| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | MERTK | MERTK_HUMAN | 7DXLA | Q12866 | 575 | 863 | 999.0 | E56:901 | Type1 | Inactive | DFGin | 5.6926 | 12.9118 | BLBplus | -151.73, -179.85 | 59.55, 33.96 | -96.78, 141.17 | 48.03, 89.29 | 122.99, -141.2 | out-out | out | 14.4061 | Saltbr-out | 11.3261 | HRD-in | -82.78, -46.78 | 71.1, -14.98 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 170.94 | APE8-dihe-out | -84.62, 44.17 | APE8-rot-na | 34.04 | APE67-dihe-in | -61.75, -10.77 | -55.95, -44.38 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.7811 | I650M | None | None | XRAY | 3.146 | 0.259 | 0.302 | A | 296.0 | 261.0 | 28 | 30 | 13 | 17 | [[587, 856]] | 1.0 | 7dxl | TYR_MERTK_HUMAN | TYR | 3.3e-92 | 314.4 | 2.0 | 261.0 | 260.0 | 740 | 741 | 742 | 744 | 746 | 619 | 637 | 641 | 720 | 722 | 721 | 723.0 | 782 | 770 | 765 | 764 | 763 | 762 | 761 | 760 | 759 | 672 | Tyrosine-protein kinase Mer |
| TYR | MERTK | MERTK_HUMAN | 7DXLB | Q12866 | 575 | 863 | 999.0 | E56:901 | Type1 | Inactive | DFGin | 6.3942 | 12.8872 | BLBplus | -154.41, 174.83 | 65.7, 46.55 | -105.06, 151.5 | 29.62, 85.97 | 72.51, 999.0 | out-out | out | 13.8732 | Saltbr-out | 12.9375 | HRD-in | -88.29, -46.43 | 62.33, -8.53 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 12.68 | APE8-rot-na | 329.13 | APE67-dihe-in | -64.23, -9.78 | -52.42, -47.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | I650M | None | None | XRAY | 3.146 | 0.259 | 0.302 | B | 296.0 | 256.0 | 33 | 30 | 11 | 19 | [[587, 856]] | 1.0 | 7dxl | TYR_MERTK_HUMAN | TYR | 3.3e-92 | 314.4 | 2.0 | 261.0 | 260.0 | 740 | 741 | 742 | 744 | 746 | 619 | 637 | 641 | 720 | 722 | 721 | 723.0 | 782 | 770 | 765 | 764 | 763 | 762 | 761 | 760 | 759 | 672 | Tyrosine-protein kinase Mer |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | MERTK | MERTK_HUMAN | 7DXLA | Q12866 | 575 | 863 | 999.0 | E56:901 | Type1 | Inactive | DFGin | 5.6926 | 12.9118 | BLBplus | -151.73, -179.85 | 59.55, 33.96 | -96.78, 141.17 | 48.03, 89.29 | 122.99, -141.2 | out-out | out | 14.4061 | Saltbr-out | 11.3261 | HRD-in | -82.78, -46.78 | 71.1, -14.98 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 170.94 | APE8-dihe-out | -84.62, 44.17 | APE8-rot-na | 34.04 | APE67-dihe-in | -61.75, -10.77 | -55.95, -44.38 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.7811 | I650M | None | None | XRAY | 3.146 | 0.259 | 0.302 | A | 296.0 | 261.0 | 28 | 30 | 13 | 17 | [[587, 856]] | 1.0 | 7dxl | Homo sapiens | TYR_MERTK_HUMAN | TYR | 3.3e-92 | 314.4 | 2.0 | 261.0 | 260.0 | 740 | 741 | 742 | 744 | 746 | 619 | 637 | 641 | 720 | 722 | 721 | 723.0 | 782 | 770 | 765 | 764 | 763 | 762 | 761 | 760 | 759 | 672 | Tyrosine-protein kinase Mer |
| TYR | MERTK | MERTK_HUMAN | 7DXLB | Q12866 | 575 | 863 | 999.0 | E56:901 | Type1 | Inactive | DFGin | 6.3942 | 12.8872 | BLBplus | -154.41, 174.83 | 65.7, 46.55 | -105.06, 151.5 | 29.62, 85.97 | 72.51, 999.0 | out-out | out | 13.8732 | Saltbr-out | 12.9375 | HRD-in | -88.29, -46.43 | 62.33, -8.53 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 12.68 | APE8-rot-na | 329.13 | APE67-dihe-in | -64.23, -9.78 | -52.42, -47.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | I650M | None | None | XRAY | 3.146 | 0.259 | 0.302 | B | 296.0 | 256.0 | 33 | 30 | 11 | 19 | [[587, 856]] | 1.0 | 7dxl | Homo sapiens | TYR_MERTK_HUMAN | TYR | 3.3e-92 | 314.4 | 2.0 | 261.0 | 260.0 | 740 | 741 | 742 | 744 | 746 | 619 | 637 | 641 | 720 | 722 | 721 | 723.0 | 782 | 770 | 765 | 764 | 763 | 762 | 761 | 760 | 759 | 672 | Tyrosine-protein kinase Mer |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|