| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 9UHCA | P11362 | 458 | 764 | 822.0 | A1EPE:60801 | Type1 | Inactive | DFGin | 5.0891 | 13.5661 | BLAplus | -99.26, 163.63 | 67.92, 18.69 | -73.13, -23.6 | 54.69, 89.65 | -94.23, 7.24 | in-in | in | 8.5804 | Saltbr-in | 2.8372 | HRD-in | -81.76, -52.28 | 81.48, -12.21 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.6895 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -93.01, 148.62 | APE9-dihe-in | -107.23, 98.65 | APE8-dihe-out | -61.69, -18.58 | APE8-rot-na | 332.39 | APE67-dihe-in | -73.38, -10.07 | -53.51, -28.36 | APE12-dist-na | 17.3301 | APE11-dist-na | 19.8276 | APE10-dist-na | 16.8879 | APE9-dist-out | 11.0839 | None | None | None | XRAY | 1.88 | 0.173 | 0.205 | A | 310.0 | 307.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 9uhc | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 9UHCB | P11362 | 458 | 763 | 822.0 | A1EPE:60801 | Type1 | Inactive | DFGin | 5.2803 | 12.9098 | BLAplus | -104.01, 159.23 | 73.73, 21.61 | -75.73, -25.49 | 53.38, 87.57 | -92.18, 7.01 | in-in | in | 7.958 | Saltbr-in | 3.2635 | HRD-in | -83.66, -52.1 | 79.1, -13.65 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -84.36, 141.0 | APE9-dihe-in | -101.25, 92.23 | APE8-dihe-out | -59.77, -24.69 | APE8-rot-na | 330.6 | APE67-dihe-in | -77.73, -0.07 | -57.66, -24.92 | APE12-dist-na | 17.3904 | APE11-dist-na | 20.1263 | APE10-dist-na | 17.1087 | APE9-dist-out | 11.2956 | None | None | None | XRAY | 1.88 | 0.173 | 0.205 | B | 310.0 | 286.0 | 20 | 30 | 23 | 7 | [[478, 756]] | 1.0 | 9uhc | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 9UHCA | P11362 | 458 | 764 | 822.0 | A1EPE:60801 | Type1 | Inactive | DFGin | 5.0891 | 13.5661 | BLAplus | -99.26, 163.63 | 67.92, 18.69 | -73.13, -23.6 | 54.69, 89.65 | -94.23, 7.24 | in-in | in | 8.5804 | Saltbr-in | 2.8372 | HRD-in | -81.76, -52.28 | 81.48, -12.21 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.6895 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -93.01, 148.62 | APE9-dihe-in | -107.23, 98.65 | APE8-dihe-out | -61.69, -18.58 | APE8-rot-na | 332.39 | APE67-dihe-in | -73.38, -10.07 | -53.51, -28.36 | APE12-dist-na | 17.3301 | APE11-dist-na | 19.8276 | APE10-dist-na | 16.8879 | APE9-dist-out | 11.0839 | None | None | None | XRAY | 1.88 | 0.173 | 0.205 | A | 310.0 | 307.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 9uhc | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 9UHCB | P11362 | 458 | 763 | 822.0 | A1EPE:60801 | Type1 | Inactive | DFGin | 5.2803 | 12.9098 | BLAplus | -104.01, 159.23 | 73.73, 21.61 | -75.73, -25.49 | 53.38, 87.57 | -92.18, 7.01 | in-in | in | 7.958 | Saltbr-in | 3.2635 | HRD-in | -83.66, -52.1 | 79.1, -13.65 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -84.36, 141.0 | APE9-dihe-in | -101.25, 92.23 | APE8-dihe-out | -59.77, -24.69 | APE8-rot-na | 330.6 | APE67-dihe-in | -77.73, -0.07 | -57.66, -24.92 | APE12-dist-na | 17.3904 | APE11-dist-na | 20.1263 | APE10-dist-na | 17.1087 | APE9-dist-out | 11.2956 | None | None | None | XRAY | 1.88 | 0.173 | 0.205 | B | 310.0 | 286.0 | 20 | 30 | 23 | 7 | [[478, 756]] | 1.0 | 9uhc | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|