| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 7OZYAAA | P21802 | 467 | 762 | 821.0 | 47I:801 | Type1 | Inactive | DFGin | 6.6178 | 14.2181 | BLAminus | -128.08, -179.64 | 55.32, 74.91 | -83.11, 15.08 | 289.1, 82.71 | -52.3, -39.22 | in-in | in | 7.5351 | Saltbr-in | 2.859 | HRD-in | -77.89, -51.81 | 75.61, -0.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.984 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.13, 18.52 | APE9-dihe-in | -94.81, 128.18 | APE8-dihe-in | -53.28, 119.61 | APE8-rot-na | 329.84 | APE67-dihe-in | -69.21, -9.08 | -65.59, -32.88 | APE12-dist-na | 10.0982 | APE11-dist-na | 10.6282 | APE10-dist-na | 7.3477 | APE9-dist-in | 4.6628 | None | None | None | XRAY | 2.28 | 0.243 | 0.296 | AAA | 303.0 | 281.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 7ozy | TYR_FGFR2_HUMAN | TYR | 2.2e-104 | 354.3 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 7OZYBBB | P21802 | 467 | 762 | 821.0 | 47I:801 | Type1 | Inactive | DFGin | 6.5249 | 14.2215 | BLAminus | -125.86, 176.96 | 60.82, 78.39 | -85.84, 17.43 | 287.27, 80.93 | -50.81, -42.13 | in-in | in | 7.4108 | Saltbr-in | 2.9245 | HRD-in | -87.72, -51.8 | 77.6, -3.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8893 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.37, 16.38 | APE9-dihe-in | -94.48, 132.52 | APE8-dihe-in | -58.52, 125.58 | APE8-rot-na | 337.9 | APE67-dihe-in | -78.03, -12.35 | -66.5, -32.9 | APE12-dist-na | 9.9376 | APE11-dist-na | 10.8072 | APE10-dist-na | 7.34 | APE9-dist-in | 4.8253 | None | None | None | XRAY | 2.28 | 0.243 | 0.296 | BBB | 303.0 | 278.0 | 18 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 7ozy | TYR_FGFR2_HUMAN | TYR | 2.2e-104 | 354.3 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 7OZYAAA | P21802 | 467 | 762 | 821.0 | 47I:801 | Type1 | Inactive | DFGin | 6.6178 | 14.2181 | BLAminus | -128.08, -179.64 | 55.32, 74.91 | -83.11, 15.08 | 289.1, 82.71 | -52.3, -39.22 | in-in | in | 7.5351 | Saltbr-in | 2.859 | HRD-in | -77.89, -51.81 | 75.61, -0.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.984 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.13, 18.52 | APE9-dihe-in | -94.81, 128.18 | APE8-dihe-in | -53.28, 119.61 | APE8-rot-na | 329.84 | APE67-dihe-in | -69.21, -9.08 | -65.59, -32.88 | APE12-dist-na | 10.0982 | APE11-dist-na | 10.6282 | APE10-dist-na | 7.3477 | APE9-dist-in | 4.6628 | None | None | None | XRAY | 2.28 | 0.243 | 0.296 | AAA | 303.0 | 281.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 7ozy | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.2e-104 | 354.3 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 7OZYBBB | P21802 | 467 | 762 | 821.0 | 47I:801 | Type1 | Inactive | DFGin | 6.5249 | 14.2215 | BLAminus | -125.86, 176.96 | 60.82, 78.39 | -85.84, 17.43 | 287.27, 80.93 | -50.81, -42.13 | in-in | in | 7.4108 | Saltbr-in | 2.9245 | HRD-in | -87.72, -51.8 | 77.6, -3.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8893 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.37, 16.38 | APE9-dihe-in | -94.48, 132.52 | APE8-dihe-in | -58.52, 125.58 | APE8-rot-na | 337.9 | APE67-dihe-in | -78.03, -12.35 | -66.5, -32.9 | APE12-dist-na | 9.9376 | APE11-dist-na | 10.8072 | APE10-dist-na | 7.34 | APE9-dist-in | 4.8253 | None | None | None | XRAY | 2.28 | 0.243 | 0.296 | BBB | 303.0 | 278.0 | 18 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 7ozy | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.2e-104 | 354.3 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|