| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8W38A | P21802 | 467 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.884 | 13.9387 | BLAminus | -141.73, -172.44 | 58.43, 85.09 | -99.65, 33.03 | 296.5, 153.04 | -60.44, -42.96 | in-in | in | 7.7157 | Saltbr-in | 2.7302 | HRD-in | -67.46, -57.27 | 77.66, 6.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8529 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.69, 6.19 | APE9-dihe-in | -92.48, 138.52 | APE8-dihe-in | -67.31, 130.89 | APE8-rot-na | 342.55 | APE67-dihe-in | -76.49, 2.73 | -63.26, -44.89 | APE12-dist-na | 9.9384 | APE11-dist-na | 10.8626 | APE10-dist-na | 7.1874 | APE9-dist-in | 4.84 | N549D,D650V | None | None | XRAY | 2.6 | 0.337 | 0.359 | A | 324.0 | 298.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8w38 | TYR_FGFR2_HUMAN | TYR | 1.5e-103 | 351.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W38B | P21802 | 467 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.9169 | 13.8673 | BLAminus | -141.61, -172.11 | 58.71, 84.88 | -99.53, 33.01 | 296.86, 151.72 | -60.67, -42.8 | in-in | in | 7.6773 | Saltbr-in | 2.7365 | HRD-in | -66.89, -57.79 | 77.67, 7.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8537 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.73, 7.76 | APE9-dihe-in | -92.14, 138.79 | APE8-dihe-in | -66.97, 130.73 | APE8-rot-na | 341.51 | APE67-dihe-in | -76.67, 2.98 | -63.37, -44.91 | APE12-dist-na | 9.7659 | APE11-dist-na | 10.7509 | APE10-dist-na | 7.1935 | APE9-dist-in | 4.8257 | N549D,D650V | None | None | XRAY | 2.6 | 0.337 | 0.359 | B | 324.0 | 288.0 | 10 | 30 | 24 | 6 | [[481, 759]] | 1.0 | 8w38 | TYR_FGFR2_HUMAN | TYR | 1.5e-103 | 351.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W38C | P21802 | 465 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.9054 | 14.0005 | BLAminus | -141.73, -172.23 | 58.36, 85.55 | -99.69, 32.51 | 297.47, 150.87 | -60.14, -43.03 | in-in | in | 7.7655 | Saltbr-in | 2.7334 | HRD-in | -67.3, -57.38 | 78.5, 5.79 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8526 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.74, 8.72 | APE9-dihe-in | -90.56, 139.47 | APE8-dihe-in | -66.09, 130.7 | APE8-rot-na | 342.51 | APE67-dihe-in | -75.82, 2.85 | -65.85, -41.6 | APE12-dist-na | 999.0 | APE11-dist-na | 10.6496 | APE10-dist-na | 7.2376 | APE9-dist-in | 4.7764 | N549D,D650V | None | None | XRAY | 2.6 | 0.337 | 0.359 | C | 324.0 | 289.0 | 11 | 30 | 19 | 11 | [[481, 759]] | 1.0 | 8w38 | TYR_FGFR2_HUMAN | TYR | 1.5e-103 | 351.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W38D | P21802 | 467 | 764 | 821.0 | TZ0:800 | Type1.5_Back | Inactive | DFGin | 5.9583 | 13.994 | BLAminus | -141.63, -172.13 | 58.59, 85.21 | -99.57, 33.16 | 297.38, 150.22 | -60.22, -43.6 | in-in | in | 7.7819 | Saltbr-in | 2.7642 | HRD-in | -66.88, -57.89 | 78.41, 5.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8509 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.9, 7.03 | APE9-dihe-in | -91.06, 139.7 | APE8-dihe-in | -66.27, 130.75 | APE8-rot-na | 343.36 | APE67-dihe-in | -75.84, 2.91 | -65.4, -41.85 | APE12-dist-na | 999.0 | APE11-dist-na | 10.7499 | APE10-dist-na | 7.2202 | APE9-dist-in | 4.7939 | N549D,D650V | None | None | XRAY | 2.6 | 0.337 | 0.359 | D | 324.0 | 271.0 | 27 | 30 | 19 | 11 | [[481, 759]] | 1.0 | 8w38 | TYR_FGFR2_HUMAN | TYR | 1.5e-103 | 351.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8W38A | P21802 | 467 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.884 | 13.9387 | BLAminus | -141.73, -172.44 | 58.43, 85.09 | -99.65, 33.03 | 296.5, 153.04 | -60.44, -42.96 | in-in | in | 7.7157 | Saltbr-in | 2.7302 | HRD-in | -67.46, -57.27 | 77.66, 6.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8529 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.69, 6.19 | APE9-dihe-in | -92.48, 138.52 | APE8-dihe-in | -67.31, 130.89 | APE8-rot-na | 342.55 | APE67-dihe-in | -76.49, 2.73 | -63.26, -44.89 | APE12-dist-na | 9.9384 | APE11-dist-na | 10.8626 | APE10-dist-na | 7.1874 | APE9-dist-in | 4.84 | N549D,D650V | None | None | XRAY | 2.6 | 0.337 | 0.359 | A | 324.0 | 298.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8w38 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 1.5e-103 | 351.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W38B | P21802 | 467 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.9169 | 13.8673 | BLAminus | -141.61, -172.11 | 58.71, 84.88 | -99.53, 33.01 | 296.86, 151.72 | -60.67, -42.8 | in-in | in | 7.6773 | Saltbr-in | 2.7365 | HRD-in | -66.89, -57.79 | 77.67, 7.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8537 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -102.73, 7.76 | APE9-dihe-in | -92.14, 138.79 | APE8-dihe-in | -66.97, 130.73 | APE8-rot-na | 341.51 | APE67-dihe-in | -76.67, 2.98 | -63.37, -44.91 | APE12-dist-na | 9.7659 | APE11-dist-na | 10.7509 | APE10-dist-na | 7.1935 | APE9-dist-in | 4.8257 | N549D,D650V | None | None | XRAY | 2.6 | 0.337 | 0.359 | B | 324.0 | 288.0 | 10 | 30 | 24 | 6 | [[481, 759]] | 1.0 | 8w38 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 1.5e-103 | 351.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W38C | P21802 | 465 | 764 | 821.0 | TZ0:801 | Type1.5_Back | Inactive | DFGin | 5.9054 | 14.0005 | BLAminus | -141.73, -172.23 | 58.36, 85.55 | -99.69, 32.51 | 297.47, 150.87 | -60.14, -43.03 | in-in | in | 7.7655 | Saltbr-in | 2.7334 | HRD-in | -67.3, -57.38 | 78.5, 5.79 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8526 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.74, 8.72 | APE9-dihe-in | -90.56, 139.47 | APE8-dihe-in | -66.09, 130.7 | APE8-rot-na | 342.51 | APE67-dihe-in | -75.82, 2.85 | -65.85, -41.6 | APE12-dist-na | 999.0 | APE11-dist-na | 10.6496 | APE10-dist-na | 7.2376 | APE9-dist-in | 4.7764 | N549D,D650V | None | None | XRAY | 2.6 | 0.337 | 0.359 | C | 324.0 | 289.0 | 11 | 30 | 19 | 11 | [[481, 759]] | 1.0 | 8w38 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 1.5e-103 | 351.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8W38D | P21802 | 467 | 764 | 821.0 | TZ0:800 | Type1.5_Back | Inactive | DFGin | 5.9583 | 13.994 | BLAminus | -141.63, -172.13 | 58.59, 85.21 | -99.57, 33.16 | 297.38, 150.22 | -60.22, -43.6 | in-in | in | 7.7819 | Saltbr-in | 2.7642 | HRD-in | -66.88, -57.89 | 78.41, 5.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8509 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -100.9, 7.03 | APE9-dihe-in | -91.06, 139.7 | APE8-dihe-in | -66.27, 130.75 | APE8-rot-na | 343.36 | APE67-dihe-in | -75.84, 2.91 | -65.4, -41.85 | APE12-dist-na | 999.0 | APE11-dist-na | 10.7499 | APE10-dist-na | 7.2202 | APE9-dist-in | 4.7939 | N549D,D650V | None | None | XRAY | 2.6 | 0.337 | 0.359 | D | 324.0 | 271.0 | 27 | 30 | 19 | 11 | [[481, 759]] | 1.0 | 8w38 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 1.5e-103 | 351.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|