| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | TTBK2 | TTBK2_HUMAN | 6U0KA | Q6IQ55 | 8 | 298 | 1244.0 | DTQ:302 | Type1 | Active | DFGin | 5.4455 | 13.0064 | BLAminus | -119.74, 158.68 | 65.44, 93.77 | -97.5, 16.58 | 303.39, 115.2 | -64.55, -24.48 | in-in | in | 7.3634 | Saltbr-in | 2.6861 | HRD-in | -77.31, -47.61 | 69.33, 3.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8535 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.86, 126.44 | APE9-dihe-na | 120.4, -155.7 | APE8-dihe-in | -106.9, 129.29 | APE8-rot-in | 301.05 | APE67-dihe-in | -61.62, -36.39 | -57.04, -41.68 | APE12-dist-in | 11.6476 | APE11-dist-in | 11.5741 | APE10-dist-in | 6.085 | APE9-dist-in | 3.8654 | None | None | None | XRAY | 1.744 | 0.193 | 0.233 | A | 300.0 | 290.0 | 1 | 34 | 34 | 0 | [[21, 282]] | 1.0 | 6u0k | CK1_TTBK2_HUMAN | CK1 | 7.8e-104 | 352.6 | 1.0 | 262.0 | 262.0 | 162 | 163 | 164 | 166 | 168 | 50 | 64 | 68 | 138 | 140 | 139 | 141.0 | 208 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 95 | Tau-tubulin kinase 2 |
| CK1 | TTBK2 | TTBK2_HUMAN | 6U0KB | Q6IQ55 | 8 | 299 | 1244.0 | DTQ:303 | Type1 | Active | DFGin | 5.539 | 12.9635 | BLAminus | -121.87, 159.25 | 66.65, 95.14 | -97.46, 15.84 | 302.12, 119.42 | -64.27, -23.46 | in-in | in | 7.473 | Saltbr-in | 2.6919 | HRD-in | -78.29, -47.84 | 69.94, 2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.843 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.42, 128.32 | APE9-dihe-na | 118.19, -156.28 | APE8-dihe-in | -104.4, 132.63 | APE8-rot-in | 299.38 | APE67-dihe-in | -60.41, -36.62 | -56.84, -43.97 | APE12-dist-in | 11.7517 | APE11-dist-in | 11.6488 | APE10-dist-in | 6.2643 | APE9-dist-in | 3.7387 | None | None | None | XRAY | 1.744 | 0.193 | 0.233 | B | 300.0 | 292.0 | 0 | 34 | 34 | 0 | [[21, 282]] | 1.0 | 6u0k | CK1_TTBK2_HUMAN | CK1 | 7.8e-104 | 352.6 | 1.0 | 262.0 | 262.0 | 162 | 163 | 164 | 166 | 168 | 50 | 64 | 68 | 138 | 140 | 139 | 141.0 | 208 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 95 | Tau-tubulin kinase 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | TTBK2 | TTBK2_HUMAN | 6U0KA | Q6IQ55 | 8 | 298 | 1244.0 | DTQ:302 | Type1 | Active | DFGin | 5.4455 | 13.0064 | BLAminus | -119.74, 158.68 | 65.44, 93.77 | -97.5, 16.58 | 303.39, 115.2 | -64.55, -24.48 | in-in | in | 7.3634 | Saltbr-in | 2.6861 | HRD-in | -77.31, -47.61 | 69.33, 3.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8535 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.86, 126.44 | APE9-dihe-na | 120.4, -155.7 | APE8-dihe-in | -106.9, 129.29 | APE8-rot-in | 301.05 | APE67-dihe-in | -61.62, -36.39 | -57.04, -41.68 | APE12-dist-in | 11.6476 | APE11-dist-in | 11.5741 | APE10-dist-in | 6.085 | APE9-dist-in | 3.8654 | None | None | None | XRAY | 1.744 | 0.193 | 0.233 | A | 300.0 | 290.0 | 1 | 34 | 34 | 0 | [[21, 282]] | 1.0 | 6u0k | Homo sapiens | CK1_TTBK2_HUMAN | CK1 | 7.8e-104 | 352.6 | 1.0 | 262.0 | 262.0 | 162 | 163 | 164 | 166 | 168 | 50 | 64 | 68 | 138 | 140 | 139 | 141.0 | 208 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 95 | Tau-tubulin kinase 2 |
| CK1 | TTBK2 | TTBK2_HUMAN | 6U0KB | Q6IQ55 | 8 | 299 | 1244.0 | DTQ:303 | Type1 | Active | DFGin | 5.539 | 12.9635 | BLAminus | -121.87, 159.25 | 66.65, 95.14 | -97.46, 15.84 | 302.12, 119.42 | -64.27, -23.46 | in-in | in | 7.473 | Saltbr-in | 2.6919 | HRD-in | -78.29, -47.84 | 69.94, 2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.843 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.42, 128.32 | APE9-dihe-na | 118.19, -156.28 | APE8-dihe-in | -104.4, 132.63 | APE8-rot-in | 299.38 | APE67-dihe-in | -60.41, -36.62 | -56.84, -43.97 | APE12-dist-in | 11.7517 | APE11-dist-in | 11.6488 | APE10-dist-in | 6.2643 | APE9-dist-in | 3.7387 | None | None | None | XRAY | 1.744 | 0.193 | 0.233 | B | 300.0 | 292.0 | 0 | 34 | 34 | 0 | [[21, 282]] | 1.0 | 6u0k | Homo sapiens | CK1_TTBK2_HUMAN | CK1 | 7.8e-104 | 352.6 | 1.0 | 262.0 | 262.0 | 162 | 163 | 164 | 166 | 168 | 50 | 64 | 68 | 138 | 140 | 139 | 141.0 | 208 | 196 | 191 | 190 | 189 | 188 | 187 | 186 | 185 | 95 | Tau-tubulin kinase 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|