| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TKL | TGFBR1 | TGFR1_HUMAN | AF-P36897-K1A | P36897 | 197 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.0972 | 12.6974 | BLAminus | -127.47, -177.39 | 59.98, 50.67 | -75.64, 9.99 | 303.25, 0.83 | -67.03, -14.65 | in-in | in | 7.7504 | Saltbr-in | 2.6308 | HRD-in | -79.18, -43.89 | 66.79, -8.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0147 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.74, 159.13 | APE9-dihe-na | 99.19, -175.01 | APE8-dihe-in | -81.52, 117.2 | APE8-rot-in | 304.32 | APE67-dihe-in | -58.11, -28.29 | -49.21, -42.7 | APE12-dist-in | 13.0338 | APE11-dist-in | 12.4755 | APE10-dist-in | 6.3484 | APE9-dist-in | 3.7811 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306.0 | 306.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | AF-P36897-K1 | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | AF-P36897-K3A | P36897 | 197 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.3884 | 12.8818 | BLAminus | -127.89, -179.35 | 58.97, 55.86 | -76.18, 6.96 | 301.47, 0.09 | -63.41, -19.74 | in-in | in | 8.0954 | Saltbr-in | 2.6745 | HRD-in | -77.05, -40.27 | 65.4, -16.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8499 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -117.36, 158.96 | APE9-dihe-na | 107.71, -175.1 | APE8-dihe-in | -94.3, 114.61 | APE8-rot-in | 303.53 | APE67-dihe-in | -61.67, -24.01 | -41.02, -46.98 | APE12-dist-in | 11.2123 | APE11-dist-in | 11.8142 | APE10-dist-in | 5.9249 | APE9-dist-in | 3.7002 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306.0 | 306.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | AF-P36897-K3 | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TKL | TGFBR1 | TGFR1_HUMAN | AF-P36897-K1A | P36897 | 197 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.0972 | 12.6974 | BLAminus | -127.47, -177.39 | 59.98, 50.67 | -75.64, 9.99 | 303.25, 0.83 | -67.03, -14.65 | in-in | in | 7.7504 | Saltbr-in | 2.6308 | HRD-in | -79.18, -43.89 | 66.79, -8.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0147 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.74, 159.13 | APE9-dihe-na | 99.19, -175.01 | APE8-dihe-in | -81.52, 117.2 | APE8-rot-in | 304.32 | APE67-dihe-in | -58.11, -28.29 | -49.21, -42.7 | APE12-dist-in | 13.0338 | APE11-dist-in | 12.4755 | APE10-dist-in | 6.3484 | APE9-dist-in | 3.7811 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306.0 | 306.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | AF-P36897-K1 | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| TKL | TGFBR1 | TGFR1_HUMAN | AF-P36897-K3A | P36897 | 197 | 502 | 503.0 | No_ligand | No_ligand | Active | DFGin | 6.3884 | 12.8818 | BLAminus | -127.89, -179.35 | 58.97, 55.86 | -76.18, 6.96 | 301.47, 0.09 | -63.41, -19.74 | in-in | in | 8.0954 | Saltbr-in | 2.6745 | HRD-in | -77.05, -40.27 | 65.4, -16.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8499 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -117.36, 158.96 | APE9-dihe-na | 107.71, -175.1 | APE8-dihe-in | -94.3, 114.61 | APE8-rot-in | 303.53 | APE67-dihe-in | -61.67, -24.01 | -41.02, -46.98 | APE12-dist-in | 11.2123 | APE11-dist-in | 11.8142 | APE10-dist-in | 5.9249 | APE9-dist-in | 3.7002 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306.0 | 306.0 | 0 | 32 | 32 | 0 | [[205, 494]] | 1.0 | AF-P36897-K3 | Homo sapiens | TKL_TGFBR1_HUMAN | TKL | 3.3e-85 | 291.7 | 3.0 | 266.0 | 264.0 | 350 | 351 | 352 | 354 | 356 | 232 | 245 | 249 | 330 | 332 | 331 | 333.0 | 400 | 382 | 377 | 376 | 375 | 374 | 373 | 372 | 371 | 281 | TGF-beta receptor type-1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|