| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | DDR1 | DDR1_HUMAN | 6Y23A | Q08345 | 574 | 907 | 913.0 | No_ligand | No_ligand | Inactive | DFGinter | 10.153 | 7.3082 | None | -140.3, -158.95 | -155.89, 34.86 | -96.49, -19.82 | 306.08, 111.29 | -54.16, -38.8 | in-out | in | 7.4307 | Saltbr-out | 4.3029 | HRD-in | -69.02, -55.97 | 80.69, 2.43 | out-out-in | SNCooi | out-in | ActLoopNT-out | 17.5924 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -133.93, 116.48 | APE9-dihe-in | -127.74, 145.71 | APE8-dihe-in | -88.51, 68.54 | APE8-rot-na | 35.64 | APE67-dihe-in | -68.64, -17.14 | -58.48, -33.24 | APE12-dist-na | 999.0 | APE11-dist-na | 12.2476 | APE10-dist-na | 7.8804 | APE9-dist-in | 7.1756 | Y569F,Y586F | None | None | XRAY | 2.58 | 0.228 | 0.27 | A | 350.0 | 305.0 | 27 | 30 | 27 | 3 | [[610, 907]] | 1.0 | 6y23 | TYR_DDR1_HUMAN | TYR | 2.2e-92 | 315.0 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | DDR1 | DDR1_HUMAN | 6Y23B | Q08345 | 574 | 910 | 913.0 | No_ligand | No_ligand | Inactive | DFGinter | 10.177 | 7.4895 | None | -147.65, -164.17 | -143.7, 24.01 | -83.51, -17.89 | 309.63, 115.78 | -53.01, -42.7 | in-out | in | 7.401 | Saltbr-out | 4.5382 | HRD-in | -62.79, -53.56 | 80.0, -6.1 | out-out-none | SNCoon | out-none | ActLoopNT-out | 17.3965 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 122.54 | APE9-dihe-in | -139.37, 143.31 | APE8-dihe-in | -88.22, 70.91 | APE8-rot-na | 34.24 | APE67-dihe-in | -65.16, -14.5 | -56.89, -35.39 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 7.7904 | APE9-dist-in | 7.2448 | Y569F,Y586F | None | None | XRAY | 2.58 | 0.228 | 0.27 | B | 350.0 | 301.0 | 30 | 30 | 25 | 5 | [[610, 907]] | 1.0 | 6y23 | TYR_DDR1_HUMAN | TYR | 2.2e-92 | 315.0 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | DDR1 | DDR1_HUMAN | 6Y23C | Q08345 | 574 | 911 | 913.0 | No_ligand | No_ligand | Inactive | DFGinter | 10.3257 | 7.4236 | None | -131.36, -161.95 | -146.38, 29.72 | -92.15, -18.74 | 310.61, 115.72 | -49.18, -37.85 | in-out | in | 7.6029 | Saltbr-out | 5.0782 | HRD-in | -65.34, -54.8 | 81.25, 2.61 | out-out-none | SNCoon | out-none | ActLoopNT-out | 17.5183 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 131.97 | APE9-dihe-in | -138.28, 145.82 | APE8-dihe-in | -85.36, 72.32 | APE8-rot-na | 34.45 | APE67-dihe-in | -71.14, -17.59 | -62.42, -29.77 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 8.1079 | APE9-dist-in | 7.1112 | Y569F,Y586F | None | None | XRAY | 2.58 | 0.228 | 0.27 | C | 350.0 | 305.0 | 33 | 30 | 25 | 5 | [[610, 907]] | 1.0 | 6y23 | TYR_DDR1_HUMAN | TYR | 2.2e-92 | 315.0 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | DDR1 | DDR1_HUMAN | 6Y23A | Q08345 | 574 | 907 | 913.0 | No_ligand | No_ligand | Inactive | DFGinter | 10.153 | 7.3082 | None | -140.3, -158.95 | -155.89, 34.86 | -96.49, -19.82 | 306.08, 111.29 | -54.16, -38.8 | in-out | in | 7.4307 | Saltbr-out | 4.3029 | HRD-in | -69.02, -55.97 | 80.69, 2.43 | out-out-in | SNCooi | out-in | ActLoopNT-out | 17.5924 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -133.93, 116.48 | APE9-dihe-in | -127.74, 145.71 | APE8-dihe-in | -88.51, 68.54 | APE8-rot-na | 35.64 | APE67-dihe-in | -68.64, -17.14 | -58.48, -33.24 | APE12-dist-na | 999.0 | APE11-dist-na | 12.2476 | APE10-dist-na | 7.8804 | APE9-dist-in | 7.1756 | Y569F,Y586F | None | None | XRAY | 2.58 | 0.228 | 0.27 | A | 350.0 | 305.0 | 27 | 30 | 27 | 3 | [[610, 907]] | 1.0 | 6y23 | Homo sapiens | TYR_DDR1_HUMAN | TYR | 2.2e-92 | 315.0 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | DDR1 | DDR1_HUMAN | 6Y23B | Q08345 | 574 | 910 | 913.0 | No_ligand | No_ligand | Inactive | DFGinter | 10.177 | 7.4895 | None | -147.65, -164.17 | -143.7, 24.01 | -83.51, -17.89 | 309.63, 115.78 | -53.01, -42.7 | in-out | in | 7.401 | Saltbr-out | 4.5382 | HRD-in | -62.79, -53.56 | 80.0, -6.1 | out-out-none | SNCoon | out-none | ActLoopNT-out | 17.3965 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 122.54 | APE9-dihe-in | -139.37, 143.31 | APE8-dihe-in | -88.22, 70.91 | APE8-rot-na | 34.24 | APE67-dihe-in | -65.16, -14.5 | -56.89, -35.39 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 7.7904 | APE9-dist-in | 7.2448 | Y569F,Y586F | None | None | XRAY | 2.58 | 0.228 | 0.27 | B | 350.0 | 301.0 | 30 | 30 | 25 | 5 | [[610, 907]] | 1.0 | 6y23 | Homo sapiens | TYR_DDR1_HUMAN | TYR | 2.2e-92 | 315.0 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| TYR | DDR1 | DDR1_HUMAN | 6Y23C | Q08345 | 574 | 911 | 913.0 | No_ligand | No_ligand | Inactive | DFGinter | 10.3257 | 7.4236 | None | -131.36, -161.95 | -146.38, 29.72 | -92.15, -18.74 | 310.61, 115.72 | -49.18, -37.85 | in-out | in | 7.6029 | Saltbr-out | 5.0782 | HRD-in | -65.34, -54.8 | 81.25, 2.61 | out-out-none | SNCoon | out-none | ActLoopNT-out | 17.5183 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 131.97 | APE9-dihe-in | -138.28, 145.82 | APE8-dihe-in | -85.36, 72.32 | APE8-rot-na | 34.45 | APE67-dihe-in | -71.14, -17.59 | -62.42, -29.77 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 8.1079 | APE9-dist-in | 7.1112 | Y569F,Y586F | None | None | XRAY | 2.58 | 0.228 | 0.27 | C | 350.0 | 305.0 | 33 | 30 | 25 | 5 | [[610, 907]] | 1.0 | 6y23 | Homo sapiens | TYR_DDR1_HUMAN | TYR | 2.2e-92 | 315.0 | 1.0 | 260.0 | 260.0 | 783 | 784 | 785 | 787 | 789 | 655 | 672 | 676 | 763 | 765 | 764 | 766.0 | 825 | 813 | 808 | 807 | 806 | 805 | 804 | 803 | 802 | 702 | Epithelial discoidin domain-containing receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|