PDB: 8W38 — TYR FGFR2_HUMAN

Total number of chains: 4
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 4 100.0% 8W38A

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
TYR FGFR2 FGFR2_HUMAN 8W38A P21802 467 764 821.0 TZ0:801 Type1.5_Back Inactive DFGin 5.884 13.9387 BLAminus -141.73, -172.44 58.43, 85.09 -99.65, 33.03 296.5, 153.04 -60.44, -42.96 in-in in 7.7157 Saltbr-in 2.7302 HRD-in -67.46, -57.27 77.66, 6.76 in-in-out SNCiio in-out ActLoopNT-in 2.8529 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -102.69, 6.19 APE9-dihe-in -92.48, 138.52 APE8-dihe-in -67.31, 130.89 APE8-rot-na 342.55 APE67-dihe-in -76.49, 2.73 -63.26, -44.89 APE12-dist-na 9.9384 APE11-dist-na 10.8626 APE10-dist-na 7.1874 APE9-dist-in 4.84 N549D,D650V None None XRAY 2.6 0.337 0.359 A 324.0 298.0 0 30 30 0 [[481, 759]] 1.0 8w38 TYR_FGFR2_HUMAN TYR 1.5e-103 351.6 1.0 260.0 260.0 643 644 645 647 649 517 534 538 623 625 624 626.0 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8W38B P21802 467 764 821.0 TZ0:801 Type1.5_Back Inactive DFGin 5.9169 13.8673 BLAminus -141.61, -172.11 58.71, 84.88 -99.53, 33.01 296.86, 151.72 -60.67, -42.8 in-in in 7.6773 Saltbr-in 2.7365 HRD-in -66.89, -57.79 77.67, 7.38 in-in-out SNCiio in-out ActLoopNT-in 2.8537 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -102.73, 7.76 APE9-dihe-in -92.14, 138.79 APE8-dihe-in -66.97, 130.73 APE8-rot-na 341.51 APE67-dihe-in -76.67, 2.98 -63.37, -44.91 APE12-dist-na 9.7659 APE11-dist-na 10.7509 APE10-dist-na 7.1935 APE9-dist-in 4.8257 N549D,D650V None None XRAY 2.6 0.337 0.359 B 324.0 288.0 10 30 24 6 [[481, 759]] 1.0 8w38 TYR_FGFR2_HUMAN TYR 1.5e-103 351.6 1.0 260.0 260.0 643 644 645 647 649 517 534 538 623 625 624 626.0 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8W38C P21802 465 764 821.0 TZ0:801 Type1.5_Back Inactive DFGin 5.9054 14.0005 BLAminus -141.73, -172.23 58.36, 85.55 -99.69, 32.51 297.47, 150.87 -60.14, -43.03 in-in in 7.7655 Saltbr-in 2.7334 HRD-in -67.3, -57.38 78.5, 5.79 in-in-out SNCiio in-out ActLoopNT-in 2.8526 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -100.74, 8.72 APE9-dihe-in -90.56, 139.47 APE8-dihe-in -66.09, 130.7 APE8-rot-na 342.51 APE67-dihe-in -75.82, 2.85 -65.85, -41.6 APE12-dist-na 999.0 APE11-dist-na 10.6496 APE10-dist-na 7.2376 APE9-dist-in 4.7764 N549D,D650V None None XRAY 2.6 0.337 0.359 C 324.0 289.0 11 30 19 11 [[481, 759]] 1.0 8w38 TYR_FGFR2_HUMAN TYR 1.5e-103 351.6 1.0 260.0 260.0 643 644 645 647 649 517 534 538 623 625 624 626.0 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8W38D P21802 467 764 821.0 TZ0:800 Type1.5_Back Inactive DFGin 5.9583 13.994 BLAminus -141.63, -172.13 58.59, 85.21 -99.57, 33.16 297.38, 150.22 -60.22, -43.6 in-in in 7.7819 Saltbr-in 2.7642 HRD-in -66.88, -57.89 78.41, 5.63 in-in-out SNCiio in-out ActLoopNT-in 2.8509 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -100.9, 7.03 APE9-dihe-in -91.06, 139.7 APE8-dihe-in -66.27, 130.75 APE8-rot-na 343.36 APE67-dihe-in -75.84, 2.91 -65.4, -41.85 APE12-dist-na 999.0 APE11-dist-na 10.7499 APE10-dist-na 7.2202 APE9-dist-in 4.7939 N549D,D650V None None XRAY 2.6 0.337 0.359 D 324.0 271.0 27 30 19 11 [[481, 759]] 1.0 8w38 TYR_FGFR2_HUMAN TYR 1.5e-103 351.6 1.0 260.0 260.0 643 644 645 647 649 517 534 538 623 625 624 626.0 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2

PDB: 8W38 — TYR FGFR2_HUMAN

Total number of chains: 4
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 4 100.0% 8W38A

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
TYR FGFR2 FGFR2_HUMAN 8W38A P21802 467 764 821.0 TZ0:801 Type1.5_Back Inactive DFGin 5.884 13.9387 BLAminus -141.73, -172.44 58.43, 85.09 -99.65, 33.03 296.5, 153.04 -60.44, -42.96 in-in in 7.7157 Saltbr-in 2.7302 HRD-in -67.46, -57.27 77.66, 6.76 in-in-out SNCiio in-out ActLoopNT-in 2.8529 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -102.69, 6.19 APE9-dihe-in -92.48, 138.52 APE8-dihe-in -67.31, 130.89 APE8-rot-na 342.55 APE67-dihe-in -76.49, 2.73 -63.26, -44.89 APE12-dist-na 9.9384 APE11-dist-na 10.8626 APE10-dist-na 7.1874 APE9-dist-in 4.84 N549D,D650V None None XRAY 2.6 0.337 0.359 A 324.0 298.0 0 30 30 0 [[481, 759]] 1.0 8w38 Homo sapiens TYR_FGFR2_HUMAN TYR 1.5e-103 351.6 1.0 260.0 260.0 643 644 645 647 649 517 534 538 623 625 624 626.0 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8W38B P21802 467 764 821.0 TZ0:801 Type1.5_Back Inactive DFGin 5.9169 13.8673 BLAminus -141.61, -172.11 58.71, 84.88 -99.53, 33.01 296.86, 151.72 -60.67, -42.8 in-in in 7.6773 Saltbr-in 2.7365 HRD-in -66.89, -57.79 77.67, 7.38 in-in-out SNCiio in-out ActLoopNT-in 2.8537 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -102.73, 7.76 APE9-dihe-in -92.14, 138.79 APE8-dihe-in -66.97, 130.73 APE8-rot-na 341.51 APE67-dihe-in -76.67, 2.98 -63.37, -44.91 APE12-dist-na 9.7659 APE11-dist-na 10.7509 APE10-dist-na 7.1935 APE9-dist-in 4.8257 N549D,D650V None None XRAY 2.6 0.337 0.359 B 324.0 288.0 10 30 24 6 [[481, 759]] 1.0 8w38 Homo sapiens TYR_FGFR2_HUMAN TYR 1.5e-103 351.6 1.0 260.0 260.0 643 644 645 647 649 517 534 538 623 625 624 626.0 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8W38C P21802 465 764 821.0 TZ0:801 Type1.5_Back Inactive DFGin 5.9054 14.0005 BLAminus -141.73, -172.23 58.36, 85.55 -99.69, 32.51 297.47, 150.87 -60.14, -43.03 in-in in 7.7655 Saltbr-in 2.7334 HRD-in -67.3, -57.38 78.5, 5.79 in-in-out SNCiio in-out ActLoopNT-in 2.8526 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -100.74, 8.72 APE9-dihe-in -90.56, 139.47 APE8-dihe-in -66.09, 130.7 APE8-rot-na 342.51 APE67-dihe-in -75.82, 2.85 -65.85, -41.6 APE12-dist-na 999.0 APE11-dist-na 10.6496 APE10-dist-na 7.2376 APE9-dist-in 4.7764 N549D,D650V None None XRAY 2.6 0.337 0.359 C 324.0 289.0 11 30 19 11 [[481, 759]] 1.0 8w38 Homo sapiens TYR_FGFR2_HUMAN TYR 1.5e-103 351.6 1.0 260.0 260.0 643 644 645 647 649 517 534 538 623 625 624 626.0 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2
TYR FGFR2 FGFR2_HUMAN 8W38D P21802 467 764 821.0 TZ0:800 Type1.5_Back Inactive DFGin 5.9583 13.994 BLAminus -141.63, -172.13 58.59, 85.21 -99.57, 33.16 297.38, 150.22 -60.22, -43.6 in-in in 7.7819 Saltbr-in 2.7642 HRD-in -66.88, -57.89 78.41, 5.63 in-in-out SNCiio in-out ActLoopNT-in 2.8509 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -100.9, 7.03 APE9-dihe-in -91.06, 139.7 APE8-dihe-in -66.27, 130.75 APE8-rot-na 343.36 APE67-dihe-in -75.84, 2.91 -65.4, -41.85 APE12-dist-na 999.0 APE11-dist-na 10.7499 APE10-dist-na 7.2202 APE9-dist-in 4.7939 N549D,D650V None None XRAY 2.6 0.337 0.359 D 324.0 271.0 27 30 19 11 [[481, 759]] 1.0 8w38 Homo sapiens TYR_FGFR2_HUMAN TYR 1.5e-103 351.6 1.0 260.0 260.0 643 644 645 647 649 517 534 538 623 625 624 626.0 685 673 668 667 666 665 664 663 662 565 Fibroblast growth factor receptor 2

PDB: 8W38 — TYR FGFR2_HUMAN

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name