| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR3 | FGFR3_HUMAN | 8UDUB | P22607 | 459 | 755 | 806.0 | WIQ:61002 | Type1.5_Front | Active | DFGin | 6.4209 | 14.4148 | BLAminus | -138.69, 176.26 | 64.2, 86.01 | -100.28, 24.84 | 287.71, 79.66 | -57.6, -41.09 | in-in | in | 8.1853 | Saltbr-in | 2.9464 | HRD-in | -71.69, -47.92 | 71.62, 0.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9471 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.88, 155.75 | APE9-dihe-in | -122.51, 89.95 | APE8-dihe-in | -81.37, 70.05 | APE8-rot-na | 30.61 | APE67-dihe-in | -66.22, -12.9 | -45.0, -50.18 | APE12-dist-na | 999.0 | APE11-dist-na | 7.6606 | APE10-dist-na | 8.4893 | APE9-dist-in | 7.717 | P572S,P573G | None | None | XRAY | 1.737 | 0.231 | 0.256 | B | 297.0 | 276.0 | 9 | 30 | 29 | 1 | [[472, 750]] | 1.0 | 8udu | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | 8UDUA | P22607 | 460 | 756 | 806.0 | WIQ:61002 | Type1.5_Back | Inactive | DFGin | 5.7614 | 13.5292 | BLBplus | -121.3, 171.32 | 71.72, 21.7 | -99.77, 166.76 | 66.11, 93.34 | 95.58, -59.45 | in-in | in | 7.9172 | Saltbr-in | 2.7343 | HRD-in | -77.2, -48.45 | 77.61, -12.83 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -71.65, 162.44 | APE9-dihe-in | -54.1, 129.25 | APE8-dihe-in | -83.64, 61.19 | APE8-rot-na | 34.62 | APE67-dihe-in | -73.43, -8.03 | -52.16, -35.97 | APE12-dist-na | 999.0 | APE11-dist-na | 14.2323 | APE10-dist-na | 17.7469 | APE9-dist-out | 8.253 | P572S,P573G | None | None | XRAY | 1.737 | 0.231 | 0.256 | A | 297.0 | 277.0 | 8 | 30 | 22 | 8 | [[472, 750]] | 1.0 | 8udu | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR3 | FGFR3_HUMAN | 8UDUB | P22607 | 459 | 755 | 806.0 | WIQ:61002 | Type1.5_Front | Active | DFGin | 6.4209 | 14.4148 | BLAminus | -138.69, 176.26 | 64.2, 86.01 | -100.28, 24.84 | 287.71, 79.66 | -57.6, -41.09 | in-in | in | 8.1853 | Saltbr-in | 2.9464 | HRD-in | -71.69, -47.92 | 71.62, 0.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9471 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.88, 155.75 | APE9-dihe-in | -122.51, 89.95 | APE8-dihe-in | -81.37, 70.05 | APE8-rot-na | 30.61 | APE67-dihe-in | -66.22, -12.9 | -45.0, -50.18 | APE12-dist-na | 999.0 | APE11-dist-na | 7.6606 | APE10-dist-na | 8.4893 | APE9-dist-in | 7.717 | P572S,P573G | None | None | XRAY | 1.737 | 0.231 | 0.256 | B | 297.0 | 276.0 | 9 | 30 | 29 | 1 | [[472, 750]] | 1.0 | 8udu | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | 8UDUA | P22607 | 460 | 756 | 806.0 | WIQ:61002 | Type1.5_Back | Inactive | DFGin | 5.7614 | 13.5292 | BLBplus | -121.3, 171.32 | 71.72, 21.7 | -99.77, 166.76 | 66.11, 93.34 | 95.58, -59.45 | in-in | in | 7.9172 | Saltbr-in | 2.7343 | HRD-in | -77.2, -48.45 | 77.61, -12.83 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -71.65, 162.44 | APE9-dihe-in | -54.1, 129.25 | APE8-dihe-in | -83.64, 61.19 | APE8-rot-na | 34.62 | APE67-dihe-in | -73.43, -8.03 | -52.16, -35.97 | APE12-dist-na | 999.0 | APE11-dist-na | 14.2323 | APE10-dist-na | 17.7469 | APE9-dist-out | 8.253 | P572S,P573G | None | None | XRAY | 1.737 | 0.231 | 0.256 | A | 297.0 | 277.0 | 8 | 30 | 22 | 8 | [[472, 750]] | 1.0 | 8udu | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|