| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8SWEA | P21802 | 468 | 765 | 821.0 | GSH:802,WXQ:803 | Allosteric,Type1 | Inactive | DFGin | 6.5842 | 14.4213 | BLAminus | -150.2, -171.84 | 53.84, 62.99 | -84.08, 24.59 | 289.03, 91.27 | -65.33, -29.69 | in-in | in | 7.6673 | Saltbr-in | 3.4776 | HRD-in | -78.34, -48.7 | 72.49, -5.74 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.935 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.6, 22.79 | APE9-dihe-in | -98.31, 134.63 | APE8-dihe-in | -56.2, 130.73 | APE8-rot-na | 335.99 | APE67-dihe-in | -78.04, -7.77 | -69.42, -32.87 | APE12-dist-na | 10.0826 | APE11-dist-na | 10.7199 | APE10-dist-na | 7.381 | APE9-dist-in | 4.8605 | None | None | None | XRAY | 2.24 | 0.212 | 0.25 | A | 316.0 | 284.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8swe | TYR_FGFR2_HUMAN | TYR | 2.6e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8SWEB | P21802 | 468 | 767 | 821.0 | WXQ:804 | Type1 | Inactive | DFGin | 6.3615 | 14.3904 | BLAminus | -138.39, -167.44 | 55.86, 63.6 | -85.72, 22.79 | 292.14, 86.9 | -64.13, -34.28 | in-out | in | 7.8403 | Saltbr-out | 3.6147 | HRD-in | -78.85, -51.07 | 77.2, -7.67 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.0233 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.42, 18.52 | APE9-dihe-in | -97.67, 132.33 | APE8-dihe-in | -56.79, 133.06 | APE8-rot-na | 333.48 | APE67-dihe-in | -69.86, -7.28 | -72.44, -38.73 | APE12-dist-na | 10.1012 | APE11-dist-na | 10.7967 | APE10-dist-na | 7.3183 | APE9-dist-in | 4.8919 | None | None | None | XRAY | 2.24 | 0.212 | 0.25 | B | 316.0 | 288.0 | 12 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8swe | TYR_FGFR2_HUMAN | TYR | 2.6e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8SWEA | P21802 | 468 | 765 | 821.0 | GSH:802,WXQ:803 | Allosteric,Type1 | Inactive | DFGin | 6.5842 | 14.4213 | BLAminus | -150.2, -171.84 | 53.84, 62.99 | -84.08, 24.59 | 289.03, 91.27 | -65.33, -29.69 | in-in | in | 7.6673 | Saltbr-in | 3.4776 | HRD-in | -78.34, -48.7 | 72.49, -5.74 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.935 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.6, 22.79 | APE9-dihe-in | -98.31, 134.63 | APE8-dihe-in | -56.2, 130.73 | APE8-rot-na | 335.99 | APE67-dihe-in | -78.04, -7.77 | -69.42, -32.87 | APE12-dist-na | 10.0826 | APE11-dist-na | 10.7199 | APE10-dist-na | 7.381 | APE9-dist-in | 4.8605 | None | None | None | XRAY | 2.24 | 0.212 | 0.25 | A | 316.0 | 284.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8swe | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.6e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8SWEB | P21802 | 468 | 767 | 821.0 | WXQ:804 | Type1 | Inactive | DFGin | 6.3615 | 14.3904 | BLAminus | -138.39, -167.44 | 55.86, 63.6 | -85.72, 22.79 | 292.14, 86.9 | -64.13, -34.28 | in-out | in | 7.8403 | Saltbr-out | 3.6147 | HRD-in | -78.85, -51.07 | 77.2, -7.67 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.0233 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.42, 18.52 | APE9-dihe-in | -97.67, 132.33 | APE8-dihe-in | -56.79, 133.06 | APE8-rot-na | 333.48 | APE67-dihe-in | -69.86, -7.28 | -72.44, -38.73 | APE12-dist-na | 10.1012 | APE11-dist-na | 10.7967 | APE10-dist-na | 7.3183 | APE9-dist-in | 4.8919 | None | None | None | XRAY | 2.24 | 0.212 | 0.25 | B | 316.0 | 288.0 | 12 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8swe | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.6e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|