| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK3 | MK03_HUMAN | AF-P27361-K1A | P27361 | 34 | 338 | 379.0 | No_ligand | No_ligand | Active | DFGin | 6.5927 | 14.8959 | BLAminus | -130.53, -179.67 | 55.56, 73.68 | -81.57, 15.4 | 283.43, 73.42 | -60.15, -27.17 | in-in | in | 9.0976 | Saltbr-in | 2.6988 | HRD-in | -71.43, -46.13 | 64.54, 6.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8631 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -74.91, 170.97 | APE9-dihe-na | 59.86, 147.58 | APE8-dihe-in | -63.62, 134.74 | APE8-rot-in | 298.27 | APE67-dihe-in | -68.94, -17.88 | -46.37, -48.07 | APE12-dist-in | 12.835 | APE11-dist-in | 11.3255 | APE10-dist-in | 6.8179 | APE9-dist-in | 3.0367 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 305.0 | 305.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | AF-P27361-K1 | CMGC_MAPK3_HUMAN | CMGC | 1.5e-87 | 299.6 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| CMGC | MAPK3 | MK03_HUMAN | AF-P27361-K3A | P27361 | 34 | 338 | 379.0 | No_ligand | No_ligand | Active | DFGin | 6.5353 | 14.6344 | BLAminus | -133.14, -176.56 | 56.67, 65.23 | -76.5, 14.43 | 283.46, 73.65 | -63.2, -17.33 | in-in | in | 9.0366 | Saltbr-in | 2.6885 | HRD-in | -77.08, -46.07 | 62.9, 16.83 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8517 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -69.1, 168.93 | APE9-dihe-na | 59.76, 143.47 | APE8-dihe-in | -62.52, 135.83 | APE8-rot-in | 298.7 | APE67-dihe-in | -69.69, -17.66 | -48.0, -47.1 | APE12-dist-in | 12.4845 | APE11-dist-in | 11.0788 | APE10-dist-in | 6.6158 | APE9-dist-in | 3.0598 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 305.0 | 305.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | AF-P27361-K3 | CMGC_MAPK3_HUMAN | CMGC | 1.5e-87 | 299.6 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK3 | MK03_HUMAN | AF-P27361-K1A | P27361 | 34 | 338 | 379.0 | No_ligand | No_ligand | Active | DFGin | 6.5927 | 14.8959 | BLAminus | -130.53, -179.67 | 55.56, 73.68 | -81.57, 15.4 | 283.43, 73.42 | -60.15, -27.17 | in-in | in | 9.0976 | Saltbr-in | 2.6988 | HRD-in | -71.43, -46.13 | 64.54, 6.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8631 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -74.91, 170.97 | APE9-dihe-na | 59.86, 147.58 | APE8-dihe-in | -63.62, 134.74 | APE8-rot-in | 298.27 | APE67-dihe-in | -68.94, -17.88 | -46.37, -48.07 | APE12-dist-in | 12.835 | APE11-dist-in | 11.3255 | APE10-dist-in | 6.8179 | APE9-dist-in | 3.0367 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 305.0 | 305.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | AF-P27361-K1 | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 1.5e-87 | 299.6 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| CMGC | MAPK3 | MK03_HUMAN | AF-P27361-K3A | P27361 | 34 | 338 | 379.0 | No_ligand | No_ligand | Active | DFGin | 6.5353 | 14.6344 | BLAminus | -133.14, -176.56 | 56.67, 65.23 | -76.5, 14.43 | 283.46, 73.65 | -63.2, -17.33 | in-in | in | 9.0366 | Saltbr-in | 2.6885 | HRD-in | -77.08, -46.07 | 62.9, 16.83 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8517 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -69.1, 168.93 | APE9-dihe-na | 59.76, 143.47 | APE8-dihe-in | -62.52, 135.83 | APE8-rot-in | 298.7 | APE67-dihe-in | -69.69, -17.66 | -48.0, -47.1 | APE12-dist-in | 12.4845 | APE11-dist-in | 11.0788 | APE10-dist-in | 6.6158 | APE9-dist-in | 3.0598 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 305.0 | 305.0 | 0 | 31 | 31 | 0 | [[42, 330]] | 1.0 | AF-P27361-K3 | Homo sapiens | CMGC_MAPK3_HUMAN | CMGC | 1.5e-87 | 299.6 | 1.0 | 301.0 | 301.0 | 183 | 184 | 185 | 187 | 189 | 71 | 88 | 92 | 163 | 165 | 164 | 166.0 | 227 | 214 | 209 | 208 | 207 | 206 | 205 | 204 | 203 | 123 | Mitogen-activated protein kinase 3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|