| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK3 | ARBK2_HUMAN | AF-P35626-K1A | P35626 | 183 | 461 | 688.0 | No_ligand | No_ligand | Active | DFGin | 5.3893 | 12.9794 | BLAminus | -119.85, -177.05 | 47.66, 71.7 | -81.78, 19.84 | 282.66, 77.07 | -60.27, -30.98 | in-in | in | 8.4444 | Saltbr-in | 2.574 | HRD-in | -79.78, -43.12 | 66.85, 1.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8539 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.85, 154.0 | APE9-dihe-na | 126.52, 172.74 | APE8-dihe-in | -77.57, 128.03 | APE8-rot-in | 302.33 | APE67-dihe-inflip | 86.21, -2.04 | -52.74, 135.57 | APE12-dist-in | 9.228 | APE11-dist-in | 12.0585 | APE10-dist-in | 6.1471 | APE9-dist-in | 3.4943 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | AF-P35626-K1 | AGC_GRK3_HUMAN | AGC | 1e-79 | 273.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | G protein-coupled receptor kinase 3 |
| AGC | GRK3 | ARBK2_HUMAN | AF-P35626-K3A | P35626 | 183 | 461 | 688.0 | No_ligand | No_ligand | Active | DFGin | 5.3365 | 12.9662 | BLAminus | -127.84, 178.42 | 53.44, 63.01 | -72.34, 17.54 | 287.43, 91.74 | -61.73, -26.86 | in-in | in | 8.5862 | Saltbr-in | 2.5735 | HRD-in | -86.58, -43.9 | 68.67, 3.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8449 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.82, 153.69 | APE9-dihe-na | 128.92, -164.53 | APE8-dihe-in | -101.52, 124.31 | APE8-rot-in | 298.48 | APE67-dihe-inflip | 88.79, 1.53 | -53.76, 131.32 | APE12-dist-in | 9.0927 | APE11-dist-in | 11.8401 | APE10-dist-in | 5.9226 | APE9-dist-in | 3.1954 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | AF-P35626-K3 | AGC_GRK3_HUMAN | AGC | 1e-79 | 273.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | G protein-coupled receptor kinase 3 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK3 | ARBK2_HUMAN | AF-P35626-K1A | P35626 | 183 | 461 | 688.0 | No_ligand | No_ligand | Active | DFGin | 5.3893 | 12.9794 | BLAminus | -119.85, -177.05 | 47.66, 71.7 | -81.78, 19.84 | 282.66, 77.07 | -60.27, -30.98 | in-in | in | 8.4444 | Saltbr-in | 2.574 | HRD-in | -79.78, -43.12 | 66.85, 1.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8539 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.85, 154.0 | APE9-dihe-na | 126.52, 172.74 | APE8-dihe-in | -77.57, 128.03 | APE8-rot-in | 302.33 | APE67-dihe-inflip | 86.21, -2.04 | -52.74, 135.57 | APE12-dist-in | 9.228 | APE11-dist-in | 12.0585 | APE10-dist-in | 6.1471 | APE9-dist-in | 3.4943 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | AF-P35626-K1 | Homo sapiens | AGC_GRK3_HUMAN | AGC | 1e-79 | 273.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | G protein-coupled receptor kinase 3 |
| AGC | GRK3 | ARBK2_HUMAN | AF-P35626-K3A | P35626 | 183 | 461 | 688.0 | No_ligand | No_ligand | Active | DFGin | 5.3365 | 12.9662 | BLAminus | -127.84, 178.42 | 53.44, 63.01 | -72.34, 17.54 | 287.43, 91.74 | -61.73, -26.86 | in-in | in | 8.5862 | Saltbr-in | 2.5735 | HRD-in | -86.58, -43.9 | 68.67, 3.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8449 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.82, 153.69 | APE9-dihe-na | 128.92, -164.53 | APE8-dihe-in | -101.52, 124.31 | APE8-rot-in | 298.48 | APE67-dihe-inflip | 88.79, 1.53 | -53.76, 131.32 | APE12-dist-in | 9.0927 | APE11-dist-in | 11.8401 | APE10-dist-in | 5.9226 | APE9-dist-in | 3.1954 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | AF-P35626-K3 | Homo sapiens | AGC_GRK3_HUMAN | AGC | 1e-79 | 273.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | G protein-coupled receptor kinase 3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|