| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 8Y22A | P11362 | 459 | 762 | 822.0 | A1LW9:801 | Type1.5_Back | Inactive | DFGin | 5.1055 | 13.1789 | BLAplus | -113.25, 160.17 | 59.08, 34.01 | -79.21, -14.36 | 51.54, 87.27 | -109.45, 13.99 | in-in | in | 7.9825 | Saltbr-in | 2.7993 | HRD-in | -70.73, -44.6 | 68.63, 0.76 | in-out-out | SNCioo | out-out | ActLoopNT-out | 9.0288 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.2, 162.84 | APE9-dihe-in | -99.13, 115.53 | APE8-dihe-out | -57.19, -22.1 | APE8-rot-na | 334.84 | APE67-dihe-in | -76.32, -7.85 | -61.99, -21.14 | APE12-dist-na | 19.6449 | APE11-dist-na | 20.8827 | APE10-dist-na | 19.4784 | APE9-dist-out | 11.673 | C584S | None | None | XRAY | 2.792 | 0.197 | 0.26 | A | 308.0 | 288.0 | 16 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 8y22 | TYR_FGFR1_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 8Y22B | P11362 | 463 | 765 | 822.0 | A1LW9:801 | Type1.5_Back | Inactive | DFGin | 4.9267 | 13.3865 | BLAplus | -106.53, 165.87 | 49.37, 36.23 | -76.81, -19.53 | 50.68, 85.1 | -111.75, 14.63 | in-in | in | 8.1525 | Saltbr-in | 2.7928 | HRD-in | -74.01, -46.1 | 72.79, 0.75 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.596 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -115.29, 150.81 | APE9-dihe-in | -94.3, 115.55 | APE8-dihe-out | -59.96, -16.81 | APE8-rot-na | 335.23 | APE67-dihe-in | -86.59, -1.86 | -68.36, -9.3 | APE12-dist-na | 19.374 | APE11-dist-na | 20.9185 | APE10-dist-na | 19.1449 | APE9-dist-out | 11.7338 | C584S | None | None | XRAY | 2.792 | 0.197 | 0.26 | B | 308.0 | 291.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 8y22 | TYR_FGFR1_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 8Y22A | P11362 | 459 | 762 | 822.0 | A1LW9:801 | Type1.5_Back | Inactive | DFGin | 5.1055 | 13.1789 | BLAplus | -113.25, 160.17 | 59.08, 34.01 | -79.21, -14.36 | 51.54, 87.27 | -109.45, 13.99 | in-in | in | 7.9825 | Saltbr-in | 2.7993 | HRD-in | -70.73, -44.6 | 68.63, 0.76 | in-out-out | SNCioo | out-out | ActLoopNT-out | 9.0288 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.2, 162.84 | APE9-dihe-in | -99.13, 115.53 | APE8-dihe-out | -57.19, -22.1 | APE8-rot-na | 334.84 | APE67-dihe-in | -76.32, -7.85 | -61.99, -21.14 | APE12-dist-na | 19.6449 | APE11-dist-na | 20.8827 | APE10-dist-na | 19.4784 | APE9-dist-out | 11.673 | C584S | None | None | XRAY | 2.792 | 0.197 | 0.26 | A | 308.0 | 288.0 | 16 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 8y22 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 8Y22B | P11362 | 463 | 765 | 822.0 | A1LW9:801 | Type1.5_Back | Inactive | DFGin | 4.9267 | 13.3865 | BLAplus | -106.53, 165.87 | 49.37, 36.23 | -76.81, -19.53 | 50.68, 85.1 | -111.75, 14.63 | in-in | in | 8.1525 | Saltbr-in | 2.7928 | HRD-in | -74.01, -46.1 | 72.79, 0.75 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.596 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -115.29, 150.81 | APE9-dihe-in | -94.3, 115.55 | APE8-dihe-out | -59.96, -16.81 | APE8-rot-na | 335.23 | APE67-dihe-in | -86.59, -1.86 | -68.36, -9.3 | APE12-dist-na | 19.374 | APE11-dist-na | 20.9185 | APE10-dist-na | 19.1449 | APE9-dist-out | 11.7338 | C584S | None | None | XRAY | 2.792 | 0.197 | 0.26 | B | 308.0 | 291.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 8y22 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|