APE11-dist-in | 8.502 | APE10-dist-in | 4.1257 | APE9-dist-in | 3.6319 | None | None | None | XRAY | 2.0 | 0.199 | 0.227 | A | 318.0 | 313.0 | 2 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 9qb5 | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.5 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 9QB5B | Q2M2I8 | 34 | 342 | 961.0 | F7I:60401 | Type1 | Active | DFGin | 6.4569 | 13.0394 | BLAminus | -136.45, 178.27 | 73.68, 94.2 | -109.77, 25.54 | 300.89, 108.71 | -73.91, -11.3 | in-in | in | 8.0922 | Saltbr-in | 2.4615 | HRD-in | -66.48, -48.55 | 75.65, -3.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9081 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.0, -6.97 | APE9-dihe-na | -121.88, 160.23 | APE8-dihe-in | -103.81, 124.81 | APE8-rot-in | 304.19 | APE67-dihe-in | -60.83, -28.74 | -52.63, -42.77 | APE12-dist-in | 12.174 | APE11-dist-in | 8.5775 | APE10-dist-in | 4.3028 | APE9-dist-in | 3.6645 | None | None | None | XRAY | 2.0 | 0.199 | 0.227 | B | 318.0 | 309.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 9qb5 | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 3.6e-41 | 147.5 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 5L4QA | Q2M2I8 | 33 | 335 | 961.0 | LKB:401 | Type1 | Active | DFGin | 6.0047 | 13.2273 | BLAminus | -132.85, -177.94 | 63.93, 92.35 | -114.27, 19.37 | 301.1, 98.45 | -80.74, -11.63 | in-in | in | 8.685 | Saltbr-in | 2.708 | HRD-in | -67.77, -48.62 | 71.48, 2.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9221 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.55, -17.02 | APE9-dihe-na | -109.84, 154.17 | APE8-dihe-in | -96.17, 123.72 | APE8-rot-in | 302.79 | APE67-dihe-in | -62.67, -23.02 | -45.97, -51.51 | APE12-dist-in | 11.9991 | APE11-dist-in | 8.3501 | APE10-dist-in | 4.067 | APE9-dist-in | 3.4826 | None | None | None | XRAY | 1.97 | 0.208 | 0.227 | A | 346.0 | 293.0 | 10 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 5l4q | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 4.8e-41 | 147.2 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 5L4QB | Q2M2I8 | 33 | 333 | 961.0 | LKB:401 | Type1 | Active | DFGin | 6.0008 | 13.2527 | BLAminus | -132.29, -178.13 | 64.06, 92.67 | -114.66, 18.46 | 300.35, 97.82 | -80.3, -11.3 | in-in | in | 8.5651 | Saltbr-in | 2.7137 | HRD-in | -67.84, -48.94 | 70.89, 2.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8784 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -107.29, -16.57 | APE9-dihe-na | -109.81, 154.98 | APE8-dihe-in | -96.35, 124.27 | APE8-rot-in | 304.05 | APE67-dihe-in | -62.49, -22.16 | -46.27, -52.25 | APE12-dist-in | 11.9555 | APE11-dist-in | 8.4008 | APE10-dist-in | 4.043 | APE9-dist-in | 3.5048 | None | None | None | XRAY | 1.97 | 0.208 | 0.227 | B | 346.0 | 287.0 | 14 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 5l4q | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 4.8e-41 | 147.2 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_HUMAN | 5TE0A | Q2M2I8 | 27 | 345 | 961.0 | XIN:60401 | Type1 | Active | DFGin | 6.1767 | 13.7286 | BLAminus | -133.95, 173.97 | 66.46, 103.31 | -110.15, 22.69 | 304.86, 94.85 | -65.74, -20.86 | in-in | in | 9.0545 | Saltbr-in | 3.4906 | HRD-in | -62.42, -46.29 | 70.69, -4.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8421 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -107.12, -11.26 | APE9-dihe-na | -114.88, 156.03 | APE8-dihe-in | -99.05, 119.5 | APE8-rot-in | 300.83 | APE67-dihe-in | -58.27, -25.82 | -45.89, -49.71 | APE12-dist-in | 12.1407 | APE11-dist-in | 8.3978 | APE10-dist-in | 4.1462 | APE9-dist-in | 3.7311 | None | None | None | XRAY | 1.9 | 0.182 | 0.199 | A | 347.0 | 315.0 | 4 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 5te0 | Homo sapiens | OTHER_AAK1_HUMAN | OTHER | 4.8e-41 | 147.2 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7LVHA | Q3UHJ0 | 34 | 328 | 959.0 | YFS:401 | Type1 | Active | DFGin | 6.3815 | 13.1586 | BLAminus | -99.27, -147.3 | 14.04, 114.8 | -121.99, 26.42 | 298.51, 87.91 | -70.89, -12.69 | in-in | in | 8.6326 | Saltbr-in | 2.9865 | HRD-in | -65.25, -42.59 | 66.7, -3.41 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9339 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.0, -6.79 | APE9-dihe-na | -118.74, 158.73 | APE8-dihe-in | -102.63, 127.81 | APE8-rot-in | 327.57 | APE67-dihe-in | -51.65, -23.05 | -49.85, -58.32 | APE12-dist-in | 12.2326 | APE11-dist-in | 8.6319 | APE10-dist-in | 4.2873 | APE9-dist-in | 3.7712 | None | None | None | XRAY | 2.65 | 0.267 | 0.299 | A | 318.0 | 284.0 | 11 | 36 | 34 | 2 | [[46, 313]] | 1.0 | 7lvh | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7LVHB | Q3UHJ0 | 35 | 329 | 959.0 | YFV:401 | Type1 | Active | DFGin | 6.305 | 13.462 | BLAminus | -109.39, -171.27 | 52.7, 102.9 | -109.75, 14.5 | 296.74, 93.05 | -60.15, -20.34 | in-in | in | 8.5725 | Saltbr-in | 2.9247 | HRD-in | -64.33, -41.66 | 66.46, -2.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.927 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.01, -10.47 | APE9-dihe-na | -112.81, 152.03 | APE8-dihe-in | -104.75, 117.86 | APE8-rot-in | 298.94 | APE67-dihe-in | -52.25, -35.41 | -40.96, -54.57 | APE12-dist-in | 12.4236 | APE11-dist-in | 8.6752 | APE10-dist-in | 4.2649 | APE9-dist-in | 3.8852 | None | None | None | XRAY | 2.65 | 0.267 | 0.299 | B | 318.0 | 281.0 | 14 | 36 | 34 | 2 | [[46, 313]] | 1.0 | 7lvh | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7LVIB | Q3UHJ0 | 35 | 330 | 959.0 | YFV:401 | Type1 | Active | DFGin | 6.5554 | 13.9557 | BLAminus | -120.74, -177.87 | 58.36, 103.46 | -109.53, 15.49 | 286.96, 91.82 | -62.65, -18.35 | in-in | in | 8.6464 | Saltbr-in | 2.9382 | HRD-in | -65.69, -47.95 | 71.36, -2.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7984 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.16, -5.91 | APE9-dihe-na | -123.61, 155.71 | APE8-dihe-in | -99.3, 117.77 | APE8-rot-in | 306.22 | APE67-dihe-in | -52.8, -28.0 | -40.05, -53.5 | APE12-dist-in | 12.1358 | APE11-dist-in | 8.5899 | APE10-dist-in | 4.2334 | APE9-dist-in | 3.7808 | None | None | None | XRAY | 2.2 | 0.219 | 0.241 | B | 318.0 | 288.0 | 8 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7lvi | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ6A | Q3UHJ0 | 26 | 330 | 959.0 | YFV:401 | Type1 | Active | DFGin | 6.5122 | 13.3768 | BLAminus | -125.62, 169.71 | 67.71, 96.16 | -104.68, 24.3 | 300.02, 93.63 | -68.93, -22.4 | in-in | in | 8.5967 | Saltbr-in | 2.7099 | HRD-in | -65.12, -47.31 | 74.51, -5.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8935 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -105.26, -12.99 | APE9-dihe-na | -116.7, 155.82 | APE8-dihe-in | -97.42, 121.54 | APE8-rot-in | 304.46 | APE67-dihe-in | -58.17, -28.42 | -45.34, -49.66 | APE12-dist-in | 12.1363 | APE11-dist-in | 8.6182 | APE10-dist-in | 4.2728 | APE9-dist-in | 3.6627 | None | None | None | XRAY | 2.132 | 0.202 | 0.215 | A | 318.0 | 305.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj6 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ6B | Q3UHJ0 | 32 | 330 | 959.0 | 5OI:401 | Type1 | Active | DFGin | 6.386 | 13.2644 | BLAminus | -136.98, -179.6 | 61.47, 90.79 | -102.58, 19.8 | 300.28, 93.44 | -74.01, -20.13 | in-in | in | 8.7043 | Saltbr-in | 2.7308 | HRD-in | -65.76, -48.0 | 74.66, -11.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8975 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.51, -10.49 | APE9-dihe-na | -120.36, 163.0 | APE8-dihe-in | -104.78, 122.31 | APE8-rot-in | 303.78 | APE67-dihe-in | -58.21, -28.47 | -45.49, -49.71 | APE12-dist-in | 11.9714 | APE11-dist-in | 8.4144 | APE10-dist-in | 4.1372 | APE9-dist-in | 3.7792 | None | None | None | XRAY | 2.132 | 0.202 | 0.215 | B | 318.0 | 299.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj6 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ7A | Q3UHJ0 | 26 | 330 | 959.0 | 5P6:401 | Type1 | Active | DFGin | 6.4175 | 13.2295 | BLAminus | -119.48, 174.96 | 57.07, 109.64 | -122.04, 21.88 | 302.38, 85.37 | -70.96, -15.13 | in-in | in | 8.8767 | Saltbr-in | 2.7471 | HRD-in | -69.47, -41.35 | 71.48, -9.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9302 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.51, -3.09 | APE9-dihe-na | -122.59, 149.49 | APE8-dihe-in | -97.34, 124.1 | APE8-rot-in | 304.72 | APE67-dihe-in | -57.28, -27.01 | -46.87, -50.73 | APE12-dist-in | 12.1476 | APE11-dist-in | 8.4871 | APE10-dist-in | 4.133 | APE9-dist-in | 3.7038 | None | None | None | XRAY | 2.124 | 0.23 | 0.241 | A | 318.0 | 304.0 | 1 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj7 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ7B | Q3UHJ0 | 31 | 330 | 959.0 | 5P6:401 | Type1 | Active | DFGin | 6.0891 | 13.1308 | BLAminus | -124.6, -178.84 | 57.9, 88.94 | -99.65, 26.07 | 303.29, 101.38 | -78.17, -15.56 | in-in | in | 8.8917 | Saltbr-in | 2.7552 | HRD-in | -71.2, -45.26 | 74.74, -14.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9313 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.73, -6.79 | APE9-dihe-na | -120.3, 157.4 | APE8-dihe-in | -99.84, 124.85 | APE8-rot-in | 305.17 | APE67-dihe-in | -58.1, -26.76 | -48.79, -48.64 | APE12-dist-in | 12.0925 | APE11-dist-in | 8.4564 | APE10-dist-in | 4.1132 | APE9-dist-in | 3.8598 | None | None | None | XRAY | 2.124 | 0.23 | 0.241 | B | 318.0 | 300.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj7 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ8A | Q3UHJ0 | 33 | 329 | 959.0 | 5QI:401,PG6:402 | Type1,Allosteric | Active | DFGin | 5.8996 | 12.8884 | BLAminus | -133.43, 178.44 | 53.42, 101.65 | -103.66, 23.97 | 304.98, 112.99 | -67.68, -29.68 | in-in | in | 8.3964 | Saltbr-in | 2.7456 | HRD-in | -63.24, -44.02 | 66.63, -0.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.5201 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.11, -10.27 | APE9-dihe-na | -117.76, 158.13 | APE8-dihe-in | -102.68, 119.66 | APE8-rot-in | 301.04 | APE67-dihe-in | -54.01, -28.74 | -43.37, -51.03 | APE12-dist-in | 12.1372 | APE11-dist-in | 8.4799 | APE10-dist-in | 4.0816 | APE9-dist-in | 3.8112 | None | None | None | XRAY | 2.59 | 0.187 | 0.222 | A | 318.0 | 297.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj8 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ8B | Q3UHJ0 | 26 | 330 | 959.0 | YFV:401,PG6:402 | Type1,Allosteric | Active | DFGin | 6.1715 | 13.5947 | BLAminus | -125.6, -179.39 | 58.59, 102.41 | -105.91, 18.84 | 291.4, 96.74 | -62.2, -32.16 | in-in | in | 8.5892 | Saltbr-in | 2.8156 | HRD-in | -63.34, -43.99 | 65.76, 0.54 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8659 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.14, -12.1 | APE9-dihe-na | -116.75, 157.99 | APE8-dihe-in | -101.55, 119.49 | APE8-rot-in | 301.75 | APE67-dihe-in | -54.59, -29.22 | -43.63, -50.74 | APE12-dist-in | 12.1253 | APE11-dist-in | 8.5316 | APE10-dist-in | 4.1081 | APE9-dist-in | 3.8064 | None | None | None | XRAY | 2.59 | 0.187 | 0.222 | B | 318.0 | 305.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj8 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7LVIA | Q3UHJ0 | 34 | 330 | 959.0 | YFY:401 | Type1 | Inactive | DFGin | 6.2747 | 13.1608 | ABAminus | -90.42, -24.8 | -129.94, 143.17 | -139.29, 27.72 | 306.54, 92.44 | -75.37, -6.08 | in-in | in | 8.7052 | Saltbr-in | 2.9639 | HRD-in | -66.79, -49.03 | 71.63, -3.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.809 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -105.14, -3.93 | APE9-dihe-na | -125.59, 156.06 | APE8-dihe-in | -100.72, 117.66 | APE8-rot-in | 307.66 | APE67-dihe-in | -52.98, -27.5 | -41.63, -52.86 | APE12-dist-in | 12.0745 | APE11-dist-in | 8.5387 | APE10-dist-in | 4.2106 | APE9-dist-in | 3.7825 | None | None | None | XRAY | 2.2 | 0.219 | 0.241 | A | 318.0 | 294.0 | 3 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7lvi | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AAK1 | AAK1_MOUSE | 7LVHA | Q3UHJ0 | 34 | 328 | 959.0 | YFS:401 | Type1 | Active | DFGin | 6.3815 | 13.1586 | BLAminus | -99.27, -147.3 | 14.04, 114.8 | -121.99, 26.42 | 298.51, 87.91 | -70.89, -12.69 | in-in | in | 8.6326 | Saltbr-in | 2.9865 | HRD-in | -65.25, -42.59 | 66.7, -3.41 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9339 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.0, -6.79 | APE9-dihe-na | -118.74, 158.73 | APE8-dihe-in | -102.63, 127.81 | APE8-rot-in | 327.57 | APE67-dihe-in | -51.65, -23.05 | -49.85, -58.32 | APE12-dist-in | 12.2326 | APE11-dist-in | 8.6319 | APE10-dist-in | 4.2873 | APE9-dist-in | 3.7712 | None | None | None | XRAY | 2.65 | 0.267 | 0.299 | A | 318.0 | 284.0 | 11 | 36 | 34 | 2 | [[46, 313]] | 1.0 | 7lvh | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7LVHB | Q3UHJ0 | 35 | 329 | 959.0 | YFV:401 | Type1 | Active | DFGin | 6.305 | 13.462 | BLAminus | -109.39, -171.27 | 52.7, 102.9 | -109.75, 14.5 | 296.74, 93.05 | -60.15, -20.34 | in-in | in | 8.5725 | Saltbr-in | 2.9247 | HRD-in | -64.33, -41.66 | 66.46, -2.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.927 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.01, -10.47 | APE9-dihe-na | -112.81, 152.03 | APE8-dihe-in | -104.75, 117.86 | APE8-rot-in | 298.94 | APE67-dihe-in | -52.25, -35.41 | -40.96, -54.57 | APE12-dist-in | 12.4236 | APE11-dist-in | 8.6752 | APE10-dist-in | 4.2649 | APE9-dist-in | 3.8852 | None | None | None | XRAY | 2.65 | 0.267 | 0.299 | B | 318.0 | 281.0 | 14 | 36 | 34 | 2 | [[46, 313]] | 1.0 | 7lvh | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7LVIB | Q3UHJ0 | 35 | 330 | 959.0 | YFV:401 | Type1 | Active | DFGin | 6.5554 | 13.9557 | BLAminus | -120.74, -177.87 | 58.36, 103.46 | -109.53, 15.49 | 286.96, 91.82 | -62.65, -18.35 | in-in | in | 8.6464 | Saltbr-in | 2.9382 | HRD-in | -65.69, -47.95 | 71.36, -2.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7984 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.16, -5.91 | APE9-dihe-na | -123.61, 155.71 | APE8-dihe-in | -99.3, 117.77 | APE8-rot-in | 306.22 | APE67-dihe-in | -52.8, -28.0 | -40.05, -53.5 | APE12-dist-in | 12.1358 | APE11-dist-in | 8.5899 | APE10-dist-in | 4.2334 | APE9-dist-in | 3.7808 | None | None | None | XRAY | 2.2 | 0.219 | 0.241 | B | 318.0 | 288.0 | 8 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7lvi | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ6A | Q3UHJ0 | 26 | 330 | 959.0 | YFV:401 | Type1 | Active | DFGin | 6.5122 | 13.3768 | BLAminus | -125.62, 169.71 | 67.71, 96.16 | -104.68, 24.3 | 300.02, 93.63 | -68.93, -22.4 | in-in | in | 8.5967 | Saltbr-in | 2.7099 | HRD-in | -65.12, -47.31 | 74.51, -5.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8935 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -105.26, -12.99 | APE9-dihe-na | -116.7, 155.82 | APE8-dihe-in | -97.42, 121.54 | APE8-rot-in | 304.46 | APE67-dihe-in | -58.17, -28.42 | -45.34, -49.66 | APE12-dist-in | 12.1363 | APE11-dist-in | 8.6182 | APE10-dist-in | 4.2728 | APE9-dist-in | 3.6627 | None | None | None | XRAY | 2.132 | 0.202 | 0.215 | A | 318.0 | 305.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj6 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ6B | Q3UHJ0 | 32 | 330 | 959.0 | 5OI:401 | Type1 | Active | DFGin | 6.386 | 13.2644 | BLAminus | -136.98, -179.6 | 61.47, 90.79 | -102.58, 19.8 | 300.28, 93.44 | -74.01, -20.13 | in-in | in | 8.7043 | Saltbr-in | 2.7308 | HRD-in | -65.76, -48.0 | 74.66, -11.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8975 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.51, -10.49 | APE9-dihe-na | -120.36, 163.0 | APE8-dihe-in | -104.78, 122.31 | APE8-rot-in | 303.78 | APE67-dihe-in | -58.21, -28.47 | -45.49, -49.71 | APE12-dist-in | 11.9714 | APE11-dist-in | 8.4144 | APE10-dist-in | 4.1372 | APE9-dist-in | 3.7792 | None | None | None | XRAY | 2.132 | 0.202 | 0.215 | B | 318.0 | 299.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj6 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ7A | Q3UHJ0 | 26 | 330 | 959.0 | 5P6:401 | Type1 | Active | DFGin | 6.4175 | 13.2295 | BLAminus | -119.48, 174.96 | 57.07, 109.64 | -122.04, 21.88 | 302.38, 85.37 | -70.96, -15.13 | in-in | in | 8.8767 | Saltbr-in | 2.7471 | HRD-in | -69.47, -41.35 | 71.48, -9.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9302 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.51, -3.09 | APE9-dihe-na | -122.59, 149.49 | APE8-dihe-in | -97.34, 124.1 | APE8-rot-in | 304.72 | APE67-dihe-in | -57.28, -27.01 | -46.87, -50.73 | APE12-dist-in | 12.1476 | APE11-dist-in | 8.4871 | APE10-dist-in | 4.133 | APE9-dist-in | 3.7038 | None | None | None | XRAY | 2.124 | 0.23 | 0.241 | A | 318.0 | 304.0 | 1 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj7 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ7B | Q3UHJ0 | 31 | 330 | 959.0 | 5P6:401 | Type1 | Active | DFGin | 6.0891 | 13.1308 | BLAminus | -124.6, -178.84 | 57.9, 88.94 | -99.65, 26.07 | 303.29, 101.38 | -78.17, -15.56 | in-in | in | 8.8917 | Saltbr-in | 2.7552 | HRD-in | -71.2, -45.26 | 74.74, -14.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9313 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.73, -6.79 | APE9-dihe-na | -120.3, 157.4 | APE8-dihe-in | -99.84, 124.85 | APE8-rot-in | 305.17 | APE67-dihe-in | -58.1, -26.76 | -48.79, -48.64 | APE12-dist-in | 12.0925 | APE11-dist-in | 8.4564 | APE10-dist-in | 4.1132 | APE9-dist-in | 3.8598 | None | None | None | XRAY | 2.124 | 0.23 | 0.241 | B | 318.0 | 300.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj7 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ8A | Q3UHJ0 | 33 | 329 | 959.0 | 5QI:401,PG6:402 | Type1,Allosteric | Active | DFGin | 5.8996 | 12.8884 | BLAminus | -133.43, 178.44 | 53.42, 101.65 | -103.66, 23.97 | 304.98, 112.99 | -67.68, -29.68 | in-in | in | 8.3964 | Saltbr-in | 2.7456 | HRD-in | -63.24, -44.02 | 66.63, -0.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.5201 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.11, -10.27 | APE9-dihe-na | -117.76, 158.13 | APE8-dihe-in | -102.68, 119.66 | APE8-rot-in | 301.04 | APE67-dihe-in | -54.01, -28.74 | -43.37, -51.03 | APE12-dist-in | 12.1372 | APE11-dist-in | 8.4799 | APE10-dist-in | 4.0816 | APE9-dist-in | 3.8112 | None | None | None | XRAY | 2.59 | 0.187 | 0.222 | A | 318.0 | 297.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj8 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7RJ8B | Q3UHJ0 | 26 | 330 | 959.0 | YFV:401,PG6:402 | Type1,Allosteric | Active | DFGin | 6.1715 | 13.5947 | BLAminus | -125.6, -179.39 | 58.59, 102.41 | -105.91, 18.84 | 291.4, 96.74 | -62.2, -32.16 | in-in | in | 8.5892 | Saltbr-in | 2.8156 | HRD-in | -63.34, -43.99 | 65.76, 0.54 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8659 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.14, -12.1 | APE9-dihe-na | -116.75, 157.99 | APE8-dihe-in | -101.55, 119.49 | APE8-rot-in | 301.75 | APE67-dihe-in | -54.59, -29.22 | -43.63, -50.74 | APE12-dist-in | 12.1253 | APE11-dist-in | 8.5316 | APE10-dist-in | 4.1081 | APE9-dist-in | 3.8064 | None | None | None | XRAY | 2.59 | 0.187 | 0.222 | B | 318.0 | 305.0 | 0 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7rj8 | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |
| AAK1 | AAK1_MOUSE | 7LVIA | Q3UHJ0 | 34 | 330 | 959.0 | YFY:401 | Type1 | Inactive | DFGin | 6.2747 | 13.1608 | ABAminus | -90.42, -24.8 | -129.94, 143.17 | -139.29, 27.72 | 306.54, 92.44 | -75.37, -6.08 | in-in | in | 8.7052 | Saltbr-in | 2.9639 | HRD-in | -66.79, -49.03 | 71.63, -3.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.809 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -105.14, -3.93 | APE9-dihe-na | -125.59, 156.06 | APE8-dihe-in | -100.72, 117.66 | APE8-rot-in | 307.66 | APE67-dihe-in | -52.98, -27.5 | -41.63, -52.86 | APE12-dist-in | 12.0745 | APE11-dist-in | 8.5387 | APE10-dist-in | 4.2106 | APE9-dist-in | 3.7825 | None | None | None | XRAY | 2.2 | 0.219 | 0.241 | A | 318.0 | 294.0 | 3 | 36 | 36 | 0 | [[46, 313]] | 1.0 | 7lvi | Mus musculus | OTHER_AAK1_MOUSE | OTHER | 6.7e-41 | 146.7 | 3.0 | 254.0 | 252.0 | 193 | 194 | 195 | 197 | 199 | 74 | 90 | 94 | 173 | 175 | 174 | 176.0 | 244 | 229 | 224 | 223 | 222 | 221 | 220 | 219 | 218 | 127 | AP2-associated protein kinase 1 |