| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8H75A | P21802 | 467 | 765 | 821.0 | KX0:1001 | Type1 | Inactive | DFGin | 7.2128 | 14.5852 | BLAminus | -154.63, 179.57 | 55.91, 54.1 | -74.79, -3.2 | 274.96, 68.76 | -58.48, -41.04 | in-out | in | 7.4173 | Saltbr-out | 4.8105 | HRD-out | -96.67, 103.01 | -67.39, -41.62 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.141 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -162.98, 72.34 | APE9-dihe-in | -137.73, 148.36 | APE8-dihe-in | -71.99, 141.14 | APE8-rot-na | 343.8 | APE67-dihe-in | -63.34, -38.73 | -70.52, -42.38 | APE12-dist-na | 13.0181 | APE11-dist-na | 9.4081 | APE10-dist-na | 7.3004 | APE9-dist-in | 6.8677 | None | PTR656 | PTR656 | XRAY | 3.75 | 0.216 | 0.238 | A | 312.0 | 285.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8h75 | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8H75B | P21802 | 467 | 764 | 821.0 | KX0:1001 | Type1 | Inactive | DFGin | 7.1136 | 15.3212 | BLAminus | -140.03, -170.55 | 50.75, 50.66 | -73.91, -10.21 | 273.73, 91.58 | -58.96, -39.4 | in-out | in | 7.4683 | Saltbr-out | 4.4362 | HRD-in | -64.7, -43.07 | 75.93, -2.73 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.3826 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -63.7, -40.57 | APE9-dihe-in | -143.97, 156.51 | APE8-dihe-in | -61.01, 137.3 | APE8-rot-na | 23.2 | APE67-dihe-in | -61.01, -38.56 | -64.05, -38.82 | APE12-dist-na | 14.0921 | APE11-dist-na | 11.2874 | APE10-dist-na | 7.4456 | APE9-dist-in | 5.7379 | None | PTR656 | PTR656 | XRAY | 3.75 | 0.216 | 0.238 | B | 312.0 | 283.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8h75 | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8H75C | P21802 | 467 | 763 | 821.0 | KX0:1001 | Type1 | Inactive | DFGin | 6.4145 | 13.9419 | BLAminus | -139.77, -171.25 | 51.94, 53.82 | -68.52, 7.4 | 288.78, 82.18 | -59.71, -35.71 | in-in | in | 7.7631 | Saltbr-in | 2.5787 | HRD-in | -64.69, -38.41 | 67.2, 3.13 | in-out-out | SNCioo | out-out | ActLoopNT-out | 3.7885 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -86.06, 23.54 | APE9-dihe-in | -123.01, 141.76 | APE8-dihe-in | -64.83, 140.92 | APE8-rot-na | 351.7 | APE67-dihe-in | -63.43, -39.45 | -65.53, -40.64 | APE12-dist-na | 10.7845 | APE11-dist-na | 10.9436 | APE10-dist-na | 7.5138 | APE9-dist-in | 5.3824 | None | PTR656 | PTR656 | XRAY | 3.75 | 0.216 | 0.238 | C | 312.0 | 275.0 | 22 | 30 | 24 | 6 | [[481, 759]] | 1.0 | 8h75 | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8H75D | P21802 | 467 | 764 | 821.0 | KX0:1001 | Type1 | Inactive | DFGin | 6.7191 | 14.0063 | BLAminus | -145.79, -169.72 | 52.31, 64.06 | -85.42, 2.67 | 285.45, 103.44 | -59.5, -38.29 | in-out | in | 7.6901 | Saltbr-out | 4.3568 | HRD-in | -66.94, -45.53 | 78.8, 0.63 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.389 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 55.78, 41.43 | APE9-dihe-in | -144.13, 151.96 | APE8-dihe-in | -70.01, 128.38 | APE8-rot-na | 29.85 | APE67-dihe-in | -54.94, -35.54 | -65.88, -42.6 | APE12-dist-na | 10.9944 | APE11-dist-na | 11.0526 | APE10-dist-na | 8.8294 | APE9-dist-in | 5.7588 | None | PTR656 | PTR656 | XRAY | 3.75 | 0.216 | 0.238 | D | 312.0 | 277.0 | 21 | 30 | 26 | 4 | [[481, 759]] | 1.0 | 8h75 | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8H75A | P21802 | 467 | 765 | 821.0 | KX0:1001 | Type1 | Inactive | DFGin | 7.2128 | 14.5852 | BLAminus | -154.63, 179.57 | 55.91, 54.1 | -74.79, -3.2 | 274.96, 68.76 | -58.48, -41.04 | in-out | in | 7.4173 | Saltbr-out | 4.8105 | HRD-out | -96.67, 103.01 | -67.39, -41.62 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.141 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -162.98, 72.34 | APE9-dihe-in | -137.73, 148.36 | APE8-dihe-in | -71.99, 141.14 | APE8-rot-na | 343.8 | APE67-dihe-in | -63.34, -38.73 | -70.52, -42.38 | APE12-dist-na | 13.0181 | APE11-dist-na | 9.4081 | APE10-dist-na | 7.3004 | APE9-dist-in | 6.8677 | None | PTR656 | PTR656 | XRAY | 3.75 | 0.216 | 0.238 | A | 312.0 | 285.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8h75 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8H75B | P21802 | 467 | 764 | 821.0 | KX0:1001 | Type1 | Inactive | DFGin | 7.1136 | 15.3212 | BLAminus | -140.03, -170.55 | 50.75, 50.66 | -73.91, -10.21 | 273.73, 91.58 | -58.96, -39.4 | in-out | in | 7.4683 | Saltbr-out | 4.4362 | HRD-in | -64.7, -43.07 | 75.93, -2.73 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.3826 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -63.7, -40.57 | APE9-dihe-in | -143.97, 156.51 | APE8-dihe-in | -61.01, 137.3 | APE8-rot-na | 23.2 | APE67-dihe-in | -61.01, -38.56 | -64.05, -38.82 | APE12-dist-na | 14.0921 | APE11-dist-na | 11.2874 | APE10-dist-na | 7.4456 | APE9-dist-in | 5.7379 | None | PTR656 | PTR656 | XRAY | 3.75 | 0.216 | 0.238 | B | 312.0 | 283.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 8h75 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8H75C | P21802 | 467 | 763 | 821.0 | KX0:1001 | Type1 | Inactive | DFGin | 6.4145 | 13.9419 | BLAminus | -139.77, -171.25 | 51.94, 53.82 | -68.52, 7.4 | 288.78, 82.18 | -59.71, -35.71 | in-in | in | 7.7631 | Saltbr-in | 2.5787 | HRD-in | -64.69, -38.41 | 67.2, 3.13 | in-out-out | SNCioo | out-out | ActLoopNT-out | 3.7885 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -86.06, 23.54 | APE9-dihe-in | -123.01, 141.76 | APE8-dihe-in | -64.83, 140.92 | APE8-rot-na | 351.7 | APE67-dihe-in | -63.43, -39.45 | -65.53, -40.64 | APE12-dist-na | 10.7845 | APE11-dist-na | 10.9436 | APE10-dist-na | 7.5138 | APE9-dist-in | 5.3824 | None | PTR656 | PTR656 | XRAY | 3.75 | 0.216 | 0.238 | C | 312.0 | 275.0 | 22 | 30 | 24 | 6 | [[481, 759]] | 1.0 | 8h75 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8H75D | P21802 | 467 | 764 | 821.0 | KX0:1001 | Type1 | Inactive | DFGin | 6.7191 | 14.0063 | BLAminus | -145.79, -169.72 | 52.31, 64.06 | -85.42, 2.67 | 285.45, 103.44 | -59.5, -38.29 | in-out | in | 7.6901 | Saltbr-out | 4.3568 | HRD-in | -66.94, -45.53 | 78.8, 0.63 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.389 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 55.78, 41.43 | APE9-dihe-in | -144.13, 151.96 | APE8-dihe-in | -70.01, 128.38 | APE8-rot-na | 29.85 | APE67-dihe-in | -54.94, -35.54 | -65.88, -42.6 | APE12-dist-na | 10.9944 | APE11-dist-na | 11.0526 | APE10-dist-na | 8.8294 | APE9-dist-in | 5.7588 | None | PTR656 | PTR656 | XRAY | 3.75 | 0.216 | 0.238 | D | 312.0 | 277.0 | 21 | 30 | 26 | 4 | [[481, 759]] | 1.0 | 8h75 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|