| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | TTBK2 | TTBK2_HUMAN | 6VRFA | Q6IQ55 | 9 | 298 | 1244.0 | ADP:301 | ATPlike | Active | DFGin | 5.3543 | 13.1161 | BLAminus | -121.29, 164.21 | 73.75, 82.24 | -97.72, 13.38 | 304.67, 116.94 | -64.06, -29.66 | in-in | in | 7.2137 | Saltbr-in | 2.7506 | HRD-in | -77.1, -49.95 | 73.69, -4.56 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8129 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.12, -30.06 | APE9-dihe-na | -84.65, -146.34 | APE8-dihe-in | -107.58, 129.44 | APE8-rot-in | 302.21 | APE67-dihe-in | -59.13, -37.2 | -56.28, -42.66 | APE12-dist-in | 11.1967 | APE11-dist-in | 11.3871 | APE10-dist-in | 5.4802 | APE9-dist-in | 3.7845 | None | None | None | XRAY | 1.5 | 0.175 | 0.209 | A | 299.0 | 287.0 | 3 | 34 | 34 | 0 | [[21, 282]] | 1.0 | 6vrf | CK1_TTBK2_HUMAN | CK1 | 7.7e-104 | 352.6 | 1.0 | 262.0 | 262.0 | 162 | 163 | 164 | 166 | 168 | 50 | 64 | 68 | 138 | 140 | 139 | 141.0 | 208 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 95 | Tau-tubulin kinase 2 |
| CK1 | TTBK2 | TTBK2_HUMAN | 6VRFB | Q6IQ55 | 9 | 298 | 1244.0 | ADP:301 | ATPlike | Active | DFGin | 5.4311 | 12.6951 | BLAminus | -121.38, 163.64 | 74.07, 85.5 | -102.64, 12.86 | 306.76, 116.33 | -62.94, -32.7 | in-in | in | 7.3455 | Saltbr-in | 2.8906 | HRD-in | -78.31, -51.54 | 73.55, 1.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8595 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -109.78, -23.36 | APE9-dihe-na | -86.88, -149.11 | APE8-dihe-in | -108.63, 128.02 | APE8-rot-in | 302.45 | APE67-dihe-in | -58.2, -36.14 | -56.96, -43.7 | APE12-dist-in | 11.0394 | APE11-dist-in | 11.2442 | APE10-dist-in | 5.3369 | APE9-dist-in | 3.7117 | None | None | None | XRAY | 1.5 | 0.175 | 0.209 | B | 299.0 | 287.0 | 3 | 34 | 34 | 0 | [[21, 282]] | 1.0 | 6vrf | CK1_TTBK2_HUMAN | CK1 | 7.7e-104 | 352.6 | 1.0 | 262.0 | 262.0 | 162 | 163 | 164 | 166 | 168 | 50 | 64 | 68 | 138 | 140 | 139 | 141.0 | 208 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 95 | Tau-tubulin kinase 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | TTBK2 | TTBK2_HUMAN | 6VRFA | Q6IQ55 | 9 | 298 | 1244.0 | ADP:301 | ATPlike | Active | DFGin | 5.3543 | 13.1161 | BLAminus | -121.29, 164.21 | 73.75, 82.24 | -97.72, 13.38 | 304.67, 116.94 | -64.06, -29.66 | in-in | in | 7.2137 | Saltbr-in | 2.7506 | HRD-in | -77.1, -49.95 | 73.69, -4.56 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8129 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.12, -30.06 | APE9-dihe-na | -84.65, -146.34 | APE8-dihe-in | -107.58, 129.44 | APE8-rot-in | 302.21 | APE67-dihe-in | -59.13, -37.2 | -56.28, -42.66 | APE12-dist-in | 11.1967 | APE11-dist-in | 11.3871 | APE10-dist-in | 5.4802 | APE9-dist-in | 3.7845 | None | None | None | XRAY | 1.5 | 0.175 | 0.209 | A | 299.0 | 287.0 | 3 | 34 | 34 | 0 | [[21, 282]] | 1.0 | 6vrf | Homo sapiens | CK1_TTBK2_HUMAN | CK1 | 7.7e-104 | 352.6 | 1.0 | 262.0 | 262.0 | 162 | 163 | 164 | 166 | 168 | 50 | 64 | 68 | 138 | 140 | 139 | 141.0 | 208 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 95 | Tau-tubulin kinase 2 |
| CK1 | TTBK2 | TTBK2_HUMAN | 6VRFB | Q6IQ55 | 9 | 298 | 1244.0 | ADP:301 | ATPlike | Active | DFGin | 5.4311 | 12.6951 | BLAminus | -121.38, 163.64 | 74.07, 85.5 | -102.64, 12.86 | 306.76, 116.33 | -62.94, -32.7 | in-in | in | 7.3455 | Saltbr-in | 2.8906 | HRD-in | -78.31, -51.54 | 73.55, 1.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8595 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -109.78, -23.36 | APE9-dihe-na | -86.88, -149.11 | APE8-dihe-in | -108.63, 128.02 | APE8-rot-in | 302.45 | APE67-dihe-in | -58.2, -36.14 | -56.96, -43.7 | APE12-dist-in | 11.0394 | APE11-dist-in | 11.2442 | APE10-dist-in | 5.3369 | APE9-dist-in | 3.7117 | None | None | None | XRAY | 1.5 | 0.175 | 0.209 | B | 299.0 | 287.0 | 3 | 34 | 34 | 0 | [[21, 282]] | 1.0 | 6vrf | Homo sapiens | CK1_TTBK2_HUMAN | CK1 | 7.7e-104 | 352.6 | 1.0 | 262.0 | 262.0 | 162 | 163 | 164 | 166 | 168 | 50 | 64 | 68 | 138 | 140 | 139 | 141.0 | 208 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 95 | Tau-tubulin kinase 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|