| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 9CD5A | P11362 | 465 | 764 | 822.0 | A1AV2:903 | Type1 | Inactive | DFGin | 5.1092 | 13.0413 | BLAplus | -119.69, 171.16 | 42.37, 48.64 | -93.51, -18.78 | 55.6, 81.67 | -108.27, 19.83 | in-in | in | 7.6418 | Saltbr-in | 3.4001 | HRD-in | -70.51, -58.43 | 92.5, -15.84 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -123.63, 147.65 | APE9-dihe-in | -93.38, 113.67 | APE8-dihe-out | -55.42, -20.8 | APE8-rot-na | 334.26 | APE67-dihe-in | -78.47, -7.11 | -58.87, -20.29 | APE12-dist-na | 21.398 | APE11-dist-na | 21.2383 | APE10-dist-na | 19.5201 | APE9-dist-out | 11.6083 | C488A,C584S | None | None | XRAY | 2.939 | 0.215 | 0.263 | A | 308.0 | 281.0 | 19 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 9cd5 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 9CD5B | P11362 | 460 | 764 | 822.0 | A1AV2:902 | Type1 | Inactive | DFGin | 5.1115 | 12.7756 | BLAplus | -119.68, 169.96 | 44.78, 47.92 | -93.2, -18.16 | 54.47, 80.79 | -103.83, 15.64 | in-in | in | 7.5897 | Saltbr-in | 3.2422 | HRD-in | -70.44, -57.93 | 92.25, -15.3 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9791 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -124.57, 148.55 | APE9-dihe-in | -93.36, 113.84 | APE8-dihe-out | -53.62, -20.73 | APE8-rot-na | 332.43 | APE67-dihe-in | -77.99, -7.05 | -59.24, -19.94 | APE12-dist-na | 21.0098 | APE11-dist-na | 20.993 | APE10-dist-na | 19.181 | APE9-dist-out | 11.5839 | C488A,C584S | None | None | XRAY | 2.939 | 0.215 | 0.263 | B | 308.0 | 289.0 | 16 | 30 | 28 | 2 | [[478, 756]] | 1.0 | 9cd5 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 9CD5A | P11362 | 465 | 764 | 822.0 | A1AV2:903 | Type1 | Inactive | DFGin | 5.1092 | 13.0413 | BLAplus | -119.69, 171.16 | 42.37, 48.64 | -93.51, -18.78 | 55.6, 81.67 | -108.27, 19.83 | in-in | in | 7.6418 | Saltbr-in | 3.4001 | HRD-in | -70.51, -58.43 | 92.5, -15.84 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -123.63, 147.65 | APE9-dihe-in | -93.38, 113.67 | APE8-dihe-out | -55.42, -20.8 | APE8-rot-na | 334.26 | APE67-dihe-in | -78.47, -7.11 | -58.87, -20.29 | APE12-dist-na | 21.398 | APE11-dist-na | 21.2383 | APE10-dist-na | 19.5201 | APE9-dist-out | 11.6083 | C488A,C584S | None | None | XRAY | 2.939 | 0.215 | 0.263 | A | 308.0 | 281.0 | 19 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 9cd5 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 9CD5B | P11362 | 460 | 764 | 822.0 | A1AV2:902 | Type1 | Inactive | DFGin | 5.1115 | 12.7756 | BLAplus | -119.68, 169.96 | 44.78, 47.92 | -93.2, -18.16 | 54.47, 80.79 | -103.83, 15.64 | in-in | in | 7.5897 | Saltbr-in | 3.2422 | HRD-in | -70.44, -57.93 | 92.25, -15.3 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9791 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -124.57, 148.55 | APE9-dihe-in | -93.36, 113.84 | APE8-dihe-out | -53.62, -20.73 | APE8-rot-na | 332.43 | APE67-dihe-in | -77.99, -7.05 | -59.24, -19.94 | APE12-dist-na | 21.0098 | APE11-dist-na | 20.993 | APE10-dist-na | 19.181 | APE9-dist-out | 11.5839 | C488A,C584S | None | None | XRAY | 2.939 | 0.215 | 0.263 | B | 308.0 | 289.0 | 16 | 30 | 28 | 2 | [[478, 756]] | 1.0 | 9cd5 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|