| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | JAK1-12 | JAK1_MOUSE | 7T6FA | P52332 | 32 | 1153 | 1153.0 | ADN:61201,ADP:61202 | Allosteric,ATPlike | Inactive | DFGin | 6.8989 | 13.8131 | None | -86.13, -125.98 | -78.37, 170.67 | -132.74, 42.36 | 300.4, 95.7 | -63.52, -44.16 | in-out | in | 8.2656 | Saltbr-out | 5.3454 | HRD-in | -74.55, -24.53 | 68.9, -7.15 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.3664 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -74.97, -30.61 | APE9-dihe-in | -69.86, 145.09 | APE8-dihe-in | -65.5, 154.45 | APE8-rot-na | 337.81 | APE67-dihe-in | -111.81, 34.03 | -69.03, -47.03 | APE12-dist-na | 13.0701 | APE11-dist-na | 13.989 | APE10-dist-na | 8.6737 | APE9-dist-in | 6.36 | None | None | None | EM | 3.6 | 999.0 | 999.0 | A | 1173.0 | 1043.0 | 23 | 31 | 31 | 0 | [[582, 846], [874, 1150]] | 2.0 | 7t6f | Mus musculus | TYR_JAK1-12_MOUSE | TYR | 7.5e-59 | 499.6 | 3.0 | 260.0 | 516.0 | 1019 | 1020 | 1021 | 1023 | 1025 | 907 | 924 | 928 | 999 | 1001 | 1000 | 1002.0 | 1062 | 1050 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 1039 | 956 | Tyrosine-protein kinase JAK1 |
| TYR | JAK1-12 | JAK1_MOUSE | 7T6FB | P52332 | 32 | 1153 | 1153.0 | ADN:61201,ADP:61202 | Allosteric,ATPlike | Inactive | DFGin | 6.8984 | 13.8132 | None | -86.09, -125.95 | -78.45, 170.72 | -132.73, 42.29 | 300.45, 95.61 | -63.42, -44.2 | in-out | in | 8.2667 | Saltbr-out | 5.3471 | HRD-in | -74.65, -24.42 | 68.9, -7.11 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.3661 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -74.91, -30.65 | APE9-dihe-in | -69.79, 145.09 | APE8-dihe-in | -65.5, 154.47 | APE8-rot-na | 337.81 | APE67-dihe-in | -111.9, 34.05 | -69.03, -46.98 | APE12-dist-na | 13.0694 | APE11-dist-na | 13.9887 | APE10-dist-na | 8.6729 | APE9-dist-in | 6.3604 | None | None | None | EM | 3.6 | 999.0 | 999.0 | B | 1173.0 | 1043.0 | 23 | 31 | 31 | 0 | [[582, 846], [874, 1150]] | 2.0 | 7t6f | Mus musculus | TYR_JAK1-12_MOUSE | TYR | 7.5e-59 | 499.6 | 3.0 | 260.0 | 516.0 | 1019 | 1020 | 1021 | 1023 | 1025 | 907 | 924 | 928 | 999 | 1001 | 1000 | 1002.0 | 1062 | 1050 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 1039 | 956 | Tyrosine-protein kinase JAK1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | JAK1-12 | JAK1_MOUSE | 7T6FA | P52332 | 32 | 1153 | 1153.0 | ADN:61201,ADP:61202 | Allosteric,ATPlike | Inactive | DFGin | 6.8989 | 13.8131 | None | -86.13, -125.98 | -78.37, 170.67 | -132.74, 42.36 | 300.4, 95.7 | -63.52, -44.16 | in-out | in | 8.2656 | Saltbr-out | 5.3454 | HRD-in | -74.55, -24.53 | 68.9, -7.15 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.3664 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -74.97, -30.61 | APE9-dihe-in | -69.86, 145.09 | APE8-dihe-in | -65.5, 154.45 | APE8-rot-na | 337.81 | APE67-dihe-in | -111.81, 34.03 | -69.03, -47.03 | APE12-dist-na | 13.0701 | APE11-dist-na | 13.989 | APE10-dist-na | 8.6737 | APE9-dist-in | 6.36 | None | None | None | EM | 3.6 | 999.0 | 999.0 | A | 1173.0 | 1043.0 | 23 | 31 | 31 | 0 | [[582, 846], [874, 1150]] | 2.0 | 7t6f | Mus musculus | TYR_JAK1-12_MOUSE | TYR | 7.5e-59 | 499.6 | 3.0 | 260.0 | 516.0 | 1019 | 1020 | 1021 | 1023 | 1025 | 907 | 924 | 928 | 999 | 1001 | 1000 | 1002.0 | 1062 | 1050 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 1039 | 956 | Tyrosine-protein kinase JAK1 |
| TYR | JAK1-12 | JAK1_MOUSE | 7T6FB | P52332 | 32 | 1153 | 1153.0 | ADN:61201,ADP:61202 | Allosteric,ATPlike | Inactive | DFGin | 6.8984 | 13.8132 | None | -86.09, -125.95 | -78.45, 170.72 | -132.73, 42.29 | 300.45, 95.61 | -63.42, -44.2 | in-out | in | 8.2667 | Saltbr-out | 5.3471 | HRD-in | -74.65, -24.42 | 68.9, -7.11 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.3661 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -74.91, -30.65 | APE9-dihe-in | -69.79, 145.09 | APE8-dihe-in | -65.5, 154.47 | APE8-rot-na | 337.81 | APE67-dihe-in | -111.9, 34.05 | -69.03, -46.98 | APE12-dist-na | 13.0694 | APE11-dist-na | 13.9887 | APE10-dist-na | 8.6729 | APE9-dist-in | 6.3604 | None | None | None | EM | 3.6 | 999.0 | 999.0 | B | 1173.0 | 1043.0 | 23 | 31 | 31 | 0 | [[582, 846], [874, 1150]] | 2.0 | 7t6f | Mus musculus | TYR_JAK1-12_MOUSE | TYR | 7.5e-59 | 499.6 | 3.0 | 260.0 | 516.0 | 1019 | 1020 | 1021 | 1023 | 1025 | 907 | 924 | 928 | 999 | 1001 | 1000 | 1002.0 | 1062 | 1050 | 1045 | 1044 | 1043 | 1042 | 1041 | 1040 | 1039 | 956 | Tyrosine-protein kinase JAK1 |